CR9598A - Moduladores no esteroides de receptor de progesterona - Google Patents
Moduladores no esteroides de receptor de progesteronaInfo
- Publication number
- CR9598A CR9598A CR9598A CR9598A CR9598A CR 9598 A CR9598 A CR 9598A CR 9598 A CR9598 A CR 9598A CR 9598 A CR9598 A CR 9598A CR 9598 A CR9598 A CR 9598A
- Authority
- CR
- Costa Rica
- Prior art keywords
- therapy
- prevention
- receptor modulators
- progesterone receptor
- steroid progesterone
- Prior art date
Links
- RJKFOVLPORLFTN-LEKSSAKUSA-N Progesterone Chemical compound C1CC2=CC(=O)CC[C@]2(C)[C@@H]2[C@@H]1[C@@H]1CC[C@H](C(=O)C)[C@@]1(C)CC2 RJKFOVLPORLFTN-LEKSSAKUSA-N 0.000 title 2
- 229960003387 progesterone Drugs 0.000 title 1
- 239000000186 progesterone Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000002265 prevention Effects 0.000 abstract 2
- 239000002379 progesterone receptor modulator Substances 0.000 abstract 2
- 229940095745 sex hormone and modulator of the genital system progesterone receptor modulator Drugs 0.000 abstract 2
- 238000002560 therapeutic procedure Methods 0.000 abstract 2
- 208000005171 Dysmenorrhea Diseases 0.000 abstract 1
- 206010013935 Dysmenorrhoea Diseases 0.000 abstract 1
- 201000009273 Endometriosis Diseases 0.000 abstract 1
- 208000032843 Hemorrhage Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 206010046798 Uterine leiomyoma Diseases 0.000 abstract 1
- 230000001419 dependent effect Effects 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 230000035558 fertility Effects 0.000 abstract 1
- 229940088597 hormone Drugs 0.000 abstract 1
- 239000005556 hormone Substances 0.000 abstract 1
- 238000002657 hormone replacement therapy Methods 0.000 abstract 1
- 201000010260 leiomyoma Diseases 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000003637 steroidlike Effects 0.000 abstract 1
- 201000007954 uterine fibroid Diseases 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/02—1,2-Oxazines; Hydrogenated 1,2-oxazines
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Pregnancy & Childbirth (AREA)
- Gynecology & Obstetrics (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
Se refiere a moduladores no-esteroides de receptor de progesterona de la formula general (I), al proceso para su preparacion, al usode los moduladores del receptor de progesterona para la produccion de medicamentos asi como tambien composiciones farmaceuticas que contienen estos compuestos. Los compuestos segun la invencion son apropiados para la terapia y la prevencion de enfermedades ginecologicas tales como endometriosis, leiomiomas de utero, hemorragias disfuncionales y dismenorrea y para la terapia y la prevencion de tumores dependientes de hormonas y para el uso para el control de la fertilidad femenina y para la terapia de reemplazo hormonal.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102005030292A DE102005030292A1 (de) | 2005-06-24 | 2005-06-24 | Nichtsteroidale Progesteronrezeptor-Modulatoren |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CR9598A true CR9598A (es) | 2008-04-09 |
Family
ID=37199176
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CR9598A CR9598A (es) | 2005-06-24 | 2007-12-17 | Moduladores no esteroides de receptor de progesterona |
Country Status (22)
| Country | Link |
|---|---|
| EP (1) | EP1902049A2 (es) |
| JP (1) | JP2008543910A (es) |
| KR (1) | KR20080030622A (es) |
| CN (1) | CN101248066A (es) |
| AR (1) | AR054519A1 (es) |
| AU (1) | AU2006261048A1 (es) |
| BR (1) | BRPI0611903A2 (es) |
| CA (1) | CA2611897A1 (es) |
| CR (1) | CR9598A (es) |
| DE (1) | DE102005030292A1 (es) |
| DO (1) | DOP2006000148A (es) |
| EA (1) | EA200702524A1 (es) |
| EC (1) | ECSP078044A (es) |
| GT (1) | GT200600271A (es) |
| IL (1) | IL188021A0 (es) |
| MX (1) | MX2008000072A (es) |
| NO (1) | NO20080440L (es) |
| PE (1) | PE20070125A1 (es) |
| TW (1) | TW200740778A (es) |
| UY (1) | UY29624A1 (es) |
| WO (1) | WO2006136461A2 (es) |
| ZA (1) | ZA200800690B (es) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UY30805A1 (es) * | 2006-12-21 | 2008-07-31 | Bayer Schering Pharma Ag | Moduladores no esteroides de receptores de progesterona |
| DE102007032800A1 (de) * | 2007-07-10 | 2009-01-15 | Bayer Schering Pharma Aktiengesellschaft | Nichtsteroidale Progesteronrezeptor-Modulatoren |
| DE102007058747A1 (de) * | 2007-12-05 | 2009-06-10 | Bayer Schering Pharma Aktiengesellschaft | Nichtsteroidale Progesteronrezeptor-Modulatoren |
| JP2011519916A (ja) * | 2008-07-02 | 2011-07-14 | ファーマコステック カンパニー リミテッド | アミド誘導体の製造方法 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19856475A1 (de) * | 1998-11-27 | 2000-05-31 | Schering Ag | Nichtsteroidale Entzündungshemmer |
| EP1344776A1 (en) * | 2002-03-11 | 2003-09-17 | Schering Aktiengesellschaft | 5- 2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino -phtalide and 6- 2-hydroxy-3-[1-(3-trifluoromethylphenyl)-cyclopropyl]-propionylamino -4-methyl-2,3-benzoxazin-1-one derivatives with progesterone receptor modulating activity for use in fertility control, hormone replacement therapy and the treatment of gynecological disorders |
| RS20050974A (sr) * | 2003-07-01 | 2007-09-21 | Schering Aktiengesellschaft, | Heterociklično supstituisani pentanol-derivati,postupak za njihovo dobijanje i njihova primena kao supresora zapaljenja |
-
2005
- 2005-06-24 DE DE102005030292A patent/DE102005030292A1/de not_active Ceased
-
2006
- 2006-06-22 EA EA200702524A patent/EA200702524A1/ru unknown
- 2006-06-22 KR KR1020087001793A patent/KR20080030622A/ko not_active Withdrawn
- 2006-06-22 EP EP06762404A patent/EP1902049A2/en not_active Withdrawn
- 2006-06-22 BR BRPI0611903-4A patent/BRPI0611903A2/pt not_active Application Discontinuation
- 2006-06-22 CN CNA2006800308707A patent/CN101248066A/zh active Pending
- 2006-06-22 WO PCT/EP2006/006531 patent/WO2006136461A2/en not_active Ceased
- 2006-06-22 AU AU2006261048A patent/AU2006261048A1/en not_active Abandoned
- 2006-06-22 MX MX2008000072A patent/MX2008000072A/es not_active Application Discontinuation
- 2006-06-22 CA CA002611897A patent/CA2611897A1/en not_active Abandoned
- 2006-06-22 JP JP2008517444A patent/JP2008543910A/ja active Pending
- 2006-06-23 TW TW095122742A patent/TW200740778A/zh unknown
- 2006-06-26 UY UY29624A patent/UY29624A1/es not_active Application Discontinuation
- 2006-06-26 DO DO2006000148A patent/DOP2006000148A/es unknown
- 2006-06-26 PE PE2006000733A patent/PE20070125A1/es not_active Application Discontinuation
- 2006-06-27 AR ARP060102750A patent/AR054519A1/es unknown
- 2006-06-28 GT GT200600271A patent/GT200600271A/es unknown
-
2007
- 2007-12-10 IL IL188021A patent/IL188021A0/en unknown
- 2007-12-17 CR CR9598A patent/CR9598A/es not_active Application Discontinuation
- 2007-12-21 EC EC2007008044A patent/ECSP078044A/es unknown
-
2008
- 2008-01-23 ZA ZA200800690A patent/ZA200800690B/xx unknown
- 2008-01-23 NO NO20080440A patent/NO20080440L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EA200702524A1 (ru) | 2008-06-30 |
| IL188021A0 (en) | 2008-03-20 |
| DOP2006000148A (es) | 2007-07-15 |
| EP1902049A2 (en) | 2008-03-26 |
| UY29624A1 (es) | 2007-01-31 |
| PE20070125A1 (es) | 2007-02-14 |
| MX2008000072A (es) | 2008-03-24 |
| KR20080030622A (ko) | 2008-04-04 |
| TW200740778A (en) | 2007-11-01 |
| ECSP078044A (es) | 2008-01-23 |
| ZA200800690B (en) | 2009-09-30 |
| DE102005030292A1 (de) | 2007-01-11 |
| GT200600271A (es) | 2007-02-05 |
| BRPI0611903A2 (pt) | 2010-10-05 |
| JP2008543910A (ja) | 2008-12-04 |
| NO20080440L (no) | 2008-03-25 |
| CN101248066A (zh) | 2008-08-20 |
| AR054519A1 (es) | 2007-06-27 |
| CA2611897A1 (en) | 2006-12-28 |
| AU2006261048A1 (en) | 2006-12-28 |
| WO2006136461A2 (en) | 2006-12-28 |
| WO2006136461A3 (en) | 2007-03-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal (granting procedure) |