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AR099567A2 - Formulación de tableta revestida que comprende saxagliptina y método de preparación - Google Patents

Formulación de tableta revestida que comprende saxagliptina y método de preparación

Info

Publication number
AR099567A2
AR099567A2 ARP150100554A ARP150100554A AR099567A2 AR 099567 A2 AR099567 A2 AR 099567A2 AR P150100554 A ARP150100554 A AR P150100554A AR P150100554 A ARP150100554 A AR P150100554A AR 099567 A2 AR099567 A2 AR 099567A2
Authority
AR
Argentina
Prior art keywords
saxagliptine
coating layer
formulation
preparation
covered
Prior art date
Application number
ARP150100554A
Other languages
English (en)
Inventor
V Li Bing
S Desai Divyakant
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34971747&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AR099567(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of AR099567A2 publication Critical patent/AR099567A2/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806—Coating materials
    • A61K9/2833—Organic macromolecular compounds
    • A61K9/284—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Reivindicación 1: Tableta revestida, caracterizada porque comprende un núcleo de tableta y a) una capa de revestimiento de sello interno cubierta en el núcleo de tableta; b) una segunda capa de revestimiento que comprende un medicamento revestido en el sello interno que contiene el núcleo de tableta; y c) opcionalmente una capa de revestimiento protector exterior, cubierta en la segunda capa de revestimiento del núcleo de tableta. Reivindicación 3: Tableta revestida como se define en la reivindicación 1, caracterizada porque el medicamento es saxaglipitina (inhibidor DPP4) de fórmula (1) o una sal del mismo farmacéuticamente aceptable.
ARP150100554A 2004-05-28 2015-02-24 Formulación de tableta revestida que comprende saxagliptina y método de preparación AR099567A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US57531904P 2004-05-28 2004-05-28

Publications (1)

Publication Number Publication Date
AR099567A2 true AR099567A2 (es) 2016-08-03

Family

ID=34971747

Family Applications (2)

Application Number Title Priority Date Filing Date
ARP050102188A AR049062A1 (es) 2004-05-28 2005-05-27 Formulacion de tableta revestida que contiene un inhibidor dpp4, como saxagliptina, y metodo
ARP150100554A AR099567A2 (es) 2004-05-28 2015-02-24 Formulación de tableta revestida que comprende saxagliptina y método de preparación

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ARP050102188A AR049062A1 (es) 2004-05-28 2005-05-27 Formulacion de tableta revestida que contiene un inhibidor dpp4, como saxagliptina, y metodo

Country Status (33)

Country Link
US (4) US7951400B2 (es)
EP (3) EP1753406B2 (es)
JP (1) JP4901727B2 (es)
KR (2) KR101290925B1 (es)
CN (2) CN102895208B (es)
AR (2) AR049062A1 (es)
AU (1) AU2005249467B2 (es)
BR (1) BRPI0510419B8 (es)
CA (1) CA2568391C (es)
CY (2) CY1117813T1 (es)
DK (2) DK2298288T4 (es)
ES (3) ES2593582T5 (es)
GE (1) GEP20094639B (es)
HR (2) HRP20160880T4 (es)
HU (2) HUE029039T2 (es)
IL (2) IL179454A (es)
LT (1) LT2298288T (es)
ME (2) ME02516B (es)
MX (1) MXPA06013711A (es)
MY (1) MY147639A (es)
NO (1) NO343907B1 (es)
NZ (1) NZ551591A (es)
PE (1) PE20060425A1 (es)
PH (1) PH12013500450A1 (es)
PL (2) PL2298288T5 (es)
PT (2) PT1753406E (es)
RS (2) RS54929B2 (es)
RU (1) RU2372894C2 (es)
SI (3) SI1753406T1 (es)
TW (2) TWI415635B (es)
UA (1) UA88168C2 (es)
WO (1) WO2005117841A1 (es)
ZA (1) ZA200609541B (es)

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