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SG11201600504TA - 1-(piperazin-1-yl)-2-([1,2,4]triazol-1-yl)-ethanone derivatives - Google Patents

1-(piperazin-1-yl)-2-([1,2,4]triazol-1-yl)-ethanone derivatives

Info

Publication number
SG11201600504TA
SG11201600504TA SG11201600504TA SG11201600504TA SG11201600504TA SG 11201600504T A SG11201600504T A SG 11201600504TA SG 11201600504T A SG11201600504T A SG 11201600504TA SG 11201600504T A SG11201600504T A SG 11201600504TA SG 11201600504T A SG11201600504T A SG 11201600504TA
Authority
SG
Singapore
Prior art keywords
piperazin
triazol
ethanone derivatives
ethanone
derivatives
Prior art date
Application number
SG11201600504TA
Other languages
English (en)
Inventor
Eva Caroff
Emmanuel Meyer
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=51225512&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG11201600504T(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of SG11201600504TA publication Critical patent/SG11201600504TA/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Epidemiology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
SG11201600504TA 2013-07-22 2014-07-21 1-(piperazin-1-yl)-2-([1,2,4]triazol-1-yl)-ethanone derivatives SG11201600504TA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IB2013056001 2013-07-22
PCT/EP2014/065639 WO2015011099A1 (en) 2013-07-22 2014-07-21 1-(piperazin-1-yl)-2-([1,2,4]triazol-1-yl)-ethanone derivatives

Publications (1)

Publication Number Publication Date
SG11201600504TA true SG11201600504TA (en) 2016-02-26

Family

ID=51225512

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201600504TA SG11201600504TA (en) 2013-07-22 2014-07-21 1-(piperazin-1-yl)-2-([1,2,4]triazol-1-yl)-ethanone derivatives

Country Status (22)

Country Link
US (1) US10259807B2 (zh)
EP (1) EP3024832B1 (zh)
JP (1) JP6330040B2 (zh)
KR (1) KR102295416B1 (zh)
CN (1) CN105658649B (zh)
AR (1) AR096984A1 (zh)
AU (1) AU2014295123B2 (zh)
BR (1) BR112016001238B1 (zh)
CA (1) CA2916338C (zh)
CL (1) CL2016000152A1 (zh)
EA (1) EA030067B1 (zh)
ES (1) ES2671323T3 (zh)
IL (1) IL243650A0 (zh)
MA (1) MA38857B1 (zh)
MX (1) MX363432B (zh)
PH (1) PH12016500134A1 (zh)
PL (1) PL3024832T3 (zh)
SA (1) SA516370398B1 (zh)
SG (1) SG11201600504TA (zh)
TR (1) TR201807959T4 (zh)
TW (1) TWI630205B (zh)
WO (1) WO2015011099A1 (zh)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR201807959T4 (tr) 2013-07-22 2018-06-21 Idorsia Pharmaceuticals Ltd 1-(Piperazın-1-il)-2- ([1,2,4] triazol-1-il)-etanon türevleri.
AR099789A1 (es) 2014-03-24 2016-08-17 Actelion Pharmaceuticals Ltd Derivados de 8-(piperazin-1-il)-1,2,3,4-tetrahidro-isoquinolina
AR103399A1 (es) * 2015-01-15 2017-05-10 Actelion Pharmaceuticals Ltd Derivados de (r)-2-metil-piperazina como moduladores del receptor cxcr3
TN2017000278A1 (en) * 2015-01-15 2019-01-16 Idorsia Pharmaceuticals Ltd Hydroxyalkyl-piperazine derivatives as cxcr3 receptor modulators
WO2018011265A1 (en) 2016-07-13 2018-01-18 Idorsia Pharmaceuticals Ltd Hydroxyalkyl-piperazine derivatives as cxcr3 receptor modulators

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Also Published As

Publication number Publication date
PL3024832T3 (pl) 2018-10-31
MX2016000938A (es) 2016-05-05
MX363432B (es) 2019-03-22
EA030067B1 (ru) 2018-06-29
KR102295416B1 (ko) 2021-08-30
CA2916338A1 (en) 2015-01-29
CA2916338C (en) 2021-07-06
BR112016001238B1 (pt) 2022-10-11
ES2671323T3 (es) 2018-06-06
WO2015011099A1 (en) 2015-01-29
TW201536778A (zh) 2015-10-01
SA516370398B1 (ar) 2017-12-14
AU2014295123A1 (en) 2016-03-10
EP3024832B1 (en) 2018-03-28
BR112016001238A8 (pt) 2017-12-26
AU2014295123B2 (en) 2018-08-02
PH12016500134B1 (en) 2016-04-18
TR201807959T4 (tr) 2018-06-21
US10259807B2 (en) 2019-04-16
BR112016001238A2 (pt) 2017-12-12
TWI630205B (zh) 2018-07-21
CN105658649A (zh) 2016-06-08
IL243650A0 (en) 2016-02-29
EA201600123A1 (ru) 2016-07-29
US20160176862A1 (en) 2016-06-23
JP2016525137A (ja) 2016-08-22
AR096984A1 (es) 2016-02-10
PH12016500134A1 (en) 2016-04-18
CL2016000152A1 (es) 2016-09-02
EP3024832A1 (en) 2016-06-01
KR20160033218A (ko) 2016-03-25
JP6330040B2 (ja) 2018-05-23
CN105658649B (zh) 2019-03-22
MA38857A1 (fr) 2018-03-30
MA38857B1 (fr) 2018-10-31

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