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EE200100639A - Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod - Google Patents

Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod

Info

Publication number
EE200100639A
EE200100639A EEP200100639A EEP200100639A EE200100639A EE 200100639 A EE200100639 A EE 200100639A EE P200100639 A EEP200100639 A EE P200100639A EE P200100639 A EEP200100639 A EE P200100639A EE 200100639 A EE200100639 A EE 200100639A
Authority
EE
Estonia
Prior art keywords
preparation
benzofuran
aminoalkyl
pharmaceutical composition
benzopyran derivatives
Prior art date
Application number
EEP200100639A
Other languages
English (en)
Inventor
Van Emelen Kristof
Frans Leopold De Bruyn Marcel
Original Assignee
Janssen Pharmaceutica N.V.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica N.V. filed Critical Janssen Pharmaceutica N.V.
Publication of EE200100639A publication Critical patent/EE200100639A/et
Publication of EE04780B1 publication Critical patent/EE04780B1/et

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nutrition Science (AREA)
  • Child & Adolescent Psychology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyrane Compounds (AREA)
EEP200100639A 1999-06-02 2000-05-23 Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod EE04780B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99201747 1999-06-02
PCT/EP2000/004746 WO2000075136A1 (en) 1999-06-02 2000-05-23 Aminoalkyl substituted (benzodioxan, benzofuran or benzopyran) derivatives

Publications (2)

Publication Number Publication Date
EE200100639A true EE200100639A (et) 2003-02-17
EE04780B1 EE04780B1 (et) 2007-02-15

Family

ID=8240260

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100639A EE04780B1 (et) 1999-06-02 2000-05-23 Aminoalküül-asendatud bensodioksaani, bensofuraani või bensopüraani derivaadid, nende valmistamismeetod, farmatseutiline kompositsioon ja selle valmistamismeetod

Country Status (33)

Country Link
US (2) US6864273B1 (et)
EP (1) EP1187829B1 (et)
JP (1) JP2003501427A (et)
KR (1) KR100699512B1 (et)
CN (1) CN1150191C (et)
AR (1) AR033334A1 (et)
AT (1) ATE256125T1 (et)
AU (1) AU773773B2 (et)
BG (1) BG65269B1 (et)
BR (1) BR0011237A (et)
CA (1) CA2374902C (et)
CZ (1) CZ20014177A3 (et)
DE (1) DE60007124T2 (et)
DK (1) DK1187829T3 (et)
EA (1) EA004645B1 (et)
EE (1) EE04780B1 (et)
ES (1) ES2212774T3 (et)
HR (1) HRP20010868A2 (et)
HU (1) HUP0201404A3 (et)
IL (2) IL146840A0 (et)
MX (1) MXPA01012330A (et)
MY (1) MY120618A (et)
NO (1) NO319953B1 (et)
NZ (1) NZ514993A (et)
PL (1) PL198552B1 (et)
PT (1) PT1187829E (et)
SI (1) SI1187829T1 (et)
SK (1) SK285619B6 (et)
TR (1) TR200103430T2 (et)
TW (1) TWI289559B (et)
UA (1) UA73122C2 (et)
WO (1) WO2000075136A1 (et)
ZA (1) ZA200109860B (et)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA004648B1 (ru) 1999-06-02 2004-06-24 Янссен Фармацевтика Н.В. Пирролидинил-, пиперидинил- или гомопиперидинилзамещенные производные, способ их получения, их применение в медицине, содержащая их фармацевтическая композиция и способ ее получения
JO2352B1 (en) 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for the treatment of non-adaptation of the bottom of the uterus
JO2654B1 (en) 2000-09-04 2012-06-17 شركة جانسين فارماسوتيكا ان. في Multiple aryl caroxa amides are useful as lipid - lowering agents
JO2409B1 (en) 2000-11-21 2007-06-17 شركة جانسين فارماسوتيكا ان. في Second-phenyl carboxy amides are useful as lipid-lowering agents
ATE522214T1 (de) * 2002-04-08 2011-09-15 Zeria Pharm Co Ltd Therapeutisches mittel für nahrungskompetenzstörungen im magen
JP2008530229A (ja) 2005-02-17 2008-08-07 ワイス シクロアルキル縮合インドール、ベンゾチオフェン、ベンゾフランおよびインデン誘導体
CN103917529B (zh) 2011-11-11 2016-08-17 辉瑞大药厂 2-硫代嘧啶酮类
MA42035A (fr) 2015-05-05 2018-03-14 Pfizer 2-thiopyrimidinones

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3910930A (en) 1973-01-04 1975-10-07 Janssen Pharmaceutica Nv 1-{55 1-{8 2-(1,4-Benzodioxan-2-yl)-2-hydroxyethyl{9 -4-piperidyl{56 -2-benzimidazolinones
US3929801A (en) 1973-11-20 1975-12-30 Janssen Pharmaceutica Nv 2-Benzimidazolinones
GR71865B (et) 1978-03-20 1983-07-07 Ciba Geigy
DE2852945A1 (de) 1978-12-07 1980-06-26 Boehringer Sohn Ingelheim Benzodioxanyl-hydroxyaethylpiperidyl- imidazolidinone, verfahren zu ihrer herstellung und diese enthaltende arzneimittel
US4329348A (en) 1979-02-26 1982-05-11 Ciba-Geigy Corporation N-Oxacyclic-alkylpiperidines as psychostimulants
DE3124366A1 (de) 1981-06-20 1982-12-30 Hoechst Ag, 6000 Frankfurt N-oxacyclyl-alkylpiperidin-derivate, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und deren verwendung
FR2533584B1 (fr) 1982-09-28 1986-03-21 Pasteur Institut Procede de detection du pouvoir mutagene de substances, susceptibles d'induire la deterioration d'adn cellulaires, mettant en jeu la production d'une reponse sos
DE3901814A1 (de) 1988-07-28 1990-02-01 Bayer Ag Substituierte aminomethylzetraline sowie ihre heterocyclischen analoga
DE4140540A1 (de) 1991-12-09 1993-06-17 Bayer Ag Neue azaheterocyclylmethyl-chromane
SI9300097B (en) 1992-02-27 2001-12-31 Janssen Pharmaceutica Nv (benzodioxan, benzofuran or benzopyran) alkylamino) alkyl substituted guanidines
DE4319038A1 (de) * 1993-06-08 1994-12-15 Bayer Ag Verwendung von teilweise bekannten substituierten Chromanen als Arzneimittel, neue Wirkstoffe und Verfahren zu ihrer Herstellung
PL181385B1 (pl) 1993-08-19 2001-07-31 Janssen Pharmaceutica Nv Nowe pochodne dihydrobenzopiranu o wlasciwosciach naczyniozwezajacych, kompozycja farmaceutyczna i sposób wytwarzania pochodnych dihydrobenzopiranu PL PL PL PL PL PL
US5541199A (en) 1995-06-02 1996-07-30 American Home Products Corporation Chroman-2-ylmethylamino derivatives
FR2744451B1 (fr) 1996-02-01 1998-04-24 Pf Medicament Nouvelles imidazolidinones, pyrimidinones, et 1,3-diazepin-2 -ones, leur preparation et leurs applications en therapeutique
US6133277A (en) 1997-12-05 2000-10-17 Janssen Pharmaceutica N.V. (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
EA004648B1 (ru) * 1999-06-02 2004-06-24 Янссен Фармацевтика Н.В. Пирролидинил-, пиперидинил- или гомопиперидинилзамещенные производные, способ их получения, их применение в медицине, содержащая их фармацевтическая композиция и способ ее получения
JO2352B1 (en) 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Compounds for the treatment of non-adaptation of the bottom of the uterus

Also Published As

Publication number Publication date
MY120618A (en) 2005-11-30
AU773773B2 (en) 2004-06-03
BR0011237A (pt) 2002-03-05
SK285619B6 (sk) 2007-05-03
CA2374902A1 (en) 2000-12-14
ES2212774T3 (es) 2004-08-01
AU5525600A (en) 2000-12-28
WO2000075136A1 (en) 2000-12-14
HRP20010868A2 (en) 2003-04-30
EP1187829A1 (en) 2002-03-20
DE60007124D1 (de) 2004-01-22
EA200101236A1 (ru) 2002-08-29
SI1187829T1 (en) 2004-04-30
TWI289559B (en) 2007-11-11
DK1187829T3 (da) 2004-04-13
US6864273B1 (en) 2005-03-08
EE04780B1 (et) 2007-02-15
US20050096378A1 (en) 2005-05-05
SK17032001A3 (sk) 2002-07-02
PL198552B1 (pl) 2008-06-30
BG106156A (en) 2002-05-31
IL146840A0 (en) 2002-07-25
DE60007124T2 (de) 2004-09-23
UA73122C2 (en) 2005-06-15
BG65269B1 (bg) 2007-11-30
KR20010110806A (ko) 2001-12-13
AR033334A1 (es) 2003-12-17
NO319953B1 (no) 2005-10-03
IL146840A (en) 2006-12-10
ATE256125T1 (de) 2003-12-15
NO20015903D0 (no) 2001-12-03
KR100699512B1 (ko) 2007-03-26
CN1150191C (zh) 2004-05-19
US7273862B2 (en) 2007-09-25
EP1187829B1 (en) 2003-12-10
JP2003501427A (ja) 2003-01-14
PL352112A1 (en) 2003-07-28
PT1187829E (pt) 2004-04-30
CA2374902C (en) 2009-09-15
MXPA01012330A (es) 2002-07-30
CN1353707A (zh) 2002-06-12
EA004645B1 (ru) 2004-06-24
CZ20014177A3 (cs) 2002-05-15
HUP0201404A3 (en) 2005-02-28
HUP0201404A2 (en) 2002-08-28
NO20015903L (no) 2001-12-03
TR200103430T2 (tr) 2002-06-21
NZ514993A (en) 2003-05-30
ZA200109860B (en) 2003-05-28

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Legal Events

Date Code Title Description
KB4A Valid patent at the end of a year

Effective date: 20071231

KB4A Valid patent at the end of a year

Effective date: 20081231

MM4A Lapsed by not paying the annual fees

Effective date: 20100523