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CN1363331A - Nano storax medicine and its preparing process - Google Patents

Nano storax medicine and its preparing process Download PDF

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Publication number
CN1363331A
CN1363331A CN 01100769 CN01100769A CN1363331A CN 1363331 A CN1363331 A CN 1363331A CN 01100769 CN01100769 CN 01100769 CN 01100769 A CN01100769 A CN 01100769A CN 1363331 A CN1363331 A CN 1363331A
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China
Prior art keywords
nanometer
nano
parts
storax
part nanometer
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Pending
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CN 01100769
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Chinese (zh)
Inventor
杨孟君
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Individual
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Individual
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Priority to CN 01100769 priority Critical patent/CN1363331A/en
Publication of CN1363331A publication Critical patent/CN1363331A/en
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  • Medicines Containing Plant Substances (AREA)

Abstract

A nano medicine "Suhexiang" is prepared from the nano powders of 15 Chinese-medicinal materials including storax, benzoin, borneol, musk, etc through proportioning, microwave extracting, vacuum concentrating and supersonic-jet spray drying. Its advantages include high biological utilization rate and high curative effect.

Description

Nano storax medicine and preparation method thereof
The present invention relates to a kind of causing resuscitation with aromatic drugs, promoting the circulation of QI to relieve pain, warming the interior cold expelling, resolving depression refreshment, ward off the turbid nano storax medicine of dirtyization, the invention still further relates to the method for this medication preparation.
Styrax Pilulae is a kind of classical Chinese patent medicine, mainly contains effects such as antiplatelet aggregation, protection cardiac muscle, inhibition vasoconstriction, is used for apoplexy, heatstroke, coma due to phlegm syncope, heart peratodynia, angina pectoris.But traditional Styrax Pilulae absorbs not exclusively, and bioavailability is not high, slow curative effect.
The object of the present invention is to provide a kind of bioavailability height, solid dispersion is good, absorbs fully the nano storax medicine of increase evident in efficacy.
Another object of the present invention provides the preparation method of this nano storax medicine.
To achieve these goals, the present invention takes following technical scheme:
Medicine of the present invention is to make (consumption is a weight portion) by following component:
Nano storax 30-70 part nanometer Benzoinum 60-140 part nanometer Borneolum Syntheticum 30-70 part
Nano musk 50-100 part nanometer terminalia flesh 60-140 part nanometer Lignum Santali Albi 60-140 part
Nanometer Lignum Aquilariae Resinatum 60-140 part nano clove 60-140 part nano cyperus tuber 60-140 part
Nanometer Radix Aucklandiae 60-140 part nanometer Olibanum 60-140 part nanometer Long Pepper 60-140 part
Nanometer Rhizoma Atractylodis Macrocephalae 60-140 part nanometer Cinnabaris 60-140 part
Nanometer Pulvis Cornus Bubali Concentratus 120-280 part
The formula optimization weight proportion scope of medicine of the present invention is:
Nano storax 40-60 part nanometer Benzoinum 80-120 part nanometer Borneolum Syntheticum 40-60 part
Nano musk 60-90 part nanometer terminalia flesh 80-120 part nanometer Lignum Santali Albi 80-120 part
Nanometer Lignum Aquilariae Resinatum 80-120 part nano clove 80-120 part nano cyperus tuber 80-120 part
Nanometer Radix Aucklandiae 80-120 part nanometer Olibanum 80-120 part nanometer Long Pepper 80-120 part
Nanometer Rhizoma Atractylodis Macrocephalae 80-120 part nanometer Cinnabaris 80-120 part
Nanometer Pulvis Cornus Bubali Concentratus 160-240 part
The optimum weight proportioning of medicine of the present invention is:
50 parts of 100 parts of nanometer Borneolum Syntheticums of 50 parts of nanometer Benzoinumes of nano storax
100 parts in 100 parts of nanometer Lignum Santali Albis of 75 parts of nanometer terminalia flesh of nano musk
100 parts of 100 parts of nano cyperus tubers of 100 parts of nano cloves of nanometer Lignum Aquilariae Resinatum
100 parts of 100 parts of nanometer Long Peppers of 100 parts of nanometer Olibanums of the nanometer Radix Aucklandiae
100 parts in 100 parts of nanometer Cinnabaris of the nanometer Rhizoma Atractylodis Macrocephalae
200 parts of nanometer Pulvis Cornus Bubali Concentratuss
Technical scheme of the present invention is based on the modern material technology.One of modern material Developing Trend in Technology is to develop to the more and more littler direction of yardstick.The granule of the past composition material, its size all are at micron or more than the millimeter magnitude, and have occurred the material to the nanoscale development now.Because extremely refinement of granule, the shared percentage by volume of crystal boundary increases, and makes some performance of material that outstanding variation take place.
The property of nano material is because the special construction of nano material---the particle size of material is less than the ultra-micro powder of 100nm, its body surface area is very big, the atom number ratio at crystal boundary place makes it to produce four big effects up to 15%-50%: i.e. small-size effect, quantum effect (containing macro quanta tunnel effect), skin effect and interfacial effect.Thereby has the not available physical and chemical performance of traditional material.Nanotechnology will bring a technological revolution of the field of Chinese medicines.
One of method of above-mentioned each component being made medicine of the present invention is:
1. divide and get the Chinese crude drug of respectively distinguishing the flavor of, add to concoct according to Chinese Pharmacopoeia one one of version in 2000 and be processed into the common Chinese decoction pieces
2. divide and get the common Chinese decoction pieces of respectively distinguishing the flavor of, be processed into the nanometer prepared slices of Chinese crude drugs, its method comprises the following steps:
1. the common Chinese decoction pieces is placed extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, promptly make the nanometer prepared slices of Chinese crude drugs with the instantaneous drying of hypersonic velocity.
3. the nanometer prepared slices of Chinese crude drugs (powder) are prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent standard, make pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution.
Two of medicine method for making of the present invention is:
1. be equipped with whole common Chinese decoction pieces in the proportioning ratio, place extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, get Styrax preparation nano powder with the instantaneous drying of hypersonic velocity jet;
4. its nano powder is made aforementioned various preparation according to Chinese Pharmacopoeia version standard preparation in 2000.
The pharmacological effect that above-mentioned two kinds of methods are made nano storax medicine is identical.
A kind of important feature of the present invention is: the made drug material of the present invention has reached nanoscale, common Styrax Pilulae preparation material is micron or the above particle diameter of millimeter, can only cross the 80-120 mesh sieve, the drug material that the present invention is made, particle diameter is at 0.1-200nm, the overwhelming majority can be crossed the 1200-1500 mesh sieve less than 100nm.
Another important feature of the present invention is: solid preparation of the present invention disintegrate rapidly, and solid dispersion is good in water, absorb fully, the bioavailability height, the pharmacological action effect that mainly contains effective constituent is significantly higher than conventional formulation.
The pharmaceutical preparation that the present invention is made does not need to add any adjuvant, and is more favourable to human body.
The present invention has also created the new drug formulation that suppository, granule, membrane, microcapsule, drop pill, aerosol, injection, medicated wine, syrup, oral solution of nano storax medicine etc. is had no precedent in the past.
Pharmaceutical preparation of the present invention can be used for treatment of conditions such as the painful biliary tract ascarid of apoplexy constipation due to cold pathogen, coma and trusted subordinate, and clinical efficacy significantly is better than traditional Styrax Pilulae.
The present invention's added solvent in microwave extracting is water or ethanol.
The present invention carries out in the concentrating under reduced pressure step at extract, and its concentrating under reduced pressure is conventional scheme.
Embodiment 1:
Prepare nano raw material by preceding method:
50 parts of 100 parts of nanometer Borneolum Syntheticums of 50 parts of nanometer Benzoinumes of nano storax
100 parts in 100 parts of nanometer Lignum Santali Albis of 75 parts of nanometer terminalia flesh of nano musk
100 parts of 100 parts of nano cyperus tubers of 100 parts of nano cloves of nanometer Lignum Aquilariae Resinatum
100 parts of 100 parts of nanometer Long Peppers of 100 parts of nanometer Olibanums of the nanometer Radix Aucklandiae
100 parts in 100 parts of nanometer Cinnabaris of the nanometer Rhizoma Atractylodis Macrocephalae
200 parts of nanometer Pulvis Cornus Bubali Concentratuss
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent capsules agent standard, do not add adjuvant, do not granulate, directly divide encapsulated with the fully-automatic capsule racking machine, make capsule, every capsules content of dispersion is the 0.1-0.6 gram, and the patient takes 1-4 time every day, each 1-5 grain.
Embodiment 2:
Prepare nano raw material by preceding method:
50 parts of 100 parts of nanometer Borneolum Syntheticums of 50 parts of nanometer Benzoinumes of nano storax
100 parts in 100 parts of nanometer Lignum Santali Albis of 75 parts of nanometer terminalia flesh of nano musk
100 parts of 100 parts of nano cyperus tubers of 100 parts of nano cloves of nanometer Lignum Aquilariae Resinatum
100 parts of 100 parts of nanometer Long Peppers of 100 parts of nanometer Olibanums of the nanometer Radix Aucklandiae
100 parts in 100 parts of nanometer Cinnabaris of the nanometer Rhizoma Atractylodis Macrocephalae
200 parts of nanometer Pulvis Cornus Bubali Concentratuss
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent powder needle injection standard, do not add any adjuvant, make the nano storax powder needle injection, every injection content is the 5-20 milligram, and each consumption is that 1-2 props up, and use 1-3 every day.
Embodiment 3:
Prepare nano raw material by preceding method:
50 parts of 100 parts of nanometer Borneolum Syntheticums of 50 parts of nanometer Benzoinumes of nano storax
100 parts in 100 parts of nanometer Lignum Santali Albis of 75 parts of nanometer terminalia flesh of nano musk
100 parts of 100 parts of nano cyperus tubers of 100 parts of nano cloves of nanometer Lignum Aquilariae Resinatum
100 parts of 100 parts of nanometer Long Peppers of 100 parts of nanometer Olibanums of the nanometer Radix Aucklandiae
100 parts in 100 parts of nanometer Cinnabaris of the nanometer Rhizoma Atractylodis Macrocephalae
200 parts of nanometer Pulvis Cornus Bubali Concentratuss
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent membrane standard, filmogen adopts polyvinyl alcohol, make the nano storax membrane, every membrane area size is the 2-100 square centimeter, and content of dispersion is the 1-50 gram, every medicine film pasted 1-7 days, pasted the medicine position: abdominal part, back, chest.

Claims (6)

1, a kind of nano storax medicine is characterized in that it is the medicament that the nano raw material of following weight proportioning is made:
Nano storax 30-70 part nanometer Benzoinum 60-140 part nanometer Borneolum Syntheticum 30-70 part
Nano musk 50-100 part nanometer terminalia flesh 60-140 part nanometer Lignum Santali Albi 60-140 part
Nanometer Lignum Aquilariae Resinatum 60-140 part nano clove 60-140 part nano cyperus tuber 60-140 part
Nanometer Radix Aucklandiae 60-140 part nanometer Olibanum 60-140 part nanometer Long Pepper 60-140 part
Nanometer Rhizoma Atractylodis Macrocephalae 60-140 part nanometer Cinnabaris 60-140 part
Nanometer Pulvis Cornus Bubali Concentratus 120-280 part
And adopt following method to make: to select the formula Chinese drug material to concoct and be processed into the prepared slices of Chinese crude drugs; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters--990 meter per seconds, promptly make the nanometer prepared slices of Chinese crude drugs.
2, nano storax medicine according to claim 1, wherein the weight proportion of each nano raw material is:
Nano storax 40-60 part nanometer Benzoinum 80-120 part nanometer Borneolum Syntheticum 40-60 part
Nano musk 60-90 part nanometer terminalia flesh 80-120 part nanometer Lignum Santali Albi 80-120 part
Nanometer Lignum Aquilariae Resinatum 80-120 part nano clove 80-120 part nano cyperus tuber 80-120 part
Nanometer Radix Aucklandiae 80-120 part nanometer Olibanum 80-120 part nanometer Long Pepper 80-120 part
Nanometer Rhizoma Atractylodis Macrocephalae 80-120 part nanometer Cinnabaris 80-120 part
Nanometer Pulvis Cornus Bubali Concentratus 160-240 part
3, nano storax medicine according to claim 1, wherein the weight proportion of each nano raw material is:
50 parts of 100 parts of nanometer Borneolum Syntheticums of 50 parts of nanometer Benzoinumes of nano storax
100 parts in 100 parts of nanometer Lignum Santali Albis of 75 parts of nanometer terminalia flesh of nano musk
100 parts of 100 parts of nano cyperus tubers of 100 parts of nano cloves of nanometer Lignum Aquilariae Resinatum
100 parts of 100 parts of nanometer Long Peppers of 100 parts of nanometer Olibanums of the nanometer Radix Aucklandiae
100 parts in 100 parts of nanometer Cinnabaris of the nanometer Rhizoma Atractylodis Macrocephalae
200 parts of nanometer Pulvis Cornus Bubali Concentratuss
4,, it is characterized in that said medicine is pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution according to claim 1 or 2 or 3 described nano storax medicines.
5,, it is characterized in that this method comprises the steps: to select the formula Chinese drug material to concoct and is processed into the prepared slices of Chinese crude drugs according to the pharmaceutical methods of claim 1 or 2 or 3 described nano storax medicines; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters--990 meter per seconds, promptly make the nanometer prepared slices of Chinese crude drugs.
6, wherein respectively distinguish the flavor of Chinese medicine in the ratio of prescription or Chinese crude drug concoct be processed into the prepared slices of Chinese crude drugs after mixing, or after making the nanometer prepared slices of Chinese crude drugs mixing.
CN 01100769 2001-01-09 2001-01-09 Nano storax medicine and its preparing process Pending CN1363331A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN 01100769 CN1363331A (en) 2001-01-09 2001-01-09 Nano storax medicine and its preparing process

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN 01100769 CN1363331A (en) 2001-01-09 2001-01-09 Nano storax medicine and its preparing process

Publications (1)

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CN1363331A true CN1363331A (en) 2002-08-14

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Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102846899A (en) * 2012-09-13 2013-01-02 李承平 Storax tablet combination
CN113116997A (en) * 2021-04-30 2021-07-16 贵州汉方药业有限公司 Preparation method of storax pills

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102846899A (en) * 2012-09-13 2013-01-02 李承平 Storax tablet combination
CN113116997A (en) * 2021-04-30 2021-07-16 贵州汉方药业有限公司 Preparation method of storax pills
CN113116997B (en) * 2021-04-30 2022-10-21 贵州汉方药业有限公司 Preparation method of storax pills

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Addressee: Yang Mengjun

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