MA63498A1 - Formes posologiques orales d'ibrutinib - Google Patents
Formes posologiques orales d'ibrutinibInfo
- Publication number
- MA63498A1 MA63498A1 MA63498A MA63498A MA63498A1 MA 63498 A1 MA63498 A1 MA 63498A1 MA 63498 A MA63498 A MA 63498A MA 63498 A MA63498 A MA 63498A MA 63498 A1 MA63498 A1 MA 63498A1
- Authority
- MA
- Morocco
- Prior art keywords
- ibrutinib
- dosage forms
- oral dosage
- acidifying agent
- cancers
- Prior art date
Links
- 239000002177 L01XE27 - Ibrutinib Substances 0.000 title abstract 4
- XYFPWWZEPKGCCK-GOSISDBHSA-N ibrutinib Chemical compound C1=2C(N)=NC=NC=2N([C@H]2CN(CCC2)C(=O)C=C)N=C1C(C=C1)=CC=C1OC1=CC=CC=C1 XYFPWWZEPKGCCK-GOSISDBHSA-N 0.000 title abstract 4
- 229960001507 ibrutinib Drugs 0.000 title abstract 4
- 239000006186 oral dosage form Substances 0.000 title abstract 2
- 239000002552 dosage form Substances 0.000 abstract 3
- 239000002535 acidifier Substances 0.000 abstract 2
- IXPNQXFRVYWDDI-UHFFFAOYSA-N 1-methyl-2,4-dioxo-1,3-diazinane-5-carboximidamide Chemical compound CN1CC(C(N)=N)C(=O)NC1=O IXPNQXFRVYWDDI-UHFFFAOYSA-N 0.000 abstract 1
- 208000009329 Graft vs Host Disease Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 239000011230 binding agent Substances 0.000 abstract 1
- 239000007884 disintegrant Substances 0.000 abstract 1
- 239000000945 filler Substances 0.000 abstract 1
- 208000024908 graft versus host disease Diseases 0.000 abstract 1
- 201000005787 hematologic cancer Diseases 0.000 abstract 1
- 208000024200 hematopoietic and lymphoid system neoplasm Diseases 0.000 abstract 1
- 239000000314 lubricant Substances 0.000 abstract 1
- 235000010413 sodium alginate Nutrition 0.000 abstract 1
- 229940005550 sodium alginate Drugs 0.000 abstract 1
- 239000000661 sodium alginate Substances 0.000 abstract 1
- 239000004094 surface-active agent Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/539—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines having two or more oxygen atoms in the same ring, e.g. dioxazines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/485—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Formes posologiques orales stables et biodisponibles d'ibrutinib, les formes posologiques comprenant de l'ibrutinib et un agent acidifiant. Les formes posologiques peuvent en outre comprendre un liant, tel que de l'alginate de sodium, un tensioactif, un lubrifiant, une charge et/ou un délitant. L'invention concerne également des procédés de traitement de cancers, en particulier de cancers du sang, et la maladie du greffon contre l'hôte comprenant l'administration à un patient qui a besoin d'une forme posologique comprenant de l'ibrutinib et un agent acidifiant.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/US2021/036712 WO2022260667A1 (fr) | 2021-06-10 | 2021-06-10 | Formes posologiques orales d'ibrutinib |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MA63498A1 true MA63498A1 (fr) | 2024-07-31 |
Family
ID=76731098
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MA63498A MA63498A1 (fr) | 2021-06-10 | 2021-06-10 | Formes posologiques orales d'ibrutinib |
Country Status (3)
| Country | Link |
|---|---|
| MA (1) | MA63498A1 (fr) |
| TN (1) | TN2023000295A1 (fr) |
| WO (1) | WO2022260667A1 (fr) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN117064862B (zh) * | 2023-04-10 | 2025-12-19 | 山东新时代药业有限公司 | 一种伊布替尼肠溶片及其制备方法 |
Citations (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012087257A2 (fr) * | 2010-12-20 | 2012-06-28 | Mahmut Bilgic | Forme galénique orale contenant de l'imatinib et production de ladite forme galénique orale |
| WO2016105582A1 (fr) * | 2014-12-24 | 2016-06-30 | Nunn Philip A | Compositions pour administration de médicaments iléo-jéjunal. |
| WO2016141068A1 (fr) * | 2015-03-03 | 2016-09-09 | Pharmacyclics Llc | Formulations pharmaceutiques d'inhibiteur de la tyrosine kinase de bruton |
| WO2017174044A1 (fr) * | 2016-04-06 | 2017-10-12 | Zentiva, K.S. | Formes solides d'ibrutinib |
| WO2018033941A2 (fr) * | 2016-08-19 | 2018-02-22 | Cipla Limited | Compositions pharmaceutiques à base d'ibrutinib |
| CN111000806A (zh) * | 2018-10-07 | 2020-04-14 | 威海云睿信息科技有限公司 | 一种依鲁替尼片剂组合物 |
| US20200171036A1 (en) * | 2015-04-06 | 2020-06-04 | Janssen Pharmaceutica Nv | Compositions Containing Ibrutinib |
| KR20200127888A (ko) * | 2019-05-03 | 2020-11-11 | 보로노이 주식회사 | 이브루티닙 또는 이의 약학적으로 허용가능한 염을 포함하는 고형 제제 형태의 경구용 약학 조성물 및 이의 제조방법 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2585902T3 (es) | 2006-09-22 | 2016-10-10 | Pharmacyclics Llc | Inhibidores de tirosina cinasa de Bruton |
| BR112014030424A8 (pt) | 2012-06-04 | 2017-07-11 | Pharmacyclics Inc | Formas cristalinas de um inibidor de quinase de tirosina de bruton |
| CN103694241A (zh) | 2013-11-27 | 2014-04-02 | 苏州晶云药物科技有限公司 | Pci-32765的新晶型a及其制备方法 |
-
2021
- 2021-06-10 TN TNP/2023/000295A patent/TN2023000295A1/en unknown
- 2021-06-10 MA MA63498A patent/MA63498A1/fr unknown
- 2021-06-10 WO PCT/US2021/036712 patent/WO2022260667A1/fr not_active Ceased
Patent Citations (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2012087257A2 (fr) * | 2010-12-20 | 2012-06-28 | Mahmut Bilgic | Forme galénique orale contenant de l'imatinib et production de ladite forme galénique orale |
| WO2016105582A1 (fr) * | 2014-12-24 | 2016-06-30 | Nunn Philip A | Compositions pour administration de médicaments iléo-jéjunal. |
| WO2016141068A1 (fr) * | 2015-03-03 | 2016-09-09 | Pharmacyclics Llc | Formulations pharmaceutiques d'inhibiteur de la tyrosine kinase de bruton |
| US20170258729A1 (en) * | 2015-03-03 | 2017-09-14 | Pharmacyclics Llc | Pharmaceutical Formulations of a Bruton's Tyrosine Kinase Inhibitor |
| US20200171036A1 (en) * | 2015-04-06 | 2020-06-04 | Janssen Pharmaceutica Nv | Compositions Containing Ibrutinib |
| WO2017174044A1 (fr) * | 2016-04-06 | 2017-10-12 | Zentiva, K.S. | Formes solides d'ibrutinib |
| WO2018033941A2 (fr) * | 2016-08-19 | 2018-02-22 | Cipla Limited | Compositions pharmaceutiques à base d'ibrutinib |
| CN111000806A (zh) * | 2018-10-07 | 2020-04-14 | 威海云睿信息科技有限公司 | 一种依鲁替尼片剂组合物 |
| KR20200127888A (ko) * | 2019-05-03 | 2020-11-11 | 보로노이 주식회사 | 이브루티닙 또는 이의 약학적으로 허용가능한 염을 포함하는 고형 제제 형태의 경구용 약학 조성물 및 이의 제조방법 |
Also Published As
| Publication number | Publication date |
|---|---|
| TN2023000295A1 (en) | 2025-07-02 |
| WO2022260667A1 (fr) | 2022-12-15 |
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