DK0874834T3 - Fremgangsmåder og mellemprodukter til fremstilling af 3-(1-piperazinyl)-1,2-benzisothiazol - Google Patents

Fremgangsmåder og mellemprodukter til fremstilling af 3-(1-piperazinyl)-1,2-benzisothiazol

Info

Publication number: DK0874834T3
Authority: DK; Denmark
Prior art keywords: benzisothiazole; piperazinyl; intermediates; preparation; methods
Prior art date: 1995-11-07

Application number

DK96931940T

Other languages

English (en)

Inventor

Darrell E Fox

John F Lambert

Terry G Sinay Jr

Stanley W Walinsky

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-11-07

Filing date

1996-10-11

Publication date

2001-02-19

1996-10-11 Application filed by Pfizer filed Critical Pfizer

2001-02-19 Application granted granted Critical

2001-02-19 Publication of DK0874834T3 publication Critical patent/DK0874834T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
- C07D295/26—Sulfur atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)

DK96931940T 1995-11-07 1996-10-11 Fremgangsmåder og mellemprodukter til fremstilling af 3-(1-piperazinyl)-1,2-benzisothiazol DK0874834T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US630195P	1995-11-07	1995-11-07
PCT/IB1996/001079 WO1997017336A1 (en)	1995-11-07	1996-10-11	Processes and intermediates for preparing 3-(1-piperazinyl)-1,2-benzisothiazole

Publications (1)

Publication Number	Publication Date
DK0874834T3 true DK0874834T3 (da)	2001-02-19

Family

ID=21720240

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK96931940T DK0874834T3 (da)	1995-11-07	1996-10-11	Fremgangsmåder og mellemprodukter til fremstilling af 3-(1-piperazinyl)-1,2-benzisothiazol

Country Status (29)

Country	Link
US (1)	US6111105A (da)
EP (1)	EP0874834B1 (da)
JP (1)	JP3152938B2 (da)
KR (1)	KR100315939B1 (da)
CN (1)	CN1071324C (da)
AR (2)	AR004279A1 (da)
AT (1)	ATE198071T1 (da)
AU (1)	AU698443B2 (da)
BR (1)	BR9611366A (da)
CA (1)	CA2236940C (da)
CO (1)	CO4480028A1 (da)
CZ (1)	CZ290600B6 (da)
DE (1)	DE69611253T2 (da)
DK (1)	DK0874834T3 (da)
ES (1)	ES2152564T3 (da)
GR (1)	GR3035215T3 (da)
HU (1)	HU225921B1 (da)
MX (1)	MX9803599A (da)
MY (1)	MY116579A (da)
NO (1)	NO309811B1 (da)
NZ (1)	NZ318844A (da)
PE (1)	PE17298A1 (da)
PL (1)	PL185048B1 (da)
PT (1)	PT874834E (da)
RU (1)	RU2147302C1 (da)
TR (1)	TR199800814T2 (da)
TW (1)	TW358807B (da)
WO (1)	WO1997017336A1 (da)
ZA (1)	ZA969315B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US20040048876A1 (en) *	2002-02-20	2004-03-11	Pfizer Inc.	Ziprasidone composition and synthetic controls
UY27668A1 (es)	2002-02-20	2003-10-31	Pfizer Prod Inc	Composición de ziprasidona y controles sintéticos
CA2543805A1 (en)	2003-10-24	2005-05-06	Gideon Pilarsky	Processes for preparation of ziprasidone
US7777037B2 (en) *	2004-10-27	2010-08-17	Dr. Reddy's Laboratories Limited	Ziprasidone process
CN105891392A (zh) *	2016-03-29	2016-08-24	北京万全德众医药生物技术有限公司	一种用液相色谱法分离测定盐酸鲁拉西酮中间体有关物质的方法
CN107064323A (zh) *	2016-12-05	2017-08-18	北京万全德众医药生物技术有限公司	一种用液相色谱法分离测定盐酸鲁拉西酮及其有关物质的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4590196A (en) *	1984-08-23	1986-05-20	Bristol-Myers Company	Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives
NZ230045A (en) *	1988-08-05	1990-11-27	Janssen Pharmaceutica Nv	3-piperazinylbenzazole derivatives and pharmaceutical compositions
JPH06220030A (ja) *	1993-01-22	1994-08-09	Sumitomo Pharmaceut Co Ltd	３−アミノ−１，２−ベンズイソチアゾール誘導体の製造法
JP3701044B2 (ja) *	1995-04-24	2005-09-28	住友精化株式会社	シアノベンゼンスルフェニルハライドおよびそれを用いる３−置換ベンゾイソチアゾールの製造方法
JP3996228B2 (ja) *	1996-10-11	2007-10-24	住友精化株式会社	３−ピペラジニルベンズイソチアゾール類の製造法

1996
- 1996-10-11 EP EP96931940A patent/EP0874834B1/en not_active Expired - Lifetime
- 1996-10-11 CA CA002236940A patent/CA2236940C/en not_active Expired - Fee Related
- 1996-10-11 RU RU98110457A patent/RU2147302C1/ru not_active IP Right Cessation
- 1996-10-11 AT AT96931940T patent/ATE198071T1/de not_active IP Right Cessation
- 1996-10-11 CN CN96198127A patent/CN1071324C/zh not_active Expired - Fee Related
- 1996-10-11 AU AU70926/96A patent/AU698443B2/en not_active Ceased
- 1996-10-11 TR TR1998/00814T patent/TR199800814T2/xx unknown
- 1996-10-11 JP JP51800597A patent/JP3152938B2/ja not_active Expired - Fee Related
- 1996-10-11 DK DK96931940T patent/DK0874834T3/da active
- 1996-10-11 PL PL96326630A patent/PL185048B1/pl not_active IP Right Cessation
- 1996-10-11 ES ES96931940T patent/ES2152564T3/es not_active Expired - Lifetime
- 1996-10-11 CZ CZ19981378A patent/CZ290600B6/cs not_active IP Right Cessation
- 1996-10-11 US US09/068,285 patent/US6111105A/en not_active Expired - Fee Related
- 1996-10-11 KR KR1019980703391A patent/KR100315939B1/ko not_active Expired - Fee Related
- 1996-10-11 PT PT96931940T patent/PT874834E/pt unknown
- 1996-10-11 BR BR9611366A patent/BR9611366A/pt not_active IP Right Cessation
- 1996-10-11 WO PCT/IB1996/001079 patent/WO1997017336A1/en not_active Ceased
- 1996-10-11 NZ NZ318844A patent/NZ318844A/en unknown
- 1996-10-11 HU HU9903765A patent/HU225921B1/hu not_active IP Right Cessation
- 1996-10-11 DE DE69611253T patent/DE69611253T2/de not_active Expired - Fee Related
- 1996-10-15 TW TW085112576A patent/TW358807B/zh not_active IP Right Cessation
- 1996-11-04 AR ARP960105036A patent/AR004279A1/es unknown
- 1996-11-04 PE PE1996000766A patent/PE17298A1/es not_active Application Discontinuation
- 1996-11-06 ZA ZA9609315A patent/ZA969315B/xx unknown
- 1996-11-06 MY MYPI96004629A patent/MY116579A/en unknown
- 1996-11-07 CO CO96058758A patent/CO4480028A1/es unknown
1998
- 1998-05-06 MX MX9803599A patent/MX9803599A/es not_active IP Right Cessation
- 1998-05-06 NO NO982051A patent/NO309811B1/no not_active IP Right Cessation
2001
- 2001-01-11 GR GR20010400030T patent/GR3035215T3/el not_active IP Right Cessation
- 2001-10-29 AR ARP010105060A patent/AR032373A2/es active IP Right Grant

Also Published As

Publication number	Publication date
HUP9903765A3 (en)	2001-12-28
CZ137898A3 (cs)	1999-03-17
HUP9903765A2 (hu)	2000-03-28
PT874834E (pt)	2001-04-30
MY116579A (en)	2004-02-28
DE69611253T2 (de)	2001-04-05
ES2152564T3 (es)	2001-02-01
US6111105A (en)	2000-08-29
PL326630A1 (en)	1998-10-12
KR100315939B1 (ko)	2002-01-16
KR19990067381A (ko)	1999-08-16
NZ318844A (en)	1999-04-29
NO982051L (no)	1998-07-03
CN1071324C (zh)	2001-09-19
AR004279A1 (es)	1998-11-04
PE17298A1 (es)	1998-04-16
CZ290600B6 (cs)	2002-08-14
ZA969315B (en)	1998-05-06
JP3152938B2 (ja)	2001-04-03
ATE198071T1 (de)	2000-12-15
CA2236940C (en)	2001-08-21
CN1201457A (zh)	1998-12-09
MX9803599A (es)	1998-09-30
CO4480028A1 (es)	1997-07-09
RU2147302C1 (ru)	2000-04-10
NO982051D0 (no)	1998-05-06
HU225921B1 (en)	2008-01-28
BR9611366A (pt)	1999-02-23
CA2236940A1 (en)	1997-05-15
TW358807B (en)	1999-05-21
EP0874834B1 (en)	2000-12-13
EP0874834A1 (en)	1998-11-04
TR199800814T2 (xx)	1998-07-21
DE69611253D1 (de)	2001-01-18
AU7092696A (en)	1997-05-29
AU698443B2 (en)	1998-10-29
NO309811B1 (no)	2001-04-02
JPH10512595A (ja)	1998-12-02
PL185048B1 (pl)	2003-02-28
WO1997017336A1 (en)	1997-05-15
GR3035215T3 (en)	2001-04-30
AR032373A2 (es)	2003-11-05

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