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CN1364514A - Nano eight ingredient motherwort medicine and its preparing method - Google Patents

Nano eight ingredient motherwort medicine and its preparing method Download PDF

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Publication number
CN1364514A
CN1364514A CN 01100499 CN01100499A CN1364514A CN 1364514 A CN1364514 A CN 1364514A CN 01100499 CN01100499 CN 01100499 CN 01100499 A CN01100499 A CN 01100499A CN 1364514 A CN1364514 A CN 1364514A
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China
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nano
nanometer
motherwort
parts
chinese
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CN 01100499
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Chinese (zh)
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杨孟君
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Individual
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Individual
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Priority to CN 01100499 priority Critical patent/CN1364514A/en
Publication of CN1364514A publication Critical patent/CN1364514A/en
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Abstract

The nano eight ingredient and motherwort medicine is prepared with nano motherwort, nano Codonopsis Pilosulae, nano prepared remannia rhizome, nano Chinese angelica, nano Radix Paeoniae Alba and other four kinds of nano Chinese medicinal materials in certain proportion as raw material. The new medicine preparation has a grain fineness of 1200-1500 mesh, rain size of 0.1-200 nm, mostly below 100 nm, and new physical property. It is prepared through microwave extraction, decompression concentration, spray drying in supersonic jet and other steps. It has high biological utilization and obvious treating effect.

Description

Nano eight ingredient motherwort medicine and preparation method thereof
The present invention relates to a kind of menstruation that fills blood, transfers, cure mainly the nano eight ingredient motherwort medicine that asthenia of qi and blood loses, the invention still further relates to the method for this medication preparation.
BAZHEN YIMU PIAN is a kind of classical Chinese patent medicine, mainly contains effects such as blood vessel dilating, anticoagulant, stimulation reticuloendothelial system phagocytic function, excited uterus, is used for women's QI and blood deficiency, unable, the menoxenia of asthenia.But traditional BAZHEN YIMU PIAN disintegrate is slower, absorbs not exclusively, and bioavailability is not high, slow curative effect.
The object of the present invention is to provide a kind of bioavailability height, solid dispersion is good, absorbs fully the nano eight ingredient motherwort medicine of increase evident in efficacy.
Another object of the present invention provides the preparation method of this nano eight ingredient motherwort medicine.
To achieve these goals, the present invention takes following technical scheme:
Medicine of the present invention is to make (consumption is a weight portion) by following component:
Nanometer motherwort 150-350 part nanometer Radix Codonopsis 40-80 part nanometer Radix Rehmanniae Preparata 80-170 part
Nano Chinese angelica 80-170 part nanometer Radix Paeoniae Alba 40-80 part nano Poria 40-80 part
Nanometer Rhizoma Atractylodis Macrocephalae 40-80 part nanometer Rhizoma Chuanxiong 40-80 part nanometer Radix Glycyrrhizae 10-50 part
The formula optimization weight proportion scope of medicine of the present invention is:
Nanometer motherwort 200-300 part nanometer Radix Codonopsis 50-70 part nanometer Radix Rehmanniae Preparata 100-150 part
Nano Chinese angelica 100-150 part nanometer Radix Paeoniae Alba 50-70 part nano Poria 50-70 part
Nanometer Rhizoma Atractylodis Macrocephalae 50-70 part nanometer Rhizoma Chuanxiong 50-70 part nanometer Radix Glycyrrhizae 20-40 part
The optimum weight proportioning of medicine of the present invention is:
123 parts of 61 parts of nanometer Radix Rehmanniae Preparata of 245 parts of nanometer Radix Codonopsis of nanometer motherwort
61 parts of 61 parts of nano Porias of 123 parts of nanometer Radix Paeoniae Albas of nano Chinese angelica
31 parts in 61 parts of nanometer Radix Glycyrrhizaes of 61 parts of nanometer Rhizoma Chuanxiongs of the nanometer Rhizoma Atractylodis Macrocephalae
Technical scheme of the present invention is based on the modern material technology.One of modern material Developing Trend in Technology is to develop to the more and more littler direction of yardstick.The granule of the past composition material, its size all are at micron or more than the millimeter magnitude, and have occurred the material to the nanoscale development now.Because extremely refinement of granule, the shared percentage by volume of crystal boundary increases, and makes some performance of material that outstanding variation take place.
The property of nano material is because the special construction of nano material---the particle size of material is less than the ultra-micro powder of 100nm, its body surface area is very big, the atom number ratio at crystal boundary place makes it to produce four big effects up to 15%-50%: i.e. small-size effect, quantum effect (containing macro quanta tunnel effect), skin effect and interfacial effect.Thereby has the not available physical and chemical performance of traditional material.Nanotechnology will bring a technological revolution of the field of Chinese medicines.
One of method of above-mentioned each component being made medicine of the present invention is:
1. divide and get the Chinese crude drug of respectively distinguishing the flavor of, add to concoct according to Chinese Pharmacopoeia one one of version in 2000 and be processed into the common Chinese decoction pieces
2. divide and get the common Chinese decoction pieces of respectively distinguishing the flavor of, be processed into the nanometer prepared slices of Chinese crude drugs, its method comprises the following steps:
1. the common Chinese decoction pieces is placed extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, promptly make the nanometer prepared slices of Chinese crude drugs with the instantaneous drying of hypersonic velocity.
3. the nanometer prepared slices of Chinese crude drugs (powder) are prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent standard, make pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution.
Two of medicine method for making of the present invention is:
1. be equipped with whole common Chinese decoction pieces in the proportioning ratio, place extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, get the eight ingredient motherwort nano powder with the instantaneous drying of hypersonic velocity jet;
4. its nano powder is made aforementioned various preparation according to Chinese Pharmacopoeia version standard preparation in 2000.
The pharmacological effect that above-mentioned two kinds of methods are made nano eight ingredient motherwort medicine is identical.
A kind of important feature of the present invention is: the made drug material of the present invention has reached nanoscale, common BAZHEN YIMU PIAN preparation material is micron or the above particle diameter of millimeter, can only cross the 80-120 mesh sieve, the drug material that the present invention is made, particle diameter is at 0.1-200nm, the overwhelming majority can be crossed the 1200-1500 mesh sieve less than 100nm.
Another important feature of the present invention is: solid preparation of the present invention disintegrate rapidly, and solid dispersion is good in water, absorb fully, the bioavailability height, the pharmacological action effect that mainly contains effective constituent is significantly higher than conventional formulation.
The pharmaceutical preparation that the present invention is made does not need to add any adjuvant, and is more favourable to human body.
The present invention has also created the new drug formulation that suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection of nano eight ingredient motherwort medicine etc. is had no precedent in the past.
Pharmaceutical preparation of the present invention can be used for treatment of conditions such as Sheehan syndrome, pigment purpura, and clinical efficacy significantly is better than traditional BAZHEN YIMU PIAN.
The present invention's added solvent in microwave extracting is water or ethanol.
The present invention carries out in the concentrating under reduced pressure step at extract, and its concentrating under reduced pressure is conventional scheme.
Embodiment 1:
Prepare nano raw material by preceding method:
123 parts of 61 parts of nanometer Radix Rehmanniae Preparata of 245 parts of nanometer Radix Codonopsis of nanometer motherwort
61 parts of 61 parts of nano Porias of 123 parts of nanometer Radix Paeoniae Albas of nano Chinese angelica
31 parts in 61 parts of nanometer Radix Glycyrrhizaes of 61 parts of nanometer Rhizoma Chuanxiongs of the nanometer Rhizoma Atractylodis Macrocephalae
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent capsules agent standard, do not add adjuvant, do not granulate, directly divide encapsulated with the fully-automatic capsule racking machine, make capsule, every capsules content of dispersion is the 0.1-0.6 gram, and the patient takes 1-4 time every day, each 1-5 grain.
Embodiment 2:
Prepare nano raw material by preceding method:
123 parts of 61 parts of nanometer Radix Rehmanniae Preparata of 245 parts of nanometer Radix Codonopsis of nanometer motherwort
61 parts of 61 parts of nano Porias of 123 parts of nanometer Radix Paeoniae Albas of nano Chinese angelica
31 parts in 61 parts of nanometer Radix Glycyrrhizaes of 61 parts of nanometer Rhizoma Chuanxiongs of the nanometer Rhizoma Atractylodis Macrocephalae
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent powder needle injection standard, do not add any adjuvant, make nanometer eight delicacies with motherwort powder needle injection, every injection content is the 5-20 milligram, and each consumption is that 1-2 props up, and use 1-3 every day.
Embodiment 3:
Prepare nano raw material by preceding method:
123 parts of 61 parts of nanometer Radix Rehmanniae Preparata of 245 parts of nanometer Radix Codonopsis of nanometer motherwort
61 parts of 61 parts of nano Porias of 123 parts of nanometer Radix Paeoniae Albas of nano Chinese angelica
31 parts in 61 parts of nanometer Radix Glycyrrhizaes of 61 parts of nanometer Rhizoma Chuanxiongs of the nanometer Rhizoma Atractylodis Macrocephalae
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent membrane standard, filmogen adopts polyvinyl alcohol, make nanometer eight delicacies with motherwort membrane, every membrane area size is the 2-100 square centimeter, and content of dispersion is the 1-50 gram, every medicine film pasted 1-7 days, pasted the medicine position: abdominal part.

Claims (6)

1, a kind of nano eight ingredient motherwort medicine is characterized in that it is the medicament that the nano raw material of following weight proportioning is made:
Nanometer motherwort 150-350 part nanometer Radix Codonopsis 40-80 part nanometer Radix Rehmanniae Preparata 80-170 part
Nano Chinese angelica 80-170 part nanometer Radix Paeoniae Alba 40-80 part nano Poria 40-80 part
Nanometer Rhizoma Atractylodis Macrocephalae 40-80 part nanometer Rhizoma Chuanxiong 40-80 part nanometer Radix Glycyrrhizae 10-50 part
And adopt following method to make: to select the formula Chinese drug material to concoct and be processed into the prepared slices of Chinese crude drugs; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters--990 meter per seconds, promptly make the nanometer prepared slices of Chinese crude drugs.
2, nano eight ingredient motherwort medicine according to claim 1, wherein the weight proportion of each nano raw material is:
Nanometer motherwort 200-300 part nanometer Radix Codonopsis 50-70 part nanometer Radix Rehmanniae Preparata 100-150 part
Nano Chinese angelica 100-150 part nanometer Radix Paeoniae Alba 50-70 part nano Poria 50-70 part
Nanometer Rhizoma Atractylodis Macrocephalae 50-70 part nanometer Rhizoma Chuanxiong 50-70 part nanometer Radix Glycyrrhizae 20-40 part
3, nano eight ingredient motherwort medicine according to claim 1, wherein the weight proportion of each nano raw material is:
123 parts of 61 parts of nanometer Radix Rehmanniae Preparata of 245 parts of nanometer Radix Codonopsis of nanometer motherwort
61 parts of 61 parts of nano Porias of 123 parts of nanometer Radix Paeoniae Albas of nano Chinese angelica
31 parts in 61 parts of nanometer Radix Glycyrrhizaes of 61 parts of nanometer Rhizoma Chuanxiongs of the nanometer Rhizoma Atractylodis Macrocephalae
4,, it is characterized in that said medicine is pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution according to claim 1 or 2 or 3 described nano eight ingredient motherwort medicines.
5,, it is characterized in that this method comprises the steps: to select the formula Chinese drug material to concoct and is processed into the prepared slices of Chinese crude drugs according to the pharmaceutical methods of claim 1 or 2 or 3 described nano eight ingredient motherwort medicines; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1-10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters--990 meter per seconds, promptly make the nanometer prepared slices of Chinese crude drugs.
6, wherein respectively distinguish the flavor of Chinese medicine in the ratio of prescription or Chinese crude drug concoct be processed into the prepared slices of Chinese crude drugs after mixing, or after making the nanometer prepared slices of Chinese crude drugs mixing.
CN 01100499 2001-01-16 2001-01-16 Nano eight ingredient motherwort medicine and its preparing method Pending CN1364514A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN 01100499 CN1364514A (en) 2001-01-16 2001-01-16 Nano eight ingredient motherwort medicine and its preparing method

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN 01100499 CN1364514A (en) 2001-01-16 2001-01-16 Nano eight ingredient motherwort medicine and its preparing method

Publications (1)

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CN1364514A true CN1364514A (en) 2002-08-21

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CN 01100499 Pending CN1364514A (en) 2001-01-16 2001-01-16 Nano eight ingredient motherwort medicine and its preparing method

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102824457A (en) * 2012-06-04 2012-12-19 江西南昌桑海制药厂 Eight-treasure motherwort active site and preparation process of capsules

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102824457A (en) * 2012-06-04 2012-12-19 江西南昌桑海制药厂 Eight-treasure motherwort active site and preparation process of capsules

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