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MA32275B1 - Preparations orales et injectables de composes de tetracycline - Google Patents

Preparations orales et injectables de composes de tetracycline

Info

Publication number
MA32275B1
MA32275B1 MA33281A MA33281A MA32275B1 MA 32275 B1 MA32275 B1 MA 32275B1 MA 33281 A MA33281 A MA 33281A MA 33281 A MA33281 A MA 33281A MA 32275 B1 MA32275 B1 MA 32275B1
Authority
MA
Morocco
Prior art keywords
oral
injectable preparations
tetracycline compounds
preparations
relates
Prior art date
Application number
MA33281A
Other languages
Arabic (ar)
English (en)
Inventor
Sean Johnston
Original Assignee
Paratek Pharm Innc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41114256&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA32275(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Paratek Pharm Innc filed Critical Paratek Pharm Innc
Publication of MA32275B1 publication Critical patent/MA32275B1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/65Tetracyclines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

La présente invention concerne des préparations injectables et orales d'un composé de tétracycline. Dans un mode de réalisation, l'invention concerne une préparation orale de composé de 9-aminométhyl tétracycline, ou de son sel, sous forme de comprimé ou de capsule. Les préparations peuvent être utilisées, par exemple, pour traiter des infections.
MA33281A 2008-03-28 2010-10-25 Preparations orales et injectables de composes de tetracycline MA32275B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4039808P 2008-03-28 2008-03-28
PCT/US2009/001973 WO2009120389A1 (fr) 2008-03-28 2009-03-30 Préparations orales et injectables de composés de tétracycline

Publications (1)

Publication Number Publication Date
MA32275B1 true MA32275B1 (fr) 2011-05-02

Family

ID=41114256

Family Applications (1)

Application Number Title Priority Date Filing Date
MA33281A MA32275B1 (fr) 2008-03-28 2010-10-25 Preparations orales et injectables de composes de tetracycline

Country Status (30)

Country Link
US (2) US9314475B2 (fr)
EP (3) EP3348258B1 (fr)
JP (8) JP2011515473A (fr)
KR (3) KR101746228B1 (fr)
CN (1) CN102046177B (fr)
AU (1) AU2009229174A1 (fr)
BR (2) BRPI0909211B8 (fr)
CA (2) CA2719751C (fr)
CL (1) CL2010000281A1 (fr)
CO (1) CO6300935A2 (fr)
CY (2) CY1120240T1 (fr)
DK (2) DK3348258T3 (fr)
EC (1) ECSP10010576A (fr)
ES (2) ES2674708T3 (fr)
HR (2) HRP20180836T1 (fr)
HU (2) HUE052201T2 (fr)
IL (1) IL208440A0 (fr)
LT (2) LT3348258T (fr)
MA (1) MA32275B1 (fr)
MX (1) MX2010010585A (fr)
NO (1) NO2271348T3 (fr)
NZ (1) NZ588428A (fr)
PL (2) PL3348258T3 (fr)
PT (2) PT2271348T (fr)
RU (1) RU2010144130A (fr)
SI (2) SI2271348T1 (fr)
TR (1) TR201806893T4 (fr)
UA (2) UA122762C2 (fr)
WO (1) WO2009120389A1 (fr)
ZA (1) ZA201007013B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BRPI0908951A2 (pt) 2008-03-05 2017-01-17 Paratek Pharm Innc compostos de minociclina e método de uso dos mesmos
TW202332671A (zh) * 2008-05-19 2023-08-16 美商Prtk Spv2公司 四環素化合物之甲苯磺酸鹽及同素異形體
ES2613738T3 (es) 2010-05-12 2017-05-25 Rempex Pharmaceuticals, Inc. Composiciones de tetraciclina
US10238670B2 (en) * 2016-05-02 2019-03-26 Paratek Pharmaceuticals, Inc. 9-aminomethyl minocycline compounds and methods of use thereof in urinary tract infection (UTI) treatment
US10166912B2 (en) 2016-08-19 2019-01-01 Sl Corporation Automotive LED driving apparatus
SG10201913599RA (en) 2016-11-01 2020-02-27 Paratek Pharm Innc 9-aminomethyl minocycline compounds and use thereof in treating community-acquired bacterial pneumonia (cabp)
CN113164456A (zh) * 2018-09-04 2021-07-23 帕拉特克药品公司 使用四环素化合物治疗分枝杆菌感染的方法
MX2022008103A (es) * 2019-12-30 2022-09-19 Deciphera Pharmaceuticals Llc Formulaciones de inhibidores de la cinasa amorfa y metodos de estas.
PT117254B (pt) 2021-05-26 2024-04-18 Hovione Farm S A Método de síntese de compostos 9-aminometil tetraciclinas

Family Cites Families (53)

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Also Published As

Publication number Publication date
PL2271348T3 (pl) 2018-08-31
UA122762C2 (uk) 2021-01-06
KR101835574B1 (ko) 2018-03-08
JP5940119B2 (ja) 2016-06-29
ES2836448T3 (es) 2021-06-25
PT2271348T (pt) 2018-04-16
JP2011515473A (ja) 2011-05-19
KR101746228B1 (ko) 2017-06-12
HRP20180836T1 (hr) 2018-07-27
BRPI0909211B8 (pt) 2021-05-25
AU2009229174A1 (en) 2009-10-01
BRPI0909211B1 (pt) 2020-08-25
JP2023144043A (ja) 2023-10-06
JP2016145260A (ja) 2016-08-12
MX2010010585A (es) 2010-11-09
EP2271348B1 (fr) 2018-03-28
CN102046177B (zh) 2012-12-19
UA109627C2 (uk) 2015-09-25
SI3348258T1 (sl) 2020-12-31
US9314475B2 (en) 2016-04-19
US20160279151A1 (en) 2016-09-29
ZA201007013B (en) 2013-11-27
JP2014221820A (ja) 2014-11-27
ES2674708T3 (es) 2018-07-03
BR122020011180B1 (pt) 2021-03-23
KR20160105532A (ko) 2016-09-06
JP6412521B2 (ja) 2018-10-24
KR20180026799A (ko) 2018-03-13
WO2009120389A1 (fr) 2009-10-01
BRPI0909211A2 (pt) 2016-11-29
CL2010000281A1 (es) 2012-03-30
NO2271348T3 (fr) 2018-08-25
CY1123382T1 (el) 2021-12-31
NZ588428A (en) 2012-08-31
ECSP10010576A (es) 2010-12-30
RU2010144130A (ru) 2012-05-10
TR201806893T4 (tr) 2018-06-21
CO6300935A2 (es) 2011-07-21
US20100056638A1 (en) 2010-03-04
WO2009120389A8 (fr) 2010-05-14
EP3348258B1 (fr) 2020-09-09
BR122020011180B8 (pt) 2021-07-27
IL208440A0 (en) 2010-12-30
DK2271348T3 (en) 2018-06-14
HUE052201T2 (hu) 2021-04-28
CY1120240T1 (el) 2019-07-10
CA2984301C (fr) 2020-10-27
CA2719751A1 (fr) 2009-10-01
JP2018203778A (ja) 2018-12-27
EP3789030A1 (fr) 2021-03-10
JP2021167355A (ja) 2021-10-21
HUE038257T2 (hu) 2018-10-29
PT3348258T (pt) 2020-11-25
CA2719751C (fr) 2018-01-02
JP6577645B2 (ja) 2019-09-18
HRP20201883T1 (hr) 2021-01-22
KR101893740B1 (ko) 2018-08-30
LT2271348T (lt) 2018-06-25
EP2271348A1 (fr) 2011-01-12
JP2025137721A (ja) 2025-09-19
CN102046177A (zh) 2011-05-04
EP3348258A1 (fr) 2018-07-18
CA2984301A1 (fr) 2009-10-01
KR20110008057A (ko) 2011-01-25
JP2019196408A (ja) 2019-11-14
LT3348258T (lt) 2020-12-10
SI2271348T1 (en) 2018-08-31
HK1257928A1 (en) 2019-11-01
EP2271348A4 (fr) 2011-05-25
PL3348258T3 (pl) 2021-03-08
DK3348258T3 (da) 2020-12-07

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