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MX2009005264A - Mimeticos de glucocorticoides, metodos para su fabricacion, composiciones farmaceuticas y usos de los mismos. - Google Patents

Mimeticos de glucocorticoides, metodos para su fabricacion, composiciones farmaceuticas y usos de los mismos.

Info

Publication number
MX2009005264A
MX2009005264A MX2009005264A MX2009005264A MX2009005264A MX 2009005264 A MX2009005264 A MX 2009005264A MX 2009005264 A MX2009005264 A MX 2009005264A MX 2009005264 A MX2009005264 A MX 2009005264A MX 2009005264 A MX2009005264 A MX 2009005264A
Authority
MX
Mexico
Prior art keywords
methods
pharmaceutical compositions
making
compounds
glucocorticoid mimetics
Prior art date
Application number
MX2009005264A
Other languages
English (en)
Inventor
Daniel Kuzmich
Hossein Razavi
Michael Jason Burke
Disalvo Darren
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of MX2009005264A publication Critical patent/MX2009005264A/es

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    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D498/04—Ortho-condensed systems
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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Abstract

Compuestos de Fórmula (IA) (ver fórmula IA) y de Fórmula (IB) (ver fórmula IB) en las que R1, R2, R3, A, B, C, D, E, G, X, Y y Z son como se definen en la presente memoria, o un tautómero, profármaco, solvato o sal de los mismos; composiciones farmacéuticas que contienen dichos compuestos, métodos para modular la función del receptor de glucocorticoides y métodos para tratar estados de enfermedad o afecciones mediadas por la función del receptor de glucocorticoides o caracterizadas por procesos inflamatorios, alérgicos o proliferativos en un paciente usando estos compuestos.
MX2009005264A 2006-12-06 2007-11-29 Mimeticos de glucocorticoides, metodos para su fabricacion, composiciones farmaceuticas y usos de los mismos. MX2009005264A (es)

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BRPI0720131A2 (pt) 2014-02-04
RU2009125614A (ru) 2011-01-20
WO2008070507A2 (en) 2008-06-12
ZA200902803B (en) 2010-05-26
WO2008070507A3 (en) 2008-09-12
CA2671990A1 (en) 2008-06-12
AU2007329548A1 (en) 2008-06-12
KR20090097908A (ko) 2009-09-16
CN101547909A (zh) 2009-09-30
JP2010512331A (ja) 2010-04-22
US8658637B2 (en) 2014-02-25
US20100197678A1 (en) 2010-08-05

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