IL155841A0 - Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same - Google Patents
Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing sameInfo
- Publication number
- IL155841A0 IL155841A0 IL15584101A IL15584101A IL155841A0 IL 155841 A0 IL155841 A0 IL 155841A0 IL 15584101 A IL15584101 A IL 15584101A IL 15584101 A IL15584101 A IL 15584101A IL 155841 A0 IL155841 A0 IL 155841A0
- Authority
- IL
- Israel
- Prior art keywords
- preparation
- compositions containing
- containing same
- piperidine derivatives
- heterocyclylalkyl piperidine
- Prior art date
Links
- -1 Heterocyclylalkyl piperidine derivatives Chemical class 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0014738A FR2816618B1 (en) | 2000-11-15 | 2000-11-15 | HETEROCYCLYLALCOYL PIPERIDINE DERIVATIVES, THEIR PREPARATION AND THE COMPOSITIONS CONTAINING THEM |
| PCT/FR2001/003559 WO2002040474A2 (en) | 2000-11-15 | 2001-11-14 | Heterocyclylalkyl piperidine derivatives and their use as antimicrobial agents |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IL155841A0 true IL155841A0 (en) | 2003-12-23 |
Family
ID=8856503
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IL15584101A IL155841A0 (en) | 2000-11-15 | 2001-11-14 | Heterocyclylalkyl piperidine derivatives, their preparation and compositions containing same |
Country Status (28)
| Country | Link |
|---|---|
| EP (2) | EP1337529B1 (en) |
| JP (1) | JP2004514661A (en) |
| KR (1) | KR100849608B1 (en) |
| CN (1) | CN1483031A (en) |
| AR (1) | AR034006A1 (en) |
| AT (1) | ATE337311T1 (en) |
| AU (2) | AU1836502A (en) |
| BG (1) | BG107793A (en) |
| BR (1) | BR0115312A (en) |
| CA (1) | CA2429311A1 (en) |
| CZ (1) | CZ20031316A3 (en) |
| DE (1) | DE60122567T2 (en) |
| DK (1) | DK1337529T3 (en) |
| EA (1) | EA200300568A1 (en) |
| EE (1) | EE200300207A (en) |
| ES (1) | ES2271119T3 (en) |
| FR (1) | FR2816618B1 (en) |
| HR (1) | HRP20030379A2 (en) |
| HU (1) | HUP0303758A3 (en) |
| IL (1) | IL155841A0 (en) |
| NO (2) | NO20032187L (en) |
| PL (1) | PL363004A1 (en) |
| PT (1) | PT1337529E (en) |
| SK (1) | SK5822003A3 (en) |
| TN (1) | TNSN01160A1 (en) |
| WO (1) | WO2002040474A2 (en) |
| YU (1) | YU46803A (en) |
| ZA (1) | ZA200303794B (en) |
Families Citing this family (38)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUP0300721A3 (en) | 2000-07-26 | 2006-02-28 | Smithkline Beecham Plc | Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity, process for producing them, pharmaceutical compositions containing them and use thereof |
| GB0101577D0 (en) | 2001-01-22 | 2001-03-07 | Smithkline Beecham Plc | Compounds |
| GB0112836D0 (en) | 2001-05-25 | 2001-07-18 | Smithkline Beecham Plc | Medicaments |
| GB0112834D0 (en) | 2001-05-25 | 2001-07-18 | Smithkline Beecham Plc | Medicaments |
| GB0118238D0 (en) * | 2001-07-26 | 2001-09-19 | Smithkline Beecham Plc | Medicaments |
| JP4508650B2 (en) | 2002-01-29 | 2010-07-21 | グラクソ グループ リミテッド | Aminopiperidine compound, process for producing the compound and pharmaceutical composition containing the compound |
| AR038240A1 (en) | 2002-01-29 | 2005-01-05 | Glaxo Group Ltd | PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE FOR PREPARATION |
| AR040336A1 (en) | 2002-06-26 | 2005-03-30 | Glaxo Group Ltd | PIPERIDINE COMPOUND, USE OF THE SAME FOR THE MANUFACTURE OF A MEDICINAL PRODUCT, PHARMACEUTICAL COMPOSITION THAT INCLUDES IT AND PROCEDURE TO PREPARE SUCH COMPOUND |
| TW200406413A (en) | 2002-06-26 | 2004-05-01 | Glaxo Group Ltd | Compounds |
| FR2842807A1 (en) * | 2002-07-23 | 2004-01-30 | Aventis Pharma Sa | QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESS AND PREPARATION INTERMEDIATES AND COMPOSITIONS COMPRISING THE SAME |
| GB0217294D0 (en) * | 2002-07-25 | 2002-09-04 | Glaxo Group Ltd | Medicaments |
| FR2844270B1 (en) * | 2002-09-11 | 2006-05-19 | Aventis Pharma Sa | QUINOLYL PROPYL PIPERIDINE DERIVATIVES, THEIR PROCESS AND PREPARATION INTERMEDIATES AND THE COMPOSITIONS CONTAINING THEM |
| FR2844268B1 (en) * | 2002-09-11 | 2004-10-22 | Aventis Pharma Sa | QUINOLYL PROPYL PIPERIDINE DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION, AND COMPOSITIONS CONTAINING THEM |
| DE10256405A1 (en) * | 2002-12-02 | 2004-06-17 | Morphochem Aktiengesellschaft für kombinatorische Chemie | New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens |
| AU2003303956A1 (en) | 2002-11-05 | 2004-11-23 | Smithkline Beecham Corporation | Antibacterial agents |
| DE60334016D1 (en) | 2002-11-05 | 2010-10-14 | Glaxo Group Ltd | ANTIBACTERIAL AGENTS |
| DE60324179D1 (en) | 2002-12-04 | 2008-11-27 | Glaxo Group Ltd | CHINOLINE AND NITROGENIC DERIVATEDAVAN AND THEIR USE AS ANTIBACTERIAL AGENTS |
| US7232833B2 (en) | 2003-03-28 | 2007-06-19 | Novexel | 4-substituted quinoline derivatives, method and intermediates for their preparation and pharmaceutical compositions containing them |
| FR2852954B1 (en) * | 2003-03-28 | 2006-07-14 | Aventis Pharma Sa | QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| FR2862301B1 (en) * | 2003-11-17 | 2007-12-21 | Aventis Pharma Sa | NEW PROCESS FOR THE PREPARATION OF 3-FLUORINATED QUINOLINES |
| FR2867472B1 (en) * | 2004-03-12 | 2008-07-18 | Aventis Pharma Sa | QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
| WO2006081178A2 (en) | 2005-01-25 | 2006-08-03 | Glaxo Group Limited | Antibacterial agents |
| JP2008528598A (en) | 2005-01-25 | 2008-07-31 | グラクソ グループ リミテッド | Antibacterial agent |
| WO2006081179A1 (en) | 2005-01-25 | 2006-08-03 | Glaxo Group Limited | Antibacterial agents |
| EP1846418A4 (en) | 2005-01-25 | 2009-12-23 | Glaxo Group Ltd | Antibacterial agents |
| BRPI0607404A2 (en) | 2005-03-01 | 2009-09-01 | Wyeth Corp | cinolin compounds and their use as hepatic x receptor modulators |
| MY150958A (en) * | 2005-06-16 | 2014-03-31 | Astrazeneca Ab | Compounds for the treatment of multi-drug resistant bacterial infections |
| JP2009524643A (en) | 2006-01-26 | 2009-07-02 | アクテリオン ファーマシューティカルズ リミテッド | Tetrahydropyran antibiotics |
| ATE481406T1 (en) | 2006-04-06 | 2010-10-15 | Glaxo Group Ltd | PYRROLOQUINOXALINONE DERIVATIVES AS ANTIBACTERIAL AGENTS |
| EP1992628A1 (en) | 2007-05-18 | 2008-11-19 | Glaxo Group Limited | Derivatives and analogs of N-ethylquinolones and N-ethylazaquinolones |
| CA2689102C (en) | 2007-06-15 | 2016-07-26 | Actelion Pharmaceuticals Ltd | 3-amino-6-(1-amino-ethyl)-tetrahydropyran derivatives |
| EP2080761A1 (en) | 2008-01-18 | 2009-07-22 | Glaxo Group Limited | Compounds |
| JP2012505866A (en) | 2008-10-17 | 2012-03-08 | グラクソ グループ リミテッド | Tricyclic nitrogen compounds used as antibacterial agents |
| ES2561631T3 (en) | 2009-01-15 | 2016-02-29 | Glaxo Group Limited | Naphthyridine-2 (1H) -one compounds useful as antibacterial agents |
| CN104619706B (en) * | 2012-08-15 | 2017-06-20 | 葛兰素集团有限公司 | chemical method |
| EP3639824A1 (en) | 2014-08-22 | 2020-04-22 | GlaxoSmithKline Intellectual Property Development Limited | Tricyclic nitrogen containing compounds for treating neisseria gonorrhoea infection |
| WO2016138988A1 (en) * | 2015-03-02 | 2016-09-09 | University Of Copenhagen | Piperazine inhibitors of bacterial gyrase and topoisomerase iv |
| TW201722965A (en) | 2015-08-16 | 2017-07-01 | 葛蘭素史密斯克藍智慧財產發展有限公司 | Compounds for use in antibacterial applications |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL7908031A (en) | 1979-11-01 | 1981-06-01 | Acf Chemiefarma Nv | NEW QUINOLINE DERIVATIVES AND PHARMACEUTICAL PREPARATIONS CONTAINING SUCH A COMPOUND AND METHOD FOR PREPARING THESE COMPOUNDS. |
| JPH0239546A (en) | 1988-07-29 | 1990-02-08 | Origin Electric Co Ltd | Manufacture of hybrid integrated circuit |
| AU623474B2 (en) | 1989-01-16 | 1992-05-14 | Laboratoire Roger Bellon | New benzo(1,8)naphthyridine derivatives, their preparation and compositions containing them |
| JP2002501061A (en) * | 1998-01-26 | 2002-01-15 | スミスクライン・ビーチャム・パブリック・リミテッド・カンパニー | Quinoline derivatives for antibacterial agents |
| WO2000043383A1 (en) * | 1999-01-20 | 2000-07-27 | Smithkline Beecham P.L.C. | Piperidinylquinolines as protein tyrosine kinase inhibitors |
| FR2852954B1 (en) * | 2003-03-28 | 2006-07-14 | Aventis Pharma Sa | QUINOLINE-4-SUBSTITUTED DERIVATIVES, METHODS AND PREPARATION INTERMEDIATES THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
-
2000
- 2000-11-15 FR FR0014738A patent/FR2816618B1/en not_active Expired - Fee Related
-
2001
- 2001-11-13 AR ARP010105289A patent/AR034006A1/en unknown
- 2001-11-14 CN CNA018210996A patent/CN1483031A/en active Pending
- 2001-11-14 AT AT01996538T patent/ATE337311T1/en not_active IP Right Cessation
- 2001-11-14 IL IL15584101A patent/IL155841A0/en unknown
- 2001-11-14 CA CA002429311A patent/CA2429311A1/en not_active Abandoned
- 2001-11-14 HU HU0303758A patent/HUP0303758A3/en unknown
- 2001-11-14 YU YU46803A patent/YU46803A/en unknown
- 2001-11-14 ES ES01996538T patent/ES2271119T3/en not_active Expired - Lifetime
- 2001-11-14 KR KR1020037006600A patent/KR100849608B1/en not_active Expired - Fee Related
- 2001-11-14 WO PCT/FR2001/003559 patent/WO2002040474A2/en not_active Ceased
- 2001-11-14 EE EEP200300207A patent/EE200300207A/en unknown
- 2001-11-14 HR HR20030379A patent/HRP20030379A2/en not_active Application Discontinuation
- 2001-11-14 PL PL01363004A patent/PL363004A1/en not_active Application Discontinuation
- 2001-11-14 EA EA200300568A patent/EA200300568A1/en unknown
- 2001-11-14 DK DK01996538T patent/DK1337529T3/en active
- 2001-11-14 SK SK582-2003A patent/SK5822003A3/en unknown
- 2001-11-14 AU AU1836502A patent/AU1836502A/en active Pending
- 2001-11-14 JP JP2002543484A patent/JP2004514661A/en active Pending
- 2001-11-14 DE DE60122567T patent/DE60122567T2/en not_active Expired - Fee Related
- 2001-11-14 BR BR0115312-9A patent/BR0115312A/en not_active Application Discontinuation
- 2001-11-14 PT PT01996538T patent/PT1337529E/en unknown
- 2001-11-14 EP EP01996538A patent/EP1337529B1/en not_active Expired - Lifetime
- 2001-11-14 EP EP06010725A patent/EP1695964A1/en not_active Withdrawn
- 2001-11-14 CZ CZ20031316A patent/CZ20031316A3/en unknown
- 2001-11-14 AU AU2002218365A patent/AU2002218365B2/en not_active Ceased
- 2001-11-14 TN TNTNSN01160A patent/TNSN01160A1/en unknown
-
2003
- 2003-05-09 BG BG107793A patent/BG107793A/en unknown
- 2003-05-14 NO NO20032187A patent/NO20032187L/en unknown
- 2003-05-15 ZA ZA200303794A patent/ZA200303794B/en unknown
-
2007
- 2007-04-25 NO NO20072142A patent/NO20072142L/en not_active Application Discontinuation
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