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MXPA05009985A - Ligandos de receptores de canabinoides. - Google Patents

Ligandos de receptores de canabinoides.

Info

Publication number
MXPA05009985A
MXPA05009985A MXPA05009985A MXPA05009985A MXPA05009985A MX PA05009985 A MXPA05009985 A MX PA05009985A MX PA05009985 A MXPA05009985 A MX PA05009985A MX PA05009985 A MXPA05009985 A MX PA05009985A MX PA05009985 A MXPA05009985 A MX PA05009985A
Authority
MX
Mexico
Prior art keywords
receptor ligands
cannabinoid receptor
compounds
disclosed
solvate
Prior art date
Application number
MXPA05009985A
Other languages
English (en)
Inventor
Neng-Yang Shin
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of MXPA05009985A publication Critical patent/MXPA05009985A/es

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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C07D213/80—Acids; Esters in position 3
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    • C07C317/22—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
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    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
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    • C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
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    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
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Abstract

Se describen compuestos de la formula I (ver formula I) un solvato o sal farmaceuticamente aceptable del compuesto, que exhiben actividad antinflamatoria e inmunomoduladora; ademas se describen composiciones farmaceuticas que contienen dichos compuestos.
MXPA05009985A 2003-03-20 2004-03-18 Ligandos de receptores de canabinoides. MXPA05009985A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US45626803P 2003-03-20 2003-03-20
PCT/US2004/008333 WO2004085385A2 (en) 2003-03-20 2004-03-18 Cannabinoid receptor ligands

Publications (1)

Publication Number Publication Date
MXPA05009985A true MXPA05009985A (es) 2005-11-04

Family

ID=33098100

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA05009985A MXPA05009985A (es) 2003-03-20 2004-03-18 Ligandos de receptores de canabinoides.

Country Status (9)

Country Link
US (1) US7642272B2 (es)
EP (1) EP1611090A2 (es)
JP (2) JP2006520795A (es)
CN (1) CN1761646A (es)
AR (1) AR043633A1 (es)
CA (1) CA2519401A1 (es)
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CN1761646A (zh) 2006-04-19
WO2004085385A2 (en) 2004-10-07
TW200505902A (en) 2005-02-16
WO2004085385A3 (en) 2004-11-25
JP2006520795A (ja) 2006-09-14
JP2007211017A (ja) 2007-08-23
EP1611090A2 (en) 2006-01-04
CA2519401A1 (en) 2004-10-07
US7642272B2 (en) 2010-01-05
US20040186148A1 (en) 2004-09-23

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