RU2010146999A - PHARMACEUTICAL COMPOSITION CONTAINING CHONDROITIN SULPHATE AND / OR HYALURONIDASE AND LIPOSOMES FOR LOCAL USE - Google Patents
PHARMACEUTICAL COMPOSITION CONTAINING CHONDROITIN SULPHATE AND / OR HYALURONIDASE AND LIPOSOMES FOR LOCAL USE Download PDFInfo
- Publication number
- RU2010146999A RU2010146999A RU2010146999/15A RU2010146999A RU2010146999A RU 2010146999 A RU2010146999 A RU 2010146999A RU 2010146999/15 A RU2010146999/15 A RU 2010146999/15A RU 2010146999 A RU2010146999 A RU 2010146999A RU 2010146999 A RU2010146999 A RU 2010146999A
- Authority
- RU
- Russia
- Prior art keywords
- pharmaceutical composition
- hyaluronidase
- liposomes
- composition according
- chondroitin sulfate
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title claims abstract 9
- 229920001287 Chondroitin sulfate Polymers 0.000 title claims abstract 7
- 108010003272 Hyaluronate lyase Proteins 0.000 title claims abstract 7
- 102000001974 Hyaluronidases Human genes 0.000 title claims abstract 7
- 229960002773 hyaluronidase Drugs 0.000 title claims abstract 7
- 239000002502 liposome Substances 0.000 title claims abstract 7
- YKPUWZUDDOIDPM-SOFGYWHQSA-N capsaicin Chemical compound COC1=CC(CNC(=O)CCCC\C=C\C(C)C)=CC=C1O YKPUWZUDDOIDPM-SOFGYWHQSA-N 0.000 claims abstract 8
- CBOJBBMQJBVCMW-BTVCFUMJSA-N (2r,3r,4s,5r)-2-amino-3,4,5,6-tetrahydroxyhexanal;hydrochloride Chemical compound Cl.O=C[C@H](N)[C@@H](O)[C@H](O)[C@H](O)CO CBOJBBMQJBVCMW-BTVCFUMJSA-N 0.000 claims abstract 6
- SQDAZGGFXASXDW-UHFFFAOYSA-N 5-bromo-2-(trifluoromethoxy)pyridine Chemical compound FC(F)(F)OC1=CC=C(Br)C=N1 SQDAZGGFXASXDW-UHFFFAOYSA-N 0.000 claims abstract 6
- 229940059329 chondroitin sulfate Drugs 0.000 claims abstract 6
- 229960001911 glucosamine hydrochloride Drugs 0.000 claims abstract 6
- 229960002504 capsaicin Drugs 0.000 claims abstract 4
- 235000017663 capsaicin Nutrition 0.000 claims abstract 4
- 239000003995 emulsifying agent Substances 0.000 claims abstract 4
- 239000000203 mixture Substances 0.000 claims abstract 4
- 239000003755 preservative agent Substances 0.000 claims abstract 4
- 230000002335 preservative effect Effects 0.000 claims abstract 4
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims abstract 4
- 239000003937 drug carrier Substances 0.000 claims abstract 2
- 239000000546 pharmaceutical excipient Substances 0.000 claims abstract 2
- 239000012049 topical pharmaceutical composition Substances 0.000 claims abstract 2
Landscapes
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
1. Фармацевтическая композиция для местного применения, содержащая хондроитин сульфат и/или гиалуронидазу и фармацевтически приемлемые носители или эксципиенты, отличающаяся тем, что она дополнительно включает в себя липосомы. ! 2. Фармацевтическая композиция по п.1, отличающаяся тем, что она дополнительно содержит глюкозамина гидрохлорид. ! 3. Фармацевтическая композиция по п.2, отличающаяся тем, что она имеет следующий состав, мас.%: ! Хондроитин сульфат 0,01-5,0 Липосомы 0,01-20,0 Гиалуронидаза 0,01-1,0 Глюкозамина гидрохлорид 0,01-10,0 Эмульгатор 0,5-10,0 Консервант 0,05-1,0Вода деминерализованная 53,0-99,41 ! 4. Фармацевтическая композиция по п.3, отличающаяся тем, что она дополнительно содержит капсаицин. ! 5. Фармацевтическая композиция по п.4, отличающаяся тем, что она имеет следующий состав, мас.%: ! Хондроитин сульфат 0,01-5,0 Липосомы 0,01-20,0 Глюкозамина гидрохлорид 0,01-10,0 Капсаицин 0,01-1,0 Гиалуронидаза 0,01-1,0 Эмульгатор 0,5-10,0 Консервант 0,05-1,0 Вода деминерализованная 52,0-99,4 1. A topical pharmaceutical composition comprising chondroitin sulfate and / or hyaluronidase and pharmaceutically acceptable carriers or excipients, characterized in that it further includes liposomes. ! 2. The pharmaceutical composition according to claim 1, characterized in that it further comprises glucosamine hydrochloride. ! 3. The pharmaceutical composition according to claim 2, characterized in that it has the following composition, wt.%:! Chondroitin sulfate 0.01-5.0 Liposomes 0.01-20.0 Hyaluronidase 0.01-1.0 Glucosamine hydrochloride 0.01-10.0 Emulsifier 0.5-10.0 Preservative 0.05-1.0 Water demineralized 53.0-99.41! 4. The pharmaceutical composition according to claim 3, characterized in that it further comprises capsaicin. ! 5. The pharmaceutical composition according to claim 4, characterized in that it has the following composition, wt.%:! Chondroitin sulfate 0.01-5.0 Liposomes 0.01-20.0 Glucosamine hydrochloride 0.01-10.0 Capsaicin 0.01-1.0 Hyaluronidase 0.01-1.0 Emulsifier 0.5-10.0 Preservative 0.05-1.0 Demineralized water 52.0-99.4
Claims (5)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2010146999/15A RU2473350C2 (en) | 2010-11-17 | 2010-11-17 | Pharmaceutical composition containing chondroitin sulphate and/or hyaluronidase and liposome for local application |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2010146999/15A RU2473350C2 (en) | 2010-11-17 | 2010-11-17 | Pharmaceutical composition containing chondroitin sulphate and/or hyaluronidase and liposome for local application |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| RU2010146999A true RU2010146999A (en) | 2012-05-27 |
| RU2473350C2 RU2473350C2 (en) | 2013-01-27 |
Family
ID=46231312
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2010146999/15A RU2473350C2 (en) | 2010-11-17 | 2010-11-17 | Pharmaceutical composition containing chondroitin sulphate and/or hyaluronidase and liposome for local application |
Country Status (1)
| Country | Link |
|---|---|
| RU (1) | RU2473350C2 (en) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2539390C1 (en) * | 2013-05-21 | 2015-01-20 | Леонид Леонидович Клопотенко | Composition containing chondroitin sulphate and hyaluronidase |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2004121471A (en) * | 2004-07-14 | 2006-01-10 | Хамзат Хамидович Арсамаков (RU) | COSMETIC COMPOSITION FOR LOCAL USE CONTAINING CHONDROITIN SULPHATE AND LIPOSOMES |
| RU2355420C2 (en) * | 2007-06-29 | 2009-05-20 | Леонид Леонидович Клопотенко | Toothpaste containing lactulose, betaine, chondroitin sulphate and enzymes: papain, lysocim, ribonuclease and lidase |
| RU2381021C2 (en) * | 2007-11-12 | 2010-02-10 | Леонид Леонидович Клопотенко | Liposome containing tooth paste |
| RU2376011C1 (en) * | 2008-05-19 | 2009-12-20 | Открытое Акционерное Общество Завод Экологической Техники И Экопитания "Диод" | Agent for care of peripheral joints and backbone area |
-
2010
- 2010-11-17 RU RU2010146999/15A patent/RU2473350C2/en not_active IP Right Cessation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2539390C1 (en) * | 2013-05-21 | 2015-01-20 | Леонид Леонидович Клопотенко | Composition containing chondroitin sulphate and hyaluronidase |
Also Published As
| Publication number | Publication date |
|---|---|
| RU2473350C2 (en) | 2013-01-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | The patent is invalid due to non-payment of fees |
Effective date: 20161118 |