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EA200801128A1 - Пери-конденсированные трициклические соединения, полезные в качестве антибактериальных средств - Google Patents

Пери-конденсированные трициклические соединения, полезные в качестве антибактериальных средств

Info

Publication number
EA200801128A1
EA200801128A1 EA200801128A EA200801128A EA200801128A1 EA 200801128 A1 EA200801128 A1 EA 200801128A1 EA 200801128 A EA200801128 A EA 200801128A EA 200801128 A EA200801128 A EA 200801128A EA 200801128 A1 EA200801128 A1 EA 200801128A1
Authority
EA
Eurasian Patent Office
Prior art keywords
peri
compounds useful
tricyclic compounds
condensed tricyclic
antibacterial means
Prior art date
Application number
EA200801128A
Other languages
English (en)
Inventor
Натали Кайо
Дэвид Томас Дэвис
Джоэль Майкл Эскен
Алан Джозеф Хеннесси
Сукумар Сентхил Кумар Кусалакумари
Роджер Эдвард Марквелл
Тимоти Джеймс Майлз
Нэйл Дэвид Пирсон
Original Assignee
Глэксо Груп Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Глэксо Груп Лимитед filed Critical Глэксо Груп Лимитед
Publication of EA200801128A1 publication Critical patent/EA200801128A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Трициклические азотсодержащие соединения формулы (I) или их фармацевтически приемлемые соли и/или сольваты
EA200801128A 2005-10-21 2006-10-17 Пери-конденсированные трициклические соединения, полезные в качестве антибактериальных средств EA200801128A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US72897505P 2005-10-21 2005-10-21
US82659006P 2006-09-22 2006-09-22
PCT/US2006/060023 WO2007081597A2 (en) 2005-10-21 2006-10-17 Peri condensed tricyclic compounds useful as antibacterial agents

Publications (1)

Publication Number Publication Date
EA200801128A1 true EA200801128A1 (ru) 2008-10-30

Family

ID=38256822

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200801128A EA200801128A1 (ru) 2005-10-21 2006-10-17 Пери-конденсированные трициклические соединения, полезные в качестве антибактериальных средств

Country Status (26)

Country Link
US (2) US20080280892A1 (ru)
EP (1) EP1954697B1 (ru)
JP (1) JP2009512695A (ru)
KR (1) KR20080064173A (ru)
AR (1) AR057981A1 (ru)
AT (1) ATE458737T1 (ru)
AU (1) AU2006335042A1 (ru)
BR (1) BRPI0617467A2 (ru)
CA (1) CA2626641A1 (ru)
CR (1) CR9930A (ru)
CY (1) CY1110137T1 (ru)
DE (1) DE602006012535D1 (ru)
DK (1) DK1954697T3 (ru)
EA (1) EA200801128A1 (ru)
ES (1) ES2340531T3 (ru)
HR (1) HRP20100194T8 (ru)
IL (1) IL190803A0 (ru)
MA (1) MA29873B1 (ru)
NO (1) NO20082191L (ru)
NZ (1) NZ567315A (ru)
PE (1) PE20070793A1 (ru)
PL (1) PL1954697T3 (ru)
PT (1) PT1954697E (ru)
SI (1) SI1954697T1 (ru)
TW (1) TW200736263A (ru)
WO (1) WO2007081597A2 (ru)

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Also Published As

Publication number Publication date
BRPI0617467A2 (pt) 2011-07-26
CR9930A (es) 2008-07-29
HRP20100194T8 (hr) 2010-06-30
WO2007081597A3 (en) 2008-06-12
NO20082191L (no) 2008-07-16
ES2340531T3 (es) 2010-06-04
DK1954697T3 (da) 2010-06-14
PT1954697E (pt) 2010-05-17
IL190803A0 (en) 2008-12-29
EP1954697A2 (en) 2008-08-13
AU2006335042A1 (en) 2007-07-19
MA29873B1 (fr) 2008-10-03
TW200736263A (en) 2007-10-01
JP2009512695A (ja) 2009-03-26
SI1954697T1 (sl) 2010-05-31
US20080280892A1 (en) 2008-11-13
HRP20100194T1 (hr) 2010-05-31
NZ567315A (en) 2011-01-28
HK1118546A1 (en) 2009-02-13
US20080221110A1 (en) 2008-09-11
AR057981A1 (es) 2008-01-09
WO2007081597A2 (en) 2007-07-19
PL1954697T3 (pl) 2010-07-30
DE602006012535D1 (de) 2010-04-08
KR20080064173A (ko) 2008-07-08
ATE458737T1 (de) 2010-03-15
PE20070793A1 (es) 2007-08-23
CY1110137T1 (el) 2015-01-14
EP1954697B1 (en) 2010-02-24
CA2626641A1 (en) 2007-07-19

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