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MX2016012041A - Formulaciones de aripiprazol que tienen mayores velocidades de inyeccion. - Google Patents

Formulaciones de aripiprazol que tienen mayores velocidades de inyeccion.

Info

Publication number
MX2016012041A
MX2016012041A MX2016012041A MX2016012041A MX2016012041A MX 2016012041 A MX2016012041 A MX 2016012041A MX 2016012041 A MX2016012041 A MX 2016012041A MX 2016012041 A MX2016012041 A MX 2016012041A MX 2016012041 A MX2016012041 A MX 2016012041A
Authority
MX
Mexico
Prior art keywords
aripiprazol
formulations
higher injection
injection speeds
speeds
Prior art date
Application number
MX2016012041A
Other languages
English (en)
Other versions
MX376057B (es
Inventor
Vandiver Jennifer
B Hickey Migali
Original Assignee
Alkermes Pharma Ireland Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alkermes Pharma Ireland Ltd filed Critical Alkermes Pharma Ireland Ltd
Publication of MX2016012041A publication Critical patent/MX2016012041A/es
Publication of MX376057B publication Critical patent/MX376057B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Organic Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Pain & Pain Management (AREA)
  • Dispersion Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La presente invención se refiere a composiciones farmacéuticas que comprenden un compuesto de fórmula (I) que son útiles para la administración intramuscular de fármacos antipsicóticos utilizando tasas de inyección rápidas.
MX2016012041A 2014-03-20 2015-03-19 Formulaciones de aripiprazol que tienen mayores velocidades de inyeccion. MX376057B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201461955976P 2014-03-20 2014-03-20
PCT/US2015/021448 WO2015143145A1 (en) 2014-03-20 2015-03-19 Aripiprazole formulations having increased injection speeds

Publications (2)

Publication Number Publication Date
MX2016012041A true MX2016012041A (es) 2017-01-19
MX376057B MX376057B (es) 2025-03-07

Family

ID=54141031

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2016012041A MX376057B (es) 2014-03-20 2015-03-19 Formulaciones de aripiprazol que tienen mayores velocidades de inyeccion.
MX2020010839A MX2020010839A (es) 2014-03-20 2016-09-15 Formulaciones de aripiprazol que tienen mayores velocidades de inyeccion.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2020010839A MX2020010839A (es) 2014-03-20 2016-09-15 Formulaciones de aripiprazol que tienen mayores velocidades de inyeccion.

Country Status (12)

Country Link
US (8) US9452131B2 (es)
EP (1) EP3119399A4 (es)
JP (2) JP6524110B2 (es)
CN (2) CN110368360A (es)
AU (2) AU2015231278B2 (es)
BR (1) BR112016021535A8 (es)
CA (1) CA2943213C (es)
IL (2) IL247517B (es)
MA (1) MA39495A (es)
MX (2) MX376057B (es)
RU (1) RU2688233C2 (es)
WO (1) WO2015143145A1 (es)

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AU2012231160B2 (en) 2011-03-18 2017-04-06 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising sorbitan esters
CA2867121C (en) 2012-03-19 2021-05-25 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
ES2764383T3 (es) 2012-03-19 2020-06-03 Alkermes Pharma Ireland Ltd Composiciones farmacéuticas que comprenden ésteres de glicerol
US9999670B2 (en) 2012-03-19 2018-06-19 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising benzyl alcohol
JP6654042B2 (ja) 2012-09-19 2020-02-26 アルカームス ファーマ アイルランド リミテッド 貯蔵安定性が改善された医薬組成物
CN110368360A (zh) 2014-03-20 2019-10-25 奥克梅斯制药爱尔兰有限公司 具有增加的注射速度的阿立哌唑制剂
US10016415B2 (en) 2014-08-18 2018-07-10 Alkermes Pharma Ireland Limited Aripiprazole prodrug compositions
EP3658540B1 (en) * 2017-07-28 2021-12-01 Interquim, S.A. Process for the preparation of aripiprazole lauroxil
CN110204488A (zh) * 2018-02-28 2019-09-06 四川科伦药物研究院有限公司 一种月桂酰阿立哌唑的制备方法
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US12312315B2 (en) * 2019-07-12 2025-05-27 Interquim, S.A. Process for the preparation of aripiprazole lauroxil

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