ZA9410003B - Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation - Google Patents

Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation

Info

Publication number: ZA9410003B
Authority: ZA; South Africa
Prior art keywords: crystalline; processes; preparation; acid derivatives; neuraminic acid
Prior art date: 1993-12-17

Application number

ZA9410003A

Other languages

English (en)

Inventor

Christopher Williamson

William James White

Vipulkumar Patel

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-12-17

Filing date

1994-12-15

Publication date

1995-07-25

1994-12-15 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

1995-07-25 Publication of ZA9410003B publication Critical patent/ZA9410003B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Health & Medical Sciences (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Virology (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrane Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

ZA9410003A 1993-12-17 1994-12-15 Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation ZA9410003B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB939325841A GB9325841D0 (en)	1993-12-17	1993-12-17	Chemical compounds

Publications (1)

Publication Number	Publication Date
ZA9410003B true ZA9410003B (en)	1995-07-25

Family

ID=10746778

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA9410003A ZA9410003B (en)	1993-12-17	1994-12-15	Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation

Country Status (43)

Country	Link
US (2)	US6294572B1 (el)
EP (1)	EP0734382B1 (el)
JP (1)	JP3317972B2 (el)
KR (1)	KR100403256B1 (el)
CN (2)	CN1132829C (el)
AP (2)	AP541A (el)
AT (1)	ATE199255T1 (el)
BG (1)	BG63338B1 (el)
BR (2)	BR9408340A (el)
CA (1)	CA2177990C (el)
CO (1)	CO4340619A1 (el)
CZ (1)	CZ289234B6 (el)
DE (1)	DE69426726T2 (el)
DK (1)	DK0734382T3 (el)
EE (1)	EE03353B1 (el)
EG (1)	EG20597A (el)
ES (1)	ES2155517T3 (el)
FI (1)	FI120453B (el)
GB (1)	GB9325841D0 (el)
GR (1)	GR3035681T3 (el)
HR (1)	HRP941001B1 (el)
HU (1)	HU221971B1 (el)
IL (1)	IL112011A (el)
IS (1)	IS4240A (el)
MA (1)	MA23396A1 (el)
MY (1)	MY116221A (el)
NO (1)	NO314759B1 (el)
NZ (1)	NZ277789A (el)
OA (2)	OA10325A (el)
PE (1)	PE31095A1 (el)
PL (1)	PL186384B1 (el)
PT (1)	PT734382E (el)
RO (1)	RO114792B1 (el)
RU (1)	RU2134690C1 (el)
SA (1)	SA94150417B1 (el)
SG (1)	SG46669A1 (el)
SI (1)	SI0734382T1 (el)
SK (1)	SK282972B6 (el)
SV (1)	SV1994000076A (el)
TW (1)	TW452577B (el)
UA (1)	UA46723C2 (el)
WO (1)	WO1995016680A1 (el)
ZA (1)	ZA9410003B (el)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9325841D0 (en) *	1993-12-17	1994-02-23	Glaxo Group Ltd	Chemical compounds
US5866601A (en) *	1995-02-27	1999-02-02	Gilead Sciences, Inc.	Carbocyclic compounds
ATE305453T1 (de) *	1995-02-27	2005-10-15	Gilead Sciences Inc	Selektive inhibitoren viraler oder bakterieller neuraminidase
US5763483A (en) *	1995-12-29	1998-06-09	Gilead Sciences, Inc.	Carbocyclic compounds
US6340702B1 (en)	1996-07-22	2002-01-22	Sankyo Company, Limited	Neuraminic acid derivatives, their preparation and their medical use
US6451766B1 (en)	1996-07-22	2002-09-17	Sankyo Company, Limited	Neuraminic acid derivatives, their preparation and their medical use
PT823428E (pt) *	1996-07-22	2002-04-29	Sankyo Co	Derivados do acido neuraminico sua preparacao e sua utilizacao em medicina
US6518438B2 (en)	1996-08-23	2003-02-11	Gilead Sciences, Inc.	Preparation of cyclohexene carboxylate derivatives
US5859284A (en)	1996-08-23	1999-01-12	Gilead Sciences, Inc.	Preparation of carbocyclic compounds
US5994377A (en)	1996-10-21	1999-11-30	Gilead Sciences, Inc.	Piperidine compounds
US5886213A (en) *	1997-08-22	1999-03-23	Gilead Sciences, Inc.	Preparation of carbocyclic compounds
TW480247B (en) *	1997-12-12	2002-03-21	Gilead Sciences Inc	Novel compounds useful as neuraminidase inhibitors and pharmaceutical compositions containing same
TWI291462B (en)	2000-04-25	2007-12-21	Daiichi Sankyo Co Ltd	Hydrate crystal of neuraminic acid compound
US20080063722A1 (en) *	2006-09-08	2008-03-13	Advanced Inhalation Research, Inc.	Composition of a Spray-Dried Powder for Pulmonary Delivery of a Long Acting Neuraminidase Inhibitor (LANI)
EP2960237A1 (en) *	2011-12-16	2015-12-30	Daiichi Sankyo Company, Limited	Method for producing neuraminic acid derivative
CN109232677B (zh) *	2018-10-18	2021-12-28	中国科学院合肥物质科学研究院	一种使n-乙酰神经氨酸水合物转化为n-乙酰神经氨酸的方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SU469694A1 (ru) *	1972-12-22	1975-05-05	Московский Ордена Трудового Красного Знамени Институт Тонкой Химической Технологии Им.М.В.Ломоносова	Способ получени 2-алкокси-6-алкил (арил)- -дигидропиранов
AP249A (en) *	1990-04-24	1993-03-17	Biota Scient Management Pty Ltd	Anti-viral compounds.
AU659501B2 (en) *	1991-10-23	1995-05-18	Biota Scientific Management Pty Ltd	Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of alpha-D-neuraminic acid
GB9126725D0 (en) *	1991-12-17	1992-02-12	Glaxo Group Ltd	Process
US5639786A (en)	1992-12-04	1997-06-17	Biota Scientific Management, Pty., Ltd.	Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of α-D-neuraninic acid
GB9325841D0 (en) *	1993-12-17	1994-02-23	Glaxo Group Ltd	Chemical compounds

1993
- 1993-12-17 GB GB939325841A patent/GB9325841D0/en active Pending
1994
- 1994-12-02 TW TW083111229A patent/TW452577B/zh not_active IP Right Cessation
- 1994-12-13 IS IS4240A patent/IS4240A/is unknown
- 1994-12-15 PT PT95904472T patent/PT734382E/pt unknown
- 1994-12-15 CN CN94194973A patent/CN1132829C/zh not_active Expired - Lifetime
- 1994-12-15 CN CNA2003101199989A patent/CN1502621A/zh active Pending
- 1994-12-15 DE DE69426726T patent/DE69426726T2/de not_active Expired - Lifetime
- 1994-12-15 BR BR9408340A patent/BR9408340A/pt not_active Application Discontinuation
- 1994-12-15 EP EP95904472A patent/EP0734382B1/en not_active Expired - Lifetime
- 1994-12-15 EG EG79094A patent/EG20597A/xx active
- 1994-12-15 AP APAP/P/1994/000705A patent/AP541A/en active
- 1994-12-15 UA UA96062328A patent/UA46723C2/uk unknown
- 1994-12-15 SI SI9430333T patent/SI0734382T1/xx unknown
- 1994-12-15 HR HR941001A patent/HRP941001B1/xx not_active IP Right Cessation
- 1994-12-15 SK SK785-96A patent/SK282972B6/sk not_active IP Right Cessation
- 1994-12-15 NZ NZ277789A patent/NZ277789A/en not_active IP Right Cessation
- 1994-12-15 SV SV1994000076A patent/SV1994000076A/es active IP Right Grant
- 1994-12-15 CA CA002177990A patent/CA2177990C/en not_active Expired - Lifetime
- 1994-12-15 JP JP51653195A patent/JP3317972B2/ja not_active Expired - Lifetime
- 1994-12-15 CZ CZ19961693A patent/CZ289234B6/cs not_active IP Right Cessation
- 1994-12-15 MY MYPI94003357A patent/MY116221A/en unknown
- 1994-12-15 ES ES95904472T patent/ES2155517T3/es not_active Expired - Lifetime
- 1994-12-15 CO CO94056728A patent/CO4340619A1/es unknown
- 1994-12-15 WO PCT/EP1994/004154 patent/WO1995016680A1/en not_active Ceased
- 1994-12-15 MA MA23724A patent/MA23396A1/fr unknown
- 1994-12-15 ZA ZA9410003A patent/ZA9410003B/xx unknown
- 1994-12-15 PL PL94315055A patent/PL186384B1/pl unknown
- 1994-12-15 PE PE1994257245A patent/PE31095A1/es not_active Application Discontinuation
- 1994-12-15 AT AT95904472T patent/ATE199255T1/de active
- 1994-12-15 RU RU96115122A patent/RU2134690C1/ru active Protection Beyond IP Right Term
- 1994-12-15 RO RO96-01195A patent/RO114792B1/ro unknown
- 1994-12-15 DK DK95904472T patent/DK0734382T3/da active
- 1994-12-15 AP APAP/P/1996/000810A patent/AP9600810A0/en unknown
- 1994-12-15 HU HU9601642A patent/HU221971B1/hu active IP Right Grant
- 1994-12-15 SG SG1996007725A patent/SG46669A1/en unknown
- 1994-12-15 EE EE9600135A patent/EE03353B1/xx unknown
- 1994-12-15 KR KR1019960703180A patent/KR100403256B1/ko not_active Expired - Lifetime
- 1994-12-16 IL IL11201194A patent/IL112011A/en not_active IP Right Cessation
- 1994-12-28 SA SA94150417A patent/SA94150417B1/ar unknown
1996
- 1996-06-13 FI FI962464A patent/FI120453B/fi not_active IP Right Cessation
- 1996-06-14 NO NO19962545A patent/NO314759B1/no not_active IP Right Cessation
- 1996-06-14 OA OA60842A patent/OA10325A/fr unknown
- 1996-07-08 BG BG100709A patent/BG63338B1/bg unknown
1997
- 1997-05-13 BR BRPP1100548-KB1A patent/BR1100548KB1/pt unknown
1999
- 1999-07-02 US US09/346,583 patent/US6294572B1/en not_active Expired - Lifetime
2000
- 2000-01-06 OA OA1200000004A patent/OA11275A/fr unknown
2001
- 2001-03-30 GR GR20010400531T patent/GR3035681T3/el unknown
- 2001-09-24 US US09/961,074 patent/US20020037865A1/en not_active Abandoned

Also Published As

Publication number	Publication date
ATE199255T1 (de)	2001-03-15
HRP941001A2 (en)	1997-06-30
FI962464L (fi)	1996-06-13
IL112011A (en)	1998-08-16
AU1314495A (en)	1995-07-03
CZ289234B6 (cs)	2001-12-12
MY116221A (en)	2003-12-31
US20020037865A1 (en)	2002-03-28
AP9600810A0 (en)	1996-07-31
OA11275A (en)	2002-11-20
NZ277789A (en)	1999-04-29
NO962545L (no)	1996-06-14
CA2177990C (en)	2000-04-25
PT734382E (pt)	2001-06-29
SK78596A3 (en)	1997-03-05
BR9408340A (pt)	1997-08-19
BG63338B1 (bg)	2001-10-31
CZ169396A3 (en)	1996-11-13
IS4240A (is)	1995-06-18
EP0734382B1 (en)	2001-02-21
EG20597A (en)	1999-09-30
HRP941001B1 (en)	2001-06-30
SI0734382T1 (en)	2001-08-31
RU2134690C1 (ru)	1999-08-20
PE31095A1 (es)	1995-10-18
HUT74938A (en)	1997-03-28
IL112011A0 (en)	1995-03-15
HK1014187A1 (en)	1999-09-24
UA46723C2 (uk)	2002-06-17
SV1994000076A (es)	1995-10-26
PL315055A1 (en)	1996-09-30
CN1132829C (zh)	2003-12-31
EP0734382A1 (en)	1996-10-02
DE69426726T2 (de)	2001-06-21
CN1142820A (zh)	1997-02-12
US6294572B1 (en)	2001-09-25
ES2155517T3 (es)	2001-05-16
OA10325A (en)	1997-10-07
AP541A (en)	1996-10-01
PL186384B1 (pl)	2004-01-30
WO1995016680A1 (en)	1995-06-22
KR100403256B1 (ko)	2004-04-30
SA94150417B1 (ar)	2005-12-18
FI120453B (fi)	2009-10-30
AP9400705A0 (en)	1995-01-31
CA2177990A1 (en)	1995-06-22
GB9325841D0 (en)	1994-02-23
BR1100548KB1 (pt)	2011-11-01
BG100709A (bg)	1997-01-31
MA23396A1 (fr)	1995-07-01
HU9601642D0 (en)	1996-08-28
TW452577B (en)	2001-09-01
EE03353B1 (et)	2001-02-15
DE69426726D1 (de)	2001-03-29
NO962545D0 (no)	1996-06-14
JPH09506601A (ja)	1997-06-30
NO314759B1 (no)	2003-05-19
DK0734382T3 (da)	2001-03-19
SG46669A1 (en)	1998-02-20
RO114792B1 (ro)	1999-07-30
HU221971B1 (hu)	2003-03-28
CN1502621A (zh)	2004-06-09
JP3317972B2 (ja)	2002-08-26
SK282972B6 (sk)	2003-01-09
AU689185B2 (en)	1998-03-26
CO4340619A1 (es)	1996-07-30
FI962464A0 (fi)	1996-06-13
GR3035681T3 (en)	2001-06-29

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SI0734382T1 (en)	2001-08-31	Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation
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