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BR9609617B1 - derivados de 7h-pirrol[2,3-d]pirimidina, e composição farmacêutica. - Google Patents

derivados de 7h-pirrol[2,3-d]pirimidina, e composição farmacêutica.

Info

Publication number
BR9609617B1
BR9609617B1 BRPI9609617-9A BR9609617A BR9609617B1 BR 9609617 B1 BR9609617 B1 BR 9609617B1 BR 9609617 A BR9609617 A BR 9609617A BR 9609617 B1 BR9609617 B1 BR 9609617B1
Authority
BR
Brazil
Prior art keywords
pct
pyrimidine derivatives
pyrrol
pharmaceutical composition
date jan
Prior art date
Application number
BRPI9609617-9A
Other languages
English (en)
Other versions
BR9609617A (pt
Inventor
Peter Traxler
Guido Bold
Wolfgang Karl-Diether Brill
Joerg Frei
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27508793&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9609617(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of BR9609617A publication Critical patent/BR9609617A/pt
Publication of BR9609617B1 publication Critical patent/BR9609617B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyrrole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Saccharide Compounds (AREA)
BRPI9609617-9A 1995-07-06 1996-06-24 derivados de 7h-pirrol[2,3-d]pirimidina, e composição farmacêutica. BR9609617B1 (pt)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
CH197695 1995-07-06
CH249895 1995-09-01
CH319895 1995-11-10
CH25596 1996-02-01
CH122496 1996-05-13
PCT/EP1996/002728 WO1997002266A1 (en) 1995-07-06 1996-06-24 Pyrrolopyrimidines and processes for the preparation thereof

Publications (2)

Publication Number Publication Date
BR9609617A BR9609617A (pt) 1999-05-25
BR9609617B1 true BR9609617B1 (pt) 2010-07-27

Family

ID=27508793

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9609617-9A BR9609617B1 (pt) 1995-07-06 1996-06-24 derivados de 7h-pirrol[2,3-d]pirimidina, e composição farmacêutica.

Country Status (25)

Country Link
US (1) US6140332A (pt)
EP (1) EP0836605B1 (pt)
JP (1) JP4146514B2 (pt)
KR (1) KR100437582B1 (pt)
CN (1) CN1100778C (pt)
AT (1) ATE212993T1 (pt)
BR (1) BR9609617B1 (pt)
CA (1) CA2224435C (pt)
CY (1) CY2365B1 (pt)
CZ (1) CZ1598A3 (pt)
DE (1) DE69619114T2 (pt)
DK (1) DK0836605T3 (pt)
EA (1) EA001428B1 (pt)
ES (1) ES2172670T3 (pt)
HU (1) HUP9900330A3 (pt)
IL (1) IL122855A (pt)
MX (1) MX9800215A (pt)
NO (1) NO310359B1 (pt)
NZ (1) NZ312665A (pt)
PL (1) PL188959B1 (pt)
PT (1) PT836605E (pt)
SI (1) SI9620103A (pt)
SK (1) SK398A3 (pt)
TR (1) TR199800012T1 (pt)
WO (1) WO1997002266A1 (pt)

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NO975956L (no) 1998-02-10
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CA2224435C (en) 2008-08-05
CY2365B1 (en) 2004-06-04
EA001428B1 (ru) 2001-02-26
CA2224435A1 (en) 1997-01-23
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JP4146514B2 (ja) 2008-09-10
NO310359B1 (no) 2001-06-25
TR199800012T1 (xx) 1998-04-21
IL122855A0 (en) 1998-08-16
CZ1598A3 (cs) 1998-04-15
DE69619114D1 (de) 2002-03-21
CN1194647A (zh) 1998-09-30
HUP9900330A2 (hu) 1999-05-28
BR9609617A (pt) 1999-05-25
US6140332A (en) 2000-10-31
CN1100778C (zh) 2003-02-05
WO1997002266A1 (en) 1997-01-23
KR19990028756A (ko) 1999-04-15
SK398A3 (en) 1998-07-08
HK1008222A1 (en) 1999-05-07
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AU707626B2 (en) 1999-07-15
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ES2172670T3 (es) 2002-10-01
KR100437582B1 (ko) 2004-12-17
AU6414896A (en) 1997-02-05
PT836605E (pt) 2002-07-31
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EP0836605B1 (en) 2002-02-06
ATE212993T1 (de) 2002-02-15
EP0836605A1 (en) 1998-04-22
PL188959B1 (pl) 2005-05-31
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EA199800116A1 (ru) 1998-10-29

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