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PE20000644A1 - Combinaciones terapeuticas que comprenden un modulador del receptor de estrogenos selectivo y hormona paratiroidea - Google Patents

Combinaciones terapeuticas que comprenden un modulador del receptor de estrogenos selectivo y hormona paratiroidea

Info

Publication number
PE20000644A1
PE20000644A1 PE1999000526A PE00052699A PE20000644A1 PE 20000644 A1 PE20000644 A1 PE 20000644A1 PE 1999000526 A PE1999000526 A PE 1999000526A PE 00052699 A PE00052699 A PE 00052699A PE 20000644 A1 PE20000644 A1 PE 20000644A1
Authority
PE
Peru
Prior art keywords
reconstruction
estrogen receptor
parathyroid hormone
receptor modulator
selective estrogen
Prior art date
Application number
PE1999000526A
Other languages
English (en)
Inventor
Hua Zhu Ke
David Duane Thompson
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of PE20000644A1 publication Critical patent/PE20000644A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22Hormones
    • A61K38/29Parathyroid hormone, i.e. parathormone; Parathyroid hormone-related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32Antioestrogens

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Investigating Or Analysing Biological Materials (AREA)

Abstract

SE REFIERE A UNA COMPOSICION QUE COMPRENDE a)UN MODULADOR DEL RECEPTOR DE ESTROGENOS SELECTIVO (SERM) TAL COMO (-)-CIS-6-FENIL-5-(4-(2-PIRROLIDIN-1-IL-ETOXI)-FENIL-5,6,7,8-TETRAHIDRONAFTALEN-2-OL O SU SAL D-TARTRATO; b)UN COMPUESTO DE HORMONA PARATIROIDEA O SUS FRAGMENTOS BIOLOGICAMENTE ACTIVOS. LA COMPOSICION PUEDE SER UTIL PARA EL TRATAMIENTO DE OSTEOPOROSIS, OSTEOTOMIA, PERDIDA OSEA IDIOPATICA DE LA INFANCIA O PERDIDA OSEA ASOCIADA A PERIODONTITIS, O PARA TRATAR UNA FRACTURA OSEA O CURACION OSEA DESPUES DE UNA RECONSTRUCCION FACIAL, RECONSTRUCCION MAXILAR, RECONSTRUCCION MANDIBULAR, FRAGILIDAD MUSCULOESQUELETICA
PE1999000526A 1998-06-16 1999-06-14 Combinaciones terapeuticas que comprenden un modulador del receptor de estrogenos selectivo y hormona paratiroidea PE20000644A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8947998P 1998-06-16 1998-06-16

Publications (1)

Publication Number Publication Date
PE20000644A1 true PE20000644A1 (es) 2000-08-02

Family

ID=22217879

Family Applications (1)

Application Number Title Priority Date Filing Date
PE1999000526A PE20000644A1 (es) 1998-06-16 1999-06-14 Combinaciones terapeuticas que comprenden un modulador del receptor de estrogenos selectivo y hormona paratiroidea

Country Status (34)

Country Link
US (1) US6132774A (es)
EP (1) EP1094808A1 (es)
JP (1) JP2002518323A (es)
KR (1) KR20010052818A (es)
CN (1) CN1305373A (es)
AP (1) AP9901580A0 (es)
AR (1) AR018867A1 (es)
AU (1) AU3725999A (es)
BG (1) BG105125A (es)
BR (1) BR9911228A (es)
CA (1) CA2335078A1 (es)
CO (1) CO5070584A1 (es)
EA (1) EA200001199A1 (es)
GT (1) GT199900066A (es)
HN (1) HN1999000063A (es)
HR (1) HRP20000858A2 (es)
HU (1) HUP0102759A3 (es)
ID (1) ID26873A (es)
IL (1) IL139588A0 (es)
IS (1) IS5719A (es)
MA (1) MA26649A1 (es)
NO (1) NO20006313L (es)
NZ (1) NZ508039A (es)
OA (1) OA11566A (es)
PA (1) PA8471201A1 (es)
PE (1) PE20000644A1 (es)
PL (1) PL344982A1 (es)
SK (1) SK18922000A3 (es)
TN (1) TNSN99119A1 (es)
TR (1) TR200003567T2 (es)
UA (1) UA60367C2 (es)
WO (1) WO1999065482A1 (es)
YU (1) YU75800A (es)
ZA (1) ZA993972B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1996000101A (es) * 1996-02-28 1997-06-26 Inc Pfizer Terapia combinada para la osteoporosis
US20020107230A1 (en) * 2000-12-22 2002-08-08 Waldon R. Forrest Methods and formulations for the treatment of female sexual dysfunction
US20030191096A1 (en) * 2002-04-03 2003-10-09 Leonard Thomas W. Method of hormonal therapy
JP2007512359A (ja) 2003-11-19 2007-05-17 メタバシス・セラピューティクス・インコーポレイテッド 新規なリン含有甲状腺ホルモン様物質
MX2007005137A (es) * 2004-11-23 2007-06-22 Warner Lambert Co Derivados del acido 7-(2h-pyrazol-3-il)-3, 5-dihidroxi-heptanoico como inhibidores de hmg co-a reductasa para el tratamiento de lipidemia.
US7790745B2 (en) 2005-10-21 2010-09-07 Bristol-Myers Squibb Company Tetrahydroisoquinoline LXR Modulators
US7741317B2 (en) 2005-10-21 2010-06-22 Bristol-Myers Squibb Company LXR modulators
US7919506B2 (en) 2006-03-10 2011-04-05 Pfizer Inc. Dibenzyl amine compounds and derivatives
WO2008070496A2 (en) 2006-12-01 2008-06-12 Bristol-Myers Squibb Company N- ( (3-benzyl) -2, 2- (bis-phenyl) -propan-1-amine derivatives as cetp inhibitors for the treatment of atherosclerosis and cardiovascular diseases
US20120046364A1 (en) 2009-02-10 2012-02-23 Metabasis Therapeutics, Inc. Novel Sulfonic Acid-Containing Thyromimetics, and Methods for Their Use
TW201043595A (en) * 2009-03-13 2010-12-16 Organon Nv Tetrahydronaphthalen-2-ol derivatives
DE102010027016A1 (de) 2010-07-09 2012-01-12 Universitätsklinikum Jena Steroid-Styrylfarbstoff-Konjugate zur Simulation und direkten lichtoptischen Detektion des Verhaltens von Steroiden im lebenden biologischen Gewebe und in Gegenwart von steroidbindenden Proteinen
CN111067907A (zh) * 2018-10-18 2020-04-28 常州大学 孕激素在抑制血管内皮生长因子表达中的应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5254595A (en) * 1988-12-23 1993-10-19 Elf Sanofi Aryloxypropanolaminotetralins, a process for their preparation and pharmaceutical compositions containing them
US5552412A (en) * 1995-01-09 1996-09-03 Pfizer Inc 5-substitued-6-cyclic-5,6,7,8-tetrahydronaphthalen2-ol compounds which are useful for treating osteoporosis
TW432073B (en) * 1995-12-28 2001-05-01 Pfizer Pyrazolopyridine compounds
HN1996000101A (es) * 1996-02-28 1997-06-26 Inc Pfizer Terapia combinada para la osteoporosis

Also Published As

Publication number Publication date
NZ508039A (en) 2003-03-28
HRP20000858A2 (en) 2001-10-31
KR20010052818A (ko) 2001-06-25
PA8471201A1 (es) 2000-09-29
IS5719A (is) 2000-11-21
AR018867A1 (es) 2001-12-12
WO1999065482A1 (en) 1999-12-23
PL344982A1 (en) 2001-11-19
YU75800A (sh) 2003-12-31
AU3725999A (en) 2000-01-05
OA11566A (en) 2004-05-26
GT199900066A (es) 2000-10-31
ID26873A (id) 2001-02-15
BG105125A (en) 2001-11-30
CO5070584A1 (es) 2001-08-28
SK18922000A3 (sk) 2001-09-11
US6132774A (en) 2000-10-17
CN1305373A (zh) 2001-07-25
JP2002518323A (ja) 2002-06-25
NO20006313D0 (no) 2000-12-12
TR200003567T2 (tr) 2001-06-21
HUP0102759A2 (hu) 2002-03-28
TNSN99119A1 (fr) 2005-11-10
IL139588A0 (en) 2002-02-10
BR9911228A (pt) 2001-02-13
HUP0102759A3 (en) 2002-12-28
HN1999000063A (es) 2000-01-12
AP9901580A0 (en) 1999-06-30
ZA993972B (en) 2000-12-15
EP1094808A1 (en) 2001-05-02
MA26649A1 (fr) 2004-12-20
CA2335078A1 (en) 1999-12-23
UA60367C2 (uk) 2003-10-15
EA200001199A1 (ru) 2001-04-23
NO20006313L (no) 2000-12-12

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