EE200300126A - Kinoliini ja kinolinooni derivaadid glutamaatretseptori antagonistidena, nende saamine ja kasutamine ravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioon - Google Patents
Kinoliini ja kinolinooni derivaadid glutamaatretseptori antagonistidena, nende saamine ja kasutamine ravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioonInfo
- Publication number
- EE200300126A EE200300126A EEP200300126A EEP200300126A EE200300126A EE 200300126 A EE200300126 A EE 200300126A EE P200300126 A EEP200300126 A EE P200300126A EE P200300126 A EEP200300126 A EE P200300126A EE 200300126 A EE200300126 A EE 200300126A
- Authority
- EE
- Estonia
- Prior art keywords
- preparation
- quinoline
- pharmaceuticals
- pharmaceutical composition
- composition containing
- Prior art date
Links
- SMWDFEZZVXVKRB-UHFFFAOYSA-N Quinoline Chemical compound N1=CC=CC2=CC=CC=C21 SMWDFEZZVXVKRB-UHFFFAOYSA-N 0.000 title 2
- 239000003814 drug Substances 0.000 title 1
- 239000003825 glutamate receptor antagonist Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- LISFMEBWQUVKPJ-UHFFFAOYSA-N quinolin-2-ol Chemical class C1=CC=C2NC(=O)C=CC2=C1 LISFMEBWQUVKPJ-UHFFFAOYSA-N 0.000 title 1
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- C07D215/04—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to the ring carbon atoms
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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- C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
- C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00203419 | 2000-10-02 | ||
| PCT/EP2001/011135 WO2002028837A1 (en) | 2000-10-02 | 2001-09-25 | Metabotropic glutamate receptor antagonists |
Publications (2)
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| EE200300126A true EE200300126A (et) | 2005-04-15 |
| EE05195B1 EE05195B1 (et) | 2009-08-17 |
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| EEP200300126A EE05195B1 (et) | 2000-10-02 | 2001-09-25 | Kinoliini ja kinolinooni derivaadid glutamaatretseptori antagonistidena, nende saamine ja kasutamine ravimite valmistamiseks ning neid sisaldav farmatseutiline kompositsioon |
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| EP (1) | EP1332133B1 (et) |
| JP (1) | JP2004510764A (et) |
| KR (1) | KR100818965B1 (et) |
| CN (1) | CN1703403A (et) |
| AR (1) | AR035065A1 (et) |
| AT (1) | ATE400558T1 (et) |
| AU (2) | AU9384701A (et) |
| BG (1) | BG107672A (et) |
| BR (1) | BR0114253A (et) |
| CA (1) | CA2421782A1 (et) |
| CZ (1) | CZ20031145A3 (et) |
| DE (1) | DE60134762D1 (et) |
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| HR (1) | HRP20030229A2 (et) |
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| US5475007A (en) * | 1993-05-28 | 1995-12-12 | The Regents Of The University Of California | 1,2,3,4-tetrahydroquinoline-2,3,4-trione-3 or 4-oximes and the use thereof |
| JPH0733743A (ja) * | 1993-07-22 | 1995-02-03 | Kyorin Pharmaceut Co Ltd | 2−アリール−4−キノリノール誘導体 |
| JPH08295690A (ja) * | 1995-04-26 | 1996-11-12 | Tokuyama Corp | クロメン化合物 |
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| EP1000015A1 (en) * | 1997-07-18 | 2000-05-17 | Georgetown University | Bicyclic metabotropic glutamate receptor ligands |
| NZ505207A (en) * | 1997-11-21 | 2003-10-31 | Nps Pharma Inc | Metabotropic glutamate receptor antagonists for treating central nervous system diseases |
| WO2000012498A1 (en) * | 1998-08-27 | 2000-03-09 | Pfizer Products Inc. | Quinolin-2-one derivatives useful as anticancer agents |
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| DE19859750A1 (de) | 1998-12-23 | 2000-06-29 | Henkel Kgaa | Mittel zum Färben von keratinhaltigen Fasern |
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| CN1340051A (zh) * | 1999-02-11 | 2002-03-13 | 辉瑞产品公司 | 可用作抗癌剂的杂芳基取代的喹啉-2-酮衍生物 |
| AU2001236100A1 (en) * | 2000-03-07 | 2001-09-17 | Takeda Chemical Industries Ltd. | Vasoactive agents |
| EP1332133B1 (en) * | 2000-10-02 | 2008-07-09 | Janssen Pharmaceutica N.V. | Metabotropic glutamate receptor antagonists |
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2001
- 2001-09-25 EP EP01974298A patent/EP1332133B1/en not_active Expired - Lifetime
- 2001-09-25 HR HR20030229A patent/HRP20030229A2/hr not_active Application Discontinuation
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- 2001-09-25 EA EA200300428A patent/EA007464B1/ru not_active IP Right Cessation
- 2001-09-25 KR KR1020037002014A patent/KR100818965B1/ko not_active Expired - Fee Related
- 2001-09-25 IL IL15516301A patent/IL155163A0/xx unknown
- 2001-09-25 WO PCT/EP2001/011135 patent/WO2002028837A1/en not_active Ceased
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- 2001-09-25 UA UA2003032796A patent/UA76726C2/uk unknown
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- 2001-09-25 AU AU9384701A patent/AU9384701A/xx active Pending
- 2001-09-25 CN CNA018167179A patent/CN1703403A/zh active Pending
- 2001-09-25 EE EEP200300126A patent/EE05195B1/et not_active IP Right Cessation
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- 2001-09-25 CA CA002421782A patent/CA2421782A1/en not_active Abandoned
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- 2001-09-25 AU AU2001293847A patent/AU2001293847B2/en not_active Ceased
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- 2001-09-25 JP JP2002532423A patent/JP2004510764A/ja active Pending
- 2001-09-25 DE DE60134762T patent/DE60134762D1/de not_active Expired - Lifetime
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- 2001-09-27 MY MYPI20014515A patent/MY147730A/en unknown
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Effective date: 20100925 |