EE200300442A - Meetod imidasoolühendite valmistamiseks - Google Patents

Meetod imidasoolühendite valmistamiseks

Info

Publication number: EE200300442A
Authority: EE; Estonia
Prior art keywords: preparation; imidazole compounds; imidazole; compounds
Prior art date: 2001-03-12

Application number

EEP200300442A

Other languages

English (en)

Inventor

Ferdinand Maria Filliers Walter

Laurent Maria Broeckx Rudy

Marcel Herman Leurs Stefan

Original Assignee

Janssen Pharmaceutica N.V.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-03-12

Filing date

2002-03-05

Publication date

2003-12-15

2002-03-05 Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.

2003-12-15 Publication of EE200300442A publication Critical patent/EE200300442A/et

2009-12-15 Publication of EE05247B1 publication Critical patent/EE05247B1/et

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Epoxy Resins (AREA)

EEP200300442A 2001-03-12 2002-03-05 Meetod imidasoolhendite valmistamiseks EE05247B1 (et)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP01200928		2001-03-12
PCT/EP2002/002459 WO2002072574A1 (en)	2001-03-12	2002-03-05	Process for the preparation of imidazole compounds

Publications (2)

Publication Number	Publication Date
EE200300442A true EE200300442A (et)	2003-12-15
EE05247B1 EE05247B1 (et)	2009-12-15

Family

ID=8180004

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200300442A EE05247B1 (et)	2001-03-12	2002-03-05	Meetod imidasoolhendite valmistamiseks

Country Status (31)

Country	Link
US (1)	US6844439B2 (et)
EP (1)	EP1373255B1 (et)
JP (1)	JP4257698B2 (et)
KR (1)	KR100849042B1 (et)
CN (1)	CN1246318C (et)
AR (1)	AR035944A1 (et)
AT (1)	ATE287882T1 (et)
AU (1)	AU2002253101B2 (et)
BR (1)	BRPI0208075B8 (et)
CA (1)	CA2438421C (et)
CZ (1)	CZ300622B6 (et)
DE (1)	DE60202755T2 (et)
DK (1)	DK1373255T3 (et)
EA (1)	EA006770B1 (et)
EE (1)	EE05247B1 (et)
ES (1)	ES2236505T3 (et)
HR (1)	HRP20030695B1 (et)
HU (1)	HU230282B1 (et)
IL (2)	IL157839A0 (et)
MX (1)	MXPA03008205A (et)
MY (1)	MY124838A (et)
NO (1)	NO324954B1 (et)
NZ (1)	NZ528620A (et)
PL (1)	PL208238B1 (et)
PT (1)	PT1373255E (et)
SI (1)	SI1373255T1 (et)
SK (1)	SK287807B6 (et)
TW (1)	TWI249532B (et)
UA (1)	UA74871C2 (et)
WO (1)	WO2002072574A1 (et)
ZA (1)	ZA200307117B (et)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CZ20032691A3 (en)	2001-03-12	2004-04-14	Avanir Pharmaceuticals	Benzimidazole compounds for modulating ige and inhibiting cellular proliferation
TWI276631B (en)	2002-09-12	2007-03-21	Avanir Pharmaceuticals	Phenyl-aza-benzimidazole compounds for modulating IgE and inhibiting cellular proliferation
AU2003270426A1 (en)	2002-09-12	2004-04-30	Avanir Pharmaceuticals	PHENYL-INDOLE COMPOUNDS FOR MODULATING IgE AND INHIBITING CELLULAR PROLIFERATION
JP2007538004A (ja) *	2004-03-18	2007-12-27	ザブライハムアンドウイメンズホスピタル，インコーポレイテッド	シヌクレイノパチーを治療する方法
ES2308486T3 (es) *	2004-05-03	2008-12-01	Janssen Pharmaceutica Nv	Proceso de sintesis diastereoselectiva para la preparacion de compuestos de imidazol.
CN100567291C (zh) *	2004-05-03	2009-12-09	詹森药业有限公司	用6-溴-4-(3-氯苯基)-2-甲氧基喹啉进行的非对映选择性合成方法
EP1758885B1 (en)	2004-05-03	2008-06-18	Janssen Pharmaceutica N.V.	Diastereoselective addition of lithiated n-methylimidazole on sulfinimines
WO2007075923A2 (en)	2005-12-23	2007-07-05	Link Medicine Corporation	Treatment of synucleinopathies
WO2009151683A2 (en) *	2008-03-12	2009-12-17	Link Medicine Corporation	Quinolinone farnesyl transferase inhibitors for the treatment of synucleinopathies and other indications
KR101044430B1 (ko) *	2009-09-25	2011-06-27	듀오백코리아 주식회사	요추받이를 포함하는 의자의 등 지지 장치
KR101107900B1 (ko) *	2009-10-21	2012-01-25	성용기업 주식회사	의자용 허리지지장치
RS62709B1 (sr)	2015-08-17	2022-01-31	Kura Oncology Inc	Postupci za lečenje pacijenata obolelih od kancera pomoću inhibitora farneziltransferaze
PL3534885T3 (pl)	2016-11-03	2021-11-15	Kura Oncology, Inc.	Inhibitory farnezylotransferazy do zastosowania w leczeniu nowotworu
CN110234639A (zh) *	2016-12-08	2019-09-13	杭州领业医药科技有限公司	替吡法尼的晶型及其制备方法及药物组合物
EP3793966A1 (en)	2018-05-18	2021-03-24	Kura Oncology, Inc.	Synthesis of tipifarnib

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW349948B (en)	1995-10-31	1999-01-11	Janssen Pharmaceutica Nv	Farnesyl transferase inhibiting 2-quinolone derivatives
BR9610745A (pt) *	1995-12-08	1999-07-13	Janssen Pharmaceutica Nv	Derivados de (imidazol-5-il) metil-2-quinolinona inibindo a transferase da proteina farnesil
TW591030B (en) *	1997-03-10	2004-06-11	Janssen Pharmaceutica Nv	Farnesyl transferase inhibiting 1,8-annelated quinolinone derivatives substituted with N- or C-linked imidazoles
NZ336233A (en) *	1997-04-25	2001-01-26	Janssen Pharmaceutica Nv	Phenyl substituted quinazolines on 4-position and 2-quinazolinone moiety bearing a carbon or nitrogen-linked imidazolyl moiety
HUP0103228A3 (en) *	1998-08-27	2003-01-28	Pfizer Prod Inc	Alkynyl-substituted quinolin-2-one derivatives useful as anticancer agents and pharmaceutical compositions containing them
WO2000012498A1 (en)	1998-08-27	2000-03-09	Pfizer Products Inc.	Quinolin-2-one derivatives useful as anticancer agents

2002
- 2002-03-05 ES ES02722184T patent/ES2236505T3/es not_active Expired - Lifetime
- 2002-03-05 SI SI200230100T patent/SI1373255T1/xx unknown
- 2002-03-05 NZ NZ528620A patent/NZ528620A/en not_active IP Right Cessation
- 2002-03-05 DE DE60202755T patent/DE60202755T2/de not_active Expired - Lifetime
- 2002-03-05 SK SK1246-2003A patent/SK287807B6/sk unknown
- 2002-03-05 AU AU2002253101A patent/AU2002253101B2/en not_active Expired
- 2002-03-05 MX MXPA03008205A patent/MXPA03008205A/es active IP Right Grant
- 2002-03-05 US US10/471,215 patent/US6844439B2/en not_active Expired - Lifetime
- 2002-03-05 IL IL15783902A patent/IL157839A0/xx unknown
- 2002-03-05 EP EP02722184A patent/EP1373255B1/en not_active Expired - Lifetime
- 2002-03-05 CZ CZ20032704A patent/CZ300622B6/cs not_active IP Right Cessation
- 2002-03-05 KR KR1020037010091A patent/KR100849042B1/ko not_active Expired - Lifetime
- 2002-03-05 HU HU0303443A patent/HU230282B1/hu unknown
- 2002-03-05 CA CA2438421A patent/CA2438421C/en not_active Expired - Lifetime
- 2002-03-05 AT AT02722184T patent/ATE287882T1/de active
- 2002-03-05 PT PT02722184T patent/PT1373255E/pt unknown
- 2002-03-05 JP JP2002571490A patent/JP4257698B2/ja not_active Expired - Lifetime
- 2002-03-05 DK DK02722184T patent/DK1373255T3/da active
- 2002-03-05 HR HR20030695A patent/HRP20030695B1/xx not_active IP Right Cessation
- 2002-03-05 BR BR0208075-3 patent/BRPI0208075B8/pt not_active IP Right Cessation
- 2002-03-05 EE EEP200300442A patent/EE05247B1/et unknown
- 2002-03-05 CN CNB02806335XA patent/CN1246318C/zh not_active Expired - Lifetime
- 2002-03-05 PL PL363263A patent/PL208238B1/pl unknown
- 2002-03-05 EA EA200300998A patent/EA006770B1/ru not_active IP Right Cessation
- 2002-03-05 WO PCT/EP2002/002459 patent/WO2002072574A1/en not_active Ceased
- 2002-03-11 AR ARP020100873A patent/AR035944A1/es active IP Right Grant
- 2002-03-11 TW TW091104444A patent/TWI249532B/zh not_active IP Right Cessation
- 2002-03-11 MY MYPI20020866A patent/MY124838A/en unknown
- 2002-05-03 UA UA2003087776A patent/UA74871C2/uk unknown
2003
- 2003-09-10 IL IL157839A patent/IL157839A/en unknown
- 2003-09-10 NO NO20034003A patent/NO324954B1/no not_active IP Right Cessation
- 2003-09-11 ZA ZA200307117A patent/ZA200307117B/en unknown

Also Published As

Publication number	Publication date
IL157839A0 (en)	2004-03-28
IL157839A (en)	2008-07-08
CN1496363A (zh)	2004-05-12
CZ300622B6 (cs)	2009-07-01
SK287807B6 (sk)	2011-10-04
KR100849042B1 (ko)	2008-07-29
DK1373255T3 (da)	2005-05-23
ES2236505T3 (es)	2005-07-16
BRPI0208075B8 (pt)	2021-05-25
NO20034003D0 (no)	2003-09-10
UA74871C2 (en)	2006-02-15
NO324954B1 (no)	2008-01-14
EA006770B1 (ru)	2006-04-28
HU230282B1 (hu)	2015-12-28
DE60202755D1 (de)	2005-03-03
HRP20030695A2 (en)	2005-02-28
HUP0303443A3 (en)	2012-09-28
SK12462003A3 (sk)	2004-06-08
TWI249532B (en)	2006-02-21
AR035944A1 (es)	2004-07-28
HK1063315A1 (zh)	2004-12-24
MXPA03008205A (es)	2004-01-29
EA200300998A1 (ru)	2004-02-26
US20040138256A1 (en)	2004-07-15
CN1246318C (zh)	2006-03-22
WO2002072574A1 (en)	2002-09-19
MY124838A (en)	2006-07-31
CZ20032704A3 (en)	2004-03-17
NO20034003L (no)	2003-10-22
JP4257698B2 (ja)	2009-04-22
KR20030079971A (ko)	2003-10-10
EP1373255B1 (en)	2005-01-26
HRP20030695B1 (hr)	2011-07-31
EP1373255A1 (en)	2004-01-02
ZA200307117B (en)	2004-09-13
PT1373255E (pt)	2005-05-31
HUP0303443A2 (hu)	2004-01-28
JP2004523575A (ja)	2004-08-05
NZ528620A (en)	2005-01-28
CA2438421C (en)	2010-05-18
EE05247B1 (et)	2009-12-15
US6844439B2 (en)	2005-01-18
PL208238B1 (pl)	2011-04-29
PL363263A1 (en)	2004-11-15
ATE287882T1 (de)	2005-02-15
BRPI0208075B1 (pt)	2018-02-14
SI1373255T1 (et)	2005-08-31
CA2438421A1 (en)	2002-09-19
BR0208075A (pt)	2004-03-02
DE60202755T2 (de)	2006-03-30
AU2002253101B2 (en)	2007-08-09

Publication	Publication Date	Title
NO20042680L (no)	2004-06-25	Fremgangsmater for fremstilling av O-demetylvenflaxine
NO20030012L (no)	2003-03-03	Fremgangsmåte for fremstilling av substituerte oktanoylamider
NO20040027L (no)	2004-01-05	Fremgangsmate for fremstillingen av escitalopram
FI20011541A0 (fi)	2001-07-13	Menetelmä massan valmistamiseksi
EE200300442A (et)	2003-12-15	Meetod imidasoolühendite valmistamiseks
NO20033433L (no)	2003-09-25	Fremgangsmåte for fremstilling av 2-(2-pyridylmetyl)sulfinyl- 1H-benzimidasol
NO20044814L (no)	2004-01-07	Fremgangsmate for fremstilling av combretastaniner
NO20035538D0 (no)	2003-12-11	Fremgangsmåte for fremstilling av zaleplon
NO20030515L (no)	2003-03-31	Fremgangsmåte for fremstilling av dinapsolin
FR2826002B1 (fr)	2004-12-03	Procede de preparation de composes bromodifluoroacetiques
NO20035586L (no)	2003-12-15	Fremgangsmate for fremstilling av cykloheksanol-derivater
NO20035136D0 (no)	2003-11-18	Fremgangsmåte til fremstilling av imipenem
NO20033147D0 (no)	2003-07-09	Fremgangsmate for fremstilling av rent ondansetronhydrogenkloriddihydrat
NO20024887L (no)	2002-10-10	FremgangsmÕte for fremstilling av benzokondenserte heterosykliske forbindelser
NO20023702D0 (no)	2002-08-06	Fremgangsmåte for fremstilling av 5-arylnikotinaldehyder
NO20035138D0 (no)	2003-11-18	Fremgangsmåte til fremstilling av amorft natriumsilastatin
NO20052396D0 (no)	2005-05-13	Fremgangsmate for fremstilling av spirolactonforbindelser
DK1565445T3 (da)	2007-01-29	Fremgangsmåde til fremstilling af imidazolylforbindelser
NO20013802D0 (no)	2001-08-02	Fremgangsmåte for fremstilling av kitosaner
NO20040149L (no)	2004-01-13	Fremgangsmåte for fremstilling av tagatose
ITMI20010771A0 (it)	2001-04-11	Processo per la preparazione di composti piridil-aril-solfonici
ITMI20010772A0 (it)	2001-04-11	Processo per la preparazione di composti aril-piridinici
FR2829492B1 (fr)	2005-01-28	Procede de preparation de la disorbitylamine
DK1274684T3 (da)	2005-09-26	Fremgangsmåde til fremstilling af aryl-pyridinylforbindelser
DK1280792T3 (da)	2004-11-15	Fremgangsmåde til fremstilling af benzo-annelerede heterocykler

Legal Events

Date	Code	Title	Description
2011-02-15	KB4A	Valid patent at the end of a year	Effective date: 20101231