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DK1309585T3 - Nye indolderivater og anvendelse af disse som lægemidler - Google Patents

Nye indolderivater og anvendelse af disse som lægemidler

Info

Publication number
DK1309585T3
DK1309585T3 DK01969522T DK01969522T DK1309585T3 DK 1309585 T3 DK1309585 T3 DK 1309585T3 DK 01969522 T DK01969522 T DK 01969522T DK 01969522 T DK01969522 T DK 01969522T DK 1309585 T3 DK1309585 T3 DK 1309585T3
Authority
DK
Denmark
Prior art keywords
pharmaceuticals
indole derivatives
new indole
new
derivatives
Prior art date
Application number
DK01969522T
Other languages
Danish (da)
English (en)
Inventor
Silke Baasner
Peter Emig
Gerald Bacher
Dietmar Reichert
Beate Aue
Bernd Nickel
Eckhard Guenther
Original Assignee
Aeterna Zentaris Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aeterna Zentaris Gmbh filed Critical Aeterna Zentaris Gmbh
Application granted granted Critical
Publication of DK1309585T3 publication Critical patent/DK1309585T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
DK01969522T 2000-07-28 2001-07-26 Nye indolderivater og anvendelse af disse som lægemidler DK1309585T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10037310A DE10037310A1 (de) 2000-07-28 2000-07-28 Neue Indolderivate und deren Verwendung als Arzneimittel
PCT/EP2001/008644 WO2002010152A2 (de) 2000-07-28 2001-07-26 Neue indolderivate und deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
DK1309585T3 true DK1309585T3 (da) 2008-06-23

Family

ID=7650860

Family Applications (1)

Application Number Title Priority Date Filing Date
DK01969522T DK1309585T3 (da) 2000-07-28 2001-07-26 Nye indolderivater og anvendelse af disse som lægemidler

Country Status (30)

Country Link
US (3) US7365081B2 (no)
EP (3) EP1309585B1 (no)
JP (1) JP5113973B2 (no)
KR (1) KR100810453B1 (no)
CN (1) CN1215066C (no)
AR (1) AR055209A1 (no)
AT (1) ATE392420T1 (no)
AU (2) AU8975801A (no)
BG (1) BG66457B1 (no)
BR (1) BR0112807A (no)
CA (3) CA2354210C (no)
CY (1) CY1108770T1 (no)
CZ (1) CZ304197B6 (no)
DE (2) DE10037310A1 (no)
DK (1) DK1309585T3 (no)
ES (1) ES2303532T3 (no)
HU (1) HU229254B1 (no)
IL (2) IL153930A0 (no)
MX (1) MXPA03000644A (no)
NO (1) NO324594B1 (no)
NZ (1) NZ524404A (no)
PL (1) PL208673B1 (no)
PT (1) PT1309585E (no)
RU (1) RU2270196C9 (no)
SI (1) SI1309585T1 (no)
SK (1) SK288085B6 (no)
TW (1) TWI291955B (no)
UA (1) UA80670C2 (no)
WO (1) WO2002010152A2 (no)
ZA (1) ZA200300584B (no)

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US7205299B2 (en) * 2003-06-05 2007-04-17 Zentaris Gmbh Indole derivatives having an apoptosis-inducing effect
EP1641777A1 (de) * 2003-06-05 2006-04-05 Zentaris GmbH Indolderivate mit apoptose induzierender wirkung
US7211588B2 (en) * 2003-07-25 2007-05-01 Zentaris Gmbh N-substituted indolyl-3-glyoxylamides, their use as medicaments and process for their preparation
US20050124623A1 (en) 2003-11-26 2005-06-09 Bender John A. Diazaindole-dicarbonyl-piperazinyl antiviral agents
US20060100432A1 (en) 2004-11-09 2006-05-11 Matiskella John D Crystalline materials of 1-(4-benzoyl-piperazin-1-yl)-2-[4-methoxy-7-(3-methyl-[1,2,4]triazol-1-yl)-1H-pyrrolo[2,3-c]pyridin-3-yl]-ethane-1,2-dione
US8399666B2 (en) 2005-11-04 2013-03-19 Panmira Pharmaceuticals, Llc 5-lipoxygenase-activating protein (FLAP) inhibitors
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US7807671B2 (en) 2006-04-25 2010-10-05 Bristol-Myers Squibb Company Diketo-piperazine and piperidine derivatives as antiviral agents
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MX2010012814A (es) 2008-05-23 2010-12-20 Amira Pharmaceuticals Inc Inhibidor de proteina activadora de 5-lipoxigenasa.
AR084433A1 (es) 2010-12-22 2013-05-15 Ironwood Pharmaceuticals Inc Inhibidores de la faah y composiciones farmaceuticas que los contienen

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Also Published As

Publication number Publication date
NZ524404A (en) 2004-08-27
ZA200300584B (en) 2003-07-18
ES2303532T3 (es) 2008-08-16
CN1215066C (zh) 2005-08-17
NO324594B1 (no) 2007-11-26
BR0112807A (pt) 2003-07-01
BG66457B1 (bg) 2014-10-31
CY1108770T1 (el) 2014-04-09
IL153930A0 (en) 2003-07-31
EP1309585A2 (de) 2003-05-14
US20080153875A1 (en) 2008-06-26
DE50113867D1 (de) 2008-05-29
JP2004505075A (ja) 2004-02-19
HUP0300677A2 (hu) 2003-11-28
JP5113973B2 (ja) 2013-01-09
UA80670C2 (en) 2007-10-25
EP2163552A1 (de) 2010-03-17
US7989453B2 (en) 2011-08-02
AR055209A1 (es) 2007-08-15
US7365081B2 (en) 2008-04-29
PL208673B1 (pl) 2011-05-31
MXPA03000644A (es) 2003-06-06
HU229254B1 (en) 2013-10-28
US20080108819A1 (en) 2008-05-08
NO20030382L (no) 2003-02-20
NO20030382D0 (no) 2003-01-24
PL361356A1 (en) 2004-10-04
CA2354210C (en) 2010-09-14
EP1939195A1 (de) 2008-07-02
WO2002010152A2 (de) 2002-02-07
SI1309585T1 (sl) 2008-08-31
US20030100597A1 (en) 2003-05-29
PT1309585E (pt) 2008-06-09
KR100810453B1 (ko) 2008-03-07
ATE392420T1 (de) 2008-05-15
CA2704693A1 (en) 2002-01-28
TWI291955B (en) 2008-01-01
DE10037310A1 (de) 2002-02-07
AU8975801A (en) 2002-02-13
CZ304197B6 (cs) 2013-12-27
WO2002010152A3 (de) 2002-08-01
AU2001289758B2 (en) 2006-07-06
HK1058201A1 (en) 2004-05-07
CZ2003500A3 (cs) 2004-03-17
IL153930A (en) 2008-11-03
SK288085B6 (sk) 2013-06-03
RU2270196C9 (ru) 2007-11-27
CA2354210A1 (en) 2002-01-28
KR20030017658A (ko) 2003-03-03
CN1447805A (zh) 2003-10-08
SK2222003A3 (en) 2004-04-06
US8008324B2 (en) 2011-08-30
CA2704691A1 (en) 2002-01-28
RU2270196C2 (ru) 2006-02-20
BG107560A (bg) 2003-10-31
EP1309585B1 (de) 2008-04-16

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