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PE20100240A1 - Metodo para producir una composicion que comprende la epotilona (1s, 3s, 7s, 10r,11s,12s,16r)7, 11hidroxi-3-(2-metil-benzotiazol-5-il)-10-(prop-2-1-il)-8,8-12,16-tetrametil-4,17dioxabiciclo[14.1.0]heptade can-5,9-diona - Google Patents

Metodo para producir una composicion que comprende la epotilona (1s, 3s, 7s, 10r,11s,12s,16r)7, 11hidroxi-3-(2-metil-benzotiazol-5-il)-10-(prop-2-1-il)-8,8-12,16-tetrametil-4,17dioxabiciclo[14.1.0]heptade can-5,9-diona

Info

Publication number
PE20100240A1
PE20100240A1 PE2010000026A PE2010000026A PE20100240A1 PE 20100240 A1 PE20100240 A1 PE 20100240A1 PE 2010000026 A PE2010000026 A PE 2010000026A PE 2010000026 A PE2010000026 A PE 2010000026A PE 20100240 A1 PE20100240 A1 PE 20100240A1
Authority
PE
Peru
Prior art keywords
epotilone
diona
benzothiazol
prop
tetramethyl
Prior art date
Application number
PE2010000026A
Other languages
English (en)
Inventor
Olaf Reer
Matthias Renz
Andreas Sachse
Claudia Sprenger
Jens Thomsen
Anka Uffrecht
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of PE20100240A1 publication Critical patent/PE20100240A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/429Thiazoles condensed with heterocyclic ring systems
    • BPERFORMING OPERATIONS; TRANSPORTING
    • B82NANOTECHNOLOGY
    • B82YSPECIFIC USES OR APPLICATIONS OF NANOSTRUCTURES; MEASUREMENT OR ANALYSIS OF NANOSTRUCTURES; MANUFACTURE OR TREATMENT OF NANOSTRUCTURES
    • B82Y5/00Nanobiotechnology or nanomedicine, e.g. protein engineering or drug delivery
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40Cyclodextrins; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6949Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
    • A61K47/6951Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/19Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles lyophilised, i.e. freeze-dried, solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Inorganic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Nanotechnology (AREA)
  • Molecular Biology (AREA)
  • General Engineering & Computer Science (AREA)
  • Medical Informatics (AREA)
  • Biotechnology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Biophysics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicinal Preparation (AREA)
  • Silicon Polymers (AREA)
  • Processes Of Treating Macromolecular Substances (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

REFERIDA A UN METODO PARA PRODUCIR UNA COMPOSICION QUE COMPRENDE UNA EPOTILONA, DONDE DICHO PROCESO CONSISTE EN: a) DISOLVER (1S,3S,7S,10R,11S,12S,16R)-7,11-DIHIDROXI-3-(2-METIL-BENZOTIAZOL-5-IL)-10-(PROP-2-EN-1-IL)-8,8,12,16-TETRAMETIL-4,17-DIOXABICICLO[14.1.0]HEPTADECAN-5,9-DIONA EN UN SOLVENTE ORGANICO TAL COMO ETANOL, b) EVAPORAR DICHO SOLVENTE ORGANICO, c) DISOLVER HIDROXIPROPIL-BETA-CICLODEXTRINA EN SOLUCION ACUOSA, d) AJUSTAR EL pH DE LA MEZCLA RESULTANTE EN b) ENTRE 5 Y 9, e) DISOLVER EL POLVO RESULTANTE DE b) EN LOS SOLVENTES REULTANTES DE c) O d) Y LUEGO REALIZAR UNA FILTRACION ESTERIL PARA OBTENER UNA SOLUCION DE LA CUAL SE ELIMINA EL SOLVENTE Y SE OBTIEN UN PRODUCTO SOLIDO
PE2010000026A 2004-12-23 2006-01-03 Metodo para producir una composicion que comprende la epotilona (1s, 3s, 7s, 10r,11s,12s,16r)7, 11hidroxi-3-(2-metil-benzotiazol-5-il)-10-(prop-2-1-il)-8,8-12,16-tetrametil-4,17dioxabiciclo[14.1.0]heptade can-5,9-diona PE20100240A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP04090516A EP1674098A1 (en) 2004-12-23 2004-12-23 Stable and tolerable parental formulations of highly reactive organic drug substances with low or no solubility in water

Publications (1)

Publication Number Publication Date
PE20100240A1 true PE20100240A1 (es) 2010-05-02

Family

ID=34928859

Family Applications (2)

Application Number Title Priority Date Filing Date
PE2006000008A PE20060839A1 (es) 2004-12-23 2006-01-03 Composicion que comprende una epotilona y metodos para producir dicha composicion
PE2010000026A PE20100240A1 (es) 2004-12-23 2006-01-03 Metodo para producir una composicion que comprende la epotilona (1s, 3s, 7s, 10r,11s,12s,16r)7, 11hidroxi-3-(2-metil-benzotiazol-5-il)-10-(prop-2-1-il)-8,8-12,16-tetrametil-4,17dioxabiciclo[14.1.0]heptade can-5,9-diona

Family Applications Before (1)

Application Number Title Priority Date Filing Date
PE2006000008A PE20060839A1 (es) 2004-12-23 2006-01-03 Composicion que comprende una epotilona y metodos para producir dicha composicion

Country Status (22)

Country Link
EP (3) EP1674098A1 (es)
JP (1) JP2008525362A (es)
KR (1) KR20070088802A (es)
CN (1) CN101137364B (es)
AR (1) AR052346A1 (es)
AU (1) AU2005318353B2 (es)
BR (1) BRPI0519441A2 (es)
CA (1) CA2591997A1 (es)
CR (1) CR9211A (es)
GT (1) GT200500386A (es)
IL (1) IL183937A0 (es)
MX (1) MX2007007780A (es)
NO (1) NO20073772L (es)
NZ (1) NZ555989A (es)
PA (1) PA8657901A1 (es)
PE (2) PE20060839A1 (es)
RU (1) RU2416407C2 (es)
SG (1) SG161207A1 (es)
TW (1) TWI367758B (es)
UA (1) UA88182C2 (es)
UY (1) UY29307A1 (es)
WO (1) WO2006066949A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2210584A1 (en) 2009-01-27 2010-07-28 Bayer Schering Pharma Aktiengesellschaft Stable polymeric composition comprising an epothilone and an amphiphilic block copolymer
DE102009034368A1 (de) 2009-07-20 2011-01-27 Bayer Schering Pharma Aktiengesellschaft 17-Hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-acyloxyalkylenphenyl-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung zur Behandlung von Krankheiten
WO2012146625A1 (en) 2011-04-28 2012-11-01 Oncopeptides Ab Lyophilized preparation of cytotoxic dipeptides
NZ708016A (en) 2012-10-26 2018-02-23 Oncopeptides Ab Lyophilized preparations of melphalan flufenamide
CN107041886A (zh) * 2016-02-06 2017-08-15 北京华昊中天生物技术有限公司 脱环氧埃坡霉素衍生物制剂、制备及其治疗肿瘤的应用

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Also Published As

Publication number Publication date
IL183937A0 (en) 2007-10-31
EP1674098A1 (en) 2006-06-28
HK1114015A1 (en) 2008-10-24
CN101137364B (zh) 2011-11-16
MX2007007780A (es) 2007-08-14
NO20073772L (no) 2007-09-21
CN101137364A (zh) 2008-03-05
PA8657901A1 (es) 2007-01-17
WO2006066949A1 (en) 2006-06-29
NZ555989A (en) 2010-12-24
AR052346A1 (es) 2007-03-14
CA2591997A1 (en) 2006-06-29
RU2416407C2 (ru) 2011-04-20
CR9211A (es) 2007-11-23
PE20060839A1 (es) 2006-09-15
EP1827428A1 (en) 2007-09-05
KR20070088802A (ko) 2007-08-29
UA88182C2 (ru) 2009-09-25
SG161207A1 (en) 2010-05-27
GT200500386A (es) 2006-08-01
UY29307A1 (es) 2006-07-31
BRPI0519441A2 (pt) 2009-01-20
JP2008525362A (ja) 2008-07-17
EP2371365A1 (en) 2011-10-05
TW200635586A (en) 2006-10-16
AU2005318353B2 (en) 2011-09-29
AU2005318353A1 (en) 2006-06-29
RU2007128068A (ru) 2009-01-27
TWI367758B (en) 2012-07-11

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