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EE03608B1 - Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid - Google Patents

Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid

Info

Publication number
EE03608B1
EE03608B1 EE9700315A EE9700315A EE03608B1 EE 03608 B1 EE03608 B1 EE 03608B1 EE 9700315 A EE9700315 A EE 9700315A EE 9700315 A EE9700315 A EE 9700315A EE 03608 B1 EE03608 B1 EE 03608B1
Authority
EE
Estonia
Prior art keywords
taxoids
preparation
pharmaceutical compositions
compositions containing
pharmaceutical
Prior art date
Application number
EE9700315A
Other languages
English (en)
Estonian (et)
Other versions
EE9700315A (et
Inventor
Bouchard Herv
Bourzat Jean-Dominique
Commer�on Alain
Original Assignee
Rh�Ne-Poulenc Rorer S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9503545A external-priority patent/FR2732340B1/fr
Priority claimed from FR9515381A external-priority patent/FR2742754B1/fr
Application filed by Rh�Ne-Poulenc Rorer S.A. filed Critical Rh�Ne-Poulenc Rorer S.A.
Publication of EE9700315A publication Critical patent/EE9700315A/xx
Publication of EE03608B1 publication Critical patent/EE03608B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
EE9700315A 1995-03-27 1996-03-25 Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid EE03608B1 (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9503545A FR2732340B1 (fr) 1995-03-27 1995-03-27 Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
FR9515381A FR2742754B1 (fr) 1995-12-22 1995-12-22 Procede de preparation de taxoides
PCT/FR1996/000440 WO1996030355A1 (fr) 1995-03-27 1996-03-25 Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number Publication Date
EE9700315A EE9700315A (et) 1998-06-15
EE03608B1 true EE03608B1 (et) 2002-02-15

Family

ID=26231838

Family Applications (2)

Application Number Title Priority Date Filing Date
EE9700323A EE03609B1 (et) 1995-03-27 1996-03-25 Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid
EE9700315A EE03608B1 (et) 1995-03-27 1996-03-25 Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EE9700323A EE03609B1 (et) 1995-03-27 1996-03-25 Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid

Country Status (41)

Country Link
US (3) US5889043A (xx)
EP (2) EP0817779B1 (xx)
JP (2) JP2941951B2 (xx)
KR (2) KR100485309B1 (xx)
CN (2) CN1152870C (xx)
AP (2) AP753A (xx)
AR (1) AR001440A1 (xx)
AT (2) ATE185562T1 (xx)
AU (2) AU703278B2 (xx)
BG (2) BG63121B1 (xx)
BR (2) BR9607930A (xx)
CA (2) CA2214321C (xx)
CO (1) CO4700576A1 (xx)
CZ (2) CZ287326B6 (xx)
DE (2) DE69604653T2 (xx)
DK (2) DK0817779T3 (xx)
DZ (1) DZ2009A1 (xx)
EA (2) EA000567B1 (xx)
EE (2) EE03609B1 (xx)
ES (2) ES2140075T3 (xx)
GE (2) GEP20002211B (xx)
GR (2) GR3031526T3 (xx)
HU (2) HU223666B1 (xx)
IL (1) IL117636A (xx)
IS (2) IS2058B (xx)
MA (1) MA23823A1 (xx)
MY (1) MY121225A (xx)
NO (2) NO316379B1 (xx)
NZ (2) NZ304901A (xx)
OA (2) OA10513A (xx)
PE (1) PE51097A1 (xx)
PL (2) PL188284B1 (xx)
PT (1) PT817779E (xx)
RO (2) RO115878B1 (xx)
SK (2) SK281928B6 (xx)
TN (1) TNSN96043A1 (xx)
TR (2) TR199701042T1 (xx)
TW (1) TW394765B (xx)
UY (2) UY24192A1 (xx)
WO (2) WO1996030356A1 (xx)
ZA (1) ZA962399B (xx)

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US6495579B1 (en) 1996-12-02 2002-12-17 Angiotech Pharmaceuticals, Inc. Method for treating multiple sclerosis
US5811452A (en) * 1997-01-08 1998-09-22 The Research Foundation Of State University Of New York Taxoid reversal agents for drug-resistance in cancer chemotherapy and pharmaceutical compositions thereof
US7288665B1 (en) * 1997-08-18 2007-10-30 Florida State University Process for selective derivatization of taxanes
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EP0982027A1 (en) * 1998-08-17 2000-03-01 Aventis Pharma S.A. Taxoid derivatives for treating abnormal cell proliferation of the brain
US6346543B1 (en) * 1998-08-17 2002-02-12 Aventis Pharma S.A. Use of a taxoid to treat abnormal cell proliferation in the brain
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EP1020188A1 (en) * 1999-01-13 2000-07-19 Aventis Pharma S.A. New use of taxoid derivatives
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US6593334B1 (en) 2002-05-02 2003-07-15 The University Of North Carolina At Chapel Hill Camptothecin-taxoid conjugates as antimitotic and antitumor agents
ES2377318T3 (es) 2002-09-06 2012-03-26 Cerulean Pharma Inc. Polímeros a base de ciclodextrina para el suministro de los agentes terapéuticos enlazados covalentemente a ellos
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US7064980B2 (en) * 2003-09-17 2006-06-20 Sandisk Corporation Non-volatile memory and method with bit line coupled compensation
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HN2005000054A (es) 2004-02-13 2009-02-18 Florida State University Foundation Inc Taxanos sustituidos con esteres de ciclopentilo en c10
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WO2006088767A2 (en) * 2005-02-14 2006-08-24 Florida State University Research Foundation, Inc. C10 cyclopropyl ester substituted taxane compositions
US8263793B2 (en) * 2005-03-31 2012-09-11 Accord Healthcare Inc. Preparation of taxanes from 9-dihydro-13-acetylbaccatin III
EP1948669B1 (en) * 2005-11-04 2013-07-10 Accord Healthcare Inc. New methods for the preparation of taxanes using chiral auxiliaries
US7847111B2 (en) * 2006-06-19 2010-12-07 Canada Inc. Semi-synthetic route for the preparation of paclitaxel, docetaxel, and 10-deacetylbaccatin III from 9-dihydro-13-acetylbaccatin III
WO2008067403A2 (en) * 2006-11-28 2008-06-05 Encore Health Llc Presbyopia treatment by lens alteration
JP2010516625A (ja) 2007-01-24 2010-05-20 インサート セラピューティクス， インコーポレイテッド 制御された薬物送達のためのテザー基を有するポリマー−薬物コンジュゲート
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US8242166B2 (en) 2008-03-31 2012-08-14 Florida State University Research Foundation, Inc. C(10) ethyl ester and C(10) cyclopropyl ester substituted taxanes
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CN104650012A (zh) 2013-11-22 2015-05-27 天士力控股集团有限公司 一种紫杉烷类化合物
CN104086514A (zh) * 2014-06-19 2014-10-08 上海应用技术学院 紫杉醇衍生物及其制备方法
JP6841772B2 (ja) 2015-02-17 2021-03-10 エラスムス・ユニヴァーシティ・メディカル・センター・ロッテルダム 前立腺癌の処置におけるカバジタキセルの使用
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MX9102128A (es) 1990-11-23 1992-07-08 Rhone Poulenc Rorer Sa Derivados de taxano,procedimiento para su preparacion y composicion farmaceutica que los contiene
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Also Published As

Publication number Publication date
MA23823A1 (fr) 1996-10-01
AU703278B2 (en) 1999-03-25
CN1152870C (zh) 2004-06-09
IS4567A (is) 1997-09-23
NZ304900A (en) 1998-09-24
PL188987B1 (pl) 2005-05-31
SK130297A3 (en) 1998-03-04
AU5278096A (en) 1996-10-16
EA199700269A1 (ru) 1998-04-30
EA000567B1 (ru) 1999-12-29
EP0817780A1 (fr) 1998-01-14
HUP9801201A3 (en) 2000-12-28
UY24370A1 (es) 2001-10-25
RO115877B1 (ro) 2000-07-28
MX9706568A (es) 1997-11-29
WO1996030356A1 (fr) 1996-10-03
AP9701093A0 (en) 1997-10-31
KR100485309B1 (ko) 2005-10-12
ATE188471T1 (de) 2000-01-15
ZA962399B (en) 1996-10-01
NO316607B1 (no) 2004-03-08
IL117636A0 (en) 1996-07-23
EE9700315A (et) 1998-06-15
HU223666B1 (hu) 2004-11-29
HUP9801204A3 (en) 2000-12-28
CZ303297A3 (cs) 1998-01-14
OA10513A (fr) 2002-04-22
JPH11502531A (ja) 1999-03-02
AU5278196A (en) 1996-10-16
NZ304901A (en) 1998-12-23
GEP20002211B (en) 2000-08-25
HU223732B1 (hu) 2004-12-28
BR9607930A (pt) 1998-06-02
AU711227B2 (en) 1999-10-07
WO1996030355A1 (fr) 1996-10-03
ES2140075T3 (es) 2000-02-16
TR199701042T1 (xx) 1998-01-21
US6331635B1 (en) 2001-12-18
HUP9801204A1 (hu) 2000-05-28
EP0817779B1 (fr) 2000-01-05
MY121225A (en) 2006-01-28
IS4536A (is) 1997-07-31
PL322499A1 (en) 1998-02-02
BG63121B1 (bg) 2001-04-30
EA000709B1 (ru) 2000-02-28
BG101918A (en) 1998-10-30
PL188284B1 (pl) 2005-01-31
CO4700576A1 (es) 1998-12-29
ES2143187T3 (es) 2000-05-01
US6387946B1 (en) 2002-05-14
NO316379B1 (no) 2004-01-19
CA2214321C (fr) 2008-01-22
BR9607929A (pt) 1998-06-02
SK281927B6 (sk) 2001-09-11
TW394765B (en) 2000-06-21
CZ287468B6 (en) 2000-12-13
DE69606028D1 (de) 2000-02-10
SK130197A3 (en) 1998-04-08
PT817779E (pt) 2000-04-28
EE03609B1 (et) 2002-02-15
UY24192A1 (es) 1996-06-14
TNSN96043A1 (fr) 2005-03-15
DK0817779T3 (da) 2000-06-19
GR3032316T3 (en) 2000-04-27
NO973922L (no) 1997-08-26
IS2058B (is) 2005-10-14
SK281928B6 (sk) 2001-09-11
RO115878B1 (ro) 2000-07-28
ATE185562T1 (de) 1999-10-15
DE69606028T2 (de) 2000-08-10
EA199700270A1 (ru) 1998-02-26
KR19980703287A (ko) 1998-10-15
BG63009B1 (bg) 2001-01-31
EP0817779A1 (fr) 1998-01-14
AP753A (en) 1999-07-21
DZ2009A1 (fr) 2002-10-23
BG101917A (en) 1998-10-30
TR199701040T1 (xx) 1998-01-21
CN1179776A (zh) 1998-04-22
NO973922D0 (no) 1997-08-26
AP785A (en) 1999-11-26
CA2214319A1 (fr) 1996-10-03
EE9700323A (et) 1998-06-15
IL117636A (en) 2004-08-31
DE69604653T2 (de) 2000-05-31
GEP20002188B (en) 2000-07-25
AP9701090A0 (en) 1997-10-31
JP2941951B2 (ja) 1999-08-30
AR001440A1 (es) 1997-10-22
PL322465A1 (en) 1998-02-02
IS2056B (is) 2005-10-14
MX9706278A (es) 1997-10-31
HUP9801201A2 (hu) 2000-05-28
US20020038038A1 (en) 2002-03-28
EP0817780B1 (fr) 1999-10-13
GR3031526T3 (en) 2000-01-31
NO973923L (no) 1997-08-26
CZ303097A3 (cs) 1998-01-14
OA10514A (fr) 2002-04-22
PE51097A1 (es) 1997-12-22
NO973923D0 (no) 1997-08-26
CN1213042C (zh) 2005-08-03
CA2214319C (fr) 2004-02-17
DE69604653D1 (de) 1999-11-18
KR100297196B1 (ko) 2001-11-22
JPH11500141A (ja) 1999-01-06
US5889043A (en) 1999-03-30
JP3790826B2 (ja) 2006-06-28
CZ287326B6 (en) 2000-10-11
CN1179775A (zh) 1998-04-22
KR19980703357A (ko) 1998-10-15
DK0817780T3 (da) 2000-03-27
CA2214321A1 (fr) 1996-10-03

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