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DK1490062T3 - Glukokortikoidmimetika, fremgangsmåder til fremstilling deraf, farmaceutiske sammensætninger og anvendelser deraf - Google Patents

Glukokortikoidmimetika, fremgangsmåder til fremstilling deraf, farmaceutiske sammensætninger og anvendelser deraf

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Publication number
DK1490062T3
DK1490062T3 DK03714339T DK03714339T DK1490062T3 DK 1490062 T3 DK1490062 T3 DK 1490062T3 DK 03714339 T DK03714339 T DK 03714339T DK 03714339 T DK03714339 T DK 03714339T DK 1490062 T3 DK1490062 T3 DK 1490062T3
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DK
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Prior art keywords
preparation
methods
pharmaceutical compositions
glucocorticoid mimetics
glucocorticoid
Prior art date
Application number
DK03714339T
Other languages
English (en)
Inventor
Y Bekkali
R Betageri
Thomas A Gilmore
T M Kirrane
D Kuzmich
J Proudfoot
H Takahashi
D Thomson
Ji Wang
R Zindell
C Harcken
D Riether
Mario G Cardozo
Hossein Razavi
Original Assignee
Boehringer Ingelheim Pharma
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Publication of DK1490062T3 publication Critical patent/DK1490062T3/da

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    • C07D209/02Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12Radicals substituted by oxygen atoms
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    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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DK03714339T 2002-03-26 2003-03-21 Glukokortikoidmimetika, fremgangsmåder til fremstilling deraf, farmaceutiske sammensætninger og anvendelser deraf DK1490062T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US36775802P 2002-03-26 2002-03-26
US43181702P 2002-12-09 2002-12-09
US44240403P 2003-01-24 2003-01-24
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