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DE602006009968D1 - N4-phenyl-chinazolin-4-aminderivate und verwandte verbindungen als inhibitoren der erbb-typ-i-rezeptortyrosinkinase zur behandlung hyperproliferativer krankheiten - Google Patents

N4-phenyl-chinazolin-4-aminderivate und verwandte verbindungen als inhibitoren der erbb-typ-i-rezeptortyrosinkinase zur behandlung hyperproliferativer krankheiten

Info

Publication number
DE602006009968D1
DE602006009968D1 DE602006009968T DE602006009968T DE602006009968D1 DE 602006009968 D1 DE602006009968 D1 DE 602006009968D1 DE 602006009968 T DE602006009968 T DE 602006009968T DE 602006009968 T DE602006009968 T DE 602006009968T DE 602006009968 D1 DE602006009968 D1 DE 602006009968D1
Authority
DE
Germany
Prior art keywords
treatment
type
inhibitors
receptortosrosine
chinazolin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602006009968T
Other languages
English (en)
Inventor
Joseph P Lyssikatos
Fredrik P Marmsater
Qian Zhao
Julie Marie Greschuk
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Array Biopharma Inc
Original Assignee
Array Biopharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38022019&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DE602006009968(D1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Array Biopharma Inc filed Critical Array Biopharma Inc
Publication of DE602006009968D1 publication Critical patent/DE602006009968D1/de
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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DE602006009968T 2005-11-15 2006-11-15 N4-phenyl-chinazolin-4-aminderivate und verwandte verbindungen als inhibitoren der erbb-typ-i-rezeptortyrosinkinase zur behandlung hyperproliferativer krankheiten Active DE602006009968D1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US73628905P 2005-11-15 2005-11-15
US81701906P 2006-06-28 2006-06-28
PCT/US2006/044431 WO2007059257A2 (en) 2005-11-15 2006-11-15 N4-phenyl-quinaz0line-4 -amine derivatives and related compounds as erbb type i receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases

Publications (1)

Publication Number Publication Date
DE602006009968D1 true DE602006009968D1 (de) 2009-12-03

Family

ID=38022019

Family Applications (2)

Application Number Title Priority Date Filing Date
DE602006021645T Active DE602006021645D1 (de) 2005-11-15 2006-11-15 Verfahren und Zwischenverbindungen zur Herstellung von N4-Phenyl-Quinazolin-4-Amin Derivaten
DE602006009968T Active DE602006009968D1 (de) 2005-11-15 2006-11-15 N4-phenyl-chinazolin-4-aminderivate und verwandte verbindungen als inhibitoren der erbb-typ-i-rezeptortyrosinkinase zur behandlung hyperproliferativer krankheiten

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DE602006021645T Active DE602006021645D1 (de) 2005-11-15 2006-11-15 Verfahren und Zwischenverbindungen zur Herstellung von N4-Phenyl-Quinazolin-4-Amin Derivaten

Country Status (28)

Country Link
US (6) US8648087B2 (de)
EP (2) EP1971601B1 (de)
JP (2) JP5134548B2 (de)
KR (1) KR101086967B1 (de)
CN (2) CN101356171A (de)
AT (2) ATE507224T1 (de)
AU (2) AU2006315383B2 (de)
BR (2) BRPI0618668B1 (de)
CA (2) CA2755268C (de)
CY (3) CY1110583T1 (de)
DE (2) DE602006021645D1 (de)
DK (2) DK1971601T3 (de)
ES (2) ES2335535T3 (de)
FI (1) FIC20210022I1 (de)
FR (1) FR21C1031I2 (de)
HU (1) HUS2100028I1 (de)
IL (2) IL239149A (de)
LT (1) LTC1971601I2 (de)
LU (1) LUC00217I2 (de)
NL (1) NL301113I2 (de)
NO (1) NO342413B1 (de)
PL (2) PL1971601T3 (de)
PT (2) PT2090575E (de)
RU (2) RU2592703C9 (de)
SG (1) SG152230A1 (de)
SI (2) SI1971601T1 (de)
WO (1) WO2007059257A2 (de)
ZA (1) ZA200804498B (de)

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DK1660090T3 (da) 2003-08-14 2012-12-17 Array Biopharma Inc Quinazolin-analoger som receptor-tyrosinkinase-inhibitorer
GB0420722D0 (en) 2004-09-17 2004-10-20 Addex Pharmaceuticals Sa Novel allosteric modulators
CN101356171A (zh) 2005-11-15 2009-01-28 阿雷生物药品公司 作为erbbi型受体酪氨酸激酶抑制剂用于治疗增殖性疾病的n4-苯基-喹唑啉-4-胺衍生物和相关化合物
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US8604044B2 (en) * 2006-09-11 2013-12-10 Curis, Inc. Quinazoline based EGFR inhibitors containing a zinc binding moiety
US7547781B2 (en) 2006-09-11 2009-06-16 Curis, Inc. Quinazoline based EGFR inhibitors containing a zinc binding moiety
CA2662937A1 (en) * 2006-09-11 2008-03-20 Curis, Inc. Multi-functional small molecules as anti-proliferative agents
TW200845978A (en) 2007-03-07 2008-12-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
TW200900065A (en) 2007-03-07 2009-01-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
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