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NO20050016L - Difenylazetidinonderivater for behandling av forstyrrelser i lipid metabolismen - Google Patents

Difenylazetidinonderivater for behandling av forstyrrelser i lipid metabolismen

Info

Publication number
NO20050016L
NO20050016L NO20050016A NO20050016A NO20050016L NO 20050016 L NO20050016 L NO 20050016L NO 20050016 A NO20050016 A NO 20050016A NO 20050016 A NO20050016 A NO 20050016A NO 20050016 L NO20050016 L NO 20050016L
Authority
NO
Norway
Prior art keywords
treatment
diphenyllazetidinone
derivatives
lipid metabolism
metabolism disorders
Prior art date
Application number
NO20050016A
Other languages
English (en)
Inventor
Ingemar Starke
Ann-Margret Lindqvist
Tore Skjaret
Malin Lemurell
Mats Peter Nordberg
Mikael Ulf Johan Dahlstrom
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20050016L publication Critical patent/NO20050016L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)

Abstract

Forbindelser med formel (I): (R')b\^ R9 R"> R" 00 (hvor variable grupper er som definert ovenfor) farmasøytisk akseptable salter, solvater, solvater av slike salter og prodroge derav og anvendelse av dem som kolesterol absorpsjonsinhibitorer for behandling av hyperlipidemi er besikrevet. Fremgangsmåter for fremstilling av dem og farmasøytiske preparater inneholdende dem er også beskrevet.
NO20050016A 2002-07-05 2005-01-03 Difenylazetidinonderivater for behandling av forstyrrelser i lipid metabolismen NO20050016L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0215579.4A GB0215579D0 (en) 2002-07-05 2002-07-05 Chemical compounds
PCT/GB2003/002811 WO2004005247A1 (en) 2002-07-05 2003-07-01 Diphenylazetidinone derivatives for treating disorders of the lipid metabolism

Publications (1)

Publication Number Publication Date
NO20050016L true NO20050016L (no) 2005-03-01

Family

ID=9939901

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20050016A NO20050016L (no) 2002-07-05 2005-01-03 Difenylazetidinonderivater for behandling av forstyrrelser i lipid metabolismen

Country Status (21)

Country Link
US (1) US7470678B2 (no)
EP (1) EP1521742A1 (no)
JP (1) JP2006501184A (no)
CN (2) CN100528842C (no)
AR (1) AR041185A1 (no)
BR (1) BR0312280A (no)
CA (1) CA2491789A1 (no)
GB (1) GB0215579D0 (no)
IL (1) IL165820A0 (no)
IS (1) IS7648A (no)
MX (1) MXPA04012936A (no)
NO (1) NO20050016L (no)
NZ (1) NZ537124A (no)
PL (1) PL374725A1 (no)
RU (2) RU2333199C2 (no)
SA (1) SA02230379B1 (no)
TW (1) TW200404058A (no)
UA (1) UA78564C2 (no)
UY (1) UY27882A1 (no)
WO (1) WO2004005247A1 (no)
ZA (1) ZA200410340B (no)

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AU2003242850A1 (en) 2004-01-23
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IL165820A0 (en) 2006-01-15
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UA78564C2 (en) 2007-04-10
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