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FR14C0083I1 - Derives de 5-amino-2,4,7-trioxo-3,4,7,8-tetrahydro-2h-pyrido°2,3-d!pyrimidine et composes apparentes pour le traitement du cancer - Google Patents

Derives de 5-amino-2,4,7-trioxo-3,4,7,8-tetrahydro-2h-pyrido°2,3-d!pyrimidine et composes apparentes pour le traitement du cancer

Info

Publication number
FR14C0083I1
FR14C0083I1 FR14C0083C FR14C0083I1 FR 14C0083 I1 FR14C0083 I1 FR 14C0083I1 FR 14C0083 C FR14C0083 C FR 14C0083C FR 14C0083 I1 FR14C0083 I1 FR 14C0083I1
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Prior art keywords
trioxo
pyrido
tetrahydro
cancer
amino
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English (en)
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Japan Tobacco Inc
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Japan Tobacco Inc
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Publication of FR14C0083I1 publication Critical patent/FR14C0083I1/fr
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Publication of FR14C0083I2 publication Critical patent/FR14C0083I2/fr
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
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    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Addiction (AREA)
  • Molecular Biology (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Biotechnology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Transplantation (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Neurosurgery (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
FR14C0083C 2004-06-11 2014-11-24 Derives de 5-amino-2,4,7-trioxo-3,4,7,8-tetrahydro-2h-pyrido°2,3-d!pyrimidine et composes apparentes pour le traitement du cancer Active FR14C0083I2 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2004174770 2004-06-11
JP2004327111 2004-11-10
PCT/JP2005/011082 WO2005121142A1 (fr) 2004-06-11 2005-06-10 Dérivés de 5-amino-2,4,7-trioxo-3,4,7,8-tétrahydro-2h-pyrido’2,3-d! pyrimidine et composés apparentés pour le traitement du cancer

Publications (2)

Publication Number Publication Date
FR14C0083I1 true FR14C0083I1 (fr) 2015-02-01
FR14C0083I2 FR14C0083I2 (fr) 2015-02-20

Family

ID=34970318

Family Applications (1)

Application Number Title Priority Date Filing Date
FR14C0083C Active FR14C0083I2 (fr) 2004-06-11 2014-11-24 Derives de 5-amino-2,4,7-trioxo-3,4,7,8-tetrahydro-2h-pyrido°2,3-d!pyrimidine et composes apparentes pour le traitement du cancer

Country Status (27)

Country Link
EP (3) EP1761528B1 (fr)
JP (3) JP4163738B2 (fr)
KR (1) KR100883289B1 (fr)
CN (2) CN101912400B (fr)
AT (1) ATE383360T1 (fr)
AU (1) AU2005252110B2 (fr)
BR (1) BRPI0511967B8 (fr)
CA (2) CA2569850C (fr)
CY (3) CY1107253T1 (fr)
DE (1) DE602005004286T2 (fr)
DK (2) DK2298768T3 (fr)
ES (2) ES2297723T3 (fr)
FR (1) FR14C0083I2 (fr)
HR (2) HRP20080018T3 (fr)
IL (1) IL179671A0 (fr)
LU (1) LU92602I2 (fr)
ME (1) ME01480B (fr)
MX (1) MXPA06014478A (fr)
NL (1) NL300701I2 (fr)
NO (2) NO338355B1 (fr)
NZ (1) NZ552090A (fr)
PL (2) PL2298768T3 (fr)
PT (2) PT2298768E (fr)
RS (2) RS50569B (fr)
RU (1) RU2364596C2 (fr)
SI (2) SI1761528T1 (fr)
WO (1) WO2005121142A1 (fr)

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PT1761528E (pt) 2008-04-15
AU2005252110A1 (en) 2005-12-22
CN101006086B (zh) 2010-09-29
JP2008201788A (ja) 2008-09-04
DE602005004286D1 (de) 2008-02-21
SI1761528T1 (sl) 2008-06-30
NL300701I1 (fr) 2015-12-29
CA2727841A1 (fr) 2005-12-22
DE602005004286T2 (de) 2009-01-02
CN101912400A (zh) 2010-12-15
BRPI0511967B1 (pt) 2019-05-07
HK1107084A1 (en) 2008-03-28
EP2298768B9 (fr) 2013-04-24
EP1761528A1 (fr) 2007-03-14
AU2005252110B2 (en) 2008-09-04
CY1113538T1 (el) 2016-06-22
RU2007101158A (ru) 2008-07-20
NL300701I2 (fr) 2015-12-29
NO338355B1 (no) 2016-08-08
ES2297723T3 (es) 2008-05-01
PL1761528T3 (pl) 2008-05-30
ME01480B (fr) 2014-04-20
EP1761528B1 (fr) 2008-01-09
JP2008501631A (ja) 2008-01-24
NO20070155L (no) 2007-02-13
RS52670B (sr) 2013-06-28
PT2298768E (pt) 2012-12-05
CY2014045I1 (el) 2019-07-10
HRP20080018T3 (en) 2008-01-31
CY2014045I2 (el) 2019-07-10
MXPA06014478A (es) 2007-03-21
BRPI0511967B8 (pt) 2021-05-25
NO2016021I2 (no) 2016-11-24
LU92602I2 (fr) 2015-10-27
CN101912400B (zh) 2013-06-26
EP2298768A1 (fr) 2011-03-23
BRPI0511967A (pt) 2008-01-22
JP5421974B2 (ja) 2014-02-19
WO2005121142A1 (fr) 2005-12-22
EP2298768B1 (fr) 2012-11-14
NZ552090A (en) 2009-06-26

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