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UY30805A1 - Moduladores no esteroides de receptores de progesterona - Google Patents

Moduladores no esteroides de receptores de progesterona

Info

Publication number
UY30805A1
UY30805A1 UY30805A UY30805A UY30805A1 UY 30805 A1 UY30805 A1 UY 30805A1 UY 30805 A UY30805 A UY 30805A UY 30805 A UY30805 A UY 30805A UY 30805 A1 UY30805 A1 UY 30805A1
Authority
UY
Uruguay
Prior art keywords
therapy
modulators
prevention
progesterone receptors
progesterone receptor
Prior art date
Application number
UY30805A
Other languages
English (en)
Inventor
Andrea Rotgeri
Carsten Moeller
Thomas Kirkland
Wolfgang Schwede
Ulrike Fuhrmann
Anja Schmidt
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE102006061913A external-priority patent/DE102006061913A1/de
Priority claimed from DE102007023614A external-priority patent/DE102007023614A1/de
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of UY30805A1 publication Critical patent/UY30805A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/02—1,2-Oxazines; Hydrogenated 1,2-oxazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)

Abstract

La presente invencion se refiere a moduladores no esteroides del receptor de la progesterona de la formula general I, al uso de moduladores del receptor de Progesterona para la preparacion de medicamentos, así como a composiciones farmacéuticas que contienen estos compuestos. Los compuestos segun la invencion son apropiados para la terapia y la prevencion de enfermedades ginecologicas tales como endometriosis, leiomiomas de utero, hemorragias disfuncionales y dismenorrea y para la terapia y la prevencion de tumores dependientes de hormonas y para el uso para el control de la fertilidad femenina y para la terapia de reemplazo hormonal.
UY30805A 2006-12-21 2007-12-18 Moduladores no esteroides de receptores de progesterona UY30805A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102006061913A DE102006061913A1 (de) 2006-12-21 2006-12-21 Nichtsteroidale Progesteronrezeptor-Modulatoren
DE102007023614A DE102007023614A1 (de) 2007-05-21 2007-05-21 Nichtsteroidale Progesteronrezeptor-Modulatoren

Publications (1)

Publication Number Publication Date
UY30805A1 true UY30805A1 (es) 2008-07-31

Family

ID=39456752

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30805A UY30805A1 (es) 2006-12-21 2007-12-18 Moduladores no esteroides de receptores de progesterona

Country Status (5)

Country Link
AR (1) AR064478A1 (es)
PE (1) PE20081397A1 (es)
TW (1) TW200835498A (es)
UY (1) UY30805A1 (es)
WO (1) WO2008077647A2 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103288669B (zh) * 2013-07-01 2015-06-24 南开大学 一种阿卓乳酸酰胺衍生物及应用
CN117402111A (zh) * 2023-10-12 2024-01-16 昆明理工大学 自由基引发烯烃与炔烃交叉偶联制备全碳季碳中心衍生物的方法

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8617653D0 (en) * 1986-07-18 1986-08-28 Ici Plc Amide derivatives
GB8617652D0 (en) * 1986-07-18 1986-08-28 Ici Plc Acylanilide derivatives
IE922316A1 (en) * 1991-07-17 1993-01-27 Smithkline Beecham Corp Retroviral protease inhibitors
US5733882A (en) * 1994-01-17 1998-03-31 Smithkline Beecham Corporation Retroviral protease inhibitors
DE19723722A1 (de) * 1997-05-30 1998-12-10 Schering Ag Nichtsteroidale Gestagene
DE19856475A1 (de) * 1998-11-27 2000-05-31 Schering Ag Nichtsteroidale Entzündungshemmer
DE10038639A1 (de) * 2000-07-28 2002-02-21 Schering Ag Nichtsteroidale Entzündungshemmer
WO2003059899A1 (en) * 2002-01-14 2003-07-24 Boehringer Ingelheim Pharmaceuticals, Inc. Glucocorticoid mimetics, methods of making them, pharmaceutical formulations containing them and uses thereof
EP1344776A1 (en) * 2002-03-11 2003-09-17 Schering Aktiengesellschaft 5- 2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino -phtalide and 6- 2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino -4-methyl-2,3-benzoxazin-1-one derivatives with progesterone receptor modulating activity for use in fertility control, hormone replacement therapy and the treatment of gynecological disorders
IL164032A0 (en) * 2002-03-11 2005-12-18 Schering Ag 5-ä2-Hydroxy-3-'1-(3-trifluoromethylphenyl)-cyclopropyl-propionylaminoü-phtalide and related compounds with progesteronepeceptor
JP2008529963A (ja) * 2003-07-01 2008-08-07 バイエル・シエーリング・ファーマ アクチエンゲゼルシャフト 複素環式−置換されたペンタノール誘導体類、それらの生成方法及び抗炎症剤としてのそれらの使用
WO2006108699A1 (en) * 2005-04-14 2006-10-19 Glaxo Group Limited Indazoles as glucocorticoid receptor ligands
DE102005030293A1 (de) * 2005-06-24 2007-01-04 Schering Ag Verwendung von nichtsteroidale Progesteronrezeptor-Modulatoren
DE102005030292A1 (de) * 2005-06-24 2007-01-11 Schering Ag Nichtsteroidale Progesteronrezeptor-Modulatoren
DE102005030294A1 (de) * 2005-06-24 2007-01-04 Schering Ag Nichtsteroidale Progesteronrezeptor-Modulatoren

Also Published As

Publication number Publication date
AR064478A1 (es) 2009-04-01
PE20081397A1 (es) 2008-12-05
WO2008077647A3 (de) 2008-10-16
WO2008077647A2 (de) 2008-07-03
TW200835498A (en) 2008-09-01

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20170802