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PE20210377A1 - Anticuerpos anti-pd-l1 y usos de los mismos - Google Patents

Anticuerpos anti-pd-l1 y usos de los mismos

Info

Publication number
PE20210377A1
PE20210377A1 PE2020001301A PE2020001301A PE20210377A1 PE 20210377 A1 PE20210377 A1 PE 20210377A1 PE 2020001301 A PE2020001301 A PE 2020001301A PE 2020001301 A PE2020001301 A PE 2020001301A PE 20210377 A1 PE20210377 A1 PE 20210377A1
Authority
PE
Peru
Prior art keywords
seq
antibodies
fragments
cdr1
cdr2
Prior art date
Application number
PE2020001301A
Other languages
English (en)
Inventor
Lei Fang
Yongqiang Wang
Zhengyi Wang
Bingshi Guo
Jingwu Zang
Original Assignee
I Mab Biopharma Us Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by I Mab Biopharma Us Ltd filed Critical I Mab Biopharma Us Ltd
Publication of PE20210377A1 publication Critical patent/PE20210377A1/es

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K16/00Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
    • C07K16/18Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans
    • C07K16/28Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants
    • C07K16/2803Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against the immunoglobulin superfamily
    • C07K16/2827Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies against material from animals or humans against receptors, cell surface antigens or cell surface determinants against the immunoglobulin superfamily against B7 molecules, e.g. CD80, CD86
    • G01N33/575
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K39/00Medicinal preparations containing antigens or antibodies
    • A61K2039/505Medicinal preparations containing antigens or antibodies comprising antibodies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/20Immunoglobulins specific features characterized by taxonomic origin
    • C07K2317/24Immunoglobulins specific features characterized by taxonomic origin containing regions, domains or residues from different species, e.g. chimeric, humanized or veneered
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/30Immunoglobulins specific features characterized by aspects of specificity or valency
    • C07K2317/33Crossreactivity, e.g. for species or epitope, or lack of said crossreactivity
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/30Immunoglobulins specific features characterized by aspects of specificity or valency
    • C07K2317/34Identification of a linear epitope shorter than 20 amino acid residues or of a conformational epitope defined by amino acid residues
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/50Immunoglobulins specific features characterized by immunoglobulin fragments
    • C07K2317/56Immunoglobulins specific features characterized by immunoglobulin fragments variable (Fv) region, i.e. VH and/or VL
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/50Immunoglobulins specific features characterized by immunoglobulin fragments
    • C07K2317/56Immunoglobulins specific features characterized by immunoglobulin fragments variable (Fv) region, i.e. VH and/or VL
    • C07K2317/565Complementarity determining region [CDR]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/50Immunoglobulins specific features characterized by immunoglobulin fragments
    • C07K2317/56Immunoglobulins specific features characterized by immunoglobulin fragments variable (Fv) region, i.e. VH and/or VL
    • C07K2317/567Framework region [FR]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/73Inducing cell death, e.g. apoptosis, necrosis or inhibition of cell proliferation
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/70Immunoglobulins specific features characterized by effect upon binding to a cell or to an antigen
    • C07K2317/76Antagonist effect on antigen, e.g. neutralization or inhibition of binding
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K2317/00Immunoglobulins specific features
    • C07K2317/90Immunoglobulins specific features characterized by (pharmaco)kinetic aspects or by stability of the immunoglobulin
    • C07K2317/92Affinity (KD), association rate (Ka), dissociation rate (Kd) or EC50 value
    • GPHYSICS
    • G01MEASURING; TESTING
    • G01NINVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2333/00Assays involving biological materials from specific organisms or of a specific nature
    • G01N2333/435Assays involving biological materials from specific organisms or of a specific nature from animals; from humans
    • G01N2333/705Assays involving receptors, cell surface antigens or cell surface determinants
    • G01N2333/70503Immunoglobulin superfamily, e.g. VCAMs, PECAM, LFA-3
    • G01N2333/70532B7 molecules, e.g. CD80, CD86

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Engineering & Computer Science (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Biotechnology (AREA)
  • Cell Biology (AREA)
  • Oncology (AREA)
  • Microbiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Food Science & Technology (AREA)
  • Physics & Mathematics (AREA)
  • Analytical Chemistry (AREA)
  • General Physics & Mathematics (AREA)
  • Pathology (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente invencion se refiere a anticuerpos anti-PD-L1 o fragmentos de los mismos que se unen especificamente al dominio C de inmunoglobulina de la proteina PD-L1, en particular los residuos de aminoacidos Y134, K162 y N183. En varios ejemplos, los anticuerpos o fragmentos de los mismos incluyen una VH CDR1 de la SEQ ID NO: 1, una VH CDR2 de la SEQ ID NO: 116, una VH CDR3 de la SEQ ID NO: 117, una VL CDR1 de la SEQ ID NO: 4, una VL CDR2 de la SEQ ID NO: 5, y una VL CDR3 de la SEQ ID NO: 6, o variantes de cada uno de los mismos, utiles en el tratamiento y diagnostico de enfermedades tales como cancer y enfermedades infecciosas. Tambien se refiere a anticuerpos biespecificos, metodos de tratamiento y composiciones que comprende el anticuerpo o fragmentos de los mismos
PE2020001301A 2018-03-29 2019-03-29 Anticuerpos anti-pd-l1 y usos de los mismos PE20210377A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CN2018081079 2018-03-29
PCT/CN2019/080458 WO2019185029A1 (en) 2018-03-29 2019-03-29 Anti-pd-l1 antibodies and uses thereof

Publications (1)

Publication Number Publication Date
PE20210377A1 true PE20210377A1 (es) 2021-03-02

Family

ID=68060946

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2020001301A PE20210377A1 (es) 2018-03-29 2019-03-29 Anticuerpos anti-pd-l1 y usos de los mismos

Country Status (18)

Country Link
US (2) US11220546B2 (es)
EP (1) EP3589660A4 (es)
JP (1) JP7124257B2 (es)
KR (2) KR102177931B1 (es)
CN (1) CN110891975B (es)
AU (1) AU2019241339B2 (es)
BR (1) BR112020019827A2 (es)
CA (1) CA3086434C (es)
CL (1) CL2020002223A1 (es)
EA (1) EA202091590A1 (es)
IL (1) IL275734B (es)
MX (1) MX2020007842A (es)
MY (1) MY188237A (es)
PE (1) PE20210377A1 (es)
PH (1) PH12020551173A1 (es)
SG (1) SG11202006008WA (es)
UA (1) UA125918C2 (es)
WO (1) WO2019185029A1 (es)

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* Cited by examiner, † Cited by third party
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MX2018015584A (es) * 2016-06-13 2019-09-18 I Mab Anticuerpos anti-pd-l1 y usos de los mismos.
WO2020020307A1 (en) * 2018-07-25 2020-01-30 I-Mab Biopharma Co., Ltd. Anti-cd73 anti-pd-l1 bispecific antibodies
AU2019326635B2 (en) * 2018-08-21 2024-05-23 Abl Bio Inc. Anti-PD-L1/anti-LAG3 bispecific antibodies and uses thereof
WO2021097800A1 (en) * 2019-11-22 2021-05-27 Abl Bio Inc. Anti-pd-l1/anti-b7-h3 multispecific antibodies and uses thereof
CN115643797A (zh) * 2020-04-30 2023-01-24 天境生物科技(上海)有限公司 包含抗cd47抗体的药物组合物
CN121319180A (zh) * 2020-07-28 2026-01-13 乐普生物科技股份有限公司 靶向PD-L1和TGF-β的双功能分子
KR20230166150A (ko) 2020-08-19 2023-12-06 젠코어 인코포레이티드 항-cd28 조성물
CN114195900B (zh) * 2020-09-17 2024-02-23 普米斯生物技术(珠海)有限公司 一种抗4-1bb/pd-l1双特异性抗体及其用途
CN114316045B (zh) * 2020-09-29 2024-07-12 英诺欧奇生物医药(苏州)有限公司 抗pd-l1抗体及其用途
CN113234162B (zh) * 2020-12-24 2022-05-13 四川大学华西医院 一种靶向cd133的嵌合抗原受体t细胞
EP4276466A4 (en) * 2021-01-08 2024-12-18 Beijing Hanmi Pharmaceutical Co., Ltd. ANTIBODY SPECIFICALLY BINDING WITH PD-L1 AND ANTIGEN-BINDING FRAGMENT OF ANTIBODY
BR112023016706A2 (pt) * 2021-02-19 2023-10-31 Seoul Nat Univ R&Db Foundation Anticorpo ou um fragmento de ligação ao antígeno do mesmo, molécula de ácido nucleico, métodos para produzir um anticorpo ou um fragmento de ligação ao antígeno do mesmo e para detectar agrupamento de diferenciação 47 ou determinar uma quantidade de agrupamento de diferenciação 47 em uma amostra, e, uso do anticorpo ou de um fragmento de ligação ao antígeno do mesmo
CN115073599B (zh) * 2021-03-16 2023-04-28 北京天广实生物技术股份有限公司 结合pd-l1的抗体及其用途
CA3252619A1 (en) 2022-02-23 2023-08-31 Xencor, Inc. Anti-CD28 and anti-PSMA antibodies
US20250215089A1 (en) * 2022-04-02 2025-07-03 Harbour Biomed (Shanghai) Co., Ltd Antigen-binding protein targeting pd-l1 and cd40, preparation therefor, and use thereof
EP4619439A1 (en) * 2022-11-15 2025-09-24 TJ Biopharma (Shanghai) Co., Ltd. Anti-pd-l1 nanobodies

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PL2161336T5 (pl) * 2005-05-09 2017-10-31 Ono Pharmaceutical Co Ludzkie przeciwciała monoklonalne przeciwko białku Programmed Death 1 (PD-1) oraz sposoby leczenia raka z zastosowaniem samych przeciwciał anty-PD-1 lub w połączeniu z innymi środkami immunoterapeutycznymi
WO2011043194A1 (en) 2009-10-09 2011-04-14 Semiconductor Energy Laboratory Co., Ltd. Semiconductor device and method for manufacturing the same
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CN110156892B (zh) 2014-07-03 2023-05-16 百济神州有限公司 抗pd-l1抗体及其作为治疗剂及诊断剂的用途
LT3789402T (lt) * 2014-11-20 2022-09-26 F. Hoffmann-La Roche Ag Kompleksinė terapija, naudojant t ląsteles aktyvinančias bispecifines antigeną surišančias molekules ir pd-1 ašį surišančius antagonistus
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MX2018015584A (es) * 2016-06-13 2019-09-18 I Mab Anticuerpos anti-pd-l1 y usos de los mismos.
CN107488229B (zh) * 2016-06-13 2020-11-17 天境生物科技(上海)有限公司 Pd-l1抗体及其用途
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Also Published As

Publication number Publication date
US11220546B2 (en) 2022-01-11
AU2019241339A1 (en) 2019-11-14
JP7124257B2 (ja) 2022-08-24
IL275734B (en) 2022-06-01
BR112020019827A2 (pt) 2021-01-05
CA3086434A1 (en) 2019-10-03
UA125918C2 (uk) 2022-07-06
CN110891975A (zh) 2020-03-17
WO2019185029A1 (en) 2019-10-03
EP3589660A4 (en) 2021-04-07
EP3589660A1 (en) 2020-01-08
MX2020007842A (es) 2020-09-25
KR102475106B1 (ko) 2022-12-08
KR102177931B1 (ko) 2020-11-13
US20220119531A1 (en) 2022-04-21
KR20190128716A (ko) 2019-11-18
CN110891975B (zh) 2023-11-10
EA202091590A1 (ru) 2021-01-21
MY188237A (en) 2021-11-24
KR20200130747A (ko) 2020-11-19
JP2020518233A (ja) 2020-06-25
AU2019241339B2 (en) 2021-08-12
CL2020002223A1 (es) 2021-01-29
PH12020551173A1 (en) 2021-05-31
SG11202006008WA (en) 2020-07-29
NZ758371A (en) 2024-10-25
CA3086434C (en) 2024-01-09
US20200157222A1 (en) 2020-05-21
IL275734A (en) 2020-08-31

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