NO982051L - FremgangsmÕter og mellomprodukter for fremstilling av 3-(1-piperazinyl)-1,2-benzisotiazol - Google Patents

FremgangsmÕter og mellomprodukter for fremstilling av 3-(1-piperazinyl)-1,2-benzisotiazol

Info

Publication number: NO982051L
Authority: NO; Norway
Prior art keywords: benzisothiazole; piperazinyl; intermediates; preparation; methods
Prior art date: 1995-11-07

Application number

NO982051A

Other languages

English (en)

Other versions

NO309811B1 (no

NO982051D0 (no

Inventor

Darrell E Fox

John F Lambert

Jr Terry G Sinay

Stanley W Walinsky

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-11-07

Filing date

1998-05-06

Publication date

1998-07-03

1998-05-06 Application filed by Pfizer filed Critical Pfizer

1998-05-06 Publication of NO982051D0 publication Critical patent/NO982051D0/no

1998-07-03 Publication of NO982051L publication Critical patent/NO982051L/no

2001-04-02 Publication of NO309811B1 publication Critical patent/NO309811B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
- C07D295/26—Sulfur atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Physical Education & Sports Medicine (AREA)
Neurology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Orthopedic Medicine & Surgery (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)

NO982051A 1995-11-07 1998-05-06 FremgangsmÕter og mellomprodukter for fremstilling av 3-(1- piperazinyl)-1,2-benzisotiazol NO309811B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US630195P	1995-11-07	1995-11-07
PCT/IB1996/001079 WO1997017336A1 (en)	1995-11-07	1996-10-11	Processes and intermediates for preparing 3-(1-piperazinyl)-1,2-benzisothiazole

Publications (3)

Publication Number	Publication Date
NO982051D0 NO982051D0 (no)	1998-05-06
NO982051L true NO982051L (no)	1998-07-03
NO309811B1 NO309811B1 (no)	2001-04-02

Family

ID=21720240

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO982051A NO309811B1 (no)	1995-11-07	1998-05-06	FremgangsmÕter og mellomprodukter for fremstilling av 3-(1- piperazinyl)-1,2-benzisotiazol

Country Status (29)

Country	Link
US (1)	US6111105A (no)
EP (1)	EP0874834B1 (no)
JP (1)	JP3152938B2 (no)
KR (1)	KR100315939B1 (no)
CN (1)	CN1071324C (no)
AR (2)	AR004279A1 (no)
AT (1)	ATE198071T1 (no)
AU (1)	AU698443B2 (no)
BR (1)	BR9611366A (no)
CA (1)	CA2236940C (no)
CO (1)	CO4480028A1 (no)
CZ (1)	CZ290600B6 (no)
DE (1)	DE69611253T2 (no)
DK (1)	DK0874834T3 (no)
ES (1)	ES2152564T3 (no)
GR (1)	GR3035215T3 (no)
HU (1)	HU225921B1 (no)
MX (1)	MX9803599A (no)
MY (1)	MY116579A (no)
NO (1)	NO309811B1 (no)
NZ (1)	NZ318844A (no)
PE (1)	PE17298A1 (no)
PL (1)	PL185048B1 (no)
PT (1)	PT874834E (no)
RU (1)	RU2147302C1 (no)
TR (1)	TR199800814T2 (no)
TW (1)	TW358807B (no)
WO (1)	WO1997017336A1 (no)
ZA (1)	ZA969315B (no)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
UY27668A1 (es)	2002-02-20	2003-10-31	Pfizer Prod Inc	Composición de ziprasidona y controles sintéticos
US20040048876A1 (en) *	2002-02-20	2004-03-11	Pfizer Inc.	Ziprasidone composition and synthetic controls
WO2005040160A2 (en)	2003-10-24	2005-05-06	Teva Pharmaceutical Industries Ltd.	Processes for preparation of ziprasidone
US7777037B2 (en) *	2004-10-27	2010-08-17	Dr. Reddy's Laboratories Limited	Ziprasidone process
CN105891392A (zh) *	2016-03-29	2016-08-24	北京万全德众医药生物技术有限公司	一种用液相色谱法分离测定盐酸鲁拉西酮中间体有关物质的方法
CN107064323A (zh) *	2016-12-05	2017-08-18	北京万全德众医药生物技术有限公司	一种用液相色谱法分离测定盐酸鲁拉西酮及其有关物质的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4590196A (en) *	1984-08-23	1986-05-20	Bristol-Myers Company	Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives
NZ230045A (en) *	1988-08-05	1990-11-27	Janssen Pharmaceutica Nv	3-piperazinylbenzazole derivatives and pharmaceutical compositions
JPH06220030A (ja) *	1993-01-22	1994-08-09	Sumitomo Pharmaceut Co Ltd	３−アミノ−１，２−ベンズイソチアゾール誘導体の製造法
JP3701044B2 (ja) *	1995-04-24	2005-09-28	住友精化株式会社	シアノベンゼンスルフェニルハライドおよびそれを用いる３−置換ベンゾイソチアゾールの製造方法
JP3996228B2 (ja) *	1996-10-11	2007-10-24	住友精化株式会社	３−ピペラジニルベンズイソチアゾール類の製造法

1996
- 1996-10-11 WO PCT/IB1996/001079 patent/WO1997017336A1/en not_active Ceased
- 1996-10-11 DK DK96931940T patent/DK0874834T3/da active
- 1996-10-11 NZ NZ318844A patent/NZ318844A/en unknown
- 1996-10-11 CN CN96198127A patent/CN1071324C/zh not_active Expired - Fee Related
- 1996-10-11 CZ CZ19981378A patent/CZ290600B6/cs not_active IP Right Cessation
- 1996-10-11 US US09/068,285 patent/US6111105A/en not_active Expired - Fee Related
- 1996-10-11 DE DE69611253T patent/DE69611253T2/de not_active Expired - Fee Related
- 1996-10-11 ES ES96931940T patent/ES2152564T3/es not_active Expired - Lifetime
- 1996-10-11 KR KR1019980703391A patent/KR100315939B1/ko not_active Expired - Fee Related
- 1996-10-11 RU RU98110457A patent/RU2147302C1/ru not_active IP Right Cessation
- 1996-10-11 EP EP96931940A patent/EP0874834B1/en not_active Expired - Lifetime
- 1996-10-11 JP JP51800597A patent/JP3152938B2/ja not_active Expired - Fee Related
- 1996-10-11 AT AT96931940T patent/ATE198071T1/de not_active IP Right Cessation
- 1996-10-11 PL PL96326630A patent/PL185048B1/pl not_active IP Right Cessation
- 1996-10-11 BR BR9611366A patent/BR9611366A/pt not_active IP Right Cessation
- 1996-10-11 AU AU70926/96A patent/AU698443B2/en not_active Ceased
- 1996-10-11 CA CA002236940A patent/CA2236940C/en not_active Expired - Fee Related
- 1996-10-11 TR TR1998/00814T patent/TR199800814T2/xx unknown
- 1996-10-11 HU HU9903765A patent/HU225921B1/hu not_active IP Right Cessation
- 1996-10-11 PT PT96931940T patent/PT874834E/pt unknown
- 1996-10-15 TW TW085112576A patent/TW358807B/zh not_active IP Right Cessation
- 1996-11-04 PE PE1996000766A patent/PE17298A1/es not_active Application Discontinuation
- 1996-11-04 AR ARP960105036A patent/AR004279A1/es unknown
- 1996-11-06 MY MYPI96004629A patent/MY116579A/en unknown
- 1996-11-06 ZA ZA9609315A patent/ZA969315B/xx unknown
- 1996-11-07 CO CO96058758A patent/CO4480028A1/es unknown
1998
- 1998-05-06 MX MX9803599A patent/MX9803599A/es not_active IP Right Cessation
- 1998-05-06 NO NO982051A patent/NO309811B1/no not_active IP Right Cessation
2001
- 2001-01-11 GR GR20010400030T patent/GR3035215T3/el not_active IP Right Cessation
- 2001-10-29 AR ARP010105060A patent/AR032373A2/es active IP Right Grant

Also Published As

Publication number	Publication date
DE69611253T2 (de)	2001-04-05
JPH10512595A (ja)	1998-12-02
PL185048B1 (pl)	2003-02-28
ES2152564T3 (es)	2001-02-01
JP3152938B2 (ja)	2001-04-03
EP0874834B1 (en)	2000-12-13
TR199800814T2 (xx)	1998-07-21
HUP9903765A2 (hu)	2000-03-28
MY116579A (en)	2004-02-28
CZ137898A3 (cs)	1999-03-17
MX9803599A (es)	1998-09-30
DE69611253D1 (de)	2001-01-18
TW358807B (en)	1999-05-21
NO309811B1 (no)	2001-04-02
ATE198071T1 (de)	2000-12-15
PE17298A1 (es)	1998-04-16
WO1997017336A1 (en)	1997-05-15
ZA969315B (en)	1998-05-06
PL326630A1 (en)	1998-10-12
BR9611366A (pt)	1999-02-23
AU698443B2 (en)	1998-10-29
CA2236940A1 (en)	1997-05-15
CN1071324C (zh)	2001-09-19
HUP9903765A3 (en)	2001-12-28
US6111105A (en)	2000-08-29
GR3035215T3 (en)	2001-04-30
AR032373A2 (es)	2003-11-05
CZ290600B6 (cs)	2002-08-14
HU225921B1 (en)	2008-01-28
CO4480028A1 (es)	1997-07-09
KR100315939B1 (ko)	2002-01-16
EP0874834A1 (en)	1998-11-04
NO982051D0 (no)	1998-05-06
PT874834E (pt)	2001-04-30
DK0874834T3 (da)	2001-02-19
RU2147302C1 (ru)	2000-04-10
CN1201457A (zh)	1998-12-09
AR004279A1 (es)	1998-11-04
KR19990067381A (ko)	1999-08-16
CA2236940C (en)	2001-08-21
NZ318844A (en)	1999-04-29
AU7092696A (en)	1997-05-29

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Legal Events

Date	Code	Title	Description
2010-05-31	MM1K	Lapsed by not paying the annual fees