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HUS1500018I1 - A Bruton-féle tirozin-kináz inhibitorai - Google Patents

A Bruton-féle tirozin-kináz inhibitorai

Info

Publication number
HUS1500018I1
HUS1500018I1 HUS1500018C HUS1500018C HUS1500018I1 HU S1500018 I1 HUS1500018 I1 HU S1500018I1 HU S1500018 C HUS1500018 C HU S1500018C HU S1500018 C HUS1500018 C HU S1500018C HU S1500018 I1 HUS1500018 I1 HU S1500018I1
Authority
HU
Hungary
Prior art keywords
disclosed
inhibitors
bruton
tyrosine kinase
compounds
Prior art date
Application number
HUS1500018C
Other languages
English (en)
Original Assignee
Pharmacyclics Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39225888&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUS1500018(I1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pharmacyclics Llc filed Critical Pharmacyclics Llc
Publication of HUS1500018I1 publication Critical patent/HUS1500018I1/hu

Links

Classifications

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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52Purines, e.g. adenine
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K39/3955Antibodies; Immunoglobulins; Immune serum, e.g. antilymphocytic serum against materials from animals against proteinaceous materials, e.g. enzymes, hormones, lymphokines
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2887Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against CD20
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Reproductive Health (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Mycology (AREA)
  • Microbiology (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pain & Pain Management (AREA)
HUS1500018C 2006-09-22 2015-04-08 A Bruton-féle tirozin-kináz inhibitorai HUS1500018I1 (hu)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US82672006P 2006-09-22 2006-09-22
US82859006P 2006-10-06 2006-10-06
EP10155834A EP2201840B1 (en) 2006-09-22 2006-12-28 Inhibitors of Bruton's Tyrosine Kinase
EP06850039.6A EP2081435B1 (en) 2006-09-22 2006-12-28 Inhibitors of bruton's tyrosine kinase

Publications (1)

Publication Number Publication Date
HUS1500018I1 true HUS1500018I1 (hu) 2017-10-30

Family

ID=39225888

Family Applications (10)

Application Number Title Priority Date Filing Date
HUE12166302A HUE036897T2 (hu) 2006-09-22 2006-12-28 Bruton tirozin kináz inhibitorok
HUE12166295A HUE028086T2 (hu) 2006-09-22 2006-12-28 Bruton tirozin-kináz gátlók
HUE12166301A HUE025459T2 (hu) 2006-09-22 2006-12-28 A Bruton-féle tirozin-kináz inhibitorai
HUE12166300A HUE033182T2 (hu) 2006-09-22 2006-12-28 Bruton tirozinkináz inhibitorok
HUE12166305A HUE028712T2 (hu) 2006-09-22 2006-12-28 Bruton tirozinkináz inhibitorok
HUE12166298A HUE031334T2 (hu) 2006-09-22 2006-12-28 Bruton-tirozinkináz inhibitorok
HUE06850039A HUE029095T2 (hu) 2006-09-22 2006-12-28 BRUTON tirozin kináz inhibitorok
HUS1500018C HUS1500018I1 (hu) 2006-09-22 2015-04-08 A Bruton-féle tirozin-kináz inhibitorai
HUS1600049C HUS1600049I1 (hu) 2006-09-22 2016-11-23 Bruton tirozinkináz inhibitorok
HUS1700012C HUS1700012I1 (hu) 2006-09-22 2017-03-24 Bruton-tirozinkináz inhibitorok

Family Applications Before (7)

Application Number Title Priority Date Filing Date
HUE12166302A HUE036897T2 (hu) 2006-09-22 2006-12-28 Bruton tirozin kináz inhibitorok
HUE12166295A HUE028086T2 (hu) 2006-09-22 2006-12-28 Bruton tirozin-kináz gátlók
HUE12166301A HUE025459T2 (hu) 2006-09-22 2006-12-28 A Bruton-féle tirozin-kináz inhibitorai
HUE12166300A HUE033182T2 (hu) 2006-09-22 2006-12-28 Bruton tirozinkináz inhibitorok
HUE12166305A HUE028712T2 (hu) 2006-09-22 2006-12-28 Bruton tirozinkináz inhibitorok
HUE12166298A HUE031334T2 (hu) 2006-09-22 2006-12-28 Bruton-tirozinkináz inhibitorok
HUE06850039A HUE029095T2 (hu) 2006-09-22 2006-12-28 BRUTON tirozin kináz inhibitorok

Family Applications After (2)

Application Number Title Priority Date Filing Date
HUS1600049C HUS1600049I1 (hu) 2006-09-22 2016-11-23 Bruton tirozinkináz inhibitorok
HUS1700012C HUS1700012I1 (hu) 2006-09-22 2017-03-24 Bruton-tirozinkináz inhibitorok

Country Status (28)

Country Link
US (49) US7514444B2 (hu)
EP (11) EP2526934B1 (hu)
JP (4) JP4934197B2 (hu)
KR (4) KR101479913B1 (hu)
CN (4) CN101805341B (hu)
AT (1) ATE531263T1 (hu)
AU (2) AU2006348662B8 (hu)
BE (1) BE2015C016I2 (hu)
BR (2) BRPI0622277A2 (hu)
CA (3) CA3180977A1 (hu)
CY (11) CY1112513T1 (hu)
DK (7) DK2081435T3 (hu)
EA (3) EA018573B1 (hu)
ES (8) ES2537399T3 (hu)
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