BRPI0907977A2 - Composto, composição farmacêutica, uso de um composto, e, método para tratar ou prevenir doenças - Google Patents

Composto, composição farmacêutica, uso de um composto, e, método para tratar ou prevenir doenças

Info

Publication number: BRPI0907977A2
Authority: BR; Brazil
Prior art keywords: compound; treating; pharmaceutical composition; preventing disease; disease
Prior art date: 2008-03-07

Application number

BRPI0907977-7A

Other languages

English (en)

Inventor

Angelo Guglielmotti

Guido Furlotti

Giorgina Mangano

Nicola Cazzolla

Barbara Garofalo

Original Assignee

Acraf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2008-03-07

Filing date

2009-03-05

Publication date

2015-08-04

2009-03-05 Application filed by Acraf filed Critical Acraf

2015-08-04 Publication of BRPI0907977A2 publication Critical patent/BRPI0907977A2/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/04—Drugs for disorders of the respiratory system for throat disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Diabetes (AREA)
Immunology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pulmonology (AREA)
Oncology (AREA)
Hematology (AREA)
Biomedical Technology (AREA)
Obesity (AREA)
Urology & Nephrology (AREA)
Dermatology (AREA)
Virology (AREA)
Endocrinology (AREA)
Heart & Thoracic Surgery (AREA)
Communicable Diseases (AREA)
Cardiology (AREA)
Rheumatology (AREA)
Vascular Medicine (AREA)
Tropical Medicine & Parasitology (AREA)
Emergency Medicine (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Child & Adolescent Psychology (AREA)
AIDS & HIV (AREA)
Pain & Pain Management (AREA)

BRPI0907977-7A 2008-03-07 2009-03-05 Composto, composição farmacêutica, uso de um composto, e, método para tratar ou prevenir doenças BRPI0907977A2 (pt)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP08425139		2008-03-07
PCT/EP2009/052590 WO2009109618A2 (en)	2008-03-07	2009-03-05	Novel 1-benzyl-3-hydroxymethylindazole derivatives and use thereof in the treatment of diseases based on the expression of mcp-1, cx3cr1 and p40

Publications (1)

Publication Number	Publication Date
BRPI0907977A2 true BRPI0907977A2 (pt)	2015-08-04

Family

ID=39671487

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
BRPI0907976-9A BRPI0907976A2 (pt)	2008-03-07	2009-03-05	Composto, composição farmacêutica, uso de um composto, e, método para tratar ou prevenir doenças
BRPI0907977-7A BRPI0907977A2 (pt)	2008-03-07	2009-03-05	Composto, composição farmacêutica, uso de um composto, e, método para tratar ou prevenir doenças

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
BRPI0907976-9A BRPI0907976A2 (pt)	2008-03-07	2009-03-05	Composto, composição farmacêutica, uso de um composto, e, método para tratar ou prevenir doenças

Country Status (25)

Country	Link
US (3)	US7919518B2 (pt)
EP (3)	EP2254870B1 (pt)
JP (2)	JP5509099B2 (pt)
KR (2)	KR101581828B1 (pt)
CN (2)	CN101945855B (pt)
AR (2)	AR070810A1 (pt)
AU (2)	AU2009221083B2 (pt)
BR (2)	BRPI0907976A2 (pt)
CA (2)	CA2712703C (pt)
CY (2)	CY1117584T1 (pt)
DK (2)	DK2254870T3 (pt)
EA (2)	EA019711B1 (pt)
ES (2)	ES2637009T3 (pt)
GE (2)	GEP20135983B (pt)
HR (2)	HRP20171208T1 (pt)
HU (1)	HUE027098T2 (pt)
IL (3)	IL206893A0 (pt)
LT (1)	LT2254869T (pt)
MX (2)	MX2010009626A (pt)
PL (2)	PL2254870T3 (pt)
PT (1)	PT2254869T (pt)
SG (1)	SG188177A1 (pt)
SI (2)	SI2254870T1 (pt)
UA (2)	UA103605C2 (pt)
WO (2)	WO2009109613A2 (pt)

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KR101581828B1 (ko) *	2008-03-07	2015-12-31	아지엔드 키미쉐 리유나이트 안젤리니 프란체스코 에이.씨.알.에이.에프. 에스.피.에이	신규한 1-벤질-3-하이드록시메틸인다졸 유도체들 및 ｍｃｐ-1, ｃｘ3ｃｒ1 및 ｐ40의 발현을 기초로 한 질환들의 치료에서 이의 용도
EA018976B1 (ru) *	2008-03-07	2013-12-30	Ацьенде Кимике Рьюните Анджелини Франческо А.К.Р.А.Ф. С.П.А.	Производные 1-бензил-3-гидроксиметилиндазола и их применение для лечения заболеваний, основанных на экспрессии мср-1, cx3cr1 и p40
CA2715065C (en)	2008-03-07	2017-06-27	Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A.	Novel 1-benzyl-3-hydroxymethylindazole derivatives and use thereof in the treatment of diseases based on the expression mcp-1 and cx3cr1
GEP20135878B (en)	2009-08-03	2013-07-10	Aziende Chimiche Riunite Angelini Francesco A C R A F S P A It	Method of 1-benzyl-3-hydroxymethyl-1h-indazole preparation, derivatives thereof, and required magnesium intermediates
UA108742C2 (uk) *	2009-09-23	2015-06-10		Фармацевтична композиція для лікування запальних захворювань, опосередкованих mcp-1
US8999292B2 (en) *	2012-05-01	2015-04-07	Translatum Medicus Inc.	Methods for treating and diagnosing blinding eye diseases
WO2013163758A1 (en) *	2012-05-01	2013-11-07	Boyd Shelley Romayne	Methods for treating and diagnosing blinding eye diseases
BR112014028406A2 (pt) *	2012-05-18	2017-06-27	Sanofi Sa	derivados de pirazol e uso dos mesmos como antagonistas de lpar5.
EP2850062B1 (en)	2012-05-18	2017-07-19	Sanofi	Pyridine derivatives and their use in the treatment of conditions associated with pathological thrombus formation
US20140134116A1 (en)	2012-11-09	2014-05-15	Colgate-Palmolive Company	Block Copolymers For Tooth Enamel Protection
EP3142664B1 (en) *	2014-05-15	2019-12-04	Translatum Medicus Inc.	Compositions and methods for treating and diagnosing ocular disorders
EP3942934A1 (en) *	2015-06-12	2022-01-26	Vettore, LLC	Mct4 inhibitors for treating disease
US20180221339A1 (en) *	2015-06-16	2018-08-09	Translatum Medicus, Inc.	Compositions and methods for treating and diagnosing ocular disorders
BR112019011825A2 (pt)	2016-12-12	2019-10-22	Vettore Llc	composto, enantiômero isolado, composição farmacêutica, método para inibir a atividade do transportador de monocarboxilato mct4, ou um mutante do mesmo, em uma amostra biológica, método para inibir a atividade do transportador de monocarboxilato mct4, ou um mutante do mesmo, em relação ao transportador de monocarboxilato mct1, ou um mutante do mesmo, em um paciente, método para tratar um distúrbio mediado por transportador de monocarboxilato mct4 em um sujeito que necessite do mesmo, uso de um composto e método para obter um efeito em um paciente
GB201811169D0 (en)	2018-07-06	2018-08-29	Kancera Ab	New compounds
WO2020026471A1 (ja) *	2018-07-31	2020-02-06	株式会社親広産業	グルコース消費促進剤および解糖系促進剤
JP6612004B1 (ja) *	2018-07-31	2019-11-27	株式会社親広産業	グルコース消費促進剤および解糖系促進剤
WO2020261158A1 (en) *	2019-06-25	2020-12-30	Translatum Medicus Inc.	Processes of making 2-((1-benzyl-1h-indazol-3-yl)methoxy)-2-methylpropanoic acid and its derivatives
CN113929627A (zh) *	2021-10-19	2022-01-14	吕梁学院	一种宾达利的合成方法
WO2024108386A1 (zh) *	2022-11-22	2024-05-30	中国科学院深圳先进技术研究院	抗mcp1中和抗体在制备治疗神经退行性疾病引起的系统性炎症药物中的应用
EP4662203A1 (en) *	2023-02-10	2025-12-17	Translatum Medicus Inc.	Bindarit conjugates, compositions and methods for treating ocular diseases or disorders

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US364371A (en) *		1887-06-07		peice
IT1230441B (it) *	1989-02-07	1991-10-23	Acraf	Eteri della serie dell'indazolo
IT1253703B (it) *	1991-04-22	1995-08-23	Angelini Francesco Ist Ricerca	Uso di acidi metossi alcanoici dell'indazolo per preparare un farmaco attivo nel trattamento di malattie autoimmunitarie
IT1293795B1 (it)	1997-07-28	1999-03-10	Angelini Ricerche Spa	Farmaco attivo nel ridurre la produzione di proteina mcp-1
AU781849C (en)	1999-06-17	2006-03-02	Synta Pharmaceuticals Corp.	Inhibitors of IL-12 production
EP1188438A1 (en)	2000-09-15	2002-03-20	Warner-Lambert Company	Pharmaceutical composition for preventing or treating a disease associated with an excess of Il-12 production
EP1199074A1 (en)	2000-09-15	2002-04-24	Warner-Lambert Company	Pharmaceutical composition for preventing or treating a disease associated with an excess of il-12 production
DE60230388D1 (de)	2001-03-15	2009-01-29	Seikagaku Kogyo Co Ltd	Mittel zur steurung der expression von il-12
CN100349876C (zh)	2001-11-30	2007-11-21	辛塔医药品有限公司	嘧啶化合物
US20070142386A1 (en)	2003-10-07	2007-06-21	Astrazeneca	New 2-substituted, 4-amino-thiazolo[4,5-d] pyrimidines, useful as chemokine receptor antagonists, esp. cx3cr1
ES2641815T3 (es) *	2004-10-29	2017-11-14	Eisai R&D Management Co., Ltd.	Tratamiento para enfermedades inflamatorias
AU2005304393B2 (en)	2004-11-10	2012-09-27	Synta Pharmaceuticals Corp.	IL-12 modulatory compounds
EP1827447A1 (en)	2004-11-19	2007-09-05	Synta Pharmaceuticals Corporation	Pyrimidine compounds and uses thereof
AR053347A1 (es)	2005-04-06	2007-05-02	Astrazeneca Ab	Derivados de [1,3]tiazolo[4,5-d]pirimidin-2(3h)-ona 5,7-sustituidos
UA90707C2 (en)	2005-04-06	2010-05-25	Астразенека Аб	Novel 5-substituted 7-amino-[1,3]thiazolo[4,5-d]pyrimidine derivatives
EA018976B1 (ru)	2008-03-07	2013-12-30	Ацьенде Кимике Рьюните Анджелини Франческо А.К.Р.А.Ф. С.П.А.	Производные 1-бензил-3-гидроксиметилиндазола и их применение для лечения заболеваний, основанных на экспрессии мср-1, cx3cr1 и p40
KR101581828B1 (ko)	2008-03-07	2015-12-31	아지엔드 키미쉐 리유나이트 안젤리니 프란체스코 에이.씨.알.에이.에프. 에스.피.에이	신규한 1-벤질-3-하이드록시메틸인다졸 유도체들 및 ｍｃｐ-1, ｃｘ3ｃｒ1 및 ｐ40의 발현을 기초로 한 질환들의 치료에서 이의 용도
CA2715065C (en)	2008-03-07	2017-06-27	Aziende Chimiche Riunite Angelini Francesco A.C.R.A.F. S.P.A.	Novel 1-benzyl-3-hydroxymethylindazole derivatives and use thereof in the treatment of diseases based on the expression mcp-1 and cx3cr1

2009
- 2009-03-05 KR KR1020107017806A patent/KR101581828B1/ko not_active Expired - Fee Related
- 2009-03-05 EA EA201071040A patent/EA019711B1/ru not_active IP Right Cessation
- 2009-03-05 EP EP09718467.5A patent/EP2254870B1/en active Active
- 2009-03-05 GE GEAP200911963A patent/GEP20135983B/en unknown
- 2009-03-05 HR HRP20171208TT patent/HRP20171208T1/hr unknown
- 2009-03-05 WO PCT/EP2009/052585 patent/WO2009109613A2/en not_active Ceased
- 2009-03-05 SI SI200931404A patent/SI2254870T1/sl unknown
- 2009-03-05 CN CN200980105073.4A patent/CN101945855B/zh not_active Expired - Fee Related
- 2009-03-05 HU HUE09718467A patent/HUE027098T2/en unknown
- 2009-03-05 ES ES09717638.2T patent/ES2637009T3/es active Active
- 2009-03-05 WO PCT/EP2009/052590 patent/WO2009109618A2/en not_active Ceased
- 2009-03-05 EA EA201071038A patent/EA018241B1/ru not_active IP Right Cessation
- 2009-03-05 PL PL09718467T patent/PL2254870T3/pl unknown
- 2009-03-05 EP EP09717638.2A patent/EP2254869B1/en active Active
- 2009-03-05 CN CN200980105556.4A patent/CN101952256B/zh not_active Expired - Fee Related
- 2009-03-05 JP JP2010549143A patent/JP5509099B2/ja active Active
- 2009-03-05 SG SG2013013123A patent/SG188177A1/en unknown
- 2009-03-05 JP JP2010549146A patent/JP5509101B2/ja active Active
- 2009-03-05 MX MX2010009626A patent/MX2010009626A/es active IP Right Grant
- 2009-03-05 DK DK09718467.5T patent/DK2254870T3/en active
- 2009-03-05 EP EP17153930.7A patent/EP3181551A1/en not_active Withdrawn
- 2009-03-05 ES ES09718467.5T patent/ES2569330T3/es active Active
- 2009-03-05 HR HRP20160462TT patent/HRP20160462T1/hr unknown
- 2009-03-05 AU AU2009221083A patent/AU2009221083B2/en not_active Ceased
- 2009-03-05 KR KR1020107017445A patent/KR101599867B1/ko not_active Expired - Fee Related
- 2009-03-05 MX MX2010009623A patent/MX2010009623A/es active IP Right Grant
- 2009-03-05 GE GEAP200911965A patent/GEP20135912B/en unknown
- 2009-03-05 LT LTEP09717638.2T patent/LT2254869T/lt unknown
- 2009-03-05 SI SI200931705T patent/SI2254869T1/sl unknown
- 2009-03-05 CA CA2712703A patent/CA2712703C/en not_active Expired - Fee Related
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- 2009-03-05 DK DK09717638.2T patent/DK2254869T3/en active
- 2009-03-05 US US12/864,767 patent/US7919518B2/en not_active Expired - Fee Related
- 2009-03-05 PT PT97176382T patent/PT2254869T/pt unknown
- 2009-03-05 US US12/865,923 patent/US8835481B2/en not_active Expired - Fee Related
- 2009-03-05 PL PL09717638T patent/PL2254869T3/pl unknown
- 2009-03-06 AR ARP090100800A patent/AR070810A1/es unknown
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- 2009-05-03 UA UAA201008883A patent/UA103605C2/uk unknown
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2010
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- 2010-07-21 IL IL207131A patent/IL207131A/en not_active IP Right Cessation
2011
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Also Published As

Publication number	Publication date
JP2011513367A (ja)	2011-04-28
CY1119252T1 (el)	2018-02-14
LT2254869T (lt)	2017-08-10
PT2254869T (pt)	2017-07-18
DK2254870T3 (en)	2016-05-17
KR101581828B1 (ko)	2015-12-31
CA2712403A1 (en)	2009-09-11
GEP20135983B (en)	2013-12-10
IL215579A (en)	2015-06-30
HRP20160462T1 (hr)	2016-06-03
EA201071038A1 (ru)	2011-02-28
EP2254869A2 (en)	2010-12-01
BRPI0907976A2 (pt)	2015-08-04
EP2254870A2 (en)	2010-12-01
US8283348B2 (en)	2012-10-09
PL2254869T3 (pl)	2017-10-31
SG188177A1 (en)	2013-03-28
WO2009109613A2 (en)	2009-09-11
EP2254869B1 (en)	2017-05-31
EA201071040A1 (ru)	2011-02-28
GEP20135912B (en)	2013-08-26
US20110003874A1 (en)	2011-01-06
CA2712703A1 (en)	2009-09-11
DK2254869T3 (en)	2017-09-04
KR101599867B1 (ko)	2016-03-04
WO2009109618A3 (en)	2009-12-10
EA019711B1 (ru)	2014-05-30
CN101952256A (zh)	2011-01-19
US20110160205A1 (en)	2011-06-30
CN101945855B (zh)	2014-12-17
IL207131A0 (en)	2010-12-30
EP3181551A1 (en)	2017-06-21
HUE027098T2 (en)	2016-08-29
IL215579A0 (en)	2011-11-30
WO2009109618A2 (en)	2009-09-11
AR070810A1 (es)	2010-05-05
HRP20171208T1 (hr)	2017-10-06
SI2254870T1 (sl)	2016-05-31
CN101945855A (zh)	2011-01-12
AU2009221089A1 (en)	2009-09-11
CA2712403C (en)	2017-06-06
AU2009221089B2 (en)	2013-12-05
CA2712703C (en)	2016-10-11
CY1117584T1 (el)	2017-04-26
US20100311744A1 (en)	2010-12-09
IL207131A (en)	2013-02-28
JP5509099B2 (ja)	2014-06-04
AR070811A1 (es)	2010-05-05
ES2637009T3 (es)	2017-10-10
KR20100133957A (ko)	2010-12-22
MX2010009623A (es)	2010-09-28
WO2009109613A3 (en)	2009-12-10
EP2254870B1 (en)	2016-02-24
US7919518B2 (en)	2011-04-05
JP5509101B2 (ja)	2014-06-04
JP2011513365A (ja)	2011-04-28
US8835481B2 (en)	2014-09-16
UA103605C2 (en)	2013-11-11
UA105170C2 (en)	2014-04-25
PL2254870T3 (pl)	2016-07-29
EA018241B1 (ru)	2013-06-28
ES2569330T3 (es)	2016-05-10
SI2254869T1 (sl)	2017-10-30
AU2009221083B2 (en)	2013-11-28
KR20100131432A (ko)	2010-12-15
AU2009221083A1 (en)	2009-09-11
IL206893A0 (en)	2010-12-30
CN101952256B (zh)	2016-03-16
MX2010009626A (es)	2010-12-20

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2019-01-02	B08F	Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]	Free format text: REFERENTE A 10A ANUIDADE.
2019-04-24	B08K	Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]	Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2504 DE 02-01-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.