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ATE340562T1 - Cgmp pde-5 inhibitor enthaltende pharmazeutische formulierungen mit verzögerter freisetzung - Google Patents

Cgmp pde-5 inhibitor enthaltende pharmazeutische formulierungen mit verzögerter freisetzung

Info

Publication number
ATE340562T1
ATE340562T1 AT99946377T AT99946377T ATE340562T1 AT E340562 T1 ATE340562 T1 AT E340562T1 AT 99946377 T AT99946377 T AT 99946377T AT 99946377 T AT99946377 T AT 99946377T AT E340562 T1 ATE340562 T1 AT E340562T1
Authority
AT
Austria
Prior art keywords
inhibitor
pharmaceutical formulations
formulations containing
delayed release
release pharmaceutical
Prior art date
Application number
AT99946377T
Other languages
English (en)
Inventor
Elizabeth King
Ross James Macrae
Original Assignee
Pfizer Ireland Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27269526&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE340562(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9823192.1A external-priority patent/GB9823192D0/en
Priority claimed from GBGB9825117.6A external-priority patent/GB9825117D0/en
Priority claimed from GBGB9826392.4A external-priority patent/GB9826392D0/en
Application filed by Pfizer Ireland Pharmaceuticals filed Critical Pfizer Ireland Pharmaceuticals
Application granted granted Critical
Publication of ATE340562T1 publication Critical patent/ATE340562T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT99946377T 1998-10-23 1999-10-04 Cgmp pde-5 inhibitor enthaltende pharmazeutische formulierungen mit verzögerter freisetzung ATE340562T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9823192.1A GB9823192D0 (en) 1998-10-23 1998-10-23 Pharmaceutical formulations
GBGB9825117.6A GB9825117D0 (en) 1998-11-16 1998-11-16 Pharmaceutical formulations
GBGB9826392.4A GB9826392D0 (en) 1998-11-27 1998-11-27 Pharmaceutical formulations

Publications (1)

Publication Number Publication Date
ATE340562T1 true ATE340562T1 (de) 2006-10-15

Family

ID=27269526

Family Applications (1)

Application Number Title Priority Date Filing Date
AT99946377T ATE340562T1 (de) 1998-10-23 1999-10-04 Cgmp pde-5 inhibitor enthaltende pharmazeutische formulierungen mit verzögerter freisetzung

Country Status (44)

Country Link
US (1) US6964780B1 (de)
EP (1) EP1123088B1 (de)
JP (1) JP2002528408A (de)
KR (1) KR20010075659A (de)
CN (1) CN1324233A (de)
AP (1) AP2001002125A0 (de)
AT (1) ATE340562T1 (de)
AU (1) AU756509B2 (de)
BG (1) BG65323B1 (de)
BR (1) BR9914718A (de)
CA (1) CA2348086C (de)
CO (1) CO5160262A1 (de)
CR (1) CR6326A (de)
CY (1) CY1106239T1 (de)
CZ (1) CZ20011427A3 (de)
DE (1) DE69933383T2 (de)
DK (1) DK1123088T3 (de)
DZ (1) DZ2923A1 (de)
EA (1) EA004068B1 (de)
EE (1) EE200100235A (de)
ES (1) ES2272082T3 (de)
GT (1) GT199900184A (de)
HK (1) HK1041818A1 (de)
HR (1) HRP20010285A2 (de)
HU (1) HUP0104318A3 (de)
ID (1) ID28232A (de)
IL (1) IL141764A (de)
IS (1) IS5865A (de)
MA (1) MA26700A1 (de)
MX (1) MXPA01004011A (de)
MY (1) MY130727A (de)
NO (1) NO20011933L (de)
NZ (1) NZ510275A (de)
OA (1) OA11664A (de)
PA (1) PA8484301A1 (de)
PE (1) PE20001286A1 (de)
PL (1) PL195789B1 (de)
PT (1) PT1123088E (de)
SK (1) SK286473B6 (de)
TR (1) TR200101103T2 (de)
TW (1) TW577756B (de)
UA (1) UA67802C2 (de)
UY (1) UY25765A1 (de)
WO (1) WO2000024383A1 (de)

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CN100518827C (zh) 2000-10-30 2009-07-29 欧罗赛铁克股份有限公司 控释氢可酮制剂
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US10675280B2 (en) 2001-10-20 2020-06-09 Sprout Pharmaceuticals, Inc. Treating sexual desire disorders with flibanserin
UA78974C2 (en) 2001-10-20 2007-05-10 Boehringer Ingelheim Pharma Use of flibanserin for treating disorders of sexual desire
ITMI20020515A1 (it) * 2002-03-12 2003-09-12 Jagotec Ag Sistema per il rilasco controllato di uno o piu' principi attivi
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DE102004023069A1 (de) * 2004-05-11 2005-12-08 Bayer Healthcare Ag Neue Darreichungsformen des PDE 5-Inhibitors Vardenafil
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DE102005001989A1 (de) * 2005-01-15 2006-07-20 Bayer Healthcare Ag Intravenöse Formulierungen von PDE-Inhibitoren
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EP1945214A1 (de) 2005-10-29 2008-07-23 Boehringer Ingelheim International GmbH Benzimidazolon-derivate zur behandlung von prämenstruellen und anderen sexuellen störungen der frau
EP1790343A1 (de) 2005-11-11 2007-05-30 Emotional Brain B.V. Pharmazeutische Zusammensetzungen und deren Verwendung zur Behandlung sexueller Störungen der Frau
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BRPI0716439B8 (pt) 2006-08-14 2021-05-25 Boehringer Ingelheim Int sistemas de liberação farmacêutico compreendendo flibanserina, processo para preparação e uso dos mesmos
JP5220746B2 (ja) 2006-08-25 2013-06-26 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 制御放出システム及びその製造方法
EP1925307A1 (de) * 2006-11-03 2008-05-28 Emotional Brain B.V. Verwendung von 3-alpha-androstanediol zur Behandlung sexueller Dysfunktion
WO2008115797A1 (en) * 2007-03-16 2008-09-25 Pavo, Inc. Therapeutic compositions and methods
CA2689638A1 (en) * 2007-06-13 2008-12-18 Bayer Schering Pharma Aktiengesellschaft Pde inhibitors for the treatment of hearing impairment
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WO2009098697A1 (en) * 2008-02-08 2009-08-13 Dexxon Ltd. Modafinil and sildenafil dosage forms
BRPI0823356A2 (pt) 2008-12-12 2015-06-16 Rhein Siegfried Sa De Cv Composição de liberação pulsátil de sildenafil e processo para prepará-la
KR101004205B1 (ko) * 2008-12-17 2010-12-24 동아제약주식회사 유데나필 함유 서방성 제제를 제조하기 위한 제어방출 조성물
EA015250B9 (ru) * 2010-11-19 2013-10-30 Тева Фармасьютикал Индастриз, Лтд. Таблетка силденафила, обеспечивающая модифицированную фармакокинетику, и способ ее изготовления
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Also Published As

Publication number Publication date
UA67802C2 (uk) 2004-07-15
HUP0104318A3 (en) 2003-12-29
DK1123088T3 (da) 2007-01-02
CO5160262A1 (es) 2002-05-30
EP1123088A1 (de) 2001-08-16
SK286473B6 (sk) 2008-11-06
AU756509B2 (en) 2003-01-16
US6964780B1 (en) 2005-11-15
DZ2923A1 (fr) 2004-03-01
WO2000024383A1 (en) 2000-05-04
TW577756B (en) 2004-03-01
DE69933383T2 (de) 2007-02-01
UY25765A1 (es) 2001-08-27
MY130727A (en) 2007-07-31
MXPA01004011A (es) 2003-03-10
EE200100235A (et) 2002-08-15
EP1123088B1 (de) 2006-09-27
DE69933383D1 (de) 2006-11-09
EA200100298A1 (ru) 2001-08-27
TR200101103T2 (tr) 2001-09-21
CY1106239T1 (el) 2011-06-08
NO20011933L (no) 2001-06-25
CN1324233A (zh) 2001-11-28
GT199900184A (es) 2001-04-14
IL141764A (en) 2008-06-05
NO20011933D0 (no) 2001-04-19
PL347476A1 (en) 2002-04-08
BG105465A (bg) 2001-12-29
IS5865A (is) 2001-02-27
PA8484301A1 (es) 2000-09-29
CA2348086C (en) 2007-01-23
CR6326A (es) 2004-02-23
IL141764A0 (en) 2002-03-10
SK5192001A3 (en) 2002-09-10
CA2348086A1 (en) 2000-05-04
HUP0104318A2 (hu) 2002-03-28
HRP20010285A2 (en) 2002-06-30
HK1041818A1 (zh) 2002-07-26
PE20001286A1 (es) 2000-11-22
ID28232A (id) 2001-05-10
PT1123088E (pt) 2007-01-31
JP2002528408A (ja) 2002-09-03
ES2272082T3 (es) 2007-04-16
AP2001002125A0 (en) 2001-04-04
EA004068B1 (ru) 2003-12-25
KR20010075659A (ko) 2001-08-09
NZ510275A (en) 2003-07-25
BR9914718A (pt) 2001-07-10
AU5878799A (en) 2000-05-15
PL195789B1 (pl) 2007-10-31
CZ20011427A3 (cs) 2001-10-17
MA26700A1 (fr) 2004-12-20
OA11664A (en) 2005-01-07
BG65323B1 (bg) 2008-02-29

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