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JPS568318A - Non oral long acting composition of haloperidol and bromperidol derivative - Google Patents

Non oral long acting composition of haloperidol and bromperidol derivative

Info

Publication number
JPS568318A
JPS568318A JP8082679A JP8082679A JPS568318A JP S568318 A JPS568318 A JP S568318A JP 8082679 A JP8082679 A JP 8082679A JP 8082679 A JP8082679 A JP 8082679A JP S568318 A JPS568318 A JP S568318A
Authority
JP
Japan
Prior art keywords
bromperidol
haloperidol
derivative
long acting
acting composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP8082679A
Other languages
Japanese (ja)
Inventor
Niimegiirusu Karurosu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceutica NV
Original Assignee
Janssen Pharmaceutica NV
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica NV filed Critical Janssen Pharmaceutica NV
Priority to JP8082679A priority Critical patent/JPS568318A/en
Priority to GB8018117A priority patent/GB2054371B/en
Priority to CY1255A priority patent/CY1255A/en
Priority to NL8003583A priority patent/NL190775C/en
Priority to BE0/201165A priority patent/BE883994A/en
Priority to FR8014443A priority patent/FR2460932A1/en
Priority to DE19803024305 priority patent/DE3024305A1/en
Publication of JPS568318A publication Critical patent/JPS568318A/en
Priority to KE3427A priority patent/KE3427A/en
Priority to HK833/84A priority patent/HK83384A/en
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Anesthesiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP8082679A 1979-06-28 1979-06-28 Non oral long acting composition of haloperidol and bromperidol derivative Pending JPS568318A (en)

Priority Applications (9)

Application Number Priority Date Filing Date Title
JP8082679A JPS568318A (en) 1979-06-28 1979-06-28 Non oral long acting composition of haloperidol and bromperidol derivative
GB8018117A GB2054371B (en) 1979-06-28 1980-06-03 Long-acting parenteral compositions of haloperidol and bromperidol derivatives
CY1255A CY1255A (en) 1979-06-28 1980-06-03 Long-acting parenteral compositions of haloperidol and bromperidol derivatives
NL8003583A NL190775C (en) 1979-06-28 1980-06-20 Pharmaceutical preparations with a psychotropic action containing an ester of substituted [(4-hydroxy-4-phenyl) piperidino] butyrophenones, and a method for preparing these preparations.
BE0/201165A BE883994A (en) 1979-06-28 1980-06-25 WERKWIJZE VOOR HET BEREIDEN VAN EEN PARENTERAAL GENEESMIDDEL VAN HALOPERIDOL- EN BROOMPERIDOL-DERIVATEN MET LANGDURIGE WERKING EN VOOR HET TOEPASSEN VAN DEZE GENEESMIDDELEN
FR8014443A FR2460932A1 (en) 1979-06-28 1980-06-27 HALOPERIDOL AND BROMPERIDOL COMPOUNDS AND LONG-EFFECTIVE PARENTERAL COMPOSITIONS CONTAINING
DE19803024305 DE3024305A1 (en) 1979-06-28 1980-06-27 PARENTERAL TRACKABLE PSYCHOTROPESIC MEDICINE WITH LONG-TERM EFFECT
KE3427A KE3427A (en) 1979-06-28 1984-07-20 Long-acting parenteral compositions of haloperidol and bromoperidol derivatives
HK833/84A HK83384A (en) 1979-06-28 1984-11-01 Long-acting parenteral compositions of haloperidol and bromperidol derivatives

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP8082679A JPS568318A (en) 1979-06-28 1979-06-28 Non oral long acting composition of haloperidol and bromperidol derivative

Publications (1)

Publication Number Publication Date
JPS568318A true JPS568318A (en) 1981-01-28

Family

ID=13729223

Family Applications (1)

Application Number Title Priority Date Filing Date
JP8082679A Pending JPS568318A (en) 1979-06-28 1979-06-28 Non oral long acting composition of haloperidol and bromperidol derivative

Country Status (9)

Country Link
JP (1) JPS568318A (en)
BE (1) BE883994A (en)
CY (1) CY1255A (en)
DE (1) DE3024305A1 (en)
FR (1) FR2460932A1 (en)
GB (1) GB2054371B (en)
HK (1) HK83384A (en)
KE (1) KE3427A (en)
NL (1) NL190775C (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6377857A (en) * 1986-09-11 1988-04-08 ハー・ルンドベツク・アクチエゼルスカベツト Acetate ester of haloperidol and its pharmaceutical composition
WO1994010982A1 (en) * 1992-11-17 1994-05-26 Yoshitomi Pharmaceutical Industries, Ltd. Sustained-release microsphere containing antipsychotic and process for producing the same

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK238190D0 (en) * 1990-10-03 1990-10-03 Lundbeck & Co As H DEPOT DERIVATIVES
EP0937053A1 (en) * 1996-10-31 1999-08-25 THE UNITED STATES OF AMERICA, as represented by the Secretary of the Department of Health and Human Services Sustained-release derivatives of hydroxylated analogs of substituted 1- 2 bis(aryl)methoxy]ethyl]-piperazines and -homopiperazines and their use as noncompetitive antagonists of dopamine reuptake
RU2178297C1 (en) * 2001-02-02 2002-01-20 Открытое акционерное общество "Химико-фармацевтический комбинат "Акрихин" Pharmaceutical composition eliciting antipsychotic and antiemetic action and method of its preparing
US8003617B2 (en) 2004-11-10 2011-08-23 Genzyme Corporation Methods of treating diabetes mellitus
US8716327B2 (en) 2006-05-09 2014-05-06 Genzyme Corporation Methods of treating fatty liver disease
EP2594563B1 (en) 2007-05-31 2018-07-18 Genzyme Corporation 2-acylaminopropanol-type glucosylceramide synthase inhibitors
WO2009045503A1 (en) 2007-10-05 2009-04-09 Genzyme Corporation Method of treating polycystic kidney diseases with ceramide derivatives
JP2011529500A (en) 2008-07-28 2011-12-08 ジェンザイム コーポレーション Glucosylceramide synthase inhibition for the treatment of collapsing glomerulopathy and other glomerular diseases
CA2738768C (en) 2008-10-03 2017-10-31 Genzyme Corporation 2-acylaminopropoanol-type glucosylceramide synthase inhibitors
LT2685979T (en) 2011-03-18 2016-12-12 Alkermes Pharma Ireland Limited Injectable pharmaceutical compositions comprising a water-insoluble anti-psychotic, sorbitan laurate and polysorbate 20
CN103301461B (en) * 2012-03-08 2018-09-07 江苏豪森药业集团有限公司 A kind of long acting injection and its preparation method and application
WO2013142198A1 (en) 2012-03-19 2013-09-26 Alkermes Pharma Ireland Limited Pharmaaceutical compositions comprising fatty acid esters
CA2867137C (en) 2012-03-19 2020-12-08 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising aripiprazole prodrugs and benzyl alcohol
ES2764383T3 (en) 2012-03-19 2020-06-03 Alkermes Pharma Ireland Ltd Pharmaceutical compositions comprising glycerol esters
NZ631345A (en) 2012-09-19 2017-06-30 Alkermes Pharma Ireland Ltd Pharmaceutical compositions having improved storage stability
BR112016021535A8 (en) 2014-03-20 2021-07-20 Alkermes Pharma Ireland Ltd kit comprising aripiprazole formulations having increased injection rates useful for the treatment of a central nervous system disorder and use
CA3092335A1 (en) 2018-03-05 2019-09-12 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy
CN113117092A (en) * 2020-01-14 2021-07-16 中国科学院上海药物研究所 Non-aqueous sustained-release drug delivery system
HUP2100259A1 (en) 2021-07-07 2023-01-28 Richter Gedeon Nyrt Controlled release injectable cariprazine formulation

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3408356A (en) * 1965-08-31 1968-10-29 Squibb & Sons Inc Long chain esters of 4'-fluoro-4-[4-hydroxy-4-(alpha, alpha, alpha-trifluorotolyl)piperi-dino]butyrophenone and the like

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1695194A1 (en) * 1966-07-11 1971-03-18 Hoffmann La Roche Process for the preparation of piperidine derivatives
US3850935A (en) * 1971-10-16 1974-11-26 Sumitomo Chemical Co Process for producing piperidine derivatives by degrading quaternary piperidinium salts

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3408356A (en) * 1965-08-31 1968-10-29 Squibb & Sons Inc Long chain esters of 4'-fluoro-4-[4-hydroxy-4-(alpha, alpha, alpha-trifluorotolyl)piperi-dino]butyrophenone and the like

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6377857A (en) * 1986-09-11 1988-04-08 ハー・ルンドベツク・アクチエゼルスカベツト Acetate ester of haloperidol and its pharmaceutical composition
WO1994010982A1 (en) * 1992-11-17 1994-05-26 Yoshitomi Pharmaceutical Industries, Ltd. Sustained-release microsphere containing antipsychotic and process for producing the same

Also Published As

Publication number Publication date
FR2460932B1 (en) 1984-11-16
DE3024305C2 (en) 1989-12-07
FR2460932A1 (en) 1981-01-30
DE3024305A1 (en) 1981-01-22
NL190775B (en) 1994-03-16
CY1255A (en) 1984-08-31
KE3427A (en) 1984-08-10
HK83384A (en) 1984-11-09
NL190775C (en) 1994-08-16
BE883994A (en) 1980-12-29
GB2054371B (en) 1983-08-03
NL8003583A (en) 1980-12-30
GB2054371A (en) 1981-02-18

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