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UA86807C2 - ПОРОШКОВАЯ КОМПОЗИЦИЯ ДЛЯ ИНГАЛЯЦИИ, КОТОРАЯ СОДЕРЖИТ ЭНАНТИОМЕРНО ЧИСТЫЕ β-АГОНИСТЫ - Google Patents

ПОРОШКОВАЯ КОМПОЗИЦИЯ ДЛЯ ИНГАЛЯЦИИ, КОТОРАЯ СОДЕРЖИТ ЭНАНТИОМЕРНО ЧИСТЫЕ β-АГОНИСТЫ

Info

Publication number
UA86807C2
UA86807C2 UAA200612950A UAA200612950A UA86807C2 UA 86807 C2 UA86807 C2 UA 86807C2 UA A200612950 A UAA200612950 A UA A200612950A UA A200612950 A UAA200612950 A UA A200612950A UA 86807 C2 UA86807 C2 UA 86807C2
Authority
UA
Ukraine
Prior art keywords
agonists
enantiomerically pure
formulations containing
powder formulations
inhalation powder
Prior art date
Application number
UAA200612950A
Other languages
English (en)
Ukrainian (uk)
Inventor
Михаэль Трунк
Йорг Шиве
Original Assignee
Бёрингер Ингельхайм Интернациональ Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35058202&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA86807(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Бёрингер Ингельхайм Интернациональ Гмбх filed Critical Бёрингер Ингельхайм Интернациональ Гмбх
Publication of UA86807C2 publication Critical patent/UA86807C2/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0075Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/5381,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Otolaryngology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

В заявке описаны порошковые композиции для ингаляции, которые содержат энантиомерно чистые соединения общей формулы (1), (1)в которой остатки R, R, Rи Rмогут иметь указанные в формуле изобретения и описании значения, необязательно в виде их фармацевтически приемлемых кислотно-аддитивных солей, а также необязательно в соединении с фармацевтически приемлемым вспомогательным веществом, а также описаны способ их получения и их применения в качестве лекарственных средств, прежде всего в качестве лекарственных средств для лечения заболеваний дыхательных путей.
UAA200612950A 2004-05-14 2005-05-11 ПОРОШКОВАЯ КОМПОЗИЦИЯ ДЛЯ ИНГАЛЯЦИИ, КОТОРАЯ СОДЕРЖИТ ЭНАНТИОМЕРНО ЧИСТЫЕ β-АГОНИСТЫ UA86807C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004024451A DE102004024451A1 (de) 2004-05-14 2004-05-14 Pulverformulierungen für die Inhalation, die Enantiomerenreine Betaagonisten enthalten

Publications (1)

Publication Number Publication Date
UA86807C2 true UA86807C2 (ru) 2009-05-25

Family

ID=35058202

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200612950A UA86807C2 (ru) 2004-05-14 2005-05-11 ПОРОШКОВАЯ КОМПОЗИЦИЯ ДЛЯ ИНГАЛЯЦИИ, КОТОРАЯ СОДЕРЖИТ ЭНАНТИОМЕРНО ЧИСТЫЕ β-АГОНИСТЫ

Country Status (24)

Country Link
EP (1) EP1809236B1 (ru)
JP (1) JP4891899B2 (ru)
KR (1) KR101270449B1 (ru)
CN (1) CN1984638A (ru)
AR (1) AR048899A1 (ru)
AU (1) AU2005244424B2 (ru)
BR (1) BRPI0511136A (ru)
CA (1) CA2565915C (ru)
DE (1) DE102004024451A1 (ru)
DK (1) DK1809236T3 (ru)
EA (1) EA012582B1 (ru)
ES (1) ES2401786T3 (ru)
IL (1) IL179215A (ru)
MX (1) MXPA06013221A (ru)
MY (1) MY145838A (ru)
NO (1) NO20065078L (ru)
PE (1) PE20060239A1 (ru)
PL (1) PL1809236T3 (ru)
SG (1) SG152258A1 (ru)
TW (1) TW200607508A (ru)
UA (1) UA86807C2 (ru)
UY (1) UY28896A1 (ru)
WO (1) WO2005110359A1 (ru)
ZA (1) ZA200607785B (ru)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102004024452A1 (de) * 2004-05-14 2005-12-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg Aerosolformulierung für die Inhalation von Betaagonisten
KR20080036632A (ko) 2005-08-08 2008-04-28 아젠터 디스커버리 리미티드 바이시클로[2.2.1]헵트-7-일아민 유도체 및 이들의 용도
GB0516313D0 (en) 2005-08-08 2005-09-14 Argenta Discovery Ltd Azole derivatives and their uses
MX2008001976A (es) 2005-08-15 2008-03-25 Boehringer Ingelheim Int Procedimiento para la preparacion de betamimeticos.
US8236786B2 (en) 2008-08-07 2012-08-07 Pulmagen Therapeutics (Inflammation) Limited Respiratory disease treatment
MX2011007036A (es) 2008-12-30 2011-07-20 Pulmagen Therapeutics Inflammation Ltd Compuestos de sulfonamida para el tratamiento de trastornos respiratorios.
WO2010150014A1 (en) 2009-06-24 2010-12-29 Pulmagen Therapeutics (Inflammation) Limited 5r- 5 -deuterated glitazones for respiratory disease treatment
GB0918922D0 (en) 2009-10-28 2009-12-16 Vantia Ltd Aminopyridine derivatives
GB0918923D0 (en) 2009-10-28 2009-12-16 Vantia Ltd Aminothiazole derivatives
GB0918924D0 (en) 2009-10-28 2009-12-16 Vantia Ltd Azaindole derivatives
WO2011098746A1 (en) 2010-02-09 2011-08-18 Pulmagen Therapeutics (Inflammation) Limited Crystalline acid addition salts of ( 5r) -enanti0mer of pioglitazone
GB201002224D0 (en) 2010-02-10 2010-03-31 Argenta Therapeutics Ltd Respiratory disease treatment
GB201002243D0 (en) 2010-02-10 2010-03-31 Argenta Therapeutics Ltd Respiratory disease treatment
JP2015533131A (ja) 2012-10-09 2015-11-19 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 咳を治療するためのベータ2−アドレナリン受容体作動薬
WO2018108669A1 (en) 2016-12-12 2018-06-21 Boehringer Ingelheim International Gmbh Nintedanib for use in methods for the treatment of interstitial lung diseases by coadministration with olodaterol

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3134590A1 (de) * 1981-09-01 1983-03-10 Boehringer Ingelheim KG, 6507 Ingelheim Neue benzo-heterocyclen
US4460581A (en) 1982-10-12 1984-07-17 Boehringer Ingelheim Kg (1-Hydroxy-2-amino-alkyl)-substituted benzoxazinones and benzoxazolinones
DE4318455A1 (de) 1993-06-03 1994-12-08 Boehringer Ingelheim Kg Kapselhalterung
NZ522677A (en) * 2000-04-27 2004-10-29 Boehringer Ingelheim Pharma Novel, slow-acting betamimetics, a method for their production and their use as medicaments
GB0107106D0 (en) * 2001-03-21 2001-05-09 Boehringer Ingelheim Pharma Powder inhaler formulations
DE10141377A1 (de) * 2001-08-23 2003-03-13 Boehringer Ingelheim Pharma Aufstreuverfahren zur Herstellung von Pulverformulierungen
DE10212264A1 (de) 2002-03-20 2003-10-02 Boehringer Ingelheim Pharma Kristallines Mikronisat, Verfahren zu dessen Herstellung und dessen Verwendung zur Herstellung eines Arzneimittels
UA80123C2 (en) 2002-04-09 2007-08-27 Boehringer Ingelheim Pharma Inhalation kit comprising inhalable powder of tiotropium
DE10253282A1 (de) * 2002-11-15 2004-05-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Arzneimittel zur Behandlung von chronisch obstruktiver Lungenerkrankung

Also Published As

Publication number Publication date
ES2401786T3 (es) 2013-04-24
AU2005244424B2 (en) 2010-12-23
EP1809236B1 (de) 2012-12-26
NO20065078L (no) 2006-11-28
CA2565915A1 (en) 2005-11-24
UY28896A1 (es) 2005-12-30
JP2007537195A (ja) 2007-12-20
PL1809236T3 (pl) 2013-05-31
DE102004024451A1 (de) 2005-12-22
MY145838A (en) 2012-04-30
PE20060239A1 (es) 2006-03-27
EP1809236A1 (de) 2007-07-25
DK1809236T3 (da) 2013-02-11
IL179215A (en) 2011-04-28
AU2005244424A1 (en) 2005-11-24
BRPI0511136A (pt) 2007-11-27
CN1984638A (zh) 2007-06-20
CA2565915C (en) 2013-12-10
AR048899A1 (es) 2006-06-07
EA200602016A1 (ru) 2007-06-29
SG152258A1 (en) 2009-05-29
TW200607508A (en) 2006-03-01
WO2005110359A1 (de) 2005-11-24
KR20070016169A (ko) 2007-02-07
EA012582B1 (ru) 2009-10-30
ZA200607785B (en) 2008-07-30
MXPA06013221A (es) 2007-02-08
JP4891899B2 (ja) 2012-03-07
KR101270449B1 (ko) 2013-06-04
IL179215A0 (en) 2007-03-08

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