SV2010003642A - Compuestos - Google Patents
CompuestosInfo
- Publication number
- SV2010003642A SV2010003642A SV2010003642A SV2010003642A SV2010003642A SV 2010003642 A SV2010003642 A SV 2010003642A SV 2010003642 A SV2010003642 A SV 2010003642A SV 2010003642 A SV2010003642 A SV 2010003642A SV 2010003642 A SV2010003642 A SV 2010003642A
- Authority
- SV
- El Salvador
- Prior art keywords
- compounds
- undecano
- adrenoreceptors
- diazaspiro
- agonists
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 208000019693 Lung disease Diseases 0.000 abstract 1
- 102000014415 Muscarinic acetylcholine receptor Human genes 0.000 abstract 1
- 108050003473 Muscarinic acetylcholine receptor Proteins 0.000 abstract 1
- 239000000556 agonist Substances 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/10—Spiro-condensed systems
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Oncology (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Pulmonology (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Dermatology (AREA)
- Neurology (AREA)
- Hematology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Reproductive Health (AREA)
- Biomedical Technology (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Obesity (AREA)
- Pain & Pain Management (AREA)
- Gynecology & Obstetrics (AREA)
- Vascular Medicine (AREA)
- Molecular Biology (AREA)
- Transplantation (AREA)
Abstract
DERIVADOS DIAZASPIRO[5.5]UNDECANO Y COMPUESTOS RELACIONADOS COMO ANTAGONISTAS DE LOS RECEPTORES MUSCARINICOS Y AGONISTAS BETA-ADRENORECEPTORES PARA EL TRATAMIENTO DE DESORDENES PULMONARES
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0802192A GB0802192D0 (en) | 2008-02-06 | 2008-02-06 | Compounds |
| GB0822437A GB0822437D0 (en) | 2008-12-09 | 2008-12-09 | Compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SV2010003642A true SV2010003642A (es) | 2011-02-07 |
Family
ID=40474981
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SV2010003642A SV2010003642A (es) | 2008-02-06 | 2010-08-09 | Compuestos |
Country Status (38)
| Country | Link |
|---|---|
| US (2) | US8148373B2 (es) |
| EP (1) | EP2242759B1 (es) |
| JP (1) | JP4934223B2 (es) |
| KR (1) | KR101273200B1 (es) |
| CN (1) | CN102083839B (es) |
| AR (1) | AR070571A1 (es) |
| AU (1) | AU2009211251B2 (es) |
| BR (1) | BRPI0908353B8 (es) |
| CA (1) | CA2713322C (es) |
| CL (1) | CL2009000271A1 (es) |
| CO (1) | CO6290662A2 (es) |
| CR (1) | CR11623A (es) |
| CU (1) | CU23911B1 (es) |
| CY (1) | CY1113734T1 (es) |
| DK (1) | DK2242759T3 (es) |
| DO (1) | DOP2010000246A (es) |
| EA (1) | EA018711B1 (es) |
| EC (1) | ECSP10010390A (es) |
| ES (1) | ES2394547T3 (es) |
| HN (1) | HN2010001563A (es) |
| HR (1) | HRP20120968T1 (es) |
| IL (1) | IL207038A (es) |
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| TWI643853B (zh) | 2013-02-27 | 2018-12-11 | 阿爾米雷爾有限公司 | 同時具有β2腎上腺素受體促效劑和M3毒蕈鹼受體拮抗劑活性之2-氨基-1-羥乙基-8-羥基喹啉-2(1H)-酮衍生物之鹽類 |
| TWI641373B (zh) | 2013-07-25 | 2018-11-21 | 阿爾米雷爾有限公司 | 具有蕈毒鹼受體拮抗劑和β2腎上腺素受體促效劑二者之活性的2-胺基-1-羥乙基-8-羥基喹啉-2(1H)-酮衍生物之鹽 |
| TW201517906A (zh) | 2013-07-25 | 2015-05-16 | Almirall Sa | 含有maba化合物和皮質類固醇之組合 |
| TW201615643A (zh) | 2014-06-02 | 2016-05-01 | 伊史帝夫博士實驗室股份有限公司 | 具有多重模式抗疼痛活性之1-氧雜-4,9-二氮雜螺十一烷化合物之烷基與芳基衍生物 |
| TW201615642A (zh) * | 2014-06-02 | 2016-05-01 | 伊史帝夫博士實驗室股份有限公司 | 具有多重模式抗疼痛活性的1-氧雜-4,9-二氮雜螺十一烷化合物之醯胺衍生物 |
| TWI685497B (zh) | 2014-06-02 | 2020-02-21 | 西班牙商伊史帝夫製藥公司 | 具有多重模式抗疼痛活性的1-氧雜-4,9-二氮雜螺十一烷化合物之烷基衍生物 |
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| EP3377500B1 (en) | 2015-11-16 | 2022-10-19 | Esteve Pharmaceuticals, S.A. | Oxadiazaspiro compounds for the treatment of drug abuse and addiction |
| CN109195975B (zh) * | 2016-09-30 | 2022-01-04 | 四川海思科制药有限公司 | 一种二氮杂螺[5.5]十一碳烷衍生物及其用途 |
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| CN108264456A (zh) * | 2016-12-30 | 2018-07-10 | 湖北尚赛光电材料有限公司 | 2,8-二溴屈的合成方法及其合成中间体 |
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