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HUP0100470A3 - Oxazolidinone derivatives and pharmaceutical compositions containing them - Google Patents

Oxazolidinone derivatives and pharmaceutical compositions containing them

Info

Publication number
HUP0100470A3
HUP0100470A3 HU0100470A HUP0100470A HUP0100470A3 HU P0100470 A3 HUP0100470 A3 HU P0100470A3 HU 0100470 A HU0100470 A HU 0100470A HU P0100470 A HUP0100470 A HU P0100470A HU P0100470 A3 HUP0100470 A3 HU P0100470A3
Authority
HU
Hungary
Prior art keywords
pharmaceutical compositions
compositions containing
oxazolidinone derivatives
oxazolidinone
derivatives
Prior art date
Application number
HU0100470A
Other languages
English (en)
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of HUP0100470A2 publication Critical patent/HUP0100470A2/hu
Publication of HUP0100470A3 publication Critical patent/HUP0100470A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU0100470A 1997-11-12 1998-10-30 Oxazolidinone derivatives and pharmaceutical compositions containing them HUP0100470A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6537697P 1997-11-12 1997-11-12

Publications (2)

Publication Number Publication Date
HUP0100470A2 HUP0100470A2 (hu) 2002-05-29
HUP0100470A3 true HUP0100470A3 (en) 2002-08-28

Family

ID=22062294

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0100470A HUP0100470A3 (en) 1997-11-12 1998-10-30 Oxazolidinone derivatives and pharmaceutical compositions containing them

Country Status (21)

Country Link
US (1) US5998406A (hu)
EP (1) EP1030852B1 (hu)
JP (1) JP2001522849A (hu)
KR (1) KR20010031953A (hu)
CN (1) CN1154644C (hu)
AT (1) ATE250054T1 (hu)
AU (1) AU739055B2 (hu)
BR (1) BR9813985A (hu)
CA (1) CA2303959A1 (hu)
DE (1) DE69818294T2 (hu)
DK (1) DK1030852T3 (hu)
ES (1) ES2207010T3 (hu)
HU (1) HUP0100470A3 (hu)
IL (1) IL136062A (hu)
NO (1) NO317291B1 (hu)
NZ (1) NZ504503A (hu)
PT (1) PT1030852E (hu)
RU (1) RU2215740C2 (hu)
SK (1) SK284577B6 (hu)
TR (1) TR200001330T2 (hu)
WO (1) WO1999024428A1 (hu)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ508174A (en) 1998-06-05 2003-10-31 Astrazeneca Ab Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
DE19962924A1 (de) 1999-12-24 2001-07-05 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
KR100355345B1 (ko) * 2000-01-21 2002-10-12 한국과학기술연구원 티오펜환을 함유한 신규한 옥사졸리디논 유도체, 그의 제조방법 및 조성물
GB0009803D0 (en) 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
DE10129725A1 (de) 2001-06-20 2003-01-02 Bayer Ag Kombinationstherapie substituierter Oxazolidinone
MXPA05001558A (es) * 2002-08-12 2005-09-08 Pharmacia & Upjohn Co Llc N-aril-2-oxazolidinonas y sus derivados.
DE10300111A1 (de) 2003-01-07 2004-07-15 Bayer Healthcare Ag Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid
WO2005019214A1 (en) * 2003-08-25 2005-03-03 Warner-Lambert Company Llc Novel antimicrobial aryloxazolidinone compounds
DE10355461A1 (de) 2003-11-27 2005-06-23 Bayer Healthcare Ag Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung
KR100854211B1 (ko) * 2003-12-18 2008-08-26 동아제약주식회사 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물
EP1819699A2 (en) * 2004-11-29 2007-08-22 Pharmacia & Upjohn Company LLC Diazepine oxazolidinones as antibacterial agents
DE102004062475A1 (de) * 2004-12-24 2006-07-06 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung
EP1685841A1 (en) 2005-01-31 2006-08-02 Bayer Health Care Aktiengesellschaft Prevention and treatment of thromboembolic disorders
ES2335307T3 (es) 2005-06-29 2010-03-24 PHARMACIA & UPJOHN COMPANY LLC Homomorfolin oxalidinonas como agentes antibacterianos.
DE102005045518A1 (de) * 2005-09-23 2007-03-29 Bayer Healthcare Ag 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung
BRPI0616801B8 (pt) 2005-10-04 2021-05-25 Bayer Healthcare Ag "forma polimórfica de 5-cloro-n-({(5s)-2-oxo-3-[4-(3-oxo-4-morfolinil)-fenil]-1,3-oxazolidin-5-il}-metil)-2-tiofenocarboxamida, seus processos de preparação e seus usos, medicamento, e processo para prevenção de coagulação de sangue in vitro
DE102005047558A1 (de) * 2005-10-04 2008-02-07 Bayer Healthcare Ag Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen
DE102005047561A1 (de) 2005-10-04 2007-04-05 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung
TW200804358A (en) 2006-03-31 2008-01-16 Res Found Itsuu Lab Novel compound having heterocycle
EP2208729A4 (en) 2007-10-02 2011-04-27 Res Found Itsuu Lab OXAZOLIDINONE DERIVATIVE WITH 7-CHAIN HETEROCYCLE
KR20130102614A (ko) 2010-11-03 2013-09-17 욱크하르트 리미티드 인산 모노-(1-[4-[(s)-5-(아세틸아미노메틸)-2-옥소-옥사졸리딘-3-일]-2,6-디플루오로페닐]-4-메톡시메틸피페리딘-4-일) 에스테르의 제조 방법
WO2015173664A1 (en) 2014-05-14 2015-11-19 Wockhardt Limited Process for the preparation of (5s)-n-{3-[3,5-difluoro-4-(4-hydroxy-4-methoxymethyl-piperidin-1-yl)-phenyl]-2-oxo-oxazolidin-5-ylmethyl}-acetamide

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
CA1320730C (en) * 1987-10-16 1993-07-27 The Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
DE3884563T2 (de) * 1987-10-21 1994-02-17 Du Pont Merck Pharma Aminomethyl-oxo-oxazolidinyl-ethenylbenzen-Derivate, nützlich als antibakterielles Mittel.
US4948801A (en) * 1988-07-29 1990-08-14 E. I. Du Pont De Nemours And Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
DE68918792T2 (de) * 1988-09-15 1995-03-30 Upjohn Co 5-Indolinyl-5-beta-amidomethyloxazolidin-2-one, 3-(substituierte kondensierte)phenyl-5-beta amidomethyloxazolidin-2-one und 3-(Nitrogen-substituierte)phenyl-5-beta-amidomethyloxazolidin-2-one.
WO1993009103A1 (en) * 1991-11-01 1993-05-13 The Upjohn Company Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents
SK283420B6 (sk) * 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
WO1995014684A1 (en) * 1993-11-22 1995-06-01 The Upjohn Company Esters of substituted-hydroxyacetyl piperazine phenyl oxazolidinones
JPH0873455A (ja) * 1994-03-15 1996-03-19 Upjohn Co:The オキサゾリジノン誘導体及びこれを有効成分とする医薬組成物
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds

Also Published As

Publication number Publication date
US5998406A (en) 1999-12-07
TR200001330T2 (tr) 2000-11-21
KR20010031953A (ko) 2001-04-16
SK284577B6 (sk) 2005-07-01
NO20002434D0 (no) 2000-05-11
ES2207010T3 (es) 2004-05-16
DE69818294D1 (de) 2003-10-23
HUP0100470A2 (hu) 2002-05-29
AU1277899A (en) 1999-05-31
SK6182000A3 (en) 2000-12-11
RU2215740C2 (ru) 2003-11-10
CN1271358A (zh) 2000-10-25
NO317291B1 (no) 2004-10-04
ATE250054T1 (de) 2003-10-15
EP1030852B1 (en) 2003-09-17
CA2303959A1 (en) 1999-05-20
DK1030852T3 (da) 2003-12-22
IL136062A0 (en) 2001-05-20
NZ504503A (en) 2002-10-25
WO1999024428A1 (en) 1999-05-20
NO20002434L (no) 2000-05-11
EP1030852A1 (en) 2000-08-30
DE69818294T2 (de) 2004-07-08
BR9813985A (pt) 2000-09-26
PT1030852E (pt) 2004-02-27
JP2001522849A (ja) 2001-11-20
CN1154644C (zh) 2004-06-23
HK1030373A1 (en) 2001-05-04
IL136062A (en) 2004-02-08
AU739055B2 (en) 2001-10-04

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