FI962464L - Kiteisiä N-asetyyliamiinihappojohdannaisia ja menetelmiä niiden valmistamiseksi - Google Patents

Kiteisiä N-asetyyliamiinihappojohdannaisia ja menetelmiä niiden valmistamiseksi Download PDF

Info

Publication number: FI962464L
Authority: FI; Finland
Prior art keywords: crystalline; preparation; methods; acid derivatives; acetylamino acid
Prior art date: 1993-12-17

Application number

FI962464A

Other languages

English (en)

Swedish (sv)

Other versions

FI962464A0 (fi

FI120453B (fi

Inventor

Christopher Williamson

William James White

Vipulkumar Pater

Original Assignee

Biota Scient Management

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-12-17

Filing date

1996-06-13

Publication date

1996-06-13

1996-06-13 Application filed by Biota Scient Management filed Critical Biota Scient Management

1996-06-13 Publication of FI962464A0 publication Critical patent/FI962464A0/fi

1996-06-13 Publication of FI962464L publication Critical patent/FI962464L/fi

2009-10-30 Application granted granted Critical

2009-10-30 Publication of FI120453B publication Critical patent/FI120453B/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Health & Medical Sciences (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Virology (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrane Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

FI962464A 1993-12-17 1996-06-13 Menetelmä kiteisten N-asetyylineuramiinihappojohdannaisten valmistamiseksi FI120453B (fi)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
GB9325841		1993-12-17
GB939325841A GB9325841D0 (en)	1993-12-17	1993-12-17	Chemical compounds
PCT/EP1994/004154 WO1995016680A1 (en)	1993-12-17	1994-12-15	Crystalline n-acetyl neuraminic acid derivatives and processes for their preparation
EP9404154		1994-12-15

Publications (3)

Publication Number	Publication Date
FI962464A0 FI962464A0 (fi)	1996-06-13
FI962464L true FI962464L (fi)	1996-06-13
FI120453B FI120453B (fi)	2009-10-30

Family

ID=10746778

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI962464A FI120453B (fi)	1993-12-17	1996-06-13	Menetelmä kiteisten N-asetyylineuramiinihappojohdannaisten valmistamiseksi

Country Status (43)

Country	Link
US (2)	US6294572B1 (fi)
EP (1)	EP0734382B1 (fi)
JP (1)	JP3317972B2 (fi)
KR (1)	KR100403256B1 (fi)
CN (2)	CN1132829C (fi)
AP (2)	AP9600810A0 (fi)
AT (1)	ATE199255T1 (fi)
BG (1)	BG63338B1 (fi)
BR (2)	BR9408340A (fi)
CA (1)	CA2177990C (fi)
CO (1)	CO4340619A1 (fi)
CZ (1)	CZ289234B6 (fi)
DE (1)	DE69426726T2 (fi)
DK (1)	DK0734382T3 (fi)
EE (1)	EE03353B1 (fi)
EG (1)	EG20597A (fi)
ES (1)	ES2155517T3 (fi)
FI (1)	FI120453B (fi)
GB (1)	GB9325841D0 (fi)
GR (1)	GR3035681T3 (fi)
HR (1)	HRP941001B1 (fi)
HU (1)	HU221971B1 (fi)
IL (1)	IL112011A (fi)
IS (1)	IS4240A (fi)
MA (1)	MA23396A1 (fi)
MY (1)	MY116221A (fi)
NO (1)	NO314759B1 (fi)
NZ (1)	NZ277789A (fi)
OA (2)	OA10325A (fi)
PE (1)	PE31095A1 (fi)
PL (1)	PL186384B1 (fi)
PT (1)	PT734382E (fi)
RO (1)	RO114792B1 (fi)
RU (1)	RU2134690C1 (fi)
SA (1)	SA94150417B1 (fi)
SG (1)	SG46669A1 (fi)
SI (1)	SI0734382T1 (fi)
SK (1)	SK282972B6 (fi)
SV (1)	SV1994000076A (fi)
TW (1)	TW452577B (fi)
UA (1)	UA46723C2 (fi)
WO (1)	WO1995016680A1 (fi)
ZA (1)	ZA9410003B (fi)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9325841D0 (en) *	1993-12-17	1994-02-23	Glaxo Group Ltd	Chemical compounds
US5866601A (en) *	1995-02-27	1999-02-02	Gilead Sciences, Inc.	Carbocyclic compounds
CN100409844C (zh) *	1995-02-27	2008-08-13	吉里德科学公司	神经氨酸苷酶抑制剂
US5763483A (en) *	1995-12-29	1998-06-09	Gilead Sciences, Inc.	Carbocyclic compounds
US6451766B1 (en)	1996-07-22	2002-09-17	Sankyo Company, Limited	Neuraminic acid derivatives, their preparation and their medical use
ATE211468T1 (de) *	1996-07-22	2002-01-15	Sankyo Co	Neuraminsäuredervate, ihre herstellung und medizinische verwendung
US6340702B1 (en)	1996-07-22	2002-01-22	Sankyo Company, Limited	Neuraminic acid derivatives, their preparation and their medical use
US6518438B2 (en)	1996-08-23	2003-02-11	Gilead Sciences, Inc.	Preparation of cyclohexene carboxylate derivatives
US5859284A (en)	1996-08-23	1999-01-12	Gilead Sciences, Inc.	Preparation of carbocyclic compounds
US5994377A (en) *	1996-10-21	1999-11-30	Gilead Sciences, Inc.	Piperidine compounds
US5886213A (en) *	1997-08-22	1999-03-23	Gilead Sciences, Inc.	Preparation of carbocyclic compounds
TW480247B (en) *	1997-12-12	2002-03-21	Gilead Sciences Inc	Novel compounds useful as neuraminidase inhibitors and pharmaceutical compositions containing same
TWI291462B (en) *	2000-04-25	2007-12-21	Daiichi Sankyo Co Ltd	Hydrate crystal of neuraminic acid compound
US20080063722A1 (en) *	2006-09-08	2008-03-13	Advanced Inhalation Research, Inc.	Composition of a Spray-Dried Powder for Pulmonary Delivery of a Long Acting Neuraminidase Inhibitor (LANI)
CA2859296C (en) *	2011-12-16	2016-10-11	Daiichi Sankyo Company, Limited	Method for manufacturing neuraminic acid derivatives
CN109232677B (zh) *	2018-10-18	2021-12-28	中国科学院合肥物质科学研究院	一种使n-乙酰神经氨酸水合物转化为n-乙酰神经氨酸的方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SU469694A1 (ru) *	1972-12-22	1975-05-05	Московский Ордена Трудового Красного Знамени Институт Тонкой Химической Технологии Им.М.В.Ломоносова	Способ получени 2-алкокси-6-алкил (арил)- -дигидропиранов
CZ288492B6 (en) *	1990-04-24	2001-06-13	Biota Scient Management	Derivatives of alpha-D-neuraminic acid, process of their preparation, their use and pharmaceutical preparations based thereon
AU659501B2 (en) *	1991-10-23	1995-05-18	Biota Scientific Management Pty Ltd	Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of alpha-D-neuraminic acid
GB9126725D0 (en) *	1991-12-17	1992-02-12	Glaxo Group Ltd	Process
US5639786A (en)	1992-12-04	1997-06-17	Biota Scientific Management, Pty., Ltd.	Antiviral 4-substituted-2-deoxy-2,3-didehydro-derivatives of α-D-neuraninic acid
GB9325841D0 (en) *	1993-12-17	1994-02-23	Glaxo Group Ltd	Chemical compounds

1993
- 1993-12-17 GB GB939325841A patent/GB9325841D0/en active Pending
1994
- 1994-12-02 TW TW083111229A patent/TW452577B/zh not_active IP Right Cessation
- 1994-12-13 IS IS4240A patent/IS4240A/is unknown
- 1994-12-15 MY MYPI94003357A patent/MY116221A/en unknown
- 1994-12-15 EG EG79094A patent/EG20597A/xx active
- 1994-12-15 WO PCT/EP1994/004154 patent/WO1995016680A1/en not_active Ceased
- 1994-12-15 JP JP51653195A patent/JP3317972B2/ja not_active Expired - Lifetime
- 1994-12-15 NZ NZ277789A patent/NZ277789A/en not_active IP Right Cessation
- 1994-12-15 CZ CZ19961693A patent/CZ289234B6/cs not_active IP Right Cessation
- 1994-12-15 SV SV1994000076A patent/SV1994000076A/es active IP Right Grant
- 1994-12-15 BR BR9408340A patent/BR9408340A/pt not_active Application Discontinuation
- 1994-12-15 HR HR941001A patent/HRP941001B1/xx not_active IP Right Cessation
- 1994-12-15 ZA ZA9410003A patent/ZA9410003B/xx unknown
- 1994-12-15 UA UA96062328A patent/UA46723C2/uk unknown
- 1994-12-15 PE PE1994257245A patent/PE31095A1/es not_active Application Discontinuation
- 1994-12-15 AP APAP/P/1996/000810A patent/AP9600810A0/en unknown
- 1994-12-15 EP EP95904472A patent/EP0734382B1/en not_active Expired - Lifetime
- 1994-12-15 SG SG1996007725A patent/SG46669A1/en unknown
- 1994-12-15 EE EE9600135A patent/EE03353B1/xx unknown
- 1994-12-15 SK SK785-96A patent/SK282972B6/sk not_active IP Right Cessation
- 1994-12-15 CN CN94194973A patent/CN1132829C/zh not_active Expired - Lifetime
- 1994-12-15 CN CNA2003101199989A patent/CN1502621A/zh active Pending
- 1994-12-15 AP APAP/P/1994/000705A patent/AP541A/en active
- 1994-12-15 CA CA002177990A patent/CA2177990C/en not_active Expired - Lifetime
- 1994-12-15 CO CO94056728A patent/CO4340619A1/es unknown
- 1994-12-15 DE DE69426726T patent/DE69426726T2/de not_active Expired - Lifetime
- 1994-12-15 AT AT95904472T patent/ATE199255T1/de active
- 1994-12-15 SI SI9430333T patent/SI0734382T1/xx unknown
- 1994-12-15 RU RU96115122A patent/RU2134690C1/ru active Protection Beyond IP Right Term
- 1994-12-15 PL PL94315055A patent/PL186384B1/pl unknown
- 1994-12-15 PT PT95904472T patent/PT734382E/pt unknown
- 1994-12-15 DK DK95904472T patent/DK0734382T3/da active
- 1994-12-15 RO RO96-01195A patent/RO114792B1/ro unknown
- 1994-12-15 HU HU9601642A patent/HU221971B1/hu active IP Right Grant
- 1994-12-15 ES ES95904472T patent/ES2155517T3/es not_active Expired - Lifetime
- 1994-12-15 KR KR1019960703180A patent/KR100403256B1/ko not_active Expired - Lifetime
- 1994-12-15 MA MA23724A patent/MA23396A1/fr unknown
- 1994-12-16 IL IL11201194A patent/IL112011A/en not_active IP Right Cessation
- 1994-12-28 SA SA94150417A patent/SA94150417B1/ar unknown
1996
- 1996-06-13 FI FI962464A patent/FI120453B/fi not_active IP Right Cessation
- 1996-06-14 NO NO19962545A patent/NO314759B1/no not_active IP Right Cessation
- 1996-06-14 OA OA60842A patent/OA10325A/fr unknown
- 1996-07-08 BG BG100709A patent/BG63338B1/bg unknown
1997
- 1997-05-13 BR BRPP1100548-KB1A patent/BR1100548KB1/pt unknown
1999
- 1999-07-02 US US09/346,583 patent/US6294572B1/en not_active Expired - Lifetime
2000
- 2000-01-06 OA OA1200000004A patent/OA11275A/fr unknown
2001
- 2001-03-30 GR GR20010400531T patent/GR3035681T3/el unknown
- 2001-09-24 US US09/961,074 patent/US20020037865A1/en not_active Abandoned

Also Published As

Publication number	Publication date
IL112011A (en)	1998-08-16
UA46723C2 (uk)	2002-06-17
SK78596A3 (en)	1997-03-05
WO1995016680A1 (en)	1995-06-22
NO962545D0 (no)	1996-06-14
ES2155517T3 (es)	2001-05-16
TW452577B (en)	2001-09-01
PL186384B1 (pl)	2004-01-30
EG20597A (en)	1999-09-30
AP541A (en)	1996-10-01
PT734382E (pt)	2001-06-29
AU1314495A (en)	1995-07-03
CN1132829C (zh)	2003-12-31
HRP941001B1 (en)	2001-06-30
PL315055A1 (en)	1996-09-30
JP3317972B2 (ja)	2002-08-26
JPH09506601A (ja)	1997-06-30
NO962545L (no)	1996-06-14
SG46669A1 (en)	1998-02-20
EE03353B1 (et)	2001-02-15
CA2177990C (en)	2000-04-25
HU221971B1 (hu)	2003-03-28
OA10325A (en)	1997-10-07
AU689185B2 (en)	1998-03-26
BG100709A (bg)	1997-01-31
BR1100548KB1 (pt)	2011-11-01
GB9325841D0 (en)	1994-02-23
HUT74938A (en)	1997-03-28
SK282972B6 (sk)	2003-01-09
CO4340619A1 (es)	1996-07-30
SI0734382T1 (en)	2001-08-31
CA2177990A1 (en)	1995-06-22
NZ277789A (en)	1999-04-29
EP0734382A1 (en)	1996-10-02
CZ289234B6 (cs)	2001-12-12
FI962464A0 (fi)	1996-06-13
GR3035681T3 (en)	2001-06-29
DK0734382T3 (da)	2001-03-19
US6294572B1 (en)	2001-09-25
KR100403256B1 (ko)	2004-04-30
SA94150417B1 (ar)	2005-12-18
IS4240A (is)	1995-06-18
US20020037865A1 (en)	2002-03-28
ZA9410003B (en)	1995-07-25
CN1142820A (zh)	1997-02-12
DE69426726D1 (de)	2001-03-29
MY116221A (en)	2003-12-31
CN1502621A (zh)	2004-06-09
PE31095A1 (es)	1995-10-18
BG63338B1 (bg)	2001-10-31
EP0734382B1 (en)	2001-02-21
NO314759B1 (no)	2003-05-19
RO114792B1 (ro)	1999-07-30
ATE199255T1 (de)	2001-03-15
SV1994000076A (es)	1995-10-26
CZ169396A3 (en)	1996-11-13
OA11275A (en)	2002-11-20
IL112011A0 (en)	1995-03-15
FI120453B (fi)	2009-10-30
AP9400705A0 (en)	1995-01-31
HRP941001A2 (en)	1997-06-30
AP9600810A0 (en)	1996-07-31
RU2134690C1 (ru)	1999-08-20
MA23396A1 (fr)	1995-07-01
DE69426726T2 (de)	2001-06-21
BR9408340A (pt)	1997-08-19
HK1014187A1 (en)	1999-09-24
HU9601642D0 (en)	1996-08-28

Publication	Publication Date	Title
FI941137A7 (fi)	1994-09-12	2-debentsoyyli-2-asyylitaksolijohdannaisia ja menetelmiä niiden valmistamiseksi
FI953981A7 (fi)	1995-08-24	2-Bentsyyli-polysykliset guaniinijohdannaiset ja menetelmä niiden valmistamiseksi
FI956270L (fi)	1995-12-27	Piperdiinijohdannaisia ja menetelmä niiden valmistamiseksi
FI945900A7 (fi)	1995-06-18	Bentseenisulfonamidijohdokset ja menetelmä näiden valmistamiseksi
FI973750L (fi)	1997-09-22	2-metyylitienobentsodiatsepiinin valmistus ja kiteiset muodot
BR9510256A (pt)	1997-11-04	Derivados de ácido 3-aril-tetrônico
FI943838A7 (fi)	1994-08-19	Vinyleeniatsaindolijohdannaiset ja menetelmä niiden valmistamiseksi
FI914723A7 (fi)	1991-10-07	17b-substituoituja 4-atsa-5a-androstan-3-oni-johdannaisia ja menetelmä niiden valmistamiseksi
FI953919A7 (fi)	1995-08-21	Pyrrolydeenimetyylijohdannaiset ja menetelmä niiden valmistamiseksi
FI945776L (fi)	1995-06-11	Yhden astian menetelmä 3-kinolonikarboksyylihaapojohdannaisten valmistamiseksi
FI962464L (fi)	1996-06-13	Kiteisiä N-asetyyliamiinihappojohdannaisia ja menetelmiä niiden valmistamiseksi
FI895910A7 (fi)	1990-06-15	Antiseptiset koostumukset ja menetelmä niiden valmistamiseksi
FI944713L (fi)	1994-12-02	4-difenyylimetyylipiperidiinijohdannaisia ja menetelmä niiden valmistamiseksi
FI892052A7 (fi)	1989-10-31	Happoadditiosuoloja ja menetelmä niiden valmistamiseksi
FI945787A7 (fi)	1994-12-09	Sulfoniumsuoloja ja menetelmä niiden valmistamiseksi
FI884747A7 (fi)	1989-04-20	Vesiliukoisia L-tyrosiinijohdannaisia ja menetelmä niiden valmistamiseksi
FI955382L (fi)	1996-05-11	Uudet kiteiset kefemihappoadditiosuolat ja menetelmä niiden valmistamiseksi
FI885942L (fi)	1989-06-26	Propoksibentseenijohdannaisia ja menetelmä niiden valmistamiseksi
FI893426L (fi)	1990-01-20	Analogiamenetelmä terapeuttisesti käyttökelpoisten BU-3608-johdannaisten ja niiden suolojen valmistamiseksi
FI885721L (fi)	1989-06-11	Makeutusaine ja menetelmä sen valmistamiseksi
FI933432A7 (fi)	1994-02-04	Kviinihapon johdokset ja menetelmä niiden valmistamiseksi
FI973434A7 (fi)	1997-08-21	Aminotetralonijohdannaisia ja menetelmä niiden valmistamiseksi
FI981359L (fi)	1998-06-12	Uudet tiomarinolin johdannaiset ja menetelmät niiden valmistamiseksi
FI932863A7 (fi)	1994-01-04	Menetelmä uusien tienotiatsiinijohdosten valmistamiseksi ja niiden käyttö
FI900270A7 (fi)	1990-07-20	Kefalosporiinijohdannaiset ja menetelmä niiden valmistamiseksi

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Date	Code	Title	Description
2009-10-30	FG	Patent granted	Ref document number: 120453 Country of ref document: FI
2015-01-15	MA	Patent expired

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2009-10-30

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2015-01-15

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