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CN1360928A - Nanometer Fuyanping medicine and its prepn - Google Patents

Nanometer Fuyanping medicine and its prepn Download PDF

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Publication number
CN1360928A
CN1360928A CN 00136924 CN00136924A CN1360928A CN 1360928 A CN1360928 A CN 1360928A CN 00136924 CN00136924 CN 00136924 CN 00136924 A CN00136924 A CN 00136924A CN 1360928 A CN1360928 A CN 1360928A
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China
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nanometer
nano
parts
fuyanping
medicine
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CN 00136924
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Chinese (zh)
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杨孟君
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Individual
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Individual
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Priority to CN 00136924 priority Critical patent/CN1360928A/en
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Abstract

The nano Fuyanping medicine is prepared with nano Radix Sophorae Flavescentis, nano Cnidium mormieri, nano indian quassiawood, nano borneol, nano berbamine and other four kinds of nano Chinese medicinal materials in certain proportion as material. It has a grain fineness of 1200-1500 mesh, grain size of 0.1-200 nm and mostly below 100 nm, and new physical property. It is prepared through microwave extraction, decompressing concentration, spray drying in supersonic jet and other steps. It has high biological utilization and high treating effect.

Description

A kind of nanometer FUYANPING preparation medicine and preparation method thereof
The present invention relates to a kind of heat-clearing and toxic substances removing, dampness leukorrhagia stopping, killing parasites for relieving itching, cure mainly the nanometer FUYANPING preparation medicine of vaginitis, cervicitis, endometritis, the invention still further relates to the method for this medication preparation.
Fuyanping capsules is a kind of classical Chinese patent medicine, mainly contains effects such as heat-clearing and toxic substances removing, dampness leukorrhagia stopping, killing parasites for relieving itching, is used for that damp invasion of lower energizer, dai channel are failed to keep an appointment, leucorrhea with red and white discharge, pudendal pruritus swell and ache, and infusorian, mycete, bacterial vaginitis, vulvitis etc.But traditional fuyanping capsules disintegrate is slower, absorbs not exclusively, and bioavailability is not high, slow curative effect.
The object of the present invention is to provide a kind of bioavailability height, solid dispersion is good, absorbs fully the nanometer FUYANPING preparation medicine of increase evident in efficacy.
Another object of the present invention provides the preparation method of this nanometer FUYANPING preparation medicine.
To achieve these goals, the present invention takes following technical scheme:
Medicine of the present invention is to make (consumption is a weight portion) by following component:
Nanometer Radix Sophorae Flavescentis 200-300 part nano-pearl layer powder 1-5 part nano berberine hydrochloride 10-30 part
Nanometer Ramulus Et Folium Picrasmae 160-240 part nanometer Borneolum Syntheticum 1-10 part nano boric acid 10-50 part
Nanometer Fructus Cnidii 160-240 part nanometer Mentholum 1-3 part nanometer dried Alumen 30-70 part
The formula optimization weight proportion scope of medicine of the present invention is:
Nanometer Radix Sophorae Flavescentis 220-270 part nano-pearl layer powder 2-3 part nano berberine hydrochloride 15-25 part
Nanometer Ramulus Et Folium Picrasmae 180-220 part nanometer Borneolum Syntheticum 3-7 part nano boric acid 20-40 part
Nanometer Fructus Cnidii 180-220 part nanometer Mentholum 1.5-2.5 part nanometer dried Alumen 40-60 part
The best important proportioning of medicine of the present invention is:
20 parts of 2.5 parts of nano berberine hydrochlorides of 250 parts of nano-pearl layers of nanometer Radix Sophorae Flavescentis powder
30 parts of 5 parts of nano boric acids of 200 parts of nanometer Borneolum Syntheticums of nanometer Ramulus Et Folium Picrasmae
50 parts of 2 parts of nanometer dried Alumens of 200 parts of nanometer Mentholums of nanometer Fructus Cnidii
Technical scheme of the present invention is based on the modern material technology.One of modern material Developing Trend in Technology is to develop to the more and more littler direction of yardstick.The granule of the past composition material, its size all are at micron or more than the millimeter magnitude, and have occurred the material to the nanoscale development now.Because extremely refinement of granule, the shared percentage by volume of crystal boundary increases, and makes some performance of material that outstanding variation take place.
The property of nano material be since special construction-----material grains size of nano material less than the ultra-micro powder of 100nm, its body surface area is very big, the atom number ratio at crystal boundary place makes it to produce four big effects up to 15%-50%: i.e. small-size effect, quantum effect (containing macro quanta tunnel effect), skin effect and interfacial effect.Thereby has the not available physical and chemical performance of traditional material.Nanotechnology will bring a technological revolution of the field of Chinese medicines.
One of method of above-mentioned each component being made medicine of the present invention is:
1. divide and get the Chinese crude drug of respectively distinguishing the flavor of, add to concoct according to Chinese Pharmacopoeia one one of version in 2000 and be processed into the common Chinese decoction pieces
2. divide and get the common Chinese decoction pieces of respectively distinguishing the flavor of, be processed into the nanometer prepared slices of Chinese crude drugs, its method comprises the following steps:
1. the common Chinese decoction pieces is placed extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, promptly make the nanometer prepared slices of Chinese crude drugs with the instantaneous drying of hypersonic velocity.
3. the nanometer prepared slices of Chinese crude drugs (powder) are prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent standard, make pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution.
Two of medicine method for making of the present invention is:
1. be equipped with whole common Chinese decoction pieces in the proportioning ratio, place extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, get FUYANPING preparation nano powder with the instantaneous drying of hypersonic velocity jet;
4. its nano powder is made aforementioned various preparation according to Chinese Pharmacopoeia version standard preparation in 2000.
The pharmacological effect that above-mentioned two kinds of methods are made nanometer FUYANPING preparation medicine is identical.
A kind of important feature of the present invention is, the made drug material of the present invention has reached nanoscale, common fuyanping capsules preparation material is micron or the above particle diameter of millimeter, can only cross the 80-120 mesh sieve, the drug material that the present invention is made, particle diameter is at 0.1-200nm, and the overwhelming majority can be crossed the 1200-1500 mesh sieve less than 100nm.
Another important feature of the present invention is, solid preparation of the present invention disintegrate rapidly, and solid dispersion is good in water, absorbs fully, and the pharmacological action effect that mainly contains effective constituent is significantly higher than conventional formulation.
The pharmaceutical preparation that the present invention is made does not need to add any adjuvant, and is more favourable to human body.
The present invention has also created the new drug formulation that pill, powder, suppository, membrane, microcapsule, drop pill, aerosol, injection, oral solution of nanometer FUYANPING preparation medicine etc. had no precedent in the past.
Pharmaceutical preparation of the present invention can be used for that damp invasion of lower energizer, dai channel are failed to keep an appointment, leucorrhea with red and white discharge, pudendal pruritus swell and ache, and treatment of conditions such as infusorian, mycete, bacterial vaginitis, vulvitis, endometritis, cervicitis, clinical efficacy significantly is better than traditional fuyanping capsules.
The present invention's added solvent in microwave extracting is water or ethanol.
The present invention carries out in the concentrating under reduced pressure step at extract, and its concentrating under reduced pressure is conventional scheme.
Embodiment 1:
Prepare nano raw material by preceding method:
20 parts of 2.5 parts of nano berberine hydrochlorides of 250 parts of nano-pearl layers of nanometer Radix Sophorae Flavescentis powder
30 parts of 5 parts of nano boric acids of 200 parts of nanometer Borneolum Syntheticums of nanometer Ramulus Et Folium Picrasmae
50 parts of 2 parts of nanometer dried Alumens of 200 parts of nanometer Mentholums of nanometer Fructus Cnidii
Production method is as follows:
In the GMP cleaning shop, the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio after, according to Chinese Pharmacopoeia version two-shift system in 2000 agent capsules agent standard, do not add adjuvant, do not granulate, directly divide encapsulatedly with the fully-automatic capsule racking machine, make capsule.Every capsules content of dispersion is the 0.1-0.6 gram, and the patient takes the 1-5 grain at every turn, and take 1-4 every day.
Embodiment 2:
Prepare nano raw material by preceding method:
20 parts of 2.5 parts of nano berberine hydrochlorides of 250 parts of nano-pearl layers of nanometer Radix Sophorae Flavescentis powder
30 parts of 5 parts of nano boric acids of 200 parts of nanometer Borneolum Syntheticums of nanometer Ramulus Et Folium Picrasmae
50 parts of 2 parts of nanometer dried Alumens of 200 parts of nanometer Mentholums of nanometer Fructus Cnidii
Production method is as follows:
In the GMP cleaning shop, with the above-mentioned nanometer prepared slices of Chinese crude drugs or powder by described mixed good after, according to 2000 editions two-shift system agent of Chinese Pharmacopoeia powder needle injection standard, do not add any adjuvant, make nanometer FUYANPING powder needle injection, every injection content is the 5-20 milligram, and each consumption is that 1-2 props up, and use 1-3 every day.
Implement sharp 3:
Prepare nano raw material by preceding method:
20 parts of 2.5 parts of nano berberine hydrochlorides of 250 parts of nano-pearl layers of nanometer Radix Sophorae Flavescentis powder
30 parts of 5 parts of nano boric acids of 200 parts of nanometer Borneolum Syntheticums of nanometer Ramulus Et Folium Picrasmae
50 parts of 2 parts of nanometer dried Alumens of 200 parts of nanometer Mentholums of nanometer Fructus Cnidii
In the GMP cleaning shop, with the above-mentioned nanometer prepared slices of Chinese crude drugs or powder by described mixed good after, according to 2000 editions two-shift system agent of Chinese Pharmacopoeia membrane standard, filmogen adopts polyvinyl alcohol, make nanometer FUYANPING membrane, every membrane area size is the 2-100 square centimeter, and content of dispersion is the 1-50 gram, every medicine film pasted 1-7 days, pasted the medicine position: abdominal part.

Claims (6)

1, a kind of nanometer FUYANPING preparation medicine is characterized in that it is the medicament that the nano raw material of following weight proportioning is made:
Nanometer Radix Sophorae Flavescentis 200-300 part nano-pearl layer powder 1-5 part nano berberine hydrochloride 10-30 part
Nanometer Ramulus Et Folium Picrasmae 160-240 part nanometer Borneolum Syntheticum 1-10 part nano boric acid 10-50 part
Nanometer Fructus Cnidii 160-240 part nanometer Mentholum 1-3 part nanometer dried Alumen 30-70 part
And adopt following method to make: to select the formula Chinese drug material to concoct and be processed into the prepared slices of Chinese crude drugs; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters-990 meter per seconds, promptly makes the nanometer prepared slices of Chinese crude drugs.
2, nanometer FUYANPING preparation medicine according to claim 1, wherein the weight proportion of each nano raw material is:
Nanometer Radix Sophorae Flavescentis 220-270 part nano-pearl layer powder 2-3 part nano berberine hydrochloride 15-25 part
Nanometer Ramulus Et Folium Picrasmae 180-220 part nanometer Borneolum Syntheticum 3-7 part nano boric acid 20-40 part
Nanometer Fructus Cnidii 180-220 part nanometer Mentholum 1.5-2.5 part nanometer dried Alumen 40-60 part
3, nanometer FUYANPING preparation medicine according to claim 1, wherein the weight proportion of each nano raw material is:
20 parts of 2.5 parts of nano berberine hydrochlorides of 250 parts of nano-pearl layers of nanometer Radix Sophorae Flavescentis powder
30 parts of 5 parts of nano boric acids of 200 parts of nanometer Borneolum Syntheticums of nanometer Ramulus Et Folium Picrasmae
50 parts of 2 parts of nanometer dried Alumens of 200 parts of nanometer Mentholums of nanometer Fructus Cnidii
4, according to claim 1 or 2 or 3 described nanometer FUYANPING preparation medicines, it is characterized in that said medicine is pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution.
5,, it is characterized in that this method comprises the steps: to select the formula Chinese drug material to concoct and is processed into the prepared slices of Chinese crude drugs according to the pharmaceutical methods of claim 1 or 2 or 3 described nanometer FUYANPING preparation medicines; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters-990 meter per seconds, promptly makes the nanometer prepared slices of Chinese crude drugs.
6, wherein respectively distinguish the flavor of Chinese medicine in the ratio of prescription or Chinese crude drug concoct be processed into the prepared slices of Chinese crude drugs after mixing, or after making the nanometer prepared slices of Chinese crude drugs mixing.
CN 00136924 2000-12-29 2000-12-29 Nanometer Fuyanping medicine and its prepn Pending CN1360928A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN 00136924 CN1360928A (en) 2000-12-29 2000-12-29 Nanometer Fuyanping medicine and its prepn

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN 00136924 CN1360928A (en) 2000-12-29 2000-12-29 Nanometer Fuyanping medicine and its prepn

Publications (1)

Publication Number Publication Date
CN1360928A true CN1360928A (en) 2002-07-31

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101455715B (en) * 2008-11-13 2011-02-16 陕西东泰制药有限公司 Suppository for treating gynecologic diseases and preparation method thereof

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101455715B (en) * 2008-11-13 2011-02-16 陕西东泰制药有限公司 Suppository for treating gynecologic diseases and preparation method thereof

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