BRPI0906245A2 - Composto, método para tratar um distúrbio cognitivo, psicótico, mediado por neurotransmissor ou um distúrbio neuronal em indivíduo, uso de um composto, composição farmacêutica e kit - Google Patents
Composto, método para tratar um distúrbio cognitivo, psicótico, mediado por neurotransmissor ou um distúrbio neuronal em indivíduo, uso de um composto, composição farmacêutica e kitInfo
- Publication number
- BRPI0906245A2 BRPI0906245A2 BRPI0906245-9A BRPI0906245A BRPI0906245A2 BR PI0906245 A2 BRPI0906245 A2 BR PI0906245A2 BR PI0906245 A BRPI0906245 A BR PI0906245A BR PI0906245 A2 BRPI0906245 A2 BR PI0906245A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- disorder
- psychotic
- cognitive
- kit
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 2
- 208000028017 Psychotic disease Diseases 0.000 title 1
- 230000001149 cognitive effect Effects 0.000 title 1
- 230000001404 mediated effect Effects 0.000 title 1
- 230000001537 neural effect Effects 0.000 title 1
- 239000002858 neurotransmitter agent Substances 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/18—Bridged systems
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Immunology (AREA)
- Hospice & Palliative Care (AREA)
- Pulmonology (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3905808P | 2008-03-24 | 2008-03-24 | |
| US14505809P | 2009-01-15 | 2009-01-15 | |
| PCT/US2009/038142 WO2009120720A1 (en) | 2008-03-24 | 2009-03-24 | Bridged heterocyclic compounds and methods of use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0906245A2 true BRPI0906245A2 (pt) | 2015-06-30 |
Family
ID=40651664
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0906245-9A BRPI0906245A2 (pt) | 2008-03-24 | 2009-03-24 | Composto, método para tratar um distúrbio cognitivo, psicótico, mediado por neurotransmissor ou um distúrbio neuronal em indivíduo, uso de um composto, composição farmacêutica e kit |
Country Status (12)
| Country | Link |
|---|---|
| US (4) | US8546381B2 (pt) |
| EP (1) | EP2274307B1 (pt) |
| JP (2) | JP5586577B2 (pt) |
| CN (1) | CN102046625B (pt) |
| AR (1) | AR071284A1 (pt) |
| AU (1) | AU2009228401B2 (pt) |
| BR (1) | BRPI0906245A2 (pt) |
| CA (1) | CA2718790A1 (pt) |
| CL (1) | CL2009000725A1 (pt) |
| PE (1) | PE20091820A1 (pt) |
| TW (1) | TWI450900B (pt) |
| WO (1) | WO2009120720A1 (pt) |
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| RU2544856C2 (ru) | 2008-01-25 | 2015-03-20 | Сергей Олегович Бачурин | НОВЫЕ ПРОИЗВОДНЫЕ 2,3,4,5-ТЕТРАГИДРО-1-ПИРИДО[4,3-b]ИНДОЛА И СПОСОБЫ ИХ ПРИМЕНЕНИЯ |
| AU2009228398B2 (en) | 2008-03-24 | 2014-07-03 | Medivation Technologies, Inc. | Pyrido [3, 4-b] indoles and methods of use |
| AU2009228401B2 (en) | 2008-03-24 | 2014-10-30 | Medivation Technologies, Inc. | Bridged heterocyclic compounds and methods of use |
| PA8843701A1 (es) * | 2008-09-29 | 2010-05-26 | Abbott Lab | Derivados de indolina y métodos para usarlos |
| US9625475B2 (en) | 2008-09-29 | 2017-04-18 | Abbvie Inc. | Indole and indoline derivatives and methods of use thereof |
| AU2009308708B2 (en) | 2008-10-31 | 2015-11-19 | Medivation Technologies, Inc. | Azepino [4, 5-b] indoles and methods of use |
| BRPI0919948A2 (pt) | 2008-10-31 | 2015-08-25 | Madivation Technologies Inc | Pirido[4,3-b]indois contendo porções rígidas |
| KR20110132564A (ko) * | 2009-02-11 | 2011-12-08 | 선오비온 파마슈티컬스 인코포레이티드 | 히스타민 ｈ3 역 작용제 및 길항제, 및 이의 사용 방법 |
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| EP2480081A4 (en) * | 2009-09-23 | 2013-03-06 | Medivation Technologies Inc | Bridged heterocyclic compounds and methods for their use |
| CA2775133A1 (en) | 2009-09-23 | 2011-03-31 | Medivation Technologies, Inc. | Pyrido[3,4-b]indoles and methods of use |
| CN102711468B (zh) * | 2009-09-23 | 2014-07-09 | 梅迪维新技术公司 | 吡啶并[4，3-b]吲哚化合物及其使用方法 |
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-
2009
- 2009-03-24 AU AU2009228401A patent/AU2009228401B2/en not_active Ceased
- 2009-03-24 CN CN200980118777.5A patent/CN102046625B/zh not_active Expired - Fee Related
- 2009-03-24 TW TW098109566A patent/TWI450900B/zh not_active IP Right Cessation
- 2009-03-24 CA CA2718790A patent/CA2718790A1/en not_active Abandoned
- 2009-03-24 US US12/410,425 patent/US8546381B2/en not_active Expired - Fee Related
- 2009-03-24 WO PCT/US2009/038142 patent/WO2009120720A1/en not_active Ceased
- 2009-03-24 JP JP2011501990A patent/JP5586577B2/ja not_active Expired - Fee Related
- 2009-03-24 EP EP09725176.3A patent/EP2274307B1/en not_active Not-in-force
- 2009-03-24 PE PE2009000436A patent/PE20091820A1/es not_active Application Discontinuation
- 2009-03-24 BR BRPI0906245-9A patent/BRPI0906245A2/pt not_active IP Right Cessation
- 2009-03-24 CL CL2009000725A patent/CL2009000725A1/es unknown
- 2009-03-25 AR ARP090101068A patent/AR071284A1/es unknown
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2013
- 2013-03-07 US US13/789,606 patent/US9034869B2/en not_active Expired - Fee Related
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- 2013-09-20 US US14/033,234 patent/US9051314B2/en not_active Expired - Fee Related
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2014
- 2014-03-11 JP JP2014047700A patent/JP2014111655A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| JP5586577B2 (ja) | 2014-09-10 |
| US20130184269A1 (en) | 2013-07-18 |
| EP2274307A1 (en) | 2011-01-19 |
| US8999977B2 (en) | 2015-04-07 |
| US9051314B2 (en) | 2015-06-09 |
| HK1153196A1 (en) | 2012-03-23 |
| CL2009000725A1 (es) | 2009-05-29 |
| JP2014111655A (ja) | 2014-06-19 |
| US9034869B2 (en) | 2015-05-19 |
| HK1157751A1 (en) | 2012-07-06 |
| JP2011515483A (ja) | 2011-05-19 |
| CN102046625A (zh) | 2011-05-04 |
| TWI450900B (zh) | 2014-09-01 |
| PE20091820A1 (es) | 2009-12-10 |
| US20140024643A1 (en) | 2014-01-23 |
| US20130190303A1 (en) | 2013-07-25 |
| TW201000483A (en) | 2010-01-01 |
| US8546381B2 (en) | 2013-10-01 |
| AU2009228401B2 (en) | 2014-10-30 |
| WO2009120720A1 (en) | 2009-10-01 |
| AR071284A1 (es) | 2010-06-09 |
| CA2718790A1 (en) | 2009-10-01 |
| AU2009228401A1 (en) | 2009-10-01 |
| CN102046625B (zh) | 2015-04-08 |
| EP2274307B1 (en) | 2015-07-29 |
| US20100099667A1 (en) | 2010-04-22 |
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