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FI944602L - Farmaseuttisesti aktiiviset bisyklis-heterosykliset amiinit - Google Patents

Farmaseuttisesti aktiiviset bisyklis-heterosykliset amiinit Download PDF

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Publication number
FI944602L
FI944602L FI944602A FI944602A FI944602L FI 944602 L FI944602 L FI 944602L FI 944602 A FI944602 A FI 944602A FI 944602 A FI944602 A FI 944602A FI 944602 L FI944602 L FI 944602L
Authority
FI
Finland
Prior art keywords
pharmaceutically active
heterocyclic amines
active bicyclic
bicyclic
heterocyclic
Prior art date
Application number
FI944602A
Other languages
English (en)
Swedish (sv)
Other versions
FI944602A0 (fi
FI944602A7 (fi
Inventor
Donald E Ayer
Gordon L Bundy
Eric Jon Jacobsen
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of FI944602A0 publication Critical patent/FI944602A0/fi
Publication of FI944602A7 publication Critical patent/FI944602A7/fi
Publication of FI944602L publication Critical patent/FI944602L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26Acyclic or carbocyclic radicals, substituted by hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Hospice & Palliative Care (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
FI944602A 1992-04-03 1993-03-16 Farmaseuttisesti aktiiviset bisyklis-heterosykliset amiinit FI944602L (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86364692A 1992-04-03 1992-04-03
PCT/US1993/002188 WO1993020078A1 (en) 1992-04-03 1993-03-16 Pharmaceutically active bicyclic-heterocyclic amines

Publications (3)

Publication Number Publication Date
FI944602A0 FI944602A0 (fi) 1994-10-03
FI944602A7 FI944602A7 (fi) 1994-10-03
FI944602L true FI944602L (fi) 1994-10-03

Family

ID=25341481

Family Applications (1)

Application Number Title Priority Date Filing Date
FI944602A FI944602L (fi) 1992-04-03 1993-03-16 Farmaseuttisesti aktiiviset bisyklis-heterosykliset amiinit

Country Status (21)

Country Link
EP (1) EP0633886B1 (fi)
JP (1) JPH08502721A (fi)
KR (1) KR100284473B1 (fi)
AT (1) ATE197051T1 (fi)
AU (1) AU675932B2 (fi)
CA (1) CA2130937A1 (fi)
CZ (1) CZ236494A3 (fi)
DE (1) DE69329574T2 (fi)
DK (1) DK0633886T3 (fi)
ES (1) ES2150941T3 (fi)
FI (1) FI944602L (fi)
GR (1) GR3035188T3 (fi)
HU (1) HUT70954A (fi)
LV (1) LV12794B (fi)
MX (1) MX9301847A (fi)
NO (1) NO303542B1 (fi)
PL (2) PL175347B1 (fi)
PT (1) PT633886E (fi)
RU (1) RU2103272C1 (fi)
SK (1) SK119194A3 (fi)
WO (1) WO1993020078A1 (fi)

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US6680322B2 (en) 1999-12-02 2004-01-20 Osi Pharmaceuticals, Inc. Compounds specific to adenosine A1 receptors and uses thereof
DE60030002T2 (de) 1999-12-02 2007-03-08 Osi Pharmaceuticals, Inc. Für den adenosin-a1-a2a-und-a3-rezeptor spezifische verbindungen und verwendungen davon
US7160890B2 (en) 1999-12-02 2007-01-09 Osi Pharmaceuticals, Inc. Compounds specific to adenosine A3 receptor and uses thereof
US6664252B2 (en) 1999-12-02 2003-12-16 Osi Pharmaceuticals, Inc. 4-aminopyrrolo[2,3-d]pyrimidine compounds specific to adenosine A2a receptor and uses thereof
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US6673802B2 (en) 2000-12-01 2004-01-06 Osi Pharmaceuticals, Inc. Compounds specific to adenosine A3 receptor and uses thereof
US6680324B2 (en) 2000-12-01 2004-01-20 Osi Pharmaceuticals, Inc. Compounds specific to adenosine A1 receptors and uses thereof
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CN101973998A (zh) 2001-12-20 2011-02-16 Osi药物公司 吡咯并嘧啶A2b选择性拮抗剂化合物
CN1620294A (zh) 2001-12-20 2005-05-25 Osi药物公司 嘧啶a2b选择性拮抗剂化合物,它们的合成及用途
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Family Cites Families (3)

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GB864145A (en) * 1959-06-02 1961-03-29 Thomae Gmbh Dr K Novel purines and a process for their manufacture
GB1268772A (en) * 1968-03-15 1972-03-29 Glaxo Lab Ltd NOVEL alpha-CARBOLINE DERIVATIVES, THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME
KR970009225B1 (ko) * 1989-09-19 1997-06-09 데이진 가부시끼가이샤 피롤로[2,3-디] 피리미딘 유도체, 그의 제조방법 및 그것을 유효성분으로 하는 의약제제

Also Published As

Publication number Publication date
DK0633886T3 (da) 2000-12-18
FI944602A0 (fi) 1994-10-03
AU675932B2 (en) 1997-02-27
NO943655D0 (no) 1994-09-30
FI944602A7 (fi) 1994-10-03
HU9402829D0 (en) 1995-02-28
MX9301847A (es) 1993-10-01
PT633886E (pt) 2001-03-30
NO303542B1 (no) 1998-07-27
WO1993020078A1 (en) 1993-10-14
LV12794B (lv) 2002-06-20
PL175327B1 (pl) 1998-12-31
SK119194A3 (en) 1995-05-10
CA2130937A1 (en) 1993-10-14
EP0633886A1 (en) 1995-01-18
CZ236494A3 (en) 1994-12-15
ATE197051T1 (de) 2000-11-15
KR100284473B1 (ko) 2001-04-02
RU94042466A (ru) 1996-07-20
DE69329574T2 (de) 2001-05-31
LV12794A (en) 2002-02-20
NO943655L (no) 1994-12-05
KR950700912A (ko) 1995-02-20
RU2103272C1 (ru) 1998-01-27
GR3035188T3 (en) 2001-04-30
HUT70954A (en) 1995-11-28
JPH08502721A (ja) 1996-03-26
EP0633886B1 (en) 2000-10-18
DE69329574D1 (de) 2000-11-23
PL175347B1 (pl) 1998-12-31
AU3917493A (en) 1993-11-08
ES2150941T3 (es) 2000-12-16

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