ZA200303794B - Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same. - Google Patents

Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.

Info

Publication number: ZA200303794B
Authority: ZA; South Africa
Prior art keywords: preparation; compositions containing; containing same; piperidine derivatives; heterocyclylalkyl piperidine
Prior art date: 2000-11-15

Application number

ZA200303794A

Other languages

English (en)

Inventor

Eric Bacque

Youssef El-Ahmad

Philippe Hubert

Serge Mignani

Michel Tabart

Jean-Christophe Carry

Michel Evers

Jean-Luc Malleron

Guy Pantel

Fabrice Viviani

Original Assignee

Aventis Pharma Sa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-15

Filing date

2003-05-15

Publication date

2004-06-29

2003-05-15 Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa

2004-06-29 Publication of ZA200303794B publication Critical patent/ZA200303794B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

ZA200303794A 2000-11-15 2003-05-15 Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same. ZA200303794B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR0014738A FR2816618B1 (fr)	2000-11-15	2000-11-15	Derives heterocyclylalcoyl piperidine, leur preparation et les compositions qui les contiennent

Publications (1)

Publication Number	Publication Date
ZA200303794B true ZA200303794B (en)	2004-06-29

Family

ID=8856503

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200303794A ZA200303794B (en)	2000-11-15	2003-05-15	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.

Country Status (28)

Country	Link
EP (2)	EP1695964A1 (et)
JP (1)	JP2004514661A (et)
KR (1)	KR100849608B1 (et)
CN (1)	CN1483031A (et)
AR (1)	AR034006A1 (et)
AT (1)	ATE337311T1 (et)
AU (2)	AU2002218365B2 (et)
BG (1)	BG107793A (et)
BR (1)	BR0115312A (et)
CA (1)	CA2429311A1 (et)
CZ (1)	CZ20031316A3 (et)
DE (1)	DE60122567T2 (et)
DK (1)	DK1337529T3 (et)
EA (1)	EA200300568A1 (et)
EE (1)	EE200300207A (et)
ES (1)	ES2271119T3 (et)
FR (1)	FR2816618B1 (et)
HR (1)	HRP20030379A2 (et)
HU (1)	HUP0303758A3 (et)
IL (1)	IL155841A0 (et)
NO (2)	NO20032187L (et)
PL (1)	PL363004A1 (et)
PT (1)	PT1337529E (et)
SK (1)	SK5822003A3 (et)
TN (1)	TNSN01160A1 (et)
WO (1)	WO2002040474A2 (et)
YU (1)	YU46803A (et)
ZA (1)	ZA200303794B (et)

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NZ523749A (en)	2000-07-26	2005-03-24	Smithkline Beecham P	Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity
GB0101577D0 (en)	2001-01-22	2001-03-07	Smithkline Beecham Plc	Compounds
GB0112834D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0112836D0 (en)	2001-05-25	2001-07-18	Smithkline Beecham Plc	Medicaments
GB0118238D0 (en) *	2001-07-26	2001-09-19	Smithkline Beecham Plc	Medicaments
JP4508650B2 (ja)	2002-01-29	2010-07-21	グラクソグループリミテッド	アミノピペリジン化合物、当該化合物の製法および当該化合物を含有する医薬組成物
EP1470125A1 (en)	2002-01-29	2004-10-27	Glaxo Group Limited	Aminopiperidine derivatives
TW200406413A (en)	2002-06-26	2004-05-01	Glaxo Group Ltd	Compounds
TW200409637A (en)	2002-06-26	2004-06-16	Glaxo Group Ltd	Compounds
FR2842807A1 (fr)	2002-07-23	2004-01-30	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, procede et intermediaires de preparation et compositions les renfermant
GB0217294D0 (en) *	2002-07-25	2002-09-04	Glaxo Group Ltd	Medicaments
FR2844270B1 (fr) *	2002-09-11	2006-05-19	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, leur procede et intermediaires de preparation et les compositions qui les contiennent
FR2844268B1 (fr)	2002-09-11	2004-10-22	Aventis Pharma Sa	Derives de la quinolyl propyl piperidine, leurs procedes et intermediaires de preparation et les compositions qui les contiennent
DE10256405A1 (de) *	2002-12-02	2004-06-17	Morphochem Aktiengesellschaft für kombinatorische Chemie	Neue Verbindungen, die Topoisomerase IV inhibieren
EP1560488B1 (en)	2002-11-05	2010-09-01	Glaxo Group Limited	Antibacterial agents
ATE461928T1 (de)	2002-11-05	2010-04-15	Glaxosmithkline Llc	Antibakterielle wirkstoffe
ATE411312T1 (de)	2002-12-04	2008-10-15	Glaxo Group Ltd	Chinoline und stickstoffhaltige derivatedavon und deren verwendung als antibakterielle mittel
FR2852954B1 (fr) *	2003-03-28	2006-07-14	Aventis Pharma Sa	Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
US7232833B2 (en)	2003-03-28	2007-06-19	Novexel	4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them
FR2862301B1 (fr) *	2003-11-17	2007-12-21	Aventis Pharma Sa	Nouveau procede de preparation de quinoleines 3-fluorees
FR2867472B1 (fr) *	2004-03-12	2008-07-18	Aventis Pharma Sa	Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent
JP2008528598A (ja)	2005-01-25	2008-07-31	グラクソグループリミテッド	抗菌剤
US7592334B2 (en)	2005-01-25	2009-09-22	Glaxo Group Limited	Antibacterial agents
US7648980B2 (en)	2005-01-25	2010-01-19	Glaxo Group Limited	Antibacterial agents
US7709472B2 (en)	2005-01-25	2010-05-04	Glaxo Group Limited	Antibacterial agents
AU2006218661A1 (en)	2005-03-01	2006-09-08	Wyeth	Cinnoline compounds and their use as liver X receptor modilators
MY150958A (en) *	2005-06-16	2014-03-31	Astrazeneca Ab	Compounds for the treatment of multi-drug resistant bacterial infections
JP2009524643A (ja)	2006-01-26	2009-07-02	アクテリオンファーマシューティカルズリミテッド	テトラヒドロピラン抗生物質
JP2009532423A (ja)	2006-04-06	2009-09-10	グラクソグループリミテッド	抗菌剤としてのピロロ−キノキサリノン誘導体
EP1992628A1 (en)	2007-05-18	2008-11-19	Glaxo Group Limited	Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones
CA2689102C (en)	2007-06-15	2016-07-26	Actelion Pharmaceuticals Ltd	3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives
EP2080761A1 (en)	2008-01-18	2009-07-22	Glaxo Group Limited	Compounds
EP2352734A1 (en)	2008-10-17	2011-08-10	Glaxo Group Limited	Tricyclic nitrogen compounds used as antibacterials
EP2379554B1 (en)	2009-01-15	2015-11-11	Glaxo Group Limited	Naphthyridin-2(1h)-one compounds useful as antibacterials
IN2015KN00323A (et) *	2012-08-15	2015-07-10	Glaxo Group Ltd
US10702521B2 (en)	2014-08-22	2020-07-07	Glaxosmithkline Intellectual Property Development Limited	Methods for treating neisseria gonorrhoeae infection with substituted 1,2-dihydro-2A,5,8A-triazaacenaphthylene-3,8-diones
WO2016138988A1 (en) *	2015-03-02	2016-09-09	University Of Copenhagen	Piperazine inhibitors of bacterial gyrase and topoisomerase iv
TW201722965A (zh)	2015-08-16	2017-07-01	葛蘭素史密斯克藍智慧財產發展有限公司	用於抗菌應用之化合物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7908031A (nl)	1979-11-01	1981-06-01	Acf Chemiefarma Nv	Nieuwe chinolinederivaten en farmaceutische preparaten die een dergelijke verbinding bevatten, alsmede werk- wijze voor het bereiden van deze verbindingen.
JPH0239546A (ja)	1988-07-29	1990-02-08	Origin Electric Co Ltd	混成集積回路の製造方法
AU623474B2 (en)	1989-01-16	1992-05-14	Laboratoire Roger Bellon	New benzo(1,8)naphthyridine derivatives, their preparation and compositions containing them
AU2717899A (en) *	1998-01-26	1999-08-09	Smithkline Beecham Plc	Quinoline derivatives as antibacterials
WO2000043383A1 (en) *	1999-01-20	2000-07-27	Smithkline Beecham P.L.C.	Piperidinylquinolines as protein tyrosine kinase inhibitors
FR2852954B1 (fr) *	2003-03-28	2006-07-14	Aventis Pharma Sa	Derives de quinoleines-4-substituees, leurs procede et intermediaires de preparation et les compositions pharmaceutiques qui les contiennent

2000
- 2000-11-15 FR FR0014738A patent/FR2816618B1/fr not_active Expired - Fee Related
2001
- 2001-11-13 AR ARP010105289A patent/AR034006A1/es unknown
- 2001-11-14 CZ CZ20031316A patent/CZ20031316A3/cs unknown
- 2001-11-14 JP JP2002543484A patent/JP2004514661A/ja active Pending
- 2001-11-14 CN CNA018210996A patent/CN1483031A/zh active Pending
- 2001-11-14 CA CA002429311A patent/CA2429311A1/en not_active Abandoned
- 2001-11-14 EA EA200300568A patent/EA200300568A1/ru unknown
- 2001-11-14 AU AU2002218365A patent/AU2002218365B2/en not_active Ceased
- 2001-11-14 YU YU46803A patent/YU46803A/sh unknown
- 2001-11-14 DE DE60122567T patent/DE60122567T2/de not_active Expired - Fee Related
- 2001-11-14 PL PL01363004A patent/PL363004A1/xx not_active Application Discontinuation
- 2001-11-14 PT PT01996538T patent/PT1337529E/pt unknown
- 2001-11-14 BR BR0115312-9A patent/BR0115312A/pt not_active Application Discontinuation
- 2001-11-14 SK SK582-2003A patent/SK5822003A3/sk unknown
- 2001-11-14 DK DK01996538T patent/DK1337529T3/da active
- 2001-11-14 AU AU1836502A patent/AU1836502A/xx active Pending
- 2001-11-14 ES ES01996538T patent/ES2271119T3/es not_active Expired - Lifetime
- 2001-11-14 EP EP06010725A patent/EP1695964A1/fr not_active Withdrawn
- 2001-11-14 IL IL15584101A patent/IL155841A0/xx unknown
- 2001-11-14 HU HU0303758A patent/HUP0303758A3/hu unknown
- 2001-11-14 HR HR20030379A patent/HRP20030379A2/hr not_active Application Discontinuation
- 2001-11-14 TN TNTNSN01160A patent/TNSN01160A1/fr unknown
- 2001-11-14 KR KR1020037006600A patent/KR100849608B1/ko not_active Expired - Fee Related
- 2001-11-14 WO PCT/FR2001/003559 patent/WO2002040474A2/fr not_active Ceased
- 2001-11-14 EE EEP200300207A patent/EE200300207A/et unknown
- 2001-11-14 AT AT01996538T patent/ATE337311T1/de not_active IP Right Cessation
- 2001-11-14 EP EP01996538A patent/EP1337529B1/fr not_active Expired - Lifetime
2003
- 2003-05-09 BG BG107793A patent/BG107793A/bg unknown
- 2003-05-14 NO NO20032187A patent/NO20032187L/no unknown
- 2003-05-15 ZA ZA200303794A patent/ZA200303794B/xx unknown
2007
- 2007-04-25 NO NO20072142A patent/NO20072142L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
TNSN01160A1 (fr)	2005-11-10
EA200300568A1 (ru)	2003-12-25
CZ20031316A3 (cs)	2003-10-15
DE60122567D1 (de)	2006-10-05
ES2271119T3 (es)	2007-04-16
CA2429311A1 (en)	2002-05-23
EP1337529A2 (fr)	2003-08-27
NO20072142L (no)	2007-04-25
AR034006A1 (es)	2004-01-21
WO2002040474A3 (fr)	2002-10-31
HUP0303758A2 (hu)	2004-03-01
NO20032187D0 (no)	2003-05-14
IL155841A0 (en)	2003-12-23
CN1483031A (zh)	2004-03-17
HRP20030379A2 (en)	2005-04-30
BG107793A (bg)	2004-08-31
NO20032187L (no)	2003-06-26
FR2816618B1 (fr)	2002-12-27
BR0115312A (pt)	2003-09-23
PT1337529E (pt)	2006-12-29
ATE337311T1 (de)	2006-09-15
FR2816618A1 (fr)	2002-05-17
DK1337529T3 (da)	2006-12-18
KR100849608B1 (ko)	2008-07-31
AU2002218365B2 (en)	2007-07-05
EP1337529B1 (fr)	2006-08-23
SK5822003A3 (en)	2004-06-08
EP1695964A1 (fr)	2006-08-30
YU46803A (sh)	2006-05-25
DE60122567T2 (de)	2007-08-23
AU1836502A (en)	2002-05-27
PL363004A1 (en)	2004-11-15
KR20030060934A (ko)	2003-07-16
WO2002040474A2 (fr)	2002-05-23
HUP0303758A3 (en)	2009-08-28
EE200300207A (et)	2003-08-15
JP2004514661A (ja)	2004-05-20

Publication	Publication Date	Title
ZA200303794B (en)	2004-06-29	Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same.
ZA200206905B (en)	2003-08-26	Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same.
IL151209A0 (en)	2003-04-10	Pharmaceutical compositions containing 3-aminoazetidine derivatives, novel derivatives and their preparation
HUP0303835A3 (en)	2009-08-28	Anti-allergic piperidine compounds, their use and pharmaceutical compositions containing them
HUP0400837A3 (en)	2007-11-28	2-phenyl-thiazole derivatives, their use and pharmaceutical compositions containing them
HUP0301573A3 (en)	2004-03-29	Substituted arylpyrazines, pharmaceutical compositions containing them and their use
HUP0204474A3 (en)	2004-07-28	1h-imidazopyridine derivatives, pharmaceutical compositions containing them and their use
HUP0400636A3 (en)	2004-09-28	Pharmaceutical compositions containing azetidine derivatives, novel azetidine derivatives and preparation thereof
HUP0204514A3 (en)	2004-07-28	Pyridinylimidazoles, pharmaceutical compositions containing them and their use
HUP0301965A3 (en)	2009-01-28	Novel phenyl-propargylether derivatives, their preparation, fungicide compositions containing them and use thereof
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AU2001237526A1 (en)	2001-11-22	Pharmaceutical compositions containing 3-amino-azetidine derivatives, novel derivatives and preparation thereof
ZA200003998B (en)	2000-08-14	Pharmaceutical compositions.
MXPA03000771A (es)	2003-06-04	Nuevas composiciones farmaceuticas.
AU2001237525A1 (en)	2001-11-22	Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
IL152448A0 (en)	2003-05-29	3-nitrogen-6, 7-dioxygen steroid derivatives and pharmaceutical compositions containing the same
HUP0302959A3 (en)	2006-04-28	Non-imidazole aryloxyalkylamines, pharmaceutical compositions containing them and their use
MXPA03007848A (es)	2003-12-11	Derivados de quinolil propil piperidina, su preparacion y las composiciones que los contienen.
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PL356911A1 (en)	2004-07-12	Novel heterocyclic derivatives, preparation method and pharmaceutical compositions containing same
MXPA03002105A (es)	2003-06-19	Composiciones farmaceuticas.