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AR042199A1 - Composicion farmaceutica liquida que comprende una cantidad terapeuticamente eficaz de al menos un compuesto de 3,7 diazabiciclo (3,3,1) nonano, metodo de tratamiento y/o profilaxis de eventos anti-arritmicos en seres humanos y producto y/o forma de presentacion farmaceutica - Google Patents

Composicion farmaceutica liquida que comprende una cantidad terapeuticamente eficaz de al menos un compuesto de 3,7 diazabiciclo (3,3,1) nonano, metodo de tratamiento y/o profilaxis de eventos anti-arritmicos en seres humanos y producto y/o forma de presentacion farmaceutica

Info

Publication number
AR042199A1
AR042199A1 ARP030104235A ARP030104235A AR042199A1 AR 042199 A1 AR042199 A1 AR 042199A1 AR P030104235 A ARP030104235 A AR P030104235A AR P030104235 A ARP030104235 A AR P030104235A AR 042199 A1 AR042199 A1 AR 042199A1
Authority
AR
Argentina
Prior art keywords
products
treatment
pharmaceutical composition
events
arritmic
Prior art date
Application number
ARP030104235A
Other languages
English (en)
Inventor
Matthias Straub
Claus Rudolf Steimborn
Werner Cautreels
Johannes Wihelmus Catharine Maria Jansen
Vries Michiel De
Original Assignee
Solvay Pharm Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Gmbh filed Critical Solvay Pharm Gmbh
Publication of AR042199A1 publication Critical patent/AR042199A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4747Quinolines; Isoquinolines spiro-condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)

Abstract

Uso de 3,7-diazabiciclo[3,3,1]nonano, preferiblemente compuestos de 9,9-alquileno-3,7-diazabiciclo[3,3,1]nonano, y con mayor preferencia al uso de tedisamil, bertosamil y sus sales de adición de ácido y/o solvatos fisiológicamente aceptables, en la forma de una composición farmacéutica líquida para el tratamiento y/o profilaxis de eventos anti-arrítmicos en pacientes humanos, preferiblemente en la conversión de reciente proceso de fibrilación auricular o flúter auricular a ritmo sinusal normal en pacientes humanos. Métodos de tratamiento preferiblemente por administración en dos etapas y productos farmacéuticos.
ARP030104235A 2002-11-18 2003-11-17 Composicion farmaceutica liquida que comprende una cantidad terapeuticamente eficaz de al menos un compuesto de 3,7 diazabiciclo (3,3,1) nonano, metodo de tratamiento y/o profilaxis de eventos anti-arritmicos en seres humanos y producto y/o forma de presentacion farmaceutica AR042199A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US42679502P 2002-11-18 2002-11-18

Publications (1)

Publication Number Publication Date
AR042199A1 true AR042199A1 (es) 2005-06-15

Family

ID=32326429

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP030104235A AR042199A1 (es) 2002-11-18 2003-11-17 Composicion farmaceutica liquida que comprende una cantidad terapeuticamente eficaz de al menos un compuesto de 3,7 diazabiciclo (3,3,1) nonano, metodo de tratamiento y/o profilaxis de eventos anti-arritmicos en seres humanos y producto y/o forma de presentacion farmaceutica

Country Status (20)

Country Link
US (2) US7087620B2 (es)
EP (1) EP1565239B8 (es)
JP (1) JP2006510613A (es)
KR (1) KR101059330B1 (es)
CN (1) CN1726062A (es)
AR (1) AR042199A1 (es)
AT (1) ATE501758T1 (es)
AU (1) AU2003296580B8 (es)
BR (1) BR0316383A (es)
CA (1) CA2506083A1 (es)
DE (1) DE60336417D1 (es)
IL (1) IL168630A (es)
MX (1) MXPA05005344A (es)
NO (1) NO20053010L (es)
RU (1) RU2358732C2 (es)
SA (1) SA04250023B1 (es)
TW (1) TW200418468A (es)
UA (1) UA85546C2 (es)
WO (1) WO2004045591A2 (es)
ZA (1) ZA200504049B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW200418468A (en) * 2002-11-18 2004-10-01 Solvay Pharm Gmbh Liquid pharmaceutical formulations containing 3,7-diazabicyclo[3,3,1]nonane compounds and method of treatments relating to anti-arrhytmic events
CA2533492A1 (en) * 2003-07-21 2005-02-10 Solvay Pharmaceuticals Gmbh Use of 3,7-diazabicyclo[3,3,1]nonane compounds for the treatment and/or prophylaxis of anti-arrhythmic events in male human patients
US20050054667A1 (en) * 2003-07-21 2005-03-10 Solvay Pharmaceuticals Gmbh Method of treating or inhibiting anti-arrhythmic events in male human patients
CA2617519A1 (en) * 2005-08-23 2007-03-01 Astellas Pharma Inc. Agent for treating atrial fibrillation
EP2149370A1 (en) * 2008-07-31 2010-02-03 Neuroscienze Pharmaness S.C. A R.L. Diazabicyclic compounds and microemulsions thereof

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4550111A (en) * 1982-01-29 1985-10-29 Imperial Chemical Industries Plc Alkanolamine derivatives
DE3234697A1 (de) * 1982-09-18 1984-03-22 Kali-Chemie Pharma Gmbh, 3000 Hannover Neue diazabicyclo-(3,3,1)-nonane
PT88381B (pt) * 1987-09-09 1995-07-06 Kali Chemie Pharma Gmbh Processo para a preparacao de novos compostos 3,7-diazabiciclo{3,3,1} nonano, e de composicoes farmaceuticas que contem estes compostos
DE4019080A1 (de) * 1990-06-15 1991-12-19 Kali Chemie Pharma Gmbh Neue 3,7-diazabicycolo (3,3,1)nonan-verbindungen enthaltende arzneimittel
DE4139763A1 (de) * 1991-12-03 1993-06-09 Kali-Chemie Pharma Gmbh, 3000 Hannover, De Kristalline fumarsaure salze von 9,9-alkylen-3,7-diazabicyclononan-verbindungen und diese verbindungen enthaltende arzneimittel
DE4402933A1 (de) * 1994-02-01 1995-08-03 Kali Chemie Pharma Gmbh Neue 3-Benzoyl-3,7-diazabicyclo[3,3,1] nonan-Verbindungen enthaltende Arzneimittel
DE4402931A1 (de) * 1994-02-01 1995-08-03 Kali Chemie Pharma Gmbh Neue 3-Phenylsulfonyl-3,7-diazabicyclo[3,3,1] nonan-Verbindungen enthaltende Arzneimittel
US5576349A (en) * 1995-11-30 1996-11-19 The General Hospital Corporation Retionoic acid treatment of cardiac arrhythmia
US6026817A (en) * 1996-11-14 2000-02-22 Clemens; Anton H. Method of treating the syndrome of coronary heart disease risk factors in humans
SE9704709D0 (sv) * 1997-12-17 1997-12-17 Astra Ab Pharmaceutically active compounds
US6790463B2 (en) * 2001-03-30 2004-09-14 Robert F. Hofmann Uses of targeted oxidative therapeutic formulation in arteriosclerosis
DE10131217A1 (de) * 2001-06-28 2003-01-09 Solvay Pharm Gmbh 3-Phenyl-3,7-diazabicyclo 3,3,1 nonan-Verbindungen sowie Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
TW200418468A (en) * 2002-11-18 2004-10-01 Solvay Pharm Gmbh Liquid pharmaceutical formulations containing 3,7-diazabicyclo[3,3,1]nonane compounds and method of treatments relating to anti-arrhytmic events

Also Published As

Publication number Publication date
ZA200504049B (en) 2006-07-26
DE60336417D1 (de) 2011-04-28
AU2003296580B2 (en) 2010-02-18
KR20050116125A (ko) 2005-12-09
US20050261300A1 (en) 2005-11-24
WO2004045591A2 (en) 2004-06-03
BR0316383A (pt) 2005-10-04
KR101059330B1 (ko) 2011-08-24
CA2506083A1 (en) 2004-06-03
SA04250023B1 (ar) 2008-12-23
RU2005119280A (ru) 2006-03-20
WO2004045591A3 (en) 2004-07-22
US7087620B2 (en) 2006-08-08
IL168630A (en) 2013-08-29
EP1565239B1 (en) 2011-03-16
CN1726062A (zh) 2006-01-25
JP2006510613A (ja) 2006-03-30
UA85546C2 (en) 2009-02-10
ATE501758T1 (de) 2011-04-15
AU2003296580A1 (en) 2004-06-15
US20040152716A1 (en) 2004-08-05
MXPA05005344A (es) 2005-08-03
RU2358732C2 (ru) 2009-06-20
EP1565239B8 (en) 2011-06-22
AU2003296580B8 (en) 2010-03-18
TW200418468A (en) 2004-10-01
NO20053010L (no) 2005-06-20
EP1565239A2 (en) 2005-08-24

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