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MX2013005008A - Derivados de carboxamida y urea heteroaromaticos sustituidos como ligandos del receptor vanilloide. - Google Patents

Derivados de carboxamida y urea heteroaromaticos sustituidos como ligandos del receptor vanilloide.

Info

Publication number
MX2013005008A
MX2013005008A MX2013005008A MX2013005008A MX2013005008A MX 2013005008 A MX2013005008 A MX 2013005008A MX 2013005008 A MX2013005008 A MX 2013005008A MX 2013005008 A MX2013005008 A MX 2013005008A MX 2013005008 A MX2013005008 A MX 2013005008A
Authority
MX
Mexico
Prior art keywords
urea derivatives
substituted heteroaromatic
receptor ligands
vanilloid receptor
heteroaromatic carboxamide
Prior art date
Application number
MX2013005008A
Other languages
English (en)
Inventor
Thomas Christoph
Robert Frank
Jeewoo Lee
Bernhard Lesch
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of MX2013005008A publication Critical patent/MX2013005008A/es

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    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

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  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Diabetes (AREA)
  • Virology (AREA)
  • Urology & Nephrology (AREA)
  • Obesity (AREA)
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  • Immunology (AREA)
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Abstract

La invención se relaciona con derivados de carboxamida y urea heteroaromáticos sustituidos, con procesos para la preparación de los mismos, con composiciones farmacéuticas que comprenden esos compuestos y también con el uso de esos compuestos para preparar composiciones farmacéuticas.
MX2013005008A 2010-11-10 2011-11-09 Derivados de carboxamida y urea heteroaromaticos sustituidos como ligandos del receptor vanilloide. MX2013005008A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP10014449 2010-11-10
PCT/EP2011/005628 WO2012062462A1 (en) 2010-11-10 2011-11-09 Substituted heteroaromatic carboxamide and urea derivatives as vanilloid receptor ligands

Publications (1)

Publication Number Publication Date
MX2013005008A true MX2013005008A (es) 2013-08-01

Family

ID=43501425

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2013005008A MX2013005008A (es) 2010-11-10 2011-11-09 Derivados de carboxamida y urea heteroaromaticos sustituidos como ligandos del receptor vanilloide.

Country Status (10)

Country Link
US (1) US20120115903A1 (es)
EP (1) EP2638034A1 (es)
JP (1) JP2013545740A (es)
AR (1) AR083817A1 (es)
AU (1) AU2011328520A1 (es)
BR (1) BR112013010768A2 (es)
CA (1) CA2816769A1 (es)
MX (1) MX2013005008A (es)
TW (1) TW201305139A (es)
WO (1) WO2012062462A1 (es)

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