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MX2011011797A - Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides. - Google Patents

Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides.

Info

Publication number
MX2011011797A
MX2011011797A MX2011011797A MX2011011797A MX2011011797A MX 2011011797 A MX2011011797 A MX 2011011797A MX 2011011797 A MX2011011797 A MX 2011011797A MX 2011011797 A MX2011011797 A MX 2011011797A MX 2011011797 A MX2011011797 A MX 2011011797A
Authority
MX
Mexico
Prior art keywords
phenylamides
substituted
phenyllureas
receptor ligands
vanilloid receptor
Prior art date
Application number
MX2011011797A
Other languages
English (en)
Inventor
Sven Frormann
Klaus Schiene
Thomas Christoph
Robert Frank
Gregor Bahrenberg
Jean De Vry
Jeewoo Lee
Nils Damann
Bernhard Lesch
Yong-Soo Kim
Myeon-Seop Kim
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40908456&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2011011797(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of MX2011011797A publication Critical patent/MX2011011797A/es

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    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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  • Veterinary Medicine (AREA)
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Abstract

La invención se refiere a fenilureas y fenilamidas sustituidas de la fórmula (I), a procesos para su preparación, a composiciones farmacéuticas que contienen estos compuestos y también al uso de estos compuestos para preparar composiciones farmacéuticas. (ver fórmula (I)).
MX2011011797A 2009-05-07 2010-05-06 Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides. MX2011011797A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17628409P 2009-05-07 2009-05-07
EP09006237 2009-05-07
PCT/EP2010/002786 WO2010127856A1 (en) 2009-05-07 2010-05-06 Substituted phenyllureas and phenylamides as vanilloid receptor ligands

Publications (1)

Publication Number Publication Date
MX2011011797A true MX2011011797A (es) 2011-11-29

Family

ID=40908456

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2011011797A MX2011011797A (es) 2009-05-07 2010-05-06 Fenilureas y fenilamidas sustituidas como ligandos del receptor de vanilloides.

Country Status (20)

Country Link
US (2) US8592471B2 (es)
EP (1) EP2427435B1 (es)
JP (1) JP5745505B2 (es)
KR (1) KR101746016B1 (es)
CN (2) CN102428071A (es)
AR (1) AR076752A1 (es)
AU (1) AU2010244685B2 (es)
BR (1) BRPI1011043B8 (es)
CA (1) CA2759951C (es)
CO (1) CO6440569A2 (es)
EC (1) ECSP11011433A (es)
ES (1) ES2640257T3 (es)
IL (1) IL215661A (es)
MX (1) MX2011011797A (es)
NZ (1) NZ595759A (es)
PE (1) PE20120374A1 (es)
RU (1) RU2553392C2 (es)
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