|
BR9712544B1
(pt)
|
1996-10-18 |
2013-10-22 |
|
Inibidores de proteases de serina, composição farmacêutica compreendendo os mesmos e seus usos
|
|
US6608027B1
(en)
|
1999-04-06 |
2003-08-19 |
Boehringer Ingelheim (Canada) Ltd |
Macrocyclic peptides active against the hepatitis C virus
|
|
PE20011350A1
(es)
|
2000-05-19 |
2002-01-15 |
Vertex Pharma |
PROFARMACO DE UN INHIBIDOR DE ENZIMA CONVERTIDORA DE INTERLEUCINA-1ß (ICE)
|
|
US7244721B2
(en)
*
|
2000-07-21 |
2007-07-17 |
Schering Corporation |
Peptides as NS3-serine protease inhibitors of hepatitis C virus
|
|
MY143322A
(en)
*
|
2000-07-21 |
2011-04-15 |
Schering Corp |
Peptides as ns3-serine protease inhibitors of hepatitis c virus
|
|
SV2003000617A
(es)
*
|
2000-08-31 |
2003-01-13 |
Lilly Co Eli |
Inhibidores de la proteasa peptidomimetica ref. x-14912m
|
|
US7473691B2
(en)
|
2000-09-15 |
2009-01-06 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compounds useful as protein kinase inhibitors
|
|
US6660731B2
(en)
|
2000-09-15 |
2003-12-09 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compounds useful as protein kinase inhibitors
|
|
CA2422367C
(fr)
|
2000-09-15 |
2010-05-18 |
Vertex Pharmaceuticals Incorporated |
Composes de pyrazole pouvant etre utilises comme inhibiteurs de la proteine kinase
|
|
GB2367816A
(en)
*
|
2000-10-09 |
2002-04-17 |
Bayer Ag |
Urea- and thiourea-containing derivatives of beta-amino acids
|
|
AU3659102A
(en)
*
|
2000-12-12 |
2002-06-24 |
Schering Corp |
Diaryl peptides as ns3-serine protease inhibitors of hepatits c virus
|
|
WO2002059111A2
(fr)
|
2000-12-21 |
2002-08-01 |
Vertex Pharmaceuticals Incorporated |
Composes de pyrazole utiles en tant qu'inhibiteurs de proteine kinase
|
|
MXPA04000293A
(es)
|
2001-07-11 |
2004-05-04 |
Vertex Pharma |
Inhibidores de serina proteasa biciclica de puente.
|
|
AU2002348414B2
(en)
*
|
2001-10-24 |
2009-10-01 |
Vertex Pharmaceuticals Incorporated |
Inhibitors of serine protease, particularly hepatitis C virus NS3-NS4A protease, incorporating a fused ring system
|
|
TWI265927B
(en)
*
|
2002-01-23 |
2006-11-11 |
Schering Corp |
Novel compounds as NS3-serine protease inhibitors of hepatitis C virus
|
|
US7119072B2
(en)
|
2002-01-30 |
2006-10-10 |
Boehringer Ingelheim (Canada) Ltd. |
Macrocyclic peptides active against the hepatitis C virus
|
|
US6642204B2
(en)
|
2002-02-01 |
2003-11-04 |
Boehringer Ingelheim International Gmbh |
Hepatitis C inhibitor tri-peptides
|
|
US7091184B2
(en)
|
2002-02-01 |
2006-08-15 |
Boehringer Ingelheim International Gmbh |
Hepatitis C inhibitor tri-peptides
|
|
RU2004133044A
(ru)
*
|
2002-04-11 |
2006-01-27 |
Вертекс Фармасьютикалз Инкорпорейтед (Us) |
Ингибиторы сериновых протеаз, в частности, протеазы ns3-ns4a hcv
|
|
MY140680A
(en)
|
2002-05-20 |
2010-01-15 |
Bristol Myers Squibb Co |
Hepatitis c virus inhibitors
|
|
MY141867A
(en)
|
2002-06-20 |
2010-07-16 |
Vertex Pharma |
Substituted pyrimidines useful as protein kinase inhibitors
|
|
US20050075279A1
(en)
|
2002-10-25 |
2005-04-07 |
Boehringer Ingelheim International Gmbh |
Macrocyclic peptides active against the hepatitis C virus
|
|
AU2011203054B2
(en)
*
|
2003-04-11 |
2012-04-26 |
Vertex Pharmaceuticals, Incorporated |
Inhibitors of Serine Proteases, Particularly HCV NS3-NS4A Protease
|
|
CN100453553C
(zh)
*
|
2003-04-11 |
2009-01-21 |
沃泰克斯药物股份有限公司 |
丝氨酸蛋白酶、特别是hcv ns3-ns4a蛋白酶的抑制剂
|
|
EP1654261B1
(fr)
|
2003-05-21 |
2007-11-14 |
Boehringer Ingelheim International GmbH |
Composes inhibiteurs de l'hepatite c
|
|
AR044694A1
(es)
|
2003-06-17 |
2005-09-21 |
Schering Corp |
Proceso y compuestos intermedios para la preparacion de (1r, 2s,5s) - 3 azabiciclo [3,1,0] hexano-2- carboxamida, n- [3- amino-1- (ciclobutilmetil) - 2, 3 - dioxopropil] -3- [ (2s) - 2 - [[ [ 1,1- dimetiletil] amino] carbonilamino] -3,3-dimetil -1- oxobutil]-6,6 dimetilo
|
|
CA2526634C
(fr)
*
|
2003-06-17 |
2012-09-18 |
Schering Corporation |
Procede et intermediaires de preparation de 3-(amino)-3-cyclobutylmethyl-2-hydroxy-propionamide ou leurs sels
|
|
JP4825129B2
(ja)
|
2003-06-17 |
2011-11-30 |
シェーリング コーポレイション |
(1r,2s,5s)−6,6−ジメチル−3−アザビシクロ[3,1,0]ヘキサン−2−カルボキシレートまたはその塩の調製のためのプロセスおよび中間体
|
|
TW200523270A
(en)
|
2003-07-18 |
2005-07-16 |
Vertex Pharma |
Inhibitors of serine proteases, particularly HCV ns3-ns4a protease
|
|
WO2005021584A2
(fr)
*
|
2003-08-26 |
2005-03-10 |
Schering Corporation |
Nouveaux inhibiteurs peptidomimetiques de la serine protease ns3 du virus de l'hepatite c
|
|
UY28500A1
(es)
|
2003-09-05 |
2005-04-29 |
Vertex Pharma |
Inhibidores de proteasas de serina, en particular proteasa ns3-ns4a del vhc.
|
|
JP4685775B2
(ja)
*
|
2003-09-18 |
2011-05-18 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
セリンプロテアーゼ、とりわけhcvns3−ns4aプロテアーゼの阻害剤
|
|
MXPA06003141A
(es)
|
2003-09-22 |
2006-06-05 |
Boehringer Ingelheim Int |
Peptidos macrociclicos activos contra el virus de la hepatitis c.
|
|
CN1894274A
(zh)
|
2003-09-26 |
2007-01-10 |
先灵公司 |
丙肝病毒ns3丝氨酸蛋白酶的大环抑制剂
|
|
TW200528472A
(en)
*
|
2003-10-10 |
2005-09-01 |
Vertex Pharma |
Inhibitors of serine proteases, particularly HCV ns3-ns4a protease
|
|
US7491794B2
(en)
*
|
2003-10-14 |
2009-02-17 |
Intermune, Inc. |
Macrocyclic compounds as inhibitors of viral replication
|
|
AU2004285019B9
(en)
|
2003-10-27 |
2011-11-24 |
Vertex Pharmaceuticals Incorporated |
HCV NS3-NS4A protease resistance mutants
|
|
EP1944042A1
(fr)
|
2003-10-27 |
2008-07-16 |
Vertex Pharmceuticals Incorporated |
Combinaisons pour le traitement HCV
|
|
US8187874B2
(en)
|
2003-10-27 |
2012-05-29 |
Vertex Pharmaceuticals Incorporated |
Drug discovery method
|
|
CA2546290A1
(fr)
|
2003-11-20 |
2005-06-09 |
Schering Corporation |
Inhibiteurs depourvus de liaisons peptidiques de la protease ns3 du virus de l'hepatite c
|
|
KR20060118532A
(ko)
|
2003-12-11 |
2006-11-23 |
쉐링 코포레이션 |
C형 간염 바이러스 ns3/ns4a 세린 프로테아제의억제제
|
|
JP4682155B2
(ja)
|
2004-01-21 |
2011-05-11 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
C型肝炎ウイルスに対して活性な大環状ペプチド
|
|
DE602005017582D1
(en)
*
|
2004-01-30 |
2009-12-24 |
Medivir Ab |
Hcv ns-3 serine protease inhibitoren
|
|
EP2311851A3
(fr)
*
|
2004-02-04 |
2011-05-25 |
Vertex Pharmaceuticals Incorporated |
Inhibitoren der Serinproteasen, insbesondere der HCV-NS3-NS4A-Protease
|
|
HRP20090250T1
(hr)
|
2004-02-24 |
2009-06-30 |
Japan Tobacco |
Kondenzirani heterociklički spojevi i njihova upotreba kao inhibitora hcv polimeraze
|
|
US20070049593A1
(en)
|
2004-02-24 |
2007-03-01 |
Japan Tobacco Inc. |
Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor
|
|
EP1730142B1
(fr)
*
|
2004-02-27 |
2011-06-29 |
Schering Corporation |
Nouveaux cetoamides a p4 cycliques en tant qu'inhibiteurs de la ns3 serine protease du virus de l'hepatite c
|
|
CA2557301A1
(fr)
*
|
2004-02-27 |
2005-09-15 |
Schering Corporation |
Groupes cyclobutenedione contenant des composes servant d'inhibiteurs a la serine protease ns3 du virus de l'hepatite c
|
|
AR048413A1
(es)
*
|
2004-02-27 |
2006-04-26 |
Schering Corp |
Compuestos prolina 3,4- (ciclopentil) - fusionados , como inhibidores de serina proteasa ns3 del virus de la hepatitis c
|
|
US7635694B2
(en)
|
2004-02-27 |
2009-12-22 |
Schering Corporation |
Cyclobutenedione-containing compounds as inhibitors of hepatitis C virus NS3 serine protease
|
|
KR101316137B1
(ko)
*
|
2004-02-27 |
2013-10-10 |
머크 샤프 앤드 돔 코포레이션 |
C형 간염 바이러스 ns3 세린 프로테아제의 억제제로서의황 화합물
|
|
AU2005222055A1
(en)
|
2004-02-27 |
2005-09-22 |
Schering Corporation |
Compounds as inhibitors of hepatitis C virus NS3 serine protease
|
|
BRPI0508186A
(pt)
|
2004-02-27 |
2007-08-14 |
Schering Corp |
compostos como inibidores de ns3 serina protease de vìrus da hepatite c
|
|
US7816326B2
(en)
|
2004-02-27 |
2010-10-19 |
Schering Corporation |
Sulfur compounds as inhibitors of hepatitis C virus NS3 serine protease
|
|
KR20060124725A
(ko)
*
|
2004-02-27 |
2006-12-05 |
쉐링 코포레이션 |
C형 간염 바이러스 ns3 프로테아제의 억제제
|
|
KR20110137409A
(ko)
*
|
2004-03-12 |
2011-12-22 |
버텍스 파마슈티칼스 인코포레이티드 |
아스파르트산 아세탈 카스파아제 억제제의 제조를 위한 방법 및 중간체
|
|
US20050249702A1
(en)
*
|
2004-05-06 |
2005-11-10 |
Schering Corporation |
(1R,2S,5S)-N-[(1S)-3-amino-1-(cyclobutylmethyl)-2,3-dioxopropyl]-3-[(2S)-2-[[[(1,1-dimethylethyl)amino]carbonyl]amino]-3,3-dimethyl-1-oxobutyl]-6,6-dimethyl-3-azabicyclo[3.1.0]hexane-2-carboxamide as inhibitor of hepatitis C virus NS3/NS4a serine protease
|
|
JP2008502718A
(ja)
*
|
2004-05-20 |
2008-01-31 |
シェーリング コーポレイション |
C型肝炎ウイルスns3セリンプロテアーゼのインヒビターとしての置換型プロリン
|
|
UY29016A1
(es)
|
2004-07-20 |
2006-02-24 |
Boehringer Ingelheim Int |
Analogos de dipeptidos inhibidores de la hepatitis c
|
|
WO2006007708A1
(fr)
|
2004-07-20 |
2006-01-26 |
Boehringer Engelheim International Gmbh |
Analogues peptidiques inhibiteurs de l'hepatite c
|
|
CA2577812A1
(fr)
|
2004-08-27 |
2006-03-09 |
Schering Corporation |
Composes d'acylsulfonamide inhibiteurs de la serine protease ns3 du virus de l'hepatite c
|
|
US7196161B2
(en)
*
|
2004-10-01 |
2007-03-27 |
Scynexis Inc. |
3-ether and 3-thioether substituted cyclosporin derivatives for the treatment and prevention of hepatitis C infection
|
|
KR20130083938A
(ko)
|
2004-10-01 |
2013-07-23 |
버텍스 파마슈티칼스 인코포레이티드 |
Hcv ns3-ns4a 프로테아제 저해
|
|
WO2006039668A2
(fr)
*
|
2004-10-01 |
2006-04-13 |
Scynexis, Inc |
Derives de cyclosporine 3-ether et 3-thioether substitues utilises dans le traitement et la prevention d'une infection par hepatite c
|
|
US7659263B2
(en)
|
2004-11-12 |
2010-02-09 |
Japan Tobacco Inc. |
Thienopyrrole compound and use thereof as HCV polymerase inhibitor
|
|
GB0426661D0
(en)
*
|
2004-12-06 |
2005-01-05 |
Isis Innovation |
Pyrrolidine compounds
|
|
WO2006130552A2
(fr)
*
|
2005-06-02 |
2006-12-07 |
Schering Corporation |
Methodes de traitement du virus de l'hepatite c
|
|
US20060281689A1
(en)
*
|
2005-06-02 |
2006-12-14 |
Schering Corporation |
Method for modulating activity of HCV protease through use of a novel HCV protease inhibitor to reduce duration of treatment period
|
|
BRPI0610737A2
(pt)
*
|
2005-06-02 |
2010-07-20 |
Schering Corp |
formulações farmacêuticas e métodos de tratamento usando as mesmas
|
|
WO2006130686A2
(fr)
|
2005-06-02 |
2006-12-07 |
Schering Corporation |
Administration d'inhibiteurs de protease du vhc en combinaison avec des aliments pour ameliorer la biodisponibilite
|
|
US20060275366A1
(en)
*
|
2005-06-02 |
2006-12-07 |
Schering Corporation |
Controlled-release formulation
|
|
US20060276407A1
(en)
*
|
2005-06-02 |
2006-12-07 |
Schering Corporation |
Methods of treating hepatitis C virus
|
|
WO2006130687A2
(fr)
*
|
2005-06-02 |
2006-12-07 |
Schering Corporation |
Taux de concentration foie/plasma pour le dosage de l'inhibiteur de protease du virus de l'hepatite c
|
|
WO2006130627A2
(fr)
*
|
2005-06-02 |
2006-12-07 |
Schering Corporation |
Methodes de traitement de l'hepatite c
|
|
WO2006130607A2
(fr)
*
|
2005-06-02 |
2006-12-07 |
Schering Corporation |
Formulation a liberation controlee
|
|
US7608592B2
(en)
*
|
2005-06-30 |
2009-10-27 |
Virobay, Inc. |
HCV inhibitors
|
|
TWI449711B
(zh)
*
|
2005-06-30 |
2014-08-21 |
Virobay Inc |
C型肝炎病毒(hcv)抑制劑
|
|
US20110104109A1
(en)
*
|
2005-07-13 |
2011-05-05 |
Frank Bennett |
Tetracyclic indole derivatives and their use for treating or preventing viral infections
|
|
EA019888B1
(ru)
*
|
2005-07-25 |
2014-07-30 |
Интермьюн, Инк. |
Промежуточное соединение для получения макроциклических ингибиторов репликации вируса гепатита с и способ его синтеза
|
|
AR055361A1
(es)
|
2005-07-29 |
2007-08-22 |
Medivir Ab |
Inhibidores macrociclicos del virus de la hepatitis c
|
|
JP5230416B2
(ja)
|
2005-07-29 |
2013-07-10 |
テイボテク・フアーマシユーチカルズ |
C型肝炎ウイルスの大員環状阻害剤
|
|
EP2256113A1
(fr)
*
|
2005-08-02 |
2010-12-01 |
Vertex Pharmaceuticals Incorporated |
Inhibiteurs de sérine protéases
|
|
BRPI0615029A2
(pt)
|
2005-08-19 |
2009-06-16 |
Vertex Pharma |
processos e intermediários
|
|
US8399615B2
(en)
|
2005-08-19 |
2013-03-19 |
Vertex Pharmaceuticals Incorporated |
Processes and intermediates
|
|
AR055395A1
(es)
|
2005-08-26 |
2007-08-22 |
Vertex Pharma |
Compuestos inhibidores de la actividad de la serina proteasa ns3-ns4a del virus de la hepatitis c
|
|
US7964624B1
(en)
*
|
2005-08-26 |
2011-06-21 |
Vertex Pharmaceuticals Incorporated |
Inhibitors of serine proteases
|
|
DE602006020152D1
(de)
*
|
2005-09-30 |
2011-03-31 |
Scynexis Inc |
Arylalkyl- und heteroarylalkyl-derivate von cyclosporin a bei der behandlung und vorbeugung einer virusinfektion
|
|
NZ567262A
(en)
*
|
2005-09-30 |
2011-12-22 |
Scynexis Inc |
Cyclosporin derivatives and their use for the treatment and prevention of hepatitis C infection
|
|
KR20080056295A
(ko)
*
|
2005-10-11 |
2008-06-20 |
인터뮨, 인크. |
C형 간염 바이러스 복제를 억제하기 위한 화합물 및 방법
|
|
BRPI0619706A2
(pt)
|
2005-11-03 |
2011-10-11 |
Vertex Pharma |
composto, composição, método para inibir a atividade da proteìna aurora quinase numa amostra biológica, método para tratar um distúrbio proliferativo num paciente, método para tratar cáncer num indivìduo
|
|
US7705138B2
(en)
|
2005-11-11 |
2010-04-27 |
Vertex Pharmaceuticals Incorporated |
Hepatitis C virus variants
|
|
EP2392590A3
(fr)
|
2005-11-11 |
2012-03-14 |
Vertex Pharmaceuticals Incorporated |
Variantes du virus de l'hépatite C
|
|
AR056805A1
(es)
|
2005-11-14 |
2007-10-24 |
Schering Corp |
Un proceso para oxidacion para la preparcion de n- (3- amino-1- ( ciclobutilmetil) -2,3- dioxopropil ) -3-(n-(( ter-butilamino) carbonil )-3- metil- l- valil) -6,6- dimetil-3- azabiciclo (3.1.0) hexano -2- carboxamida y compuestos ralacionados
|
|
EP1963267B1
(fr)
*
|
2005-12-22 |
2013-08-14 |
Merck Sharp & Dohme Corp. |
Procede pour la preparation de composes 6, 6-dimethyl-3-azabicyclo-[3.1.0]-hexane et leurs sels enantiomeriques
|
|
SG170767A1
(en)
|
2005-12-23 |
2011-05-30 |
Zealand Pharma As |
Modified lysine-mimetic compounds
|
|
US7816348B2
(en)
|
2006-02-03 |
2010-10-19 |
Boehringer Ingelheim International Gmbh |
Viral polymerase inhibitors
|
|
TW200808308A
(en)
*
|
2006-02-09 |
2008-02-16 |
Schering Corp |
Novel HCV inhibitor combinations and methods
|
|
EP1981524A2
(fr)
*
|
2006-02-09 |
2008-10-22 |
Schering Corporation |
Combinaisons comprenant un ou plusieurs inhibiteurs de protéase du vhc et un ou plusieurs inhibiteurs de polymérase du vhc, et méthodes de traitement associées
|
|
US8039475B2
(en)
*
|
2006-02-27 |
2011-10-18 |
Vertex Pharmaceuticals Incorporated |
Co-crystals and pharmaceutical compositions comprising the same
|
|
EP1998765A2
(fr)
*
|
2006-03-03 |
2008-12-10 |
Schering Corporation |
Combinaisons therapeutiques contenant des inhibiteurs du protease de l'hcv et de l'ires de l'hcv
|
|
JP5646814B2
(ja)
*
|
2006-03-06 |
2014-12-24 |
アッヴィ・インコーポレイテッド |
Hcvを治療するためのリトナビルの組成物及び使用方法
|
|
EP2194039A1
(fr)
|
2006-03-16 |
2010-06-09 |
Vertex Pharmceuticals Incorporated |
Procédé de préparation de composés optiquement actifs
|
|
EP2007789B1
(fr)
*
|
2006-04-11 |
2015-05-20 |
Novartis AG |
Inhibiteurs spirocycliques du VIH/du virus de l'hépatite C
|
|
US20080045530A1
(en)
*
|
2006-04-11 |
2008-02-21 |
Trixi Brandl |
Organic Compounds and Their Uses
|
|
MX2008013125A
(es)
*
|
2006-04-11 |
2008-10-21 |
Novartis Ag |
Compuestos organicos y sus usos.
|
|
US8017612B2
(en)
|
2006-04-18 |
2011-09-13 |
Japan Tobacco Inc. |
Piperazine compound and use thereof as a HCV polymerase inhibitor
|
|
EP2012753A2
(fr)
*
|
2006-04-28 |
2009-01-14 |
Schering Corporation |
Procédé de précipitation et d'isolement de 6,6-diméthyl-3-aza-bicyclo[3.1.0]hexane-amides par précipitation contrôlée et formules pharmaceutiques les contenant
|
|
US8420122B2
(en)
*
|
2006-04-28 |
2013-04-16 |
Merck Sharp & Dohme Corp. |
Process for the precipitation and isolation of 6,6-dimethyl-3-aza-bicyclo [3.1.0] hexane-amide compounds by controlled precipitation and pharmaceutical formulations containing same
|
|
CN101495095B
(zh)
*
|
2006-04-28 |
2013-05-29 |
默沙东公司 |
通过受控的沉淀来沉淀和分离6,6-二甲基-3-氮杂-双环[3.1.0]己烷-酰胺化合物的方法和含有其的药学制剂
|
|
AU2007254148B2
(en)
|
2006-05-19 |
2013-02-07 |
Scynexis, Inc. |
Method for the treatment and prevention of ocular disorders
|
|
WO2007137080A2
(fr)
|
2006-05-23 |
2007-11-29 |
Irm Llc |
Composés et compositions en tant qu'inhibiteurs de protéases activatrices de canal
|
|
DE602007013387D1
(de)
*
|
2006-05-23 |
2011-05-05 |
Irm Llc |
Verbindungen und zusammensetzungen als kanalaktivierende protease-hemmer
|
|
WO2007141395A1
(fr)
*
|
2006-06-02 |
2007-12-13 |
Claude Annie Perrichon |
Gestion des electrons actifs
|
|
KR20090024834A
(ko)
*
|
2006-07-05 |
2009-03-09 |
인터뮨, 인크. |
C형 간염 바이러스 복제의 신규 억제제
|
|
EP2049474B1
(fr)
|
2006-07-11 |
2015-11-04 |
Bristol-Myers Squibb Company |
Inhibiteurs du virus de l'hépatite c
|
|
EP1886685A1
(fr)
|
2006-08-11 |
2008-02-13 |
INSERM (Institut National de la Santé et de la Recherche Médicale) |
Méthodes, utilisations et compositions pour la modulation de la réplication du HCV par activation ou inhibition du récepteur farnesoid X
|
|
MX2009000882A
(es)
|
2006-08-17 |
2009-02-04 |
Boehringer Ingelheim Int |
Inhibidores de la polimerasa virica.
|
|
WO2008024763A2
(fr)
*
|
2006-08-25 |
2008-02-28 |
Wyeth |
Identification et caractérisation de variants de réplicons du virus de l'hépatite c présentant une sensibilité réduite à hcv-796, et procédés correspondants
|
|
KR20090049600A
(ko)
*
|
2006-09-13 |
2009-05-18 |
노파르티스 아게 |
마크로시클릭 hcv 억제제 및 그의 용도
|
|
US8343477B2
(en)
|
2006-11-01 |
2013-01-01 |
Bristol-Myers Squibb Company |
Inhibitors of hepatitis C virus
|
|
US7772180B2
(en)
|
2006-11-09 |
2010-08-10 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
US8003604B2
(en)
|
2006-11-16 |
2011-08-23 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
US7763584B2
(en)
|
2006-11-16 |
2010-07-27 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
US7888464B2
(en)
|
2006-11-16 |
2011-02-15 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
WO2008069917A2
(fr)
|
2006-11-20 |
2008-06-12 |
Scynexis, Inc. |
Nouveaux peptides cycliques
|
|
TW200827368A
(en)
*
|
2006-11-21 |
2008-07-01 |
Genelabs Tech Inc |
Amido anti-viral compounds
|
|
US20100055071A1
(en)
*
|
2006-11-21 |
2010-03-04 |
Martin Robert Leivers |
Anti-Viral Compounds
|
|
JP2010512317A
(ja)
*
|
2006-12-07 |
2010-04-22 |
シェーリング コーポレイション |
pH感受性マトリクス処方物
|
|
MX2009006477A
(es)
*
|
2006-12-15 |
2009-06-26 |
Schering Corp |
Purificacion de bisulfito de una alfa-ceto amida.
|
|
PL2121605T3
(pl)
*
|
2006-12-20 |
2014-05-30 |
Merck Sharp & Dohme |
Sposób otrzymywania (1R,2S,5S)-N-[(1S)-3-amino-1-(cyklobutylo-metylo)-2,3-dioksypropylo]-3-[(2S)-2-[[[(1,1-dimetyloetylo)amino]-karbonylo]amino]-3,3-dimetylo-1-oksybutylo]-6,6-dimetylo-3-azabicyklo[3.1.0]heksano-2-karboksyamidu
|
|
EP2074087A2
(fr)
|
2006-12-21 |
2009-07-01 |
Wyeth |
Synthese de composes de pyrrolidine
|
|
AU2007339382B2
(en)
|
2006-12-22 |
2013-05-02 |
Merck Sharp & Dohme Llc |
4,5-ring annulated indole derivatives for treating or preventing of HCV and related viral infections
|
|
MX2009006877A
(es)
|
2006-12-22 |
2009-09-28 |
Schering Corp |
Derivados indolicos con anillo unido en las posiciones 5,6 y metodos de uso de los mismos.
|
|
CN101611002A
(zh)
*
|
2006-12-22 |
2009-12-23 |
先灵公司 |
用于治疗或预防hcv和相关病毒感染的4,5-环化吲哚衍生物
|
|
US20080161254A1
(en)
*
|
2007-01-03 |
2008-07-03 |
Virobay, Inc. |
Hcv inhibitors
|
|
EA016327B1
(ru)
|
2007-02-09 |
2012-04-30 |
Айрм Ллк |
Соединения и композиции в качестве ингибиторов протеазы, активирующей каналы
|
|
AU2008219704A1
(en)
*
|
2007-02-27 |
2008-09-04 |
Vertex Pharmaceuticals Incorporated |
Inhibitors of serine proteases
|
|
KR20090115970A
(ko)
*
|
2007-02-27 |
2009-11-10 |
버텍스 파마슈티칼스 인코포레이티드 |
공-결정 및 그를 포함하는 제약 조성물
|
|
WO2009008913A2
(fr)
*
|
2007-03-23 |
2009-01-15 |
Schering Corporation |
Inhibiteurs de cétoamides de p1 non épimérisables de protéase de ns3 du virus de l'hépatite c (vhc)
|
|
JP2010528987A
(ja)
*
|
2007-05-03 |
2010-08-26 |
インターミューン・インコーポレーテッド |
C型肝炎ウイルス複製の新規大環状阻害剤
|
|
ES2381410T3
(es)
|
2007-05-04 |
2012-05-28 |
Vertex Pharmceuticals Incorporated |
Terapia de combinación paa el tratamiento de infecciones por VHC
|
|
BRPI0811447A2
(pt)
*
|
2007-05-10 |
2014-10-29 |
Intermune Inc |
Compostos, composição farmacêutica e métodos de inibição da atividade da protease ns3/ns4, de tratamento da fibrose hepática e de intensificação da função hepática num indivíduo tendo infecção de vírus da hepatite c.
|
|
CA2693997C
(fr)
|
2007-08-03 |
2013-01-15 |
Pierre L. Beaulieu |
Inhibiteurs de polymerase virale
|
|
CN101842353A
(zh)
*
|
2007-08-29 |
2010-09-22 |
先灵公司 |
用于治疗病毒感染的2,3-取代的吲哚衍生物
|
|
AU2008295484B2
(en)
|
2007-08-29 |
2013-09-26 |
Merck Sharp & Dohme Llc |
Substituted indole derivatives and methods of use thereof
|
|
AR068108A1
(es)
*
|
2007-08-29 |
2009-11-04 |
Schering Corp |
Derivados azaindol 2,3-sustituidos y una composicion farmaceutica
|
|
ATE530546T1
(de)
|
2007-08-30 |
2011-11-15 |
Vertex Pharma |
Kokristalle und pharmazeutische zusammensetzungen damit
|
|
CN101883590A
(zh)
|
2007-09-14 |
2010-11-10 |
先灵公司 |
治疗丙型肝炎患者的方法
|
|
MX2010003916A
(es)
|
2007-10-10 |
2010-05-05 |
Novartis Ag |
Espiro-pirrolidinas y su uso contra infeccion por el virus de hepatitis c (hcv) y por el virus de inmunodeficiencia humana (vih).
|
|
US8419332B2
(en)
*
|
2007-10-19 |
2013-04-16 |
Atlas Bolt & Screw Company Llc |
Non-dimpling fastener
|
|
JP5416708B2
(ja)
*
|
2007-11-16 |
2014-02-12 |
メルク・シャープ・アンド・ドーム・コーポレーション |
3−アミノスルホニル置換インドール誘導体およびそれらの使用方法
|
|
MX2010005356A
(es)
*
|
2007-11-16 |
2010-05-27 |
Schering Corp |
Derivados de indol 3-heterociclico sustituidos y metodos de uso de los mismos.
|
|
CN101910130A
(zh)
*
|
2007-11-28 |
2010-12-08 |
先灵公司 |
制备用于形成6,6-二甲基-3-氮杂双环[3.1.0]己烷化合物的中间体的脱卤化氢方法
|
|
CA2708324C
(fr)
|
2007-12-19 |
2013-03-05 |
Boehringer Ingelheim International Gmbh |
Inhibiteurs de polymerase virale
|
|
US8202996B2
(en)
|
2007-12-21 |
2012-06-19 |
Bristol-Myers Squibb Company |
Crystalline forms of N-(tert-butoxycarbonyl)-3-methyl-L-valyl-(4R)-4-((7-chloro-4-methoxy-1-isoquinolinyl)oxy)-N- ((1R,2S)-1-((cyclopropylsulfonyl)carbamoyl)-2-vinylcyclopropyl)-L-prolinamide
|
|
CN102089274B
(zh)
*
|
2007-12-21 |
2014-09-10 |
默沙东公司 |
合成3-氨基-3-环丁基甲基-2-羟基丙酰胺或其盐的方法
|
|
JP5574982B2
(ja)
|
2008-02-04 |
2014-08-20 |
イデニク プハルマセウティカルス,インコーポレイテッド |
大環状セリンプロテアーゼ阻害剤
|
|
KR20110005869A
(ko)
*
|
2008-04-15 |
2011-01-19 |
인터뮨, 인크. |
C형 간염 바이러스 복제의 신규한 마크로사이클릭 억제제
|
|
US8163921B2
(en)
|
2008-04-16 |
2012-04-24 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
US8044023B2
(en)
|
2008-05-29 |
2011-10-25 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
US7964560B2
(en)
|
2008-05-29 |
2011-06-21 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
EP2280989B1
(fr)
*
|
2008-06-06 |
2016-02-10 |
Scynexis, Inc. |
Analogues de la cyclosporine et leur utilisation dans le traitement d'infections par le vhc
|
|
US20090306033A1
(en)
*
|
2008-06-06 |
2009-12-10 |
Keqiang Li |
Novel cyclic peptides
|
|
CA2727620A1
(fr)
*
|
2008-06-13 |
2009-12-17 |
Schering Corporation |
Derives d'indole tricycliques et procedes d'utilisation de ceux-ci
|
|
CA2728226A1
(fr)
|
2008-06-24 |
2010-01-21 |
Codexis, Inc. |
Procedes biocatalytiques pour la preparation de composes de proline bicycliques condenses sensiblement purs sur le plan stereo-isomerique
|
|
US8188137B2
(en)
|
2008-08-15 |
2012-05-29 |
Avila Therapeutics, Inc. |
HCV protease inhibitors and uses thereof
|
|
TW201019939A
(en)
|
2008-08-20 |
2010-06-01 |
Schering Corp |
Azo-substituted pyridine and pyrimidine derivatives and their use in treating viral infections
|
|
JP5674661B2
(ja)
|
2008-08-20 |
2015-02-25 |
メルク・シャープ・アンド・ドーム・コーポレーションMerck Sharp & Dohme Corp. |
エチニル置換ピリジンおよびピリミジン誘導体ならびにそれらのウイルス感染の治療における使用
|
|
TW201020238A
(en)
|
2008-08-20 |
2010-06-01 |
Schering Corp |
Ethenyl-substituted pyridine and pyrimidine derivatives and their use in treating viral infections
|
|
JP5731976B2
(ja)
|
2008-08-20 |
2015-06-10 |
メルク・シャープ・アンド・ドーム・コーポレーションMerck Sharp & Dohme Corp. |
置換ピリジン誘導体および置換ピリミジン誘導体ならびにそれらのウイルス感染の治療における使用
|
|
US8207341B2
(en)
|
2008-09-04 |
2012-06-26 |
Bristol-Myers Squibb Company |
Process or synthesizing substituted isoquinolines
|
|
US8563505B2
(en)
|
2008-09-29 |
2013-10-22 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
US8044087B2
(en)
|
2008-09-29 |
2011-10-25 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
EP2358736A1
(fr)
*
|
2008-10-15 |
2011-08-24 |
Intermune, Inc. |
Peptides antiviraux therapeutiques
|
|
US8283310B2
(en)
|
2008-12-15 |
2012-10-09 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
EP2376524B1
(fr)
*
|
2008-12-31 |
2017-03-15 |
Cypralis Limited |
Dérivés de cyclosporine a
|
|
CN102271699A
(zh)
|
2009-01-07 |
2011-12-07 |
西尼克斯公司 |
用于治疗hcv和hiv感染的环孢菌素衍生物
|
|
GB0900914D0
(en)
|
2009-01-20 |
2009-03-04 |
Angeletti P Ist Richerche Bio |
Antiviral agents
|
|
US8102720B2
(en)
*
|
2009-02-02 |
2012-01-24 |
Qualcomm Incorporated |
System and method of pulse generation
|
|
AR075584A1
(es)
*
|
2009-02-27 |
2011-04-20 |
Intermune Inc |
COMPOSICIONES TERAPEUTICAS QUE COMPRENDEN beta-D-2'-DESOXI-2'-FLUORO-2'-C-METILCITIDINA Y UN DERIVADO DE ACIDO ISOINDOL CARBOXILICO Y SUS USOS. COMPUESTO.
|
|
JP5690286B2
(ja)
|
2009-03-04 |
2015-03-25 |
イデニク プハルマセウティカルス,インコーポレイテッド |
ホスホチオフェン及びホスホチアゾールhcvポリメラーゼ阻害剤
|
|
EP2417134B1
(fr)
|
2009-04-08 |
2017-05-17 |
Idenix Pharmaceuticals LLC. |
Inhibiteurs macrocycliques de la sérine protéase
|
|
US8512690B2
(en)
|
2009-04-10 |
2013-08-20 |
Novartis Ag |
Derivatised proline containing peptide compounds as protease inhibitors
|
|
US20110182850A1
(en)
*
|
2009-04-10 |
2011-07-28 |
Trixi Brandl |
Organic compounds and their uses
|
|
WO2010138889A1
(fr)
|
2009-05-28 |
2010-12-02 |
Concert Pharmaceuticals, Inc. |
Peptides destinés au traitement des infections par le vhc
|
|
AU2010253791A1
(en)
|
2009-05-29 |
2011-11-24 |
Merck Sharp & Dohme Corp. |
Antiviral compounds composed of three linked Aryl moieties to treat diseases such as Hepatitis C
|
|
AR077139A1
(es)
|
2009-06-23 |
2011-08-03 |
Gilead Sciences Inc |
Composiciones farmaceuticas utiles para tratar el vch
|
|
US20110034469A1
(en)
|
2009-08-04 |
2011-02-10 |
Takeda Pharmaceutical Company Limited |
Heterocyclic Compound
|
|
CA2769652A1
(fr)
|
2009-08-05 |
2011-02-10 |
Idenix Pharmaceuticals, Inc. |
Inhibiteurs macrocycliques de la serine protease macrocyclique utiles contre les infections virales, en particulier le virus de l?hepatite c
|
|
US9156818B2
(en)
|
2009-09-11 |
2015-10-13 |
Enanta Pharmaceuticals, Inc. |
Hepatitis C virus inhibitors
|
|
US20110081315A1
(en)
*
|
2009-09-28 |
2011-04-07 |
Intermune, Inc. |
Novel macrocyclic inhibitors of hepatitis c virus replication
|
|
US20110082182A1
(en)
*
|
2009-10-01 |
2011-04-07 |
Intermune, Inc. |
Therapeutic antiviral peptides
|
|
US20110117055A1
(en)
|
2009-11-19 |
2011-05-19 |
Macdonald James E |
Methods of Treating Hepatitis C Virus with Oxoacetamide Compounds
|
|
CA2782024A1
(fr)
|
2009-11-25 |
2011-06-03 |
Schering Corporation |
Composes tricycliques fusionnes et leurs derives utiles pour le traitement de maladies virales
|
|
KR20120118008A
(ko)
|
2009-12-18 |
2012-10-25 |
아이데닉스 파마슈티칼스, 인코포레이티드 |
5,5-융합 아릴렌 또는 헤테로아릴렌 간염 c 바이러스 억제제
|
|
EP2516430B1
(fr)
|
2009-12-22 |
2014-11-05 |
Merck Sharp & Dohme Corp. |
Composés tricycliques fusionnés et leurs méthodes d'utilisation pour le traitement de maladies virales
|
|
US9433621B2
(en)
|
2010-02-18 |
2016-09-06 |
Merck Sharp & Dohme Corp. |
Substituted pyridine and pyrimidine derivatives and their use in treating viral infections
|
|
MX2012009927A
(es)
*
|
2010-02-25 |
2012-10-05 |
Vereniging Voor Christelijk Hoger Onderwijs Wetenschappelijk Onderzoek En Patientenzorg |
Proceso para la preparacion de alfa-aciloxibeta-formamida amidas.
|
|
EA201290882A1
(ru)
|
2010-03-09 |
2013-04-30 |
Мерк Шарп Энд Домэ Корп. |
Конденсированные трициклические силильные соединения и способы их применения для лечения вирусных заболеваний
|
|
JP2013541499A
(ja)
|
2010-07-26 |
2013-11-14 |
メルク・シャープ・エンド・ドーム・コーポレイション |
置換されたビフェニレン化合物およびウイルス性疾患の治療のためのその使用方法
|
|
WO2012050848A1
(fr)
|
2010-09-29 |
2012-04-19 |
Schering Corporation |
Dérivés tétracycliques condensés et procédés d'utilisation de ceux-ci dans le traitement de maladies virales
|
|
WO2012109398A1
(fr)
|
2011-02-10 |
2012-08-16 |
Idenix Pharmaceuticals, Inc. |
Inhibiteurs macrocycliques de sérine protéase, compositions pharmaceutiques les contenant et leur utilisation pour le traitement des infections par le vhc
|
|
WO2012107589A1
(fr)
|
2011-02-11 |
2012-08-16 |
INSERM (Institut National de la Santé et de la Recherche Médicale) |
Méthodes et compositions pharmaceutiques pour le traitement et la prévention des infections à vhc
|
|
US20120252721A1
(en)
|
2011-03-31 |
2012-10-04 |
Idenix Pharmaceuticals, Inc. |
Methods for treating drug-resistant hepatitis c virus infection with a 5,5-fused arylene or heteroarylene hepatitis c virus inhibitor
|
|
US9061041B2
(en)
|
2011-04-13 |
2015-06-23 |
Merck Sharp & Dohme Corp. |
2′-substituted nucleoside derivatives and methods of use thereof for the treatment of viral diseases
|
|
WO2012142075A1
(fr)
|
2011-04-13 |
2012-10-18 |
Merck Sharp & Dohme Corp. |
Dérivés de nucléosides à substitution 2'-azido et leurs procédés d'utilisation pour le traitement de maladies virales
|
|
US8957203B2
(en)
|
2011-05-05 |
2015-02-17 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
US8691757B2
(en)
|
2011-06-15 |
2014-04-08 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
WO2013033899A1
(fr)
|
2011-09-08 |
2013-03-14 |
Merck Sharp & Dohme Corp. |
Composés benzofuranes substitués et leur procédés d'utilisation pour le traitement de maladies virales
|
|
WO2013033900A1
(fr)
|
2011-09-08 |
2013-03-14 |
Merck Sharp & Dohme Corp. |
Composés hétérocycliques tétracycliques et leurs procédés d'utilisation pour le traitement de maladies virales
|
|
WO2013033901A1
(fr)
|
2011-09-08 |
2013-03-14 |
Merck Sharp & Dohme Corp. |
Dérivés benzofuranes substitués par un hétérocycle et leurs procédés d'utilisation pour le traitement de maladies virales
|
|
WO2013039876A1
(fr)
|
2011-09-14 |
2013-03-21 |
Merck Sharp & Dohme Corp. |
Composés hétérocycliques contenant un silyle et méthodes d'utilisation desdits composés pour traiter les maladies virales
|
|
US8492386B2
(en)
|
2011-10-21 |
2013-07-23 |
Abbvie Inc. |
Methods for treating HCV
|
|
AR088463A1
(es)
|
2011-10-21 |
2014-06-11 |
Abbvie Inc |
Metodos para el tratamiento de hcv
|
|
US8466159B2
(en)
|
2011-10-21 |
2013-06-18 |
Abbvie Inc. |
Methods for treating HCV
|
|
CN104436197A
(zh)
|
2011-10-21 |
2015-03-25 |
艾伯维公司 |
至少两种直接作用抗病毒剂的组合产品
|
|
US20130123325A1
(en)
|
2011-11-14 |
2013-05-16 |
Sven Ruf |
Use of boceprevir and related compounds in atherosclerosis, heart failure, renal diseases, liver diseases or inflammatory diseases
|
|
AR091192A1
(es)
*
|
2012-05-30 |
2015-01-21 |
Chemo Iberica Sa |
Procedimiento multicomponente para la preparacion de compuestos biciclicos
|
|
CN103508918B
(zh)
*
|
2012-06-18 |
2015-09-09 |
上海医药工业研究院 |
带有环丁基的α-羟基β-氨基酯类化合物及其制备方法
|
|
WO2014053533A1
(fr)
|
2012-10-05 |
2014-04-10 |
Sanofi |
Utilisation de dérivés substitués de l'acide 3-hétéroaroylamino-propionique en tant que produits pharmaceutiques destinés à la prévention/au traitement de la fibrillation auriculaire
|
|
WO2014061034A1
(fr)
*
|
2012-10-18 |
2014-04-24 |
Msn Laboratories Limited |
Procédé de préparation de boceprevir et de ses intermédiaires
|
|
JP6154474B2
(ja)
|
2012-10-19 |
2017-06-28 |
ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company |
C型肝炎ウイルス阻害剤
|
|
KR102186030B1
(ko)
|
2012-10-29 |
2020-12-03 |
시플라 리미티드 |
항 바이러스성 포스포네이트 유사체 및 이의 제조를 위한 방법
|
|
US9598433B2
(en)
|
2012-11-02 |
2017-03-21 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
EP2914598B1
(fr)
|
2012-11-02 |
2017-10-18 |
Bristol-Myers Squibb Company |
Inhibiteurs du virus de l'hépatite c
|
|
US9643999B2
(en)
|
2012-11-02 |
2017-05-09 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
|
EP2914614B1
(fr)
|
2012-11-05 |
2017-08-16 |
Bristol-Myers Squibb Company |
Inhibiteurs du virus de l'hépatite c
|
|
WO2014083575A2
(fr)
|
2012-11-29 |
2014-06-05 |
Mylan Laboratories Ltd |
Procédé amélioré de préparation d'intermédiaire de bocéprévir
|
|
CN103936652B
(zh)
*
|
2013-01-18 |
2016-07-06 |
上海医药工业研究院 |
抗丙肝药物Boceprevir的中间体IV及其制备方法和应用
|
|
CN103936818B
(zh)
*
|
2013-01-18 |
2017-09-29 |
上海医药工业研究院 |
抗丙肝药物Boceprevir的中间体Ⅰ及其制备方法和应用
|
|
CN103936627B
(zh)
*
|
2013-01-18 |
2016-08-31 |
上海医药工业研究院 |
抗丙肝药物Boceprevir的中间体Ⅶ及其制备方法和应用
|
|
JP6342922B2
(ja)
|
2013-03-07 |
2018-06-13 |
ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company |
C型肝炎ウイルス阻害剤
|
|
DK2970225T3
(en)
|
2013-03-14 |
2018-09-24 |
Onyx Therapeutics Inc |
DIPEPTIDE AND TRIPEPTIDE AS EPOXY-KETONE PROTEASE INHIBITORS
|
|
AR095426A1
(es)
|
2013-03-14 |
2015-10-14 |
Onyx Therapeutics Inc |
Inhibidores tripeptídicos de la epoxicetona proteasa
|
|
EP3184095A1
(fr)
|
2013-05-23 |
2017-06-28 |
IP Gesellschaft für Management mbH |
Unitées d'administration comprennante une polymorphe 1 de 2-(2-methylamino-pyrimidin-4-yl]-1h-indole-5-carboxylic acid [(s)-1-carbamoyl-2-(phenyl-pyrimidin-2-yl-amino)-ethyl]-amide
|
|
CN103387510B
(zh)
*
|
2013-08-08 |
2015-09-09 |
苏州永健生物医药有限公司 |
一种β-氨基-alpha-羟基环丁基丁酰胺盐酸盐的合成方法
|
|
WO2015042375A1
(fr)
|
2013-09-20 |
2015-03-26 |
Idenix Pharmaceuticals, Inc. |
Inhibiteurs du virus de l'hépatite c
|
|
MX2016004492A
(es)
*
|
2013-10-24 |
2016-06-16 |
Squibb Bristol Myers Co |
Inhibidores de la replicacion del virus de inmunodeficiencia humana (vih).
|
|
WO2015065817A1
(fr)
|
2013-10-30 |
2015-05-07 |
Merck Sharp & Dohme Corp. |
Pseudopolymorphes d'un inhibiteur de la protéine ns5a du vhc et leurs utilisations
|
|
EP2899207A1
(fr)
|
2014-01-28 |
2015-07-29 |
Amikana.Biologics |
Nouveau procédé pour tester l'inhibition de la protéase du HCV
|
|
WO2015134561A1
(fr)
|
2014-03-05 |
2015-09-11 |
Idenix Pharmaceuticals, Inc. |
Compositions pharmaceutiques comprenant un inhibiteur de flaviviridae hétéroarylène fusionné en 5,5 et son utilisation pour le traitement ou la prévention d'une infection par les flaviviridae
|
|
EP3114122A1
(fr)
|
2014-03-05 |
2017-01-11 |
Idenix Pharmaceuticals LLC |
Formes solides d'un composé inhibiteur des virus de la famille des flaviviridae et sels de celui-ci
|
|
CN106810485A
(zh)
*
|
2015-11-27 |
2017-06-09 |
上海现代制药股份有限公司 |
一种手性联苯吡咯烷酮的制备方法及其中间体
|
|
US11192914B2
(en)
|
2016-04-28 |
2021-12-07 |
Emory University |
Alkyne containing nucleotide and nucleoside therapeutic compositions and uses related thereto
|
|
US10730832B2
(en)
*
|
2016-06-21 |
2020-08-04 |
Orion Ophthalmology LLC |
Aliphatic prolinamide derivatives
|
|
EP3472151A4
(fr)
|
2016-06-21 |
2020-03-04 |
Orion Ophthalmology LLC |
Dérivés de prolinamide carbocycliques
|
|
AU2017282651B2
(en)
*
|
2016-06-21 |
2021-08-12 |
Orion Ophthalmology LLC |
Heterocyclic prolinamide derivatives
|
|
WO2018073110A1
(fr)
|
2016-10-20 |
2018-04-26 |
Basf Se |
Composés de quinoléine en tant que fongicides
|
|
BR112019014061A2
(pt)
|
2017-01-23 |
2020-02-04 |
Basf Se |
compostos de fórmula i, intermediários b, intermediários c, intermediários ii e intermediários d, composição, uso, método para combater fungos fitopatogênicos, semente e processo para a síntese dos compostos de fórmula i
|
|
CN110475772A
(zh)
|
2017-04-06 |
2019-11-19 |
巴斯夫欧洲公司 |
吡啶化合物
|
|
WO2018202865A1
(fr)
|
2017-05-05 |
2018-11-08 |
Zealand Pharma A/S |
Modulateurs de la communication intercellulaire par les jonctions lacunaires et leur utilisation pour le traitement d'une maladie oculaire diabétique
|
|
EP3927703B1
(fr)
|
2019-02-19 |
2023-04-05 |
Univerza V Ljubljani |
Antibactériens à base de fragments monocycliques couplés à un échafaudage de naphtyridine aminopipéridine
|
|
WO2021209563A1
(fr)
|
2020-04-16 |
2021-10-21 |
Som Innovation Biotech, S.A. |
Composés destinés à être utilisés dans le traitement d'infections virales par un coronavirus associé au syndrome respiratoire
|
|
GB2619610B
(en)
*
|
2020-07-20 |
2025-04-09 |
Enanta Pharm Inc |
Functionalized Peptides as Antiviral Agents
|
|
US11351149B2
(en)
|
2020-09-03 |
2022-06-07 |
Pfizer Inc. |
Nitrile-containing antiviral compounds
|
|
US12083099B2
(en)
|
2020-10-28 |
2024-09-10 |
Accencio LLC |
Methods of treating symptoms of coronavirus infection with viral protease inhibitors
|
|
US11976084B2
(en)
|
2020-11-23 |
2024-05-07 |
Enanta Pharmaceuticals, Inc. |
Spiropyrrolidine derived antiviral agents
|
|
US12540141B2
(en)
|
2020-11-23 |
2026-02-03 |
Enanta Pharmaceuticals, Inc. |
Spiropyrrolidine derived antiviral agents
|
|
MY200435A
(en)
*
|
2021-04-16 |
2023-12-26 |
Fujian Akeylink Biotechnology Co Ltd |
Ring-modified proline short peptide compound and use thereof
|
|
US11970502B2
(en)
|
2021-05-04 |
2024-04-30 |
Enanta Pharmaceuticals, Inc. |
Macrocyclic antiviral agents
|
|
US12398147B2
(en)
|
2021-05-11 |
2025-08-26 |
Enanta Pharmaceuticals, Inc. |
Macrocyclic spiropyrrolidine derived antiviral agents
|
|
CA3224494A1
(fr)
|
2021-07-09 |
2023-01-12 |
Koen Vandyck |
Composes anti-viraux
|
|
US12479854B2
(en)
|
2021-07-29 |
2025-11-25 |
Enanta Pharmaceuticals, Inc. |
Spiropyrrolidine derived antiviral agents
|
|
US12065428B2
(en)
|
2021-09-17 |
2024-08-20 |
Aligos Therapeutics, Inc. |
Anti-viral compounds
|
|
US11912714B2
(en)
|
2021-11-12 |
2024-02-27 |
Enanta Pharmaceuticals, Inc. |
Spiropyrrolidine derived antiviral agents
|
|
WO2023086400A1
(fr)
|
2021-11-12 |
2023-05-19 |
Enanta Pharmaceuticals, Inc. |
Nouveaux agents antiviraux dérivés de spiropyrrolidine
|
|
WO2023086350A1
(fr)
|
2021-11-12 |
2023-05-19 |
Enanta Pharmaceuticals, Inc. |
Agents antiviraux contenant des alcynes
|
|
US11993600B2
(en)
|
2021-12-08 |
2024-05-28 |
Enanta Pharmaceuticals, Inc. |
Saturated spirocyclics as antiviral agents
|
|
WO2023107417A1
(fr)
|
2021-12-08 |
2023-06-15 |
Enanta Pharmaceuticals, Inc. |
Agents antiviraux hétérocycliques
|
|
CN114133350B
(zh)
*
|
2021-12-16 |
2023-05-23 |
浙江乐普药业股份有限公司 |
一种抗新冠药物Paxlovid中间体的制备方法
|
|
WO2023149981A1
(fr)
*
|
2022-02-07 |
2023-08-10 |
Purdue Research Foundation |
Composés pour le traitement du sars
|
|
US12145942B2
(en)
|
2022-04-05 |
2024-11-19 |
Enanta Pharmaceuticals, Inc. |
Spiropyrrolidine derived antiviral agents
|
|
CN114736151B
(zh)
*
|
2022-04-13 |
2023-04-21 |
湖南复瑞生物医药技术有限责任公司 |
一种帕罗韦德关键中间体制备方法及化合物的结构式
|
|
CN115160205B
(zh)
*
|
2022-07-08 |
2024-06-07 |
上海皓鸿生物医药科技有限公司 |
一种制备(s)-1-(叔丁氧羰基)-2,5-二氢-1h-吡咯-2-羧酸及盐的方法
|