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NO940039L - Chinolon- og naftyridonkarboksylsyrederivater - Google Patents

Chinolon- og naftyridonkarboksylsyrederivater

Info

Publication number
NO940039L
NO940039L NO940039A NO940039A NO940039L NO 940039 L NO940039 L NO 940039L NO 940039 A NO940039 A NO 940039A NO 940039 A NO940039 A NO 940039A NO 940039 L NO940039 L NO 940039L
Authority
NO
Norway
Prior art keywords
carboxylic acid
halogen
amino
methyl
acid derivatives
Prior art date
Application number
NO940039A
Other languages
English (en)
Other versions
NO940039D0 (no
Inventor
Stephan Bartel
Andreas Krebs
Franz Kunisch
Uwe Petersen
Thomas Schenke
Klaus Grohe
Michael Schriewer
Klaus Dieter Bremm
Rainer Endermann
Karl-Georg Metzger
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of NO940039D0 publication Critical patent/NO940039D0/no
Publication of NO940039L publication Critical patent/NO940039L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C10PETROLEUM, GAS OR COKE INDUSTRIES; TECHNICAL GASES CONTAINING CARBON MONOXIDE; FUELS; LUBRICANTS; PEAT
    • C10MLUBRICATING COMPOSITIONS; USE OF CHEMICAL SUBSTANCES EITHER ALONE OR AS LUBRICATING INGREDIENTS IN A LUBRICATING COMPOSITION
    • C10M133/00Lubricating compositions characterised by the additive being an organic non-macromolecular compound containing nitrogen
    • C10M133/02Lubricating compositions characterised by the additive being an organic non-macromolecular compound containing nitrogen having a carbon chain of less than 30 atoms
    • C10M133/38Heterocyclic nitrogen compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Fodder In General (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Det blir beskrevet nye chlnolon- og naftyridonkarboks- ylsyrederlvater med formel (I) R1 står for rettkjedet eller forgrenet C1-C4-alkyl, som eventuelt er substituert med hydroksy, halogen eller C1-C3-alkoksy, for C3-C6-cykloalkyl som eventuelt er substituert med C1-C3-alkyl eller halogen, C2-C4- alkenyl, foruten for C1-C3-alkoksy, araino, monoal- kylamino med l til 3 C-atomer, dialkylamino med l til 3 C-atomer pr. alkylgruppe eller for fenyl som eventuelt er substituert en eller opptil tre ganger med halogen, R2 står for hydrogen, alkyl med l til 4 karbonatomer som eventuelt er substituert med hydroksy, metoksy, amlno, metylamino eller dlmetylamino, eller (5-. metyl-2-okso-l,3-dioksol-4-yl)-metyl, X1 står for hydrogen, halogen, amino, metyl eller trifluormetyl, Z står for en rest med strukturen R5 l ,N -B A står for N eller C-R9. N- Det blir dessuten beskrevet en fremgangsmåte for frem- stilling av disse såvel som deres anvendelse som antl- bakterielt middel og fortilsetningsstoff.
NO940039A 1993-01-19 1994-01-05 Chinolon- og naftyridonkarboksylsyrederivater NO940039L (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4301246A DE4301246A1 (de) 1993-01-19 1993-01-19 Chinolon- und Naphthyridoncarbonsäurederivate

Publications (2)

Publication Number Publication Date
NO940039D0 NO940039D0 (no) 1994-01-05
NO940039L true NO940039L (no) 1994-07-20

Family

ID=6478454

Family Applications (1)

Application Number Title Priority Date Filing Date
NO940039A NO940039L (no) 1993-01-19 1994-01-05 Chinolon- og naftyridonkarboksylsyrederivater

Country Status (21)

Country Link
US (1) US5457104A (no)
EP (1) EP0607825A1 (no)
JP (1) JPH06247962A (no)
KR (1) KR940018380A (no)
CN (1) CN1097423A (no)
AU (2) AU667757B2 (no)
CA (1) CA2113513A1 (no)
CZ (1) CZ10094A3 (no)
DE (1) DE4301246A1 (no)
FI (1) FI940216A7 (no)
HU (1) HUT68455A (no)
IL (1) IL108347A (no)
MX (1) MX9400341A (no)
MY (1) MY110747A (no)
NO (1) NO940039L (no)
NZ (1) NZ250681A (no)
PL (1) PL301928A1 (no)
RU (1) RU2114832C1 (no)
SK (1) SK5394A3 (no)
TW (1) TW266213B (no)
ZA (1) ZA94332B (no)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3906365A1 (de) * 1988-07-15 1990-01-18 Bayer Ag 7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe
DE4230804A1 (de) * 1992-09-15 1994-03-17 Bayer Ag 7-Isoindolinyl-chinolon- und -naphthyridon-Derivate
DE4427530A1 (de) * 1994-08-04 1996-02-08 Bayer Ag Chinolon- und Naphthyridoncarbonsäure-Derivate
DE19506535A1 (de) * 1995-02-09 1996-08-14 Bayer Ag 1,6-Naphthyridoncarbonsäurederivate
ES2158963T3 (es) * 1995-02-09 2001-09-16 Bayer Ag Derivados de acidos 1,6-naftiridoncarboxilicos.
KR100276477B1 (ko) * 1996-02-09 2000-12-15 나카노 가쓰히코 퀴놀론카복실산유도체또는그의염
KR100531967B1 (ko) * 1996-10-25 2005-11-30 다이이찌 세이야꾸 가부시기가이샤 트리사이클릭 아민 유도체, 이를 포함하는 항균제 및 퀴놀론 화합물의 제조방법
US6387928B1 (en) 1997-09-15 2002-05-14 The Procter & Gamble Co. Antimicrobial quinolones, their compositions and uses
AU735186B2 (en) 1997-09-15 2001-07-05 Warner Chilcott Company, Llc Antimicrobial quinolones, their compositions and uses
PT1070713E (pt) * 1998-04-06 2006-12-29 Toyama Chemical Co Ltd Derivados de ácido quinolonocarboxílico ou seus sais
HUP0303457A3 (en) 2000-12-14 2008-05-28 Procter & Gamble Antimicrobial 2-pyridones, compositions containing them and their use
ES2249489T3 (es) 2000-12-14 2006-04-01 THE PROCTER & GAMBLE COMPANY Quinolonas antimicrobianas.
DE10108750A1 (de) * 2001-02-23 2002-09-05 Bayer Ag Verbessertes Verfahren zur Herstellung von Fluorchinoloncarbonsäuren
AU2007230630B2 (en) * 2006-03-28 2012-12-20 Taigen Biotechnology Co., Ltd Malate salts, and polymorphs of (3S,5S)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid
EP1999125A2 (en) * 2006-03-28 2008-12-10 The Procter and Gamble Company A coupling process for preparing quinolone intermediates
EP1999106B1 (en) * 2006-03-28 2012-06-27 TaiGen Biotechnology Co., Ltd. A hydride reduction process for preparing quinolone intermediates
NZ610978A (en) 2009-05-15 2014-11-28 Redx Pharma Ltd Redox drug derivatives
JP6030146B2 (ja) 2011-11-08 2016-11-24 アクテリオン ファーマシューティカルズ リミテッドActelion Pharmaceuticals Ltd 2−オキソ−オキサゾリジン−3,5−ジイル抗生物質誘導体
CA3030204A1 (en) 2016-07-11 2018-01-18 Bayer Pharma Aktiengesellschaft 7-substituted 1-pyridyl-naphthyridine-3-carboxylic acid amides and use thereof
JOP20190045A1 (ar) 2016-09-14 2019-03-14 Bayer Ag مركبات أميد حمض 1- أريل-نفثيريدين-3-كربوكسيليك مستبدلة في الموضع 7 واستخدامها.
EP3296298A1 (de) 2016-09-14 2018-03-21 Bayer Pharma Aktiengesellschaft 7-substituierte 1-aryl-naphthyridin-3-carbonsäureamide und ihre verwendung
CN109942488A (zh) * 2019-04-04 2019-06-28 山东省联合农药工业有限公司 一种喹啉羧酸酯类化合物及其制备方法与用途
AU2020289459A1 (en) 2019-06-07 2022-01-06 Elanco Tiergesundheit Ag Bicyclic derivatives for treating endoparasites
EP4424804B1 (en) * 2019-08-14 2025-12-24 Valvoline Licensing and Intellectual Property, LLC Lubricant composition containing ashless tbn molecules
CN115251064B (zh) * 2021-04-29 2023-08-29 山东省联合农药工业有限公司 一种杀菌杀虫组合物及其应用
CN113929579A (zh) * 2021-11-22 2022-01-14 南京一苇医药科技有限公司 一种克林沙星关键中间体的制备方法

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Publication number Priority date Publication date Assignee Title
US4416884A (en) * 1978-04-12 1983-11-22 Otsuka Pharmaceutical Co., Ltd. Piperazinylbenzoheterocyclic compounds
JPS604820B2 (ja) * 1979-02-26 1985-02-06 大塚製薬株式会社 キノリンカルボン酸誘導体
DE3441788A1 (de) * 1984-11-15 1986-05-15 Bayer Ag, 5090 Leverkusen Alkyl-1-cyclopropyl-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
DE3615767A1 (de) * 1986-05-10 1987-11-12 Bayer Ag Verfahren zur herstellung von 4-hydroxy-chinolin-3-carbonsaeuren
US5270340A (en) * 1988-12-27 1993-12-14 Bayer Aktiengesellschaft Substituted 2-cyclohexen-1-yl-amine fungicidal and herbicidal agents
CA2012681A1 (en) * 1989-03-31 1990-09-30 Masayasu Okuhira Quinolone derivatives, preparation processes thereof, and antibacterial agents containing the same
CA2030217A1 (en) * 1989-11-21 1991-05-22 Jun Imose Pyridone-carboxylic acid derivatives useful as veterinary medicines
WO1992012146A1 (en) * 1990-12-27 1992-07-23 Banyu Pharmaceutical Co., Ltd. Pyridonecarboxylic acid derivative
DE4120646A1 (de) * 1991-06-22 1992-12-24 Bayer Ag 7-isoindolinyl-chinolon- und naphthyridoncarbonsaeure-derivate
TW209865B (no) * 1992-01-10 1993-07-21 Bayer Ag
DE4230804A1 (de) * 1992-09-15 1994-03-17 Bayer Ag 7-Isoindolinyl-chinolon- und -naphthyridon-Derivate

Also Published As

Publication number Publication date
JPH06247962A (ja) 1994-09-06
US5457104A (en) 1995-10-10
TW266213B (no) 1995-12-21
FI940216A0 (fi) 1994-01-17
AU4203396A (en) 1996-04-04
KR940018380A (ko) 1994-08-16
MX9400341A (es) 1994-08-31
MY110747A (en) 1999-02-27
SK5394A3 (en) 1994-12-07
EP0607825A1 (de) 1994-07-27
CZ10094A3 (en) 1995-03-15
PL301928A1 (en) 1994-07-25
AU5256193A (en) 1994-07-28
FI940216A7 (fi) 1994-07-20
NO940039D0 (no) 1994-01-05
DE4301246A1 (de) 1994-07-21
RU2114832C1 (ru) 1998-07-10
CN1097423A (zh) 1995-01-18
HU9400143D0 (en) 1994-05-30
IL108347A (en) 1998-02-22
CA2113513A1 (en) 1994-07-20
HUT68455A (en) 1995-06-28
ZA94332B (en) 1994-08-26
NZ250681A (en) 1995-06-27
AU667757B2 (en) 1996-04-04
IL108347A0 (en) 1994-04-12

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