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UY27552A1 - 17a- alquil- 17b- oxi-estratrienos y productos intermediarios para su preparacinn, uso de los 17a-alquil-17b-oxi-estratrienos para obtener medicamentos y preparados farmacéuticos. - Google Patents

17a- alquil- 17b- oxi-estratrienos y productos intermediarios para su preparacinn, uso de los 17a-alquil-17b-oxi-estratrienos para obtener medicamentos y preparados farmacéuticos.

Info

Publication number
UY27552A1
UY27552A1 UY27552A UY27552A UY27552A1 UY 27552 A1 UY27552 A1 UY 27552A1 UY 27552 A UY27552 A UY 27552A UY 27552 A UY27552 A UY 27552A UY 27552 A1 UY27552 A1 UY 27552A1
Authority
UY
Uruguay
Prior art keywords
stratriens
oxi
rent
preparation
preparations
Prior art date
Application number
UY27552A
Other languages
English (en)
Inventor
Rolf Jautelat
Orlin Petrov
Rolf Bohlmann
Nikolaus Heinrich
Jorg Kroll
Andreas Reichel
Jens Hoffmann
Rosemarie Lichtner
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of UY27552A1 publication Critical patent/UY27552A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16—Masculine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/14—Drugs for dermatological disorders for baldness or alopecia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32—Antioestrogens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Gynecology & Obstetrics (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Pregnancy & Childbirth (AREA)
  • Urology & Nephrology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Se proponen los 17a-alquil-17b-oxi-estra-1,3,5(10)-trienos de la fórmula general I. Además, la invención también se refiere a los 17-oxo-estra-1,3,5(10)-trienos, así como a los 17b-hidroxi-estra-1,3,5(10)-trienos como productos intermediarios en la preparación de los estratrieno de la invención. Por otra parte, la invención se refiere al uso de los 17a- alquil-17b-oxi-estratrienos para obtener medicamentos y preparados farmacéuticos, que contienen al menos un 17a- alquil-17b- oxi-estratrieno,así como al menos un soporte de tolerancia farmacéutica.
UY27552A 2001-11-27 2002-11-27 17a- alquil- 17b- oxi-estratrienos y productos intermediarios para su preparacinn, uso de los 17a-alquil-17b-oxi-estratrienos para obtener medicamentos y preparados farmacéuticos. UY27552A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10159217A DE10159217A1 (de) 2001-11-27 2001-11-27 17alpha-Alkyl-17ß-oxy-estratriene und Zwischenprodukte zu deren Herstellung, Verwendung der 17alpha-Alkyl-17ß-oxy-estratriene zur Herstellung von Arzneimitteln sowie pharmazeutische Präparate

Publications (1)

Publication Number Publication Date
UY27552A1 true UY27552A1 (es) 2003-06-30

Family

ID=7707804

Family Applications (1)

Application Number Title Priority Date Filing Date
UY27552A UY27552A1 (es) 2001-11-27 2002-11-27 17a- alquil- 17b- oxi-estratrienos y productos intermediarios para su preparacinn, uso de los 17a-alquil-17b-oxi-estratrienos para obtener medicamentos y preparados farmacéuticos.

Country Status (25)

Country Link
US (2) US7018994B2 (es)
EP (2) EP1916254A3 (es)
JP (3) JP2005513039A (es)
KR (1) KR100956912B1 (es)
CN (2) CN100558741C (es)
AR (1) AR037674A1 (es)
AT (1) ATE396198T1 (es)
AU (1) AU2002360949A1 (es)
BR (1) BR0214469A (es)
CA (1) CA2468412C (es)
CY (1) CY1108279T1 (es)
DE (2) DE10159217A1 (es)
DK (1) DK1448591T3 (es)
ES (1) ES2307819T3 (es)
IL (2) IL162200A0 (es)
MX (1) MXPA04005015A (es)
NO (2) NO326241B1 (es)
PE (1) PE20030727A1 (es)
PL (1) PL207955B1 (es)
PT (1) PT1448591E (es)
RU (2) RU2339643C2 (es)
TW (1) TWI256891B (es)
UY (1) UY27552A1 (es)
WO (1) WO2003045972A1 (es)
ZA (2) ZA200405029B (es)

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DE102007023614A1 (de) 2007-05-21 2008-11-27 Bayer Schering Pharma Aktiengesellschaft Nichtsteroidale Progesteronrezeptor-Modulatoren
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Also Published As

Publication number Publication date
DE50212302D1 (de) 2008-07-03
DK1448591T3 (da) 2008-09-29
KR100956912B1 (ko) 2010-05-11
RU2285009C2 (ru) 2006-10-10
US7538100B2 (en) 2009-05-26
NO20044192L (no) 2004-10-04
ES2307819T3 (es) 2008-12-01
JP2005513039A (ja) 2005-05-12
ZA200407868B (en) 2005-04-26
EP1448591A1 (de) 2004-08-25
RU2339643C2 (ru) 2008-11-27
PL369171A1 (en) 2005-04-18
NO20042694L (no) 2004-07-22
BR0214469A (pt) 2004-10-13
EP1916254A2 (de) 2008-04-30
DE10159217A1 (de) 2003-06-05
AU2002360949A1 (en) 2003-06-10
NO326241B1 (no) 2008-10-27
CN1617879A (zh) 2005-05-18
PT1448591E (pt) 2008-09-19
US20060009436A1 (en) 2006-01-12
CN1325507C (zh) 2007-07-11
TW200305426A (en) 2003-11-01
ZA200405029B (en) 2009-07-29
WO2003045972A1 (de) 2003-06-05
MXPA04005015A (es) 2005-04-08
CA2468412A1 (en) 2003-06-05
KR20040063158A (ko) 2004-07-12
EP1448591B1 (de) 2008-05-21
PL207955B1 (pl) 2011-02-28
TWI256891B (en) 2006-06-21
US20030191099A1 (en) 2003-10-09
RU2004119437A (ru) 2005-07-10
HK1079215A1 (en) 2006-03-31
CY1108279T1 (el) 2014-02-12
HK1077832A1 (en) 2006-02-24
CN100558741C (zh) 2009-11-11
CN1637015A (zh) 2005-07-13
JP2005120110A (ja) 2005-05-12
JP4335820B2 (ja) 2009-09-30
IL162200A0 (en) 2005-11-20
PE20030727A1 (es) 2003-09-18
US7018994B2 (en) 2006-03-28
RU2006120215A (ru) 2008-01-10
IL162200A (en) 2010-06-30
EP1916254A3 (de) 2012-11-14
ATE396198T1 (de) 2008-06-15
CA2468412C (en) 2010-01-12
AR037674A1 (es) 2004-12-01
JP2006306896A (ja) 2006-11-09

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