RU2012128102A - PHARMACEUTICAL COMPOSITION CONTAINING EPIRUBICIN OR MITOXANTRON OR OR MITOMYCIN AND LIPOSOMA OR BETA-CYCLODEXTRIN - Google Patents
PHARMACEUTICAL COMPOSITION CONTAINING EPIRUBICIN OR MITOXANTRON OR OR MITOMYCIN AND LIPOSOMA OR BETA-CYCLODEXTRIN Download PDFInfo
- Publication number
- RU2012128102A RU2012128102A RU2012128102/15A RU2012128102A RU2012128102A RU 2012128102 A RU2012128102 A RU 2012128102A RU 2012128102/15 A RU2012128102/15 A RU 2012128102/15A RU 2012128102 A RU2012128102 A RU 2012128102A RU 2012128102 A RU2012128102 A RU 2012128102A
- Authority
- RU
- Russia
- Prior art keywords
- pharmaceutical composition
- mitomycin
- composition according
- beta
- following composition
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title claims abstract 13
- AOJJSUZBOXZQNB-VTZDEGQISA-N 4'-epidoxorubicin Chemical compound O([C@H]1C[C@@](O)(CC=2C(O)=C3C(=O)C=4C=CC=C(C=4C(=O)C3=C(O)C=21)OC)C(=O)CO)[C@H]1C[C@H](N)[C@@H](O)[C@H](C)O1 AOJJSUZBOXZQNB-VTZDEGQISA-N 0.000 title claims abstract 5
- 229920000858 Cyclodextrin Polymers 0.000 title claims abstract 5
- HTIJFSOGRVMCQR-UHFFFAOYSA-N Epirubicin Natural products COc1cccc2C(=O)c3c(O)c4CC(O)(CC(OC5CC(N)C(=O)C(C)O5)c4c(O)c3C(=O)c12)C(=O)CO HTIJFSOGRVMCQR-UHFFFAOYSA-N 0.000 title claims abstract 5
- 229930192392 Mitomycin Natural products 0.000 title claims abstract 5
- NWIBSHFKIJFRCO-WUDYKRTCSA-N Mytomycin Chemical compound C1N2C(C(C(C)=C(N)C3=O)=O)=C3[C@@H](COC(N)=O)[C@@]2(OC)[C@@H]2[C@H]1N2 NWIBSHFKIJFRCO-WUDYKRTCSA-N 0.000 title claims abstract 5
- WHGYBXFWUBPSRW-FOUAGVGXSA-N beta-cyclodextrin Chemical compound OC[C@H]([C@H]([C@@H]([C@H]1O)O)O[C@H]2O[C@@H]([C@@H](O[C@H]3O[C@H](CO)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](CO)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](CO)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](CO)[C@H]([C@@H]([C@H]3O)O)O3)[C@H](O)[C@H]2O)CO)O[C@@H]1O[C@H]1[C@H](O)[C@@H](O)[C@@H]3O[C@@H]1CO WHGYBXFWUBPSRW-FOUAGVGXSA-N 0.000 title claims abstract 5
- 235000011175 beta-cyclodextrine Nutrition 0.000 title claims abstract 5
- 229960001904 epirubicin Drugs 0.000 title claims abstract 5
- 229960004857 mitomycin Drugs 0.000 title claims abstract 5
- KKZJGLLVHKMTCM-UHFFFAOYSA-N mitoxantrone Chemical compound O=C1C2=C(O)C=CC(O)=C2C(=O)C2=C1C(NCCNCCO)=CC=C2NCCNCCO KKZJGLLVHKMTCM-UHFFFAOYSA-N 0.000 title claims abstract 5
- 239000001116 FEMA 4028 Substances 0.000 title claims 3
- 229960004853 betadex Drugs 0.000 title claims 3
- 239000000203 mixture Substances 0.000 claims abstract 12
- 239000002502 liposome Substances 0.000 claims abstract 6
- 229960001156 mitoxantrone Drugs 0.000 claims abstract 4
- 239000003937 drug carrier Substances 0.000 claims abstract 2
- 239000000546 pharmaceutical excipient Substances 0.000 claims abstract 2
- 239000012049 topical pharmaceutical composition Substances 0.000 claims abstract 2
- 239000003995 emulsifying agent Substances 0.000 claims 6
- 239000003755 preservative agent Substances 0.000 claims 6
- 230000002335 preservative effect Effects 0.000 claims 6
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 claims 6
- 229920000036 polyvinylpyrrolidone Polymers 0.000 claims 5
- 235000013855 polyvinylpyrrolidone Nutrition 0.000 claims 5
- 239000001267 polyvinylpyrrolidone Substances 0.000 claims 5
- NIXOWILDQLNWCW-UHFFFAOYSA-N Acrylic acid Chemical compound OC(=O)C=C NIXOWILDQLNWCW-UHFFFAOYSA-N 0.000 claims 1
- 229920002125 Sokalan® Polymers 0.000 claims 1
- 229960001631 carbomer Drugs 0.000 claims 1
Landscapes
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
1. Фармацевтическая композиция для местного применения, содержащая эпирубицин или митоксантрон, или митомицин и фармацевтически приемлемые носители, или эксципиенты, отличающаяся тем, что она дополнительно включает в себя липосомы или бета-циклодекстрины.2. Фармацевтическая композиция по п.1, отличающаяся тем, что она имеет следующий состав, мас.%:3. Фармацевтическая композиция по п.1, отличающаяся тем, что она имеет следующий состав, мас.%:4. Фармацевтическая композиция по п.1, отличающаяся тем, что она имеет следующий состав, мас.%:5. Фармацевтическая композиция по п.1, отличающаяся тем, что она имеет следующий состав, мас.%:6. Фармацевтическая композиция по п.1, отличающаяся тем, что она имеет следующий состав, мас.%:7. Фармацевтическая композиция по п.1, отличающаяся тем, что она имеет следующий состав, мас.%:1. A topical pharmaceutical composition comprising epirubicin or mitoxantrone or mitomycin and pharmaceutically acceptable carriers or excipients, characterized in that it further comprises liposomes or beta-cyclodextrins. The pharmaceutical composition according to claim 1, characterized in that it has the following composition, wt.%: 3. The pharmaceutical composition according to claim 1, characterized in that it has the following composition, wt.%: 4. The pharmaceutical composition according to claim 1, characterized in that it has the following composition, wt.%: 5. The pharmaceutical composition according to claim 1, characterized in that it has the following composition, wt.%: 6. The pharmaceutical composition according to claim 1, characterized in that it has the following composition, wt.%: 7. The pharmaceutical composition according to claim 1, characterized in that it has the following composition, wt.%:
Claims (7)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2012128102/15A RU2012128102A (en) | 2012-07-03 | 2012-07-03 | PHARMACEUTICAL COMPOSITION CONTAINING EPIRUBICIN OR MITOXANTRON OR OR MITOMYCIN AND LIPOSOMA OR BETA-CYCLODEXTRIN |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| RU2012128102/15A RU2012128102A (en) | 2012-07-03 | 2012-07-03 | PHARMACEUTICAL COMPOSITION CONTAINING EPIRUBICIN OR MITOXANTRON OR OR MITOMYCIN AND LIPOSOMA OR BETA-CYCLODEXTRIN |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| RU2012128102A true RU2012128102A (en) | 2014-01-20 |
Family
ID=49944672
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| RU2012128102/15A RU2012128102A (en) | 2012-07-03 | 2012-07-03 | PHARMACEUTICAL COMPOSITION CONTAINING EPIRUBICIN OR MITOXANTRON OR OR MITOMYCIN AND LIPOSOMA OR BETA-CYCLODEXTRIN |
Country Status (1)
| Country | Link |
|---|---|
| RU (1) | RU2012128102A (en) |
-
2012
- 2012-07-03 RU RU2012128102/15A patent/RU2012128102A/en unknown
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