[go: up one dir, main page]

CN1362241A - Nano gastrodia and sharpleaf gambirplant medicine and its preparation - Google Patents

Nano gastrodia and sharpleaf gambirplant medicine and its preparation Download PDF

Info

Publication number
CN1362241A
CN1362241A CN 01100743 CN01100743A CN1362241A CN 1362241 A CN1362241 A CN 1362241A CN 01100743 CN01100743 CN 01100743 CN 01100743 A CN01100743 A CN 01100743A CN 1362241 A CN1362241 A CN 1362241A
Authority
CN
China
Prior art keywords
nano
nanometer
parts
gastrodia
ramulus uncariae
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CN 01100743
Other languages
Chinese (zh)
Inventor
杨孟君
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Priority to CN 01100743 priority Critical patent/CN1362241A/en
Publication of CN1362241A publication Critical patent/CN1362241A/en
Pending legal-status Critical Current

Links

Landscapes

  • Medicines Containing Plant Substances (AREA)
  • Medicinal Preparation (AREA)

Abstract

The present invention discloses a nano gastrodis uncaria preparation medicine. It is made up by using 11 Chinese medicinal materials of nano gastrodia, nano uncarina, nano abalone shell, nano gardenia, nano astragalus and others as raw material through the processes of microwave extraction, reduced pressure concentration and supersonic jet spray drying. Its grain fineness is up to 1200-1500 meshes, grain size is 0.1-200 nm, in which most of grain size is less than 100 nm. Said medicine is high in biological utilization rate and obvious in therapeutic effect.

Description

Nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine and preparation method thereof
The present invention relates to the nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine of a kind of suppressing the hyperactive liver to relieve the wind syndrome, heat clearing and blood circulation promoting, liver and kidney tonifying, the invention still further relates to the method for this medication preparation.
The TIANMAGOUTENG granule is a kind of classical Chinese patent medicine, mainly contains blood pressure lowering, regulates the central nervous system, the effects such as generation of antiplatelet aggregation, inhibition lipid peroxide, is used for that liver-yang is high partially, disturbs on the liver-wind, diseases such as headache, dizzy, insomnia.But traditional TIANMAGOUTENG granule absorbs not exclusively, and bioavailability is not high, slow curative effect.
The object of the present invention is to provide a kind of bioavailability height, solid dispersion is good, absorbs fully the nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine of increase evident in efficacy.
Another object of the present invention provides the preparation method of this nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine.
To achieve these goals, the present invention takes following technical scheme:
Medicine of the present invention is to make (consumption is a weight portion) by following component:
Nano gastrodia 5-50 part nanometer Ramulus Uncariae Cum Uncis 10-60 part nano abalone shell 5-50 part
Nanometer Fructus Gardeniae 5-50 part nano astragalus 10-60 part nanometer Radix Cyathulae 5-50 part
Nanometer Cortex Eucommiae 5-50 part nanometer motherwort 5-60 part nanometer Herba Taxilli 5-50 part
Nano fleece flower root rattan 5-50 part nano Poria 3-40 part
The formula optimization weight proportion scope of medicine of the present invention is:
Nano gastrodia 15-40 part nanometer Ramulus Uncariae Cum Uncis 20-50 part nano abalone shell 10-30 part
Nanometer Fructus Gardeniae 15-40 part nano astragalus 20-50 part nanometer Radix Cyathulae 15-40 part
Nanometer Cortex Eucommiae 10-40 part nanometer motherwort 10-40 part nanometer Herba Taxilli 10-40 part
Nano fleece flower root rattan 10-40 part nano Poria 8-30 part
The optimum weight proportioning of medicine of the present invention is:
20 parts of 28 parts of nano abalone shells of 25 parts of nanometer Ramulus Uncariae Cum Uncis of nano gastrodia
25 parts of 30 parts of nanometer Radix Cyathulaes of 25 parts of nano astragalus of nanometer Fructus Gardeniae
26 parts of 20 parts of nanometer Herba Taxillis of 20 parts of nanometer motherworts of the nanometer Cortex Eucommiae
15 parts of 20 parts of nano Porias of nano fleece flower root rattan
Technical scheme of the present invention is based on the modern material technology.One of modern material Developing Trend in Technology is to develop to the more and more littler direction of yardstick.The granule of the past composition material, its size all are at micron or more than the millimeter magnitude, and have occurred the material to the nanoscale development now.Because extremely refinement of granule, the shared percentage by volume of crystal boundary increases, and makes some performance of material that outstanding variation take place.
The property of nano material is because the special construction of nano material---the particle size of material is less than the ultra-micro powder of 100nm, its body surface area is very big, the atom number ratio at crystal boundary place makes it to produce four big effects up to 15%-50%: i.e. small-size effect, quantum effect (containing macro quanta tunnel effect), skin effect and interfacial effect.Thereby has the not available physical and chemical performance of traditional material.Nanotechnology will bring a technological revolution of the field of Chinese medicines.
One of method of above-mentioned each component being made medicine of the present invention is:
1. divide and get the Chinese crude drug of respectively distinguishing the flavor of, add to concoct according to Chinese Pharmacopoeia one one of version in 2000 and be processed into the common Chinese decoction pieces
2. divide and get the common Chinese decoction pieces of respectively distinguishing the flavor of, be processed into the nanometer prepared slices of Chinese crude drugs, its method comprises the following steps:
1. the common Chinese decoction pieces is placed extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, promptly make the nanometer prepared slices of Chinese crude drugs with the instantaneous drying of hypersonic velocity.
3. the nanometer prepared slices of Chinese crude drugs (powder) are prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent standard, make pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution.
Two of medicine method for making of the present invention is:
1. be equipped with whole common Chinese decoction pieces in the proportioning ratio, place extraction pot, solubilizer also imports microwave extracting, makes its speed with 20-30 hundred million times/second do the change in polarity motion, and the temperature of its microwave extracting is 30 ℃-60 ℃, time 1-10 hour;
2. above-mentioned extract is carried out concentrating under reduced pressure, temperature is 30 ℃-60 ℃, and the time is 3-72 hour, collects volatile material in the Chinese medicine simultaneously in addition;
3. decompressed concentrate and volatile material merging are placed spray drying tower, use the supersonic jet technology, 330 meters-990 meter per seconds of effluxvelocity, 30 ℃ of-60 ℃ of temperature, under 0 to the 0.05MPa pressure,, get TIANMAGOUTENG preparation nano powder with the instantaneous drying of hypersonic velocity jet;
4. its nano powder is made aforementioned various preparation according to Chinese Pharmacopoeia version standard preparation in 2000.
The pharmacological effect that above-mentioned two kinds of methods are made nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine is identical.
A kind of important feature of the present invention is: the made drug material of the present invention has reached nanoscale, common TIANMAGOUTENG granular preparation material is micron or the above particle diameter of millimeter, can only cross the 80-120 mesh sieve, the drug material that the present invention is made, particle diameter is at 0.1-200nm, the overwhelming majority can be crossed the 1200-1500 mesh sieve less than 100nm.
Another important feature of the present invention is: solid preparation of the present invention disintegrate rapidly, and solid dispersion is good in water, absorb fully, the bioavailability height, the pharmacological action effect that mainly contains effective constituent is significantly higher than conventional formulation.
The pharmaceutical preparation that the present invention is made does not need to add any adjuvant, and is more favourable to human body.
The present invention has also created the new drug formulation that suppository, membrane, microcapsule, drop pill, aerosol, injection, medicated wine, syrup of nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine etc. is had no precedent in the past.
Pharmaceutical preparation of the present invention can be used for treatment of conditions such as hypertension, interior M, trigeminal neuralgia, facial spasm, contusion and laceration of brain, and clinical efficacy significantly is better than traditional TIANMAGOUTENG granule.
The present invention's added solvent in microwave extracting is water or ethanol.
The present invention carries out in the concentrating under reduced pressure step at extract, and its concentrating under reduced pressure is conventional scheme.
Embodiment 1:
Prepare nano raw material by preceding method:
20 parts of 28 parts of nano abalone shells of 25 parts of nanometer Ramulus Uncariae Cum Uncis of nano gastrodia
25 parts of 30 parts of nanometer Radix Cyathulaes of 25 parts of nano astragalus of nanometer Fructus Gardeniae
26 parts of 20 parts of nanometer Herba Taxillis of 20 parts of nanometer motherworts of the nanometer Cortex Eucommiae
15 parts of 20 parts of nano Porias of nano fleece flower root rattan
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent capsules agent standard, do not add adjuvant, do not granulate, directly divide encapsulated with the fully-automatic capsule racking machine, make capsule, every capsules content of dispersion is the 0.1-0.6 gram, and the patient takes 1-4 time every day, each 1-5 grain.
Embodiment 2:
Prepare nano raw material by preceding method:
20 parts of 28 parts of nano abalone shells of 25 parts of nanometer Ramulus Uncariae Cum Uncis of nano gastrodia
25 parts of 30 parts of nanometer Radix Cyathulaes of 25 parts of nano astragalus of nanometer Fructus Gardeniae
26 parts of 20 parts of nanometer Herba Taxillis of 20 parts of nanometer motherworts of the nanometer Cortex Eucommiae
15 parts of 20 parts of nano Porias of nano fleece flower root rattan
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent powder needle injection standard, do not add any adjuvant, make nano gastrodia Ramulus Uncariae Cum Uncis powder needle injection, every injection content is the 5-20 milligram, and each consumption is that 1-2 props up, and use 1-3 every day.
Embodiment 3:
Prepare nano raw material by preceding method:
20 parts of 28 parts of nano abalone shells of 25 parts of nanometer Ramulus Uncariae Cum Uncis of nano gastrodia
25 parts of 30 parts of nanometer Radix Cyathulaes of 25 parts of nano astragalus of nanometer Fructus Gardeniae
26 parts of 20 parts of nanometer Herba Taxillis of 20 parts of nanometer motherworts of the nanometer Cortex Eucommiae
15 parts of 20 parts of nano Porias of nano fleece flower root rattan
Production method is as follows:
In the GMP cleaning shop, after the above-mentioned nanometer prepared slices of Chinese crude drugs or powder prepared mixing in described ratio, according to Chinese Pharmacopoeia version two-shift system in 2000 agent membrane standard, filmogen adopts polyvinyl alcohol, make nano gastrodia Ramulus Uncariae Cum Uncis membrane, every membrane area size is the 2-100 square centimeter, and content of dispersion is the 1-50 gram, every medicine film pasted 1-7 days, pasted the medicine position: abdominal part, back, chest, cervical region.

Claims (6)

1, a kind of nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine is characterized in that it is the medicament that the nano raw material of following weight proportioning is made:
Nano gastrodia 5-50 part nanometer Ramulus Uncariae Cum Uncis 10-60 part nano abalone shell 5-50 part
Nanometer Fructus Gardeniae 5-50 part nano astragalus 10-60 part nanometer Radix Cyathulae 5-50 part
Nanometer Cortex Eucommiae 5-50 part nanometer motherwort 5-60 part nanometer Herba Taxilli 5-50 part
Nano fleece flower root rattan 5-50 part nano Poria 3-40 part
And adopt following method to make: to select the formula Chinese drug material to concoct and be processed into the prepared slices of Chinese crude drugs; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters--990 meter per seconds, promptly make the nanometer prepared slices of Chinese crude drugs.
2, nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine according to claim 1, wherein the weight proportion of each nano raw material is:
Nano gastrodia 15-40 part nanometer Ramulus Uncariae Cum Uncis 20-50 part nano abalone shell 10-30 part
Nanometer Fructus Gardeniae 15-40 part nano astragalus 20-50 part nanometer Radix Cyathulae 15-40 part
Nanometer Cortex Eucommiae 10-40 part nanometer motherwort 10-40 part nanometer Herba Taxilli 10-40 part
Nano fleece flower root rattan 10-40 part nano Poria 8-30 part
3, nano gastrodia Ramulus Uncariae Cum Uncis preparation medicine according to claim 1, wherein the weight proportion of each nano raw material is:
20 parts of 28 parts of nano abalone shells of 25 parts of nanometer Ramulus Uncariae Cum Uncis of nano gastrodia
25 parts of 30 parts of nanometer Radix Cyathulaes of 25 parts of nano astragalus of nanometer Fructus Gardeniae
26 parts of 20 parts of nanometer Herba Taxillis of 20 parts of nanometer motherworts of the nanometer Cortex Eucommiae
15 parts of 20 parts of nano Porias of nano fleece flower root rattan
4, according to claim 1 or 2 or 3 described nano gastrodia Ramulus Uncariae Cum Uncis preparation medicines, it is characterized in that said medicine is pill, powder, tablet, suppository, granule, membrane, capsule, microcapsule, drop pill, aerosol, injection, unguentum, medicated wine, syrup, oral solution.
5,, it is characterized in that this method comprises the steps: to select the formula Chinese drug material to concoct and is processed into the prepared slices of Chinese crude drugs according to the pharmaceutical methods of claim 1 or 2 or 3 described nano gastrodia Ramulus Uncariae Cum Uncis preparation medicines; Place extraction pot, solubilizer also imports microwave extracting, makes it do the change in polarity motion with hundred million times/second speed of 20--30, and the temperature of its microwave extracting is 30--60 ℃, time 1--10 hour; Above-mentioned extract is carried out concentrating under reduced pressure, and temperature is 30--60 ℃, and the time is 3--72 hour, collects volatile material in the Chinese medicine simultaneously in addition; Decompressed concentrate and volatile material merging are placed spray drying tower, use the Supersonic fluidics, 30--60 ℃ of temperature, under 0 to the 0.05MPa pressure, with hypersonic velocity instantaneous jet drying, wherein supersonic jet speed is 330 meters--990 meter per seconds, promptly make the nanometer prepared slices of Chinese crude drugs.
6, wherein respectively distinguish the flavor of Chinese medicine in the ratio of prescription or Chinese crude drug concoct be processed into the prepared slices of Chinese crude drugs after mixing, or after making the nanometer prepared slices of Chinese crude drugs mixing.
CN 01100743 2001-01-08 2001-01-08 Nano gastrodia and sharpleaf gambirplant medicine and its preparation Pending CN1362241A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN 01100743 CN1362241A (en) 2001-01-08 2001-01-08 Nano gastrodia and sharpleaf gambirplant medicine and its preparation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN 01100743 CN1362241A (en) 2001-01-08 2001-01-08 Nano gastrodia and sharpleaf gambirplant medicine and its preparation

Publications (1)

Publication Number Publication Date
CN1362241A true CN1362241A (en) 2002-08-07

Family

ID=4651847

Family Applications (1)

Application Number Title Priority Date Filing Date
CN 01100743 Pending CN1362241A (en) 2001-01-08 2001-01-08 Nano gastrodia and sharpleaf gambirplant medicine and its preparation

Country Status (1)

Country Link
CN (1) CN1362241A (en)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007006203A1 (en) * 2005-07-07 2007-01-18 Shirong Duan A capsule formulation for treating hypertension and coronary heart disease and process for preparation thereof
CN102091239A (en) * 2011-01-07 2011-06-15 孙建英 Uncaria abalone sour soup for treating trigeminal neuralgia
CN102526530A (en) * 2012-02-20 2012-07-04 迟建波 Chinese medicine for treating hypertension and preparation method for Chinese medicine
CN103055164A (en) * 2012-12-26 2013-04-24 中国中医科学院中医临床基础医学研究所 Traditional Chinese medicine composition for treating isolated diastolic hypertension

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007006203A1 (en) * 2005-07-07 2007-01-18 Shirong Duan A capsule formulation for treating hypertension and coronary heart disease and process for preparation thereof
CN102091239A (en) * 2011-01-07 2011-06-15 孙建英 Uncaria abalone sour soup for treating trigeminal neuralgia
CN102091239B (en) * 2011-01-07 2012-07-04 孙建英 Uncaria abalone sour soup for treating trigeminal neuralgia
CN102526530A (en) * 2012-02-20 2012-07-04 迟建波 Chinese medicine for treating hypertension and preparation method for Chinese medicine
CN102526530B (en) * 2012-02-20 2014-02-26 迟建波 Chinese medicine for treating hypertension and preparation method for Chinese medicine
CN103055164A (en) * 2012-12-26 2013-04-24 中国中医科学院中医临床基础医学研究所 Traditional Chinese medicine composition for treating isolated diastolic hypertension

Similar Documents

Publication Publication Date Title
CN1362241A (en) Nano gastrodia and sharpleaf gambirplant medicine and its preparation
CN1362160A (en) Nano Heavn king tonic medicine for mental discomfort and its preparation
CN1368181A (en) Nano medicine 'Shufeng Dingtong' and its preparing process
CN1362075A (en) Nano blood stasis dispersing medicine and its preparation
CN1368235A (en) Nano medicine for treating leukoderma and its preparing process
CN1366915A (en) Nano brain-benefiting blood pressure-reducing preparation medicine and preparation method
CN1362167A (en) Nano Zhengtian medicine and its preparation
CN1365746A (en) Nano medicine 'Sizheng' and its preparing process
CN1362207A (en) Nano healthy energy restoring agastachis medicine and its preparation
CN1362122A (en) Nano fracture-setting traumatic medicine and its preparation
CN1360939A (en) Nanometer eyesight-improving and health-clearing medicine and its prepn
CN1363331A (en) Nano storax medicine and its preparing process
CN1368087A (en) Nano medicine for treating cerebral thrombus and its preparing process
CN1362139A (en) Nano Pingxiao medicine and its preparation
CN1368357A (en) Nano medicine 'Weitongding' and its preparing process
CN1362136A (en) Nano Jingfukang medicine and its preparation
CN1362247A (en) Nano stomach-nourishing medicine of Aucklandiae and Amino and its preparation
CN1364537A (en) Nano China Ganling medicine and its preparing method
CN1362220A (en) Nano Anemarrhenae, phellodendri and Rehmanniae medicine and its preparation
CN1362246A (en) Nano Bupleuric medicine for regulating Shaoyang and it spreparation
CN1362138A (en) Nano influenza treating decoction and its preparation
CN1362152A (en) Nano hypertension-treating bezoar medicine and its preparation
CN1362222A (en) Nanometer blood-nourishing and transquilizing medicine and its preparation
CN1362223A (en) Nano Xinmaitong medicine and its preparation
CN1362204A (en) Nanometer medicine for invigorating gallbadder and exhausting stone and its preparation

Legal Events

Date Code Title Description
C06 Publication
PB01 Publication
C02 Deemed withdrawal of patent application after publication (patent law 2001)
WD01 Invention patent application deemed withdrawn after publication